Title: Testosterone metabolism of equine single CYPs of the 3A subfamily compared to the human CYP3A4.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20170601
Title: Metabolic-induced cytotoxicity of diosbulbin B in CYP3A4-expressing cells.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20170201
Title: Identification of vitamin D(3) target genes in human breast cancer tissue.
Journal: The Journal of steroid biochemistry and molecular biology 20161101
Title: In vitro evaluation of hepatotoxic drugs in human hepatocytes from multiple donors: Identification of P450 activity as a potential risk factor for drug-induced liver injuries.
Journal: Chemico-biological interactions 20160805
Title: Modulation of 17β-estradiol induced estrogenic responses in male goldfish (Carassius auratus) by benzo[a]pyrene and ketoconazole.
Journal: Environmental science and pollution research international 20160501
Title: Metabolic activation of furan moiety makes Diosbulbin B hepatotoxic.
Journal: Archives of toxicology 20160401
Title: Ketoconazole Stereoisomers Differentially Induce Cytochrome P450 1A1 Between Human Hepatoma HepG2 and Mouse Hepatoma Hepa1c1c7 Cells.
Journal: Journal of pharmaceutical sciences 20160301
Title: Establishment of a mouse model for amiodarone-induced liver injury and analyses of its hepatotoxic mechanism.
Journal: Journal of applied toxicology : JAT 20160101
Title: Changes in plasma concentrations of corticosterone and its precursors after ketoconazole administration in rats: An application of simultaneous measurement of multiple steroids using LC-MS/MS.
Journal: Experimental and toxicologic pathology : official journal of the Gesellschaft fur Toxikologische Pathologie 20160101
Title: Cytotoxicity of luteolin in primary rat hepatocytes: the role of CYP3A-mediated ortho-benzoquinone metabolite formation and glutathione depletion.
Journal: Journal of applied toxicology : JAT 20151101
Title: Ketoconazole induces apoptosis in rat cardiomyocytes through reactive oxygen species-mediated parkin overexpression.
Journal: Archives of toxicology 20151001
Title: Testotoxicosis: Report of Two Cases, One with a Novel Mutation in LHCGR Gene.
Journal: Journal of clinical research in pediatric endocrinology 20150901
Title: Ketoconazole Treatment Decreases the Viability of Immortalized Pituitary Cell Lines Associated with an Increased Expression of Apoptosis-Related Genes and Cell Cycle Inhibitors.
Journal: Journal of neuroendocrinology 20150701
Title: Therapy of endocrine disease: steroidogenesis enzyme inhibitors in Cushing's syndrome.
Journal: European journal of endocrinology 20150601
Title: Demethylation of neferine in human liver microsomes and formation of quinone methide metabolites mediated by CYP3A4 accentuates its cytotoxicity.
Journal: Chemico-biological interactions 20141205
Title: Baboon syndrome induced by ketoconazole.
Journal: Cutaneous and ocular toxicology 20141201
Title: Clinical CYP3A inhibitor alternatives to ketoconazole, clarithromycin and itraconazole, are not transported into the liver by hepatic organic anion transporting polypeptides and organic cation transporter 1.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20141101
Title: Effects of rifampin and ketoconazole on pharmacokinetics of morinidazole in healthy chinese subjects.
Journal: Antimicrobial agents and chemotherapy 20141001
Title: Inhibition of cytochrome P450s enhances (+)-usnic acid cytotoxicity in primary cultured rat hepatocytes.
Journal: Journal of applied toxicology : JAT 20140801
Title: CYP3A4 activity reduces the cytotoxic effects of okadaic acid in HepaRG cells.
Journal: Archives of toxicology 20140801
Title: Studies on the antileishmanial mechanism of action of the arylimidamide DB766: azole interactions and role of CYP5122A1.
Journal: Antimicrobial agents and chemotherapy 20140801
Title: Investigation of a novel series of 2-hydroxyisoquinoline-1,3(2H,4H)-diones as human immunodeficiency virus type 1 integrase inhibitors.
Journal: Journal of medicinal chemistry 20140612
Title: Combination antiretroviral therapy (cART) component ritonavir significantly alters docetaxel exposure.
Journal: Cancer chemotherapy and pharmacology 20140401
Title: In vivo production of novel vitamin D2 hydroxy-derivatives by human placentas, epidermal keratinocytes, Caco-2 colon cells and the adrenal gland.
Journal: Molecular and cellular endocrinology 20140305
Title: Synthesis and biological evaluation of thiazoline derivatives as new antimicrobial and anticancer agents.
Journal: European journal of medicinal chemistry 20140303
Title: Synthesis, antifungal activities and molecular docking studies of novel 2-(2,4-difluorophenyl)-2-hydroxy-3-(1H-1,2,4-triazol-1-yl)propyl dithiocarbamates.
Journal: European journal of medicinal chemistry 20140303
Title: Molecular identification and antifungal susceptibility of yeast isolates causing fungemia collected in a population-based study in Spain in 2010 and 2011.
Journal: Antimicrobial agents and chemotherapy 20140301
Title: Targeted androgen pathway suppression in localized prostate cancer: a pilot study.
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20140120
Title: Human variation and CYP enzyme contribution in benfuracarb metabolism in human in vitro hepatic models.
Journal: Toxicology letters 20140113
Title: Synthesis and biological evaluation of novel N-substituted 1H-dibenzo[a,c]carbazole derivatives of dehydroabietic acid as potential antimicrobial agents.
Journal: Bioorganic & medicinal chemistry letters 20140101
Title: Vitamin D up-regulates the vitamin D receptor by protecting it from proteasomal degradation in human CD4+ T cells.
Journal: PloS one 20140101
Title: Enantiospecific effects of ketoconazole on aryl hydrocarbon receptor.
Journal: PloS one 20140101
Title: Dual effects of ketoconazole cis-enantiomers on CYP3A4 in human hepatocytes and HepG2 Cells.
Journal: PloS one 20140101
Title: Capsaicin pretreatment increased the bioavailability of cyclosporin in rats: involvement of P-glycoprotein and CYP 3A inhibition.
Journal: Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association 20131201
Title: Hytramycins V and I, anti-Mycobacterium tuberculosis hexapeptides from a Streptomyces hygroscopicus strain.
Journal: Journal of natural products 20131122
Title: 3-Aryl-4-acyloxyethoxyfuran-2(5H)-ones as inhibitors of tyrosyl-tRNA synthetase: synthesis, molecular docking and antibacterial evaluation.
Journal: Bioorganic & medicinal chemistry 20130901
Title: Synthesis, in vitro antifungal activity and in silico study of 3-(1,2,4-triazol-1-yl)flavanones.
Journal: European journal of medicinal chemistry 20130801
Title: Interaction of 17β-estradiol and ketoconazole on endocrine function in goldfish (Carassius auratus).
Journal: Aquatic toxicology (Amsterdam, Netherlands) 20130515
Title: Novel yeast-based strategy unveils antagonist binding regions on the nuclear xenobiotic receptor PXR.
Journal: The Journal of biological chemistry 20130510
Title: Effect of ketoconazole on the pharmacokinetics of the 11β-hydroxysteroid dehydrogenase type 1 inhibitor ABT-384 and its two active metabolites in healthy volunteers: population analysis of data from a drug-drug interaction study.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20130501
Title: Synthesis and evaluation of non-dimeric HCV NS5A inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20130401
Title: Coordinated roles of pregnane X receptor and constitutive androstane receptor in autoinduction of voriconazole metabolism in mice.
Journal: Antimicrobial agents and chemotherapy 20130301
Title: Transport inhibition of digoxin using several common P-gp expressing cell lines is not necessarily reporting only on inhibitor binding to P-gp.
Journal: PloS one 20130101
Title: Fluconazole inhibits human adrenocortical steroidogenesis in vitro.
Journal: The Journal of endocrinology 20121201
Title: Inhibition of CYP3A4 by 6',7'-dihydroxybergamottin in human CYP3A4 over-expressed hepG2 cells.
Journal: The Journal of pharmacy and pharmacology 20121201
Title: Binding processes determine the stereoselective intestinal and hepatic extraction of verapamil in vivo.
Journal: Molecular pharmaceutics 20121105
Title: A reappraisal of the medical therapy with steroidogenesis inhibitors in Cushing's syndrome.
Journal: Clinical endocrinology 20121101
Title: Catecholaminergic signalling through thymic nerve fibres, thymocytes and stromal cells is dependent on both circulating and locally synthesized glucocorticoids.
Journal: Experimental physiology 20121101
Title: Impact of nonlinear midazolam pharmacokinetics on the magnitude of the midazolam-ketoconazole interaction in rats.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20121101
Title: Assessment of the drug interaction risk for remogliflozin etabonate, a sodium-dependent glucose cotransporter-2 inhibitor: evidence from in vitro, human mass balance, and ketoconazole interaction studies.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20121101
Title: Synthesis and antifungal activity of diverse C-2 pyridinyl and pyridinylvinyl substituted quinolines.
Journal: Bioorganic & medicinal chemistry 20121101
Title: Synthesis, characterization and biological evaluation of some novel 2,4-thiazolidinediones as potential cytotoxic, antimicrobial and antihyperglycemic agents.
Journal: Bioorganic & medicinal chemistry letters 20121015
Title: Structure-activity relationship study of nitrosopyrimidines acting as antifungal agents.
Journal: Bioorganic & medicinal chemistry 20121015
Title: Evaluation of the effects of rifampicin, ketoconazole and erythromycin on the steady-state pharmacokinetics of the components of a novel oral contraceptive containing estradiol valerate and dienogest in healthy postmenopausal women.
Journal: Contraception 20121001
Title: Human aldosterone synthase: recombinant expression in E. coli and purification enables a detailed biochemical analysis of the protein on the molecular level.
Journal: The Journal of steroid biochemistry and molecular biology 20121001
Title: Course of pregnancies in women with Cushing's disease treated by gamma-knife.
Journal: Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology 20121001
Title: The effects on metabolic clearance when administering a potent CYP3A autoinducer with the prototypic CYP3A inhibitor, ketoconazole.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20121001
Title: Prototheca wickerhamii as a cause of neuroinfection in a child with congenital hydrocephalus. First case of human protothecosis in Poland.
Journal: Diagnostic microbiology and infectious disease 20121001
Title: Mouse precision-cut liver slices as an ex vivo model to study idiosyncratic drug-induced liver injury.
Journal: Chemical research in toxicology 20120917
Title: Identification of priority pharmaceuticals in the water environment of China.
Journal: Chemosphere 20120901
Title: Discovery of a highly selective CYP3A4 inhibitor suitable for reaction phenotyping studies and differentiation of CYP3A4 and CYP3A5.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20120901
Title: Studies on the mechanisms of superagonistic pro-differentiating activities of side-chain modified analogs of vitamin D2.
Journal: Oncology reports 20120901
Title: Involvement of the neurosteroid 7α-hydroxypregnenolone in the courtship behavior of the male newt Cynops pyrrhogaster.
Journal: Hormones and behavior 20120901
Title: Laurene-type sesquiterpenes from the Red Sea red alga Laurencia obtusa as potential antitumor-antimicrobial agents.
Journal: European journal of medicinal chemistry 20120901
Title: Effect of ketoconazole on the pharmacokinetic profile of buprenorphine following administration of a once-weekly buprenorphine transdermal system.
Journal: Clinical drug investigation 20120901
Title: Phase I studies of sirolimus alone or in combination with pharmacokinetic modulators in advanced cancer patients.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20120901
Title: Ascending single-dose study of the safety profile, tolerability, and pharmacokinetics of bosutinib coadministered with ketoconazole to healthy adult subjects.
Journal: Clinical therapeutics 20120901
Title: The prognostic factors of effective ketoconazole treatment for metastatic castration-resistant prostate cancer: who can benefit from ketoconazole therapy?
Journal: Asian journal of andrology 20120901
Title: Isolated Cushing's syndrome in early infancy due to left adrenal adenoma: an unusual aetiology.
Journal: Journal of clinical research in pediatric endocrinology 20120901
Title: Differentiating mucosal and hepatic metabolism of budesonide by local pretreatment with increasing doses of ketoconazole in the proximal jejunum.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20120815
Title: Evaluation of saliva flow rates, Candida colonization and susceptibility of Candida strains after head and neck radiation.
Journal: Clinical oral investigations 20120801
Title: A randomized, crossover, placebo- and moxifloxacin-controlled study to evaluate the effects of bosutinib (SKI-606), a dual Src/Abl tyrosine kinase inhibitor, on cardiac repolarization in healthy adult subjects.
Journal: International journal of cancer 20120801
Title: In vitro activities of antifungal agents against clinical isolates of dermatophytes from animals.
Journal: The Journal of veterinary medical science 20120801
Title: Drug-drug interactions and cooperative effects detected in electrochemically driven human cytochrome P450 3A4.
Journal: Bioelectrochemistry (Amsterdam, Netherlands) 20120801
Title: Synthesis, antimicrobial and cytotoxic activities of sulfone linked bis heterocycles.
Journal: European journal of medicinal chemistry 20120801
Title: Synthesis and evaluation of novel potent HCV NS5A inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20120715
Title: Influence of Pluronic 85 and ketoconazole on disposition and efficacy of ivermectin in sheep infected with a multiple resistant Haemonchus contortus isolate.
Journal: Veterinary parasitology 20120706
Title: Synthesis of benzimidazolyl-1,3,4-oxadiazol-2ylthio-N-phenyl (benzothiazolyl) acetamides as antibacterial, antifungal and antituberculosis agents.
Journal: European journal of medicinal chemistry 20120701
Title: The fatty acid 8,11-diol synthase of Aspergillus fumigatus is inhibited by imidazole derivatives and unrelated to PpoB.
Journal: Lipids 20120701
Title: Bioactive briarane diterpenoids from the South China Sea gorgonian Dichotella gemmacea.
Journal: Bioorganic & medicinal chemistry letters 20120701
Title: CDR4 is the major contributor to azole resistance among four Pdr5p-like ABC transporters in Neurospora crassa.
Journal: Fungal biology 20120701
Title: Identification, synthesis, and biological evaluation of the metabolites of 3-amino-6-(3'-aminopropyl)-5H-indeno[1,2-c]isoquinoline-5,11-(6H)dione (AM6-36), a promising rexinoid lead compound for the development of cancer chemotherapeutic and chemopreventive agents.
Journal: Journal of medicinal chemistry 20120628
Title: Cytochrome P450 3A4 inhibition by ketoconazole: tackling the problem of ligand cooperativity using molecular dynamics simulations and free-energy calculations.
Journal: Journal of chemical information and modeling 20120625
Title: A time-course analysis of effects of the steroidogenesis inhibitor ketoconazole on components of the hypothalamic-pituitary-gonadal axis of fathead minnows.
Journal: Aquatic toxicology (Amsterdam, Netherlands) 20120615
Title: CYP3A-mediated apoptosis of dauricine in cultured human bronchial epithelial cells and in lungs of CD-1 mice.
Journal: Toxicology and applied pharmacology 20120615
Title: The effect of CYP3A4 inhibition or induction on the pharmacokinetics and pharmacodynamics of orally administered ruxolitinib (INCB018424 phosphate) in healthy volunteers.
Journal: Journal of clinical pharmacology 20120601
Title: Lack of significant effect of bilastine administered at therapeutic and supratherapeutic doses and concomitantly with ketoconazole on ventricular repolarization: results of a thorough QT study (TQTS) with QT-concentration analysis.
Journal: Journal of clinical pharmacology 20120601
Title: Tolbutamide hydroxylation by hepatic microsomes from Atlantic salmon (Salmo salar L.).
Journal: Molecular biology reports 20120601
Title: Design and synthesis of new 4-pyrazolin-3-yl-1,2,3-triazoles and 1,2,3-triazol-4-yl-pyrazolin-1-ylthiazoles as potential antimicrobial agents.
Journal: European journal of medicinal chemistry 20120601
Title: Distribution, behavior and fate of azole antifungals during mechanical, biological, and chemical treatments in sewage treatment plants in China.
Journal: The Science of the total environment 20120601
Title: Apparent triclabendazole-resistant human Fasciola hepatica infection, the Netherlands.
Journal: Emerging infectious diseases 20120601
Title: Influence of P-glycoprotein modulation on plasma concentrations and pharmacokinetics of orally administered prednisolone in dogs.
Journal: American journal of veterinary research 20120601
Title: Fluconazole exposure rather than clonal spreading is correlated with the emergence of Candida glabrata with cross-resistance to triazole antifungal agents.
Journal: The Kaohsiung journal of medical sciences 20120601
Title: Implication of free cholesterol in LC-MS response enhancement.
Journal: Bioanalysis 20120601
Title: Therapeutic effectiveness of Ageratina pichinchensis on the treatment of chronic interdigital tinea pedis: a randomized, double-blind clinical trial.
Journal: Journal of alternative and complementary medicine (New York, N.Y.) 20120601
Title: Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
Journal: Journal of medicinal chemistry 20120524
Title: Effects of ketoconazole and valproic acid on the pharmacokinetics of the next generation NNRTI, lersivirine (UK-453,061), in healthy adult subjects.
Journal: British journal of clinical pharmacology 20120501
Title: Drug-drug interactions between ketoconazole and berberine in rats: pharmacokinetic effects benefit pharmacodynamic synergism.
Journal: Phytotherapy research : PTR 20120501
Title: The effect of multiple doses of rifampin and ketoconazole on the single-dose pharmacokinetics of ridaforolimus.
Journal: Cancer chemotherapy and pharmacology 20120501
Title: Human testis steroidogenesis is inhibited by phthalates.
Journal: Human reproduction (Oxford, England) 20120501
Title: Synthesis of novel spirooxindole derivatives by one pot multicomponent reaction and their antimicrobial activity.
Journal: European journal of medicinal chemistry 20120501
Title: Preclinical metabolism of LB42908, a novel farnesyl transferase inhibitor, and its effects on the cytochrome P450 isozyme activities.
Journal: Bioorganic & medicinal chemistry letters 20120501
Title: The stepwise selection for ketoconazole resistance induces upregulation of C14-demethylase (CYP51) in Leishmania amazonensis.
Journal: Memorias do Instituto Oswaldo Cruz 20120501
Title: Stereoselective metabolism of tetrahydropalmatine enantiomers in rat liver microsomes.
Journal: Chirality 20120501
Title: Effects of ketoconazole and rifampicin on the pharmacokinetics of gemigliptin, a dipeptidyl peptidase-IV inhibitor: a crossover drug-drug interaction study in healthy male Korean volunteers.
Journal: Clinical therapeutics 20120501
Title: Hydrogel of ketoconazole and PAMAM dendrimers: formulation and antifungal activity.
Journal: Molecules (Basel, Switzerland) 20120418
Title: New triazole derivatives as antifungal agents: synthesis via click reaction, in vitro evaluation and molecular docking studies.
Journal: Bioorganic & medicinal chemistry letters 20120415
Title: Development of a new class of aromatase inhibitors: design, synthesis and inhibitory activity of 3-phenylchroman-4-one (isoflavanone) derivatives.
Journal: Bioorganic & medicinal chemistry 20120415
Title: Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal: Journal of medicinal chemistry 20120412
Title: Effect of cytochrome P450 3A4 inhibitor ketoconazole on risperidone pharmacokinetics in healthy volunteers.
Journal: Journal of clinical pharmacy and therapeutics 20120401
Title: Involvement of P-glycoprotein and cytochrome P450 3A in the metabolism of florfenicol of rabbits.
Journal: Journal of veterinary pharmacology and therapeutics 20120401
Title: Effects of CYP3A4 inhibition and induction on the pharmacokinetics and pharmacodynamics of tolvaptan, a non-peptide AVP antagonist in healthy subjects.
Journal: British journal of clinical pharmacology 20120401
Title: Iatrogenic heart block during treatment of a patient with Cushing's syndrome: report of a case.
Journal: Endocrine 20120401
Title: Orteronel (TAK-700), a novel non-steroidal 17,20-lyase inhibitor: effects on steroid synthesis in human and monkey adrenal cells and serum steroid levels in cynomolgus monkeys.
Journal: The Journal of steroid biochemistry and molecular biology 20120401
Title: The hypercoagulable state in Cushing's disease is associated with increased levels of procoagulant factors and impaired fibrinolysis, but is not reversible after short-term biochemical remission induced by medical therapy.
Journal: The Journal of clinical endocrinology and metabolism 20120401
Title: Predicting drug candidate victims of drug-drug interactions, using microdosing.
Journal: Clinical pharmacokinetics 20120401
Title: Increasing evidence for and regulation of a human placental endogenous digitalis-like factor.
Journal: Reproductive sciences (Thousand Oaks, Calif.) 20120401
Title: Regioselective synthesis and antimicrobial activities of some novel aryloxyacetic acid derivatives.
Journal: European journal of medicinal chemistry 20120401
Title: Comparison of three fluorescent CYP3A substrates in two vertebrate models: pig and Atlantic salmon.
Journal: Animal : an international journal of animal bioscience 20120401
Title: In vitro antifungal susceptibility of Malassezia pachydermatis from dogs with and without skin lesions.
Journal: Veterinary microbiology 20120323
Title: Contemporary experience with ketoconazole in patients with metastatic castration-resistant prostate cancer: clinical factors associated with PSA response and disease progression.
Journal: The Prostate 20120301
Title: Pharmacokinetic interaction between domperidone and ketoconazole leads to QT prolongation in healthy volunteers: a randomized, placebo-controlled, double-blind, crossover study.
Journal: British journal of clinical pharmacology 20120301
Title: H295R cells as a model for steroidogenic disruption: a broader perspective using simultaneous chemical analysis of 7 key steroid hormones.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20120301
Title: Hypercalcemia, hypercalciuria, and elevated calcitriol concentrations with autosomal dominant transmission due to CYP24A1 mutations: effects of ketoconazole therapy.
Journal: The Journal of clinical endocrinology and metabolism 20120301
Title: Take another CYP: confirming a novel mechanism for 'idiopathic' hypercalcemia.
Journal: The Journal of clinical endocrinology and metabolism 20120301
Title: An Aruban man with fever, abdominal mass and eosinophilia.
Journal: The Netherlands journal of medicine 20120301
Title: Potentiation of triclabendazole action in vivo against a triclabendazole-resistant isolate of Fasciola hepatica following its co-administration with the metabolic inhibitor, ketoconazole.
Journal: Veterinary parasitology 20120227
Title: Tocol modified glycol chitosan for the oral delivery of poorly soluble drugs.
Journal: International journal of pharmaceutics 20120227
Title: [Efficacy of low dose ketoconazole therapy for Chinese patients with castration resistant prostate cancer].
Journal: Zhonghua yi xue za zhi 20120227
Title: Synthesis of novel brassinosteroid biosynthesis inhibitors based on the ketoconazole scaffold.
Journal: Bioorganic & medicinal chemistry letters 20120215
Title: Synthesis of novel sulfonamide-1,2,4-triazoles, 1,3,4-thiadiazoles and 1,3,4-oxadiazoles, as potential antibacterial and antifungal agents. Biological evaluation and conformational analysis studies.
Journal: Bioorganic & medicinal chemistry 20120215
Title: Effect of ketoconazole on the pharmacokinetics of axitinib in healthy volunteers.
Journal: Investigational new drugs 20120201
Title: Malformation spectrum induced by ketoconazole after single administration to pregnant rats during the critical period - comparison with vitamin A-induced malformation spectrum.
Journal: Journal of applied toxicology : JAT 20120201
Title: Enhancement of β-carotene production by over-expression of HMG-CoA reductase coupled with addition of ergosterol biosynthesis inhibitors in recombinant Saccharomyces cerevisiae.
Journal: Current microbiology 20120201
Title: Synthesis and biological evaluation of some thiazolidinones as antimicrobial agents.
Journal: European journal of medicinal chemistry 20120201
Title: Ketoconazole-associated preferential increase in dopamine D2 receptor occupancy in striatum compared to pituitary in vivo: role for drug transporters?
Journal: Journal of clinical psychopharmacology 20120201
Title: Effects of efonidipine on the pharmacokinetics and pharmacodynamics of repaglinide: possible role of CYP3A4 and P-glycoprotein inhibition by efonidipine.
Journal: Journal of pharmacokinetics and pharmacodynamics 20120201
Title: [Blastomycosis in Morocco: imported mycosis].
Journal: Revue de pneumologie clinique 20120201
Title: Advances in medical therapies for Cushing's syndrome.
Journal: Discovery medicine 20120201
Title: [Transport of limonin in rat intestine in situ and Caco-2 cells in vitro].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20120201
Title: Tinea versicolor: understanding effective treatment options.
Journal: The Nurse practitioner 20120119
Title: Synthesis, characterization and in vitro biological evaluation of some novel diarylsulfonylureas as potential cytotoxic and antimicrobial agents.
Journal: Bioorganic & medicinal chemistry letters 20120115
Title: Radiation port dermatophytosis: tinea corporis occurring at the site of irradiated skin.
Journal: Dermatology online journal 20120115
Title: Determination of metabolic profile of anti-malarial trioxane CDRI 99/411 in rat liver microsomes using HPLC.
Journal: Biomedical chromatography : BMC 20120101
Title: Identification of ketoconazole as an AhR-Nrf2 activator in cultured human keratinocytes: the basis of its anti-inflammatory effect.
Journal: The Journal of investigative dermatology 20120101
Title: Application of PBPK modelling in drug discovery and development at Pfizer.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20120101
Title: Ultrasound-enhanced surfactant-assisted dispersive liquid-liquid microextraction and high-performance liquid chromatography for determination of ketoconazole and econazole nitrate in human blood.
Journal: Analytical and bioanalytical chemistry 20120101
Title: Discovery of a novel class of aldol-derived 1,2,3-triazoles: potent and selective inhibitors of human cytochrome P450 19A1 (aromatase).
Journal: Bioorganic & medicinal chemistry letters 20120101
Title: Antifungal activities of novel non-azole molecules against S. cerevisiae and C. albicans.
Journal: European journal of medicinal chemistry 20120101
Title: Synthesis, antimicrobial, antimycobacterial and structure-activity relationship of substituted pyrazolo-, isoxazolo-, pyrimido- and mercaptopyrimidocyclohepta[b]indoles.
Journal: European journal of medicinal chemistry 20120101
Title: Isoxazoles incorporated N-substituted decahydroquinolines: a precursor to the next generation antimicrobial drug.
Journal: European journal of medicinal chemistry 20120101
Title: The AhR-Nrf2 pathway in keratinocytes: on the road to chemoprevention?
Journal: The Journal of investigative dermatology 20120101
Title: Lack of drug interaction between the migraine drug MAP0004 (orally inhaled dihydroergotamine) and a CYP3A4 inhibitor in humans.
Journal: Cephalalgia : an international journal of headache 20120101
Title: Comparison of the effect of non-antifungal and antifungal agents on Candida isolates from the gastrointestinal tract.
Journal: Archives of Iranian medicine 20120101
Title: Efficacy and safety of venous thromboembolism prophylaxis with apixaban in major orthopedic surgery.
Journal: Therapeutics and clinical risk management 20120101
Title: Roles of adapalene in the treatment of pityriasis versicolor.
Journal: Dermatology (Basel, Switzerland) 20120101
Title: The effect of ketoconazole on post-burn inflammation, hypermetabolism and clinical outcomes.
Journal: PloS one 20120101
Title: Disappearance of pituitary macro adenoma with combination of ketoconazole and cabergoline treatment: an unusual case of Cushing's syndrome with interesting findings.
Journal: BMJ case reports 20120101
Title: Stimulation of human monocytic THP-1 cells by metabolic activation of hepatotoxic drugs.
Journal: Drug metabolism and pharmacokinetics 20120101
Title: Retigeric acid B enhances the efficacy of azoles combating the virulence and biofilm formation of Candida albicans.
Journal: Biological & pharmaceutical bulletin 20120101
Title: Comparison between two culture media for in vitro evaluation of antifungal susceptibility of the Sporothrix schenckii complex.
Journal: Anais brasileiros de dermatologia 20120101
Title: Telaprevir: pharmacokinetics and drug interactions.
Journal: Antiviral therapy 20120101
Title: Blockade of K+ and Ca2+ channels by azole antifungal agents in neonatal rat ventricular myocytes.
Journal: Biological & pharmaceutical bulletin 20120101
Title: The cytochrome P450 inhibitor, ketoconazole, inhibits oxidized linoleic acid metabolite-mediated peripheral inflammatory pain.
Journal: Molecular pain 20120101
Title: Synthesis and antileishmanial evaluation of 1-aryl-4-(4,5-dihydro-1H-imidazol-2-yl)-1H-pyrazole derivatives.
Journal: Bioorganic & medicinal chemistry letters 20111215
Title: A new antifungal briarane diterpenoid from the gorgonian Junceella juncea Pallas.
Journal: Bioorganic & medicinal chemistry letters 20111215
Title: Novel (E)-1-(4-methyl-2-(alkylamino)thiazol-5-yl)-3-arylprop-2-en-1-ones as potent antimicrobial agents.
Journal: Bioorganic & medicinal chemistry 20111215
Title: Effect of ketoconazole on the pharmacokinetics of oral bosutinib in healthy subjects.
Journal: Journal of clinical pharmacology 20111201
Title: Precipitation in and supersaturation of contents of the upper small intestine after administration of two weak bases to fasted adults.
Journal: Pharmaceutical research 20111201
Title: Cytotoxicity of 3-(3,5-dichlorophenyl)-2,4-thiazolidinedione (DCPT) and analogues in wild type and CYP3A4 stably transfected HepG2 cells.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20111201
Title: Translating clinical findings into knowledge in drug safety evaluation--drug induced liver injury prediction system (DILIps).
Journal: PLoS computational biology 20111201
Title: Effect of different durations and formulations of diltiazem on the single-dose pharmacokinetics of midazolam: how long do we go?
Journal: Journal of clinical pharmacology 20111101
Title: Effect of hyperlipidemia on ketoconazole-midazolam drug-drug interaction in rat.
Journal: Journal of pharmaceutical sciences 20111101
Title: A random comparative study of terbinafine versus griseofulvin in patients with tinea capitis in Western China.
Journal: Mycopathologia 20111101
Title: Antifungal susceptibility and virulence attributes of bloodstream isolates of Candida from Hong Kong and Finland.
Journal: Mycopathologia 20111101
Title: Synthesis and antimicrobial activity of amido linked pyrrolyl and pyrazolyl-oxazoles, thiazoles and imidazoles.
Journal: European journal of medicinal chemistry 20111101
Title: Synthesis and biological evaluation of some novel triazol-3-ones as antimicrobial agents.
Journal: Bioorganic & medicinal chemistry letters 20111101
Title: Synthesis and anticandidal activity of new triazolothiadiazine derivatives.
Journal: European journal of medicinal chemistry 20111101
Title: The influence of modulation of P-glycoprotein and /or cytochrome P450 3A on the pharmacokinetics and pharmacodynamics of orally administered morphine in dogs.
Journal: Journal of veterinary pharmacology and therapeutics 20111001
Title: Exploring the possible metabolism mediated interaction of Glycyrrhiza glabra extract with CYP3A4 and CYP2D6.
Journal: Phytotherapy research : PTR 20111001
Title: Inhibition of triclabendazole metabolism in vitro by ketoconazole increases disruption to the tegument of a triclabendazole-resistant isolate of Fasciola hepatica.
Journal: Parasitology research 20111001
Title: Overt immune dysfunction after Cushing's syndrome remission: a consecutive case series and review of the literature.
Journal: The Journal of clinical endocrinology and metabolism 20111001
Title: Tyrosyl-tRNA synthetase inhibitors as antibacterial agents: synthesis, molecular docking and structure-activity relationship analysis of 3-aryl-4-arylaminofuran-2(5H)-ones.
Journal: European journal of medicinal chemistry 20111001
Title: Enantioselective capillary electrophoresis for the assessment of CYP3A4-mediated ketamine demethylation and inhibition in vitro.
Journal: Electrophoresis 20111001
Title: Effects of CYP inhibitors on precocene I metabolism and toxicity in rat liver slices.
Journal: Chemico-biological interactions 20110905
Title: Therapeutic efficacy of topical OLEOZON® in patients suffering from onychomycosis.
Journal: Mycoses 20110901
Title: Successful outcome of pregnancy in a patient with Cushing's disease under treatment with ketoconazole during the first trimester of gestation.
Journal: Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology 20110901
Title: Investigating the effect of moisture protection on solid-state stability and dissolution of fenofibrate and ketoconazole solid dispersions using PXRD, HSDSC and Raman microscopy.
Journal: Drug development and industrial pharmacy 20110901
Title: Arachidonic acid products in airway nociceptor activation during acute lung injury.
Journal: Experimental physiology 20110901
Title: Molecular complexes of ketaconazole and oxatomide with p-chloranil: spectroscopic and spectrofluorimetric studies.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20110901
Title: Design, synthesis and antimicrobial activity of chiral 2-(substituted-hydroxyl)-3-(benzo[d]oxazol-5-yl)propanoic acid derivatives.
Journal: European journal of medicinal chemistry 20110901
Title: A novel biotransformation of alkyl aminopyrrolidine to aminopiperidine ring by human CYP3A.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20110901
Title: Effect of ketoconazole-mediated CYP3A4 inhibition on clinical pharmacokinetics of panobinostat (LBH589), an orally active histone deacetylase inhibitor.
Journal: Cancer chemotherapy and pharmacology 20110901
Title: Mitotane, metyrapone, and ketoconazole combination therapy as an alternative to rescue adrenalectomy for severe ACTH-dependent Cushing's syndrome.
Journal: The Journal of clinical endocrinology and metabolism 20110901
Title: A phase II clinical trial of neoadjuvant ketoconazole and docetaxel chemotherapy before radical prostatectomy in high risk patients.
Journal: The Journal of urology 20110901
Title: Editorial comment.
Journal: The Journal of urology 20110901
Title: Synthesis and studies of novel 2-(4-cyano-3-trifluoromethylphenyl amino)-4-(quinoline-4-yloxy)-6-(piperazinyl/piperidinyl)-s-triazines as potential antimicrobial, antimycobacterial and anticancer agents.
Journal: European journal of medicinal chemistry 20110901
Title: Pulmonary histoplasmosis presenting with the reversed halo sign on high-resolution CT scan.
Journal: Chest 20110901
Title: In vitro susceptibility of fluconazole-susceptible and -resistant isolates of Malassezia pachydermatis against azoles.
Journal: Veterinary microbiology 20110826
Title: Cytotoxic bipyridines from the marine-derived actinomycete Actinoalloteichus cyanogriseus WH1-2216-6.
Journal: Journal of natural products 20110826
Title: Hydroxylation of DHEA, androstenediol and epiandrosterone by Mortierella isabellina AM212. Evidence indicating that both constitutive and inducible hydroxylases catalyze 7α- as well as 7β-hydroxylations of 5-ene substrates.
Journal: Organic & biomolecular chemistry 20110807
Title: The effect of vitamin D3 and ketoconazole combination on VDR-mediated P-gp expression and function in human colon adenocarcinoma cells: implications in drug disposition and resistance.
Journal: Basic & clinical pharmacology & toxicology 20110801
Title: Effects of strong CYP2D6 and 3A4 inhibitors, paroxetine and ketoconazole, on the pharmacokinetics and cardiovascular safety of tamsulosin.
Journal: British journal of clinical pharmacology 20110801
Title: Substrate specificity and ligand interactions of CYP26A1, the human liver retinoic acid hydroxylase.
Journal: Molecular pharmacology 20110801
Title: Hepatic cytochrome P450s attenuate the cytotoxicity induced by leflunomide and its active metabolite A77 1726 in primary cultured rat hepatocytes.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20110801
Title: Synthesis and antimicrobial evaluation of new benzofuran derivatives.
Journal: European journal of medicinal chemistry 20110801
Title: The pharmacological inhibition of sterol biosynthesis in Leishmania is counteracted by enhancement of LDL endocytosis.
Journal: Acta tropica 20110801
Title: Improved treatment of visceral leishmaniasis (kala-azar) by using combination of ketoconazole, miltefosine with an immunomodulator-Picroliv.
Journal: Acta tropica 20110801
Title: Higher throughput human hepatocyte assays for the evaluation of time-dependent inhibition of CYP3A4.
Journal: Drug metabolism letters 20110801
Title: Auto-inhibition of verapamil metabolism in rat hepatocytes of gel entrapment culture.
Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie 20110801
Title: Bioactive 11,20-epoxy-3,5(16)-diene briarane diterpenoids from the South China Sea gorgonian Dichotella gemmacea.
Journal: Journal of natural products 20110722
Title: Spanlastics--a novel nanovesicular carrier system for ocular delivery.
Journal: International journal of pharmaceutics 20110715
Title: Bioavailability considerations in evaluating drug-drug interactions using the population pharmacokinetic approach.
Journal: Journal of clinical pharmacology 20110701
Title: Low dose of ketoconazole in patients with prostate adenocarcinoma resistant to pharmacological castration.
Journal: BJU international 20110701
Title: Nanoparticle formation and growth during in vitro dissolution of ketoconazole solid dispersion.
Journal: Journal of pharmaceutical sciences 20110701
Title: Fenretinide metabolism in humans and mice: utilizing pharmacological modulation of its metabolic pathway to increase systemic exposure.
Journal: British journal of pharmacology 20110701
Title: Secondary hormonal manipulations in the treatment of castration refractory prostate cancer.
Journal: BJU international 20110701
Title: Design, synthesis and antifungal activities of novel 1,2,4-triazole derivatives.
Journal: European journal of medicinal chemistry 20110701
Title: Antifungal quinazolinones from marine-derived Bacillus cereus and their preparation.
Journal: Bioorganic & medicinal chemistry letters 20110701
Title: Practical synthesis, anticonvulsant, and antimicrobial activity of N-allyl and N-propargyl di(indolyl)indolin-2-ones.
Journal: Bioorganic & medicinal chemistry letters 20110701
Title: 4-alkoxy-3-arylfuran-2(5H)-ones as inhibitors of tyrosyl-tRNA synthetase: synthesis, molecular docking and antibacterial evaluation.
Journal: Bioorganic & medicinal chemistry 20110701
Title: Efficacious and safe management of moderate to severe scalp seborrhoeic dermatitis using clobetasol propionate shampoo 0·05% combined with ketoconazole shampoo 2%: a randomized, controlled study.
Journal: The British journal of dermatology 20110701
Title: Synergistic effects of tetrandrine on the antifungal activity of topical ketoconazole cream in the treatment of dermatophytoses: a clinical trial.
Journal: Chinese journal of integrative medicine 20110701
Title: Drug metabolism of CYP3A4, CYP2C9 and CYP2D6 substrates in pigs and humans.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20110614
Title: Investigating effect of microemulsion components: In vitro permeation of ketoconazole.
Journal: Pharmaceutical development and technology 20110601
Title: Prevalence and antifungal resistance profile of Candida spp. oral isolates from patients with type 1 and 2 diabetes mellitus.
Journal: Archives of oral biology 20110601
Title: Cushing's syndrome due to a pancreatic neuroendocrine tumor metastatic to the ovaries: a clinicopathological description of a case.
Journal: Endocrine pathology 20110601
Title: Melatonin and steroid hormones activate intermembrane Cu,Zn-superoxide dismutase by means of mitochondrial cytochrome P450.
Journal: Free radical biology & medicine 20110601
Title: Tinea capitis versus acne keloidalis nuchae with Trichophyton violaceum superinfection.
Journal: Giornale italiano di dermatologia e venereologia : organo ufficiale, Societa italiana di dermatologia e sifilografia 20110601
Title: [Bilateral conjunctival oedema as a symptom of adrenal adenocarcinoma].
Journal: Archivos de la Sociedad Espanola de Oftalmologia 20110601
Title: Pseudotumor cerebri during Cushing's disease treatment with ketoconazole.
Journal: Arquivos brasileiros de endocrinologia e metabologia 20110601
Title: Thiazole-based chalcones as potent antimicrobial agents. Synthesis and biological evaluation.
Journal: Bioorganic & medicinal chemistry 20110515
Title: Enhancement of triclabendazole action in vivo against a triclabendazole-resistant isolate of Fasciola hepatica by co-treatment with ketoconazole.
Journal: Veterinary parasitology 20110511
Title: In vivo investigation in pigs of intestinal absorption, hepatobiliary disposition, and metabolism of the 5α-reductase inhibitor finasteride and the effects of coadministered ketoconazole.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20110501
Title: Synthesis, antimicrobial, antioxidant, anti-hemolytic and cytotoxic evaluation of new imidazole-based heterocycles.
Journal: European journal of medicinal chemistry 20110501
Title: Assessment of milling-induced disorder of two pharmaceutical compounds.
Journal: Journal of pharmaceutical sciences 20110501
Title: Management of pituitary tumors in pregnancy.
Journal: Nature reviews. Endocrinology 20110501
Title: Antifungal, cytotoxic and SAR studies of a series of N-alkyl, N-aryl and N-alkylphenyl-1,4-pyrrolediones and related compounds.
Journal: Bioorganic & medicinal chemistry 20110501
Title: The effects of concurrent administration of cytochrome P-450 inhibitors on the pharmacokinetics of oral methadone in healthy dogs.
Journal: Veterinary anaesthesia and analgesia 20110501
Title: [Management of invasive fungal infections in children].
Journal: Archives de pediatrie : organe officiel de la Societe francaise de pediatrie 20110501
Title: An azole-resistant isolate of Malassezia pachydermatis.
Journal: Veterinary microbiology 20110421
Title: Fine-tuning the selectivity of aldosterone synthase inhibitors: structure-activity and structure-selectivity insights from studies of heteroaryl substituted 1,2,5,6-tetrahydropyrrolo[3,2,1-ij]quinolin-4-one derivatives.
Journal: Journal of medicinal chemistry 20110414
Title: Synthesis and biological activity of 2-(bis((1,3,4-oxadiazolyl/1,3,4-thiadiazolyl)methylthio)methylene)malononitriles.
Journal: European journal of medicinal chemistry 20110401
Title: Concurrent assessment of hepatic and intestinal cytochrome P450 3A activities using deuterated alfentanil.
Journal: Clinical pharmacology and therapeutics 20110401
Title: Pharmacokinetics of oral neratinib during co-administration of ketoconazole in healthy subjects.
Journal: British journal of clinical pharmacology 20110401
Title: Pharmacokinetic interactions between alitretinoin and ketoconazole or simvastatin or ciclosporin A.
Journal: Clinical and experimental dermatology 20110401
Title: Inhibitory effects of ketoconazole and rifampin on OAT1 and OATP1B1 transport activities: considerations on drug-drug interactions.
Journal: Biopharmaceutics & drug disposition 20110401
Title: Nonhealing scalp wound infected with Aspergillus niger in an elderly patient.
Journal: Cutis 20110401
Title: Low dose of ketoconazole in patients with prostate adenocarcinoma resistant to pharmacological castration.
Journal: BJU international 20110401
Title: Design, synthesis, and biological evaluation of imidazolyl derivatives of 4,7-disubstituted coumarins as aromatase inhibitors selective over 17-α-hydroxylase/C17-20 lyase.
Journal: Journal of medicinal chemistry 20110324
Title: Marginal increase of sunitinib exposure by grapefruit juice.
Journal: Cancer chemotherapy and pharmacology 20110301
Title: Crucial role of cytochrome P450 in hepatotoxicity induced by 2,3-dimethoxy-1,4-naphthoquinone in rats.
Journal: Journal of applied toxicology : JAT 20110301
Title: Evaluation of the origin of a sample of Sporothrix schenckii that caused contamination of a researcher in Southern Brazil.
Journal: Mycopathologia 20110301
Title: CYP3A-mediated generation of aldehyde and hydrazine in atazanavir metabolism.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20110301
Title: Synthesis, structure, molecular docking, and structure-activity relationship analysis of enamines: 3-aryl-4-alkylaminofuran-2(5H)-ones as potential antibacterials.
Journal: Bioorganic & medicinal chemistry 20110301
Title: [Castration resistant prostate cancer 2011].
Journal: Aktuelle Urologie 20110301
Title: First description of onychomycosis caused by Chrysosporium keratinophilum in captive Bennett's wallabies (Macropus rufogriseus rufogriseus).
Journal: Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians 20110301
Title: Unexpected effect of rifampin on the pharmacokinetics of linezolid: in silico and in vitro approaches to explain its mechanism.
Journal: Journal of clinical pharmacology 20110201
Title: Effects of ketoconazole on the in vivo biotransformation and hepatobiliary transport of the thrombin inhibitor AZD0837 in pigs.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20110201
Title: The effect of increased lipoprotein levels on the pharmacokinetics of ketoconazole enantiomers in the rat.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20110201
Title: Application of validated RP-HPLC method for simultaneous determination of docetaxel and ketoconazole in solid lipid nanoparticles.
Journal: Journal of chromatographic science 20110201
Title: Mechanism of cytochrome P450-3A inhibition by ketoconazole.
Journal: The Journal of pharmacy and pharmacology 20110201
Title: [Evaluation of efficacy of ketoconazole 800 mg-clindamycin 100 mg tablets vaginal against ketoconazole 800 mg- clindamycin 100 mg vaginal capsules in candida vaginitis and vaginosis].
Journal: Ginecologia y obstetricia de Mexico 20110201
Title: Cytochrome P450 3A4 inhibitory constituents of the wood of Taxus yunnanensis.
Journal: Journal of natural products 20110128
Title: Radical scavenging and antioxidant activities of isocoumarins and a phthalide from the endophytic fungus Colletotrichum sp.
Journal: Journal of natural products 20110128
Title: New drug-like hydroxyphenylnaphthol steroidomimetics as potent and selective 17β-hydroxysteroid dehydrogenase type 1 inhibitors for the treatment of estrogen-dependent diseases.
Journal: Journal of medicinal chemistry 20110127
Title: A species-specific approach to the use of non-antimony treatments for cutaneous leishmaniasis.
Journal: The American journal of tropical medicine and hygiene 20110105
Title: A case of kerion celsi caused by Microsporum gypseum in a boy following dermatoplasty for a scalp wound from a road accident.
Journal: Medical mycology 20110101
Title: Effects of rifampin and ketoconazole on the pharmacokinetics of nilotinib in healthy participants.
Journal: Journal of clinical pharmacology 20110101
Title: Effect of the inhibition of CYP3A4 or CYP2D6 on the pharmacokinetics and pharmacodynamics of oxycodone.
Journal: European journal of clinical pharmacology 20110101
Title: Identification of human liver cytochrome P450 enzymes involved in the metabolism of SCH 530348 (Vorapaxar), a potent oral thrombin protease-activated receptor 1 antagonist.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20110101
Title: Ketoconazole and miconazole alter potassium homeostasis in Saccharomyces cerevisiae.
Journal: Biochimica et biophysica acta 20110101
Title: N-(Pyridin-3-yl)benzamides as selective inhibitors of human aldosterone synthase (CYP11B2).
Journal: Bioorganic & medicinal chemistry letters 20110101
Title: 3-[Benzimidazo- and 3-[benzothiadiazoleimidazo-(1,2-c)quinazolin-5-yl]-2H-chromene-2-ones as potent antimicrobial agents.
Journal: Bioorganic & medicinal chemistry letters 20110101
Title: CYP1A2-mediated biotransformation of cardioactive 2-thienylidene-3,4-methylenedioxybenzoylhydrazine (LASSBio-294) by rat liver microsomes and human recombinant CYP enzymes.
Journal: European journal of medicinal chemistry 20110101
Title: Fixed drug eruptions induced by cross-reactive imidazoles.
Journal: Allergologia et immunopathologia 20110101
Title: [Onychomycosis-causing yeasts in four Mexican dermatology centers and their antifungal susceptibility to azolic compounds].
Journal: Revista iberoamericana de micologia 20110101
Title: Evaluation of the pharmacokinetic interaction of midazolam with ursodeoxycholic acid, ketoconazole and dexamethasone by brain benzodiazepine receptor occupancy.
Journal: The Journal of pharmacy and pharmacology 20110101
Title: Inhibitory effects of Phyllanthus amarus and its major lignans on human microsomal cytochrome P450 activities: evidence for CYP3A4 mechanism-based inhibition.
Journal: Drug metabolism and pharmacokinetics 20110101
Title: In vitro antifungal susceptibility of Candida spp. oral isolates from HIV-positive patients and control individuals.
Journal: Brazilian oral research 20110101
Title: Patient preferences and treatment safety for uncomplicated vulvovaginal candidiasis in primary health care.
Journal: BMC public health 20110101
Title: Oropharyngeal histoplasmosis: report of eleven cases and review of the literature.
Journal: Revista da Sociedade Brasileira de Medicina Tropical 20110101
Title: [Determination of hemolytic activity and in vitro antifungal susceptibility of Trichophyton rubrum clinical strains].
Journal: Mikrobiyoloji bulteni 20110101
Title: Disturbance in hemoglobin metabolism and in vivo antimalarial activity of azole antimycotics.
Journal: Revista do Instituto de Medicina Tropical de Sao Paulo 20110101
Title: Physicochemical characterization and dissolution study of solid dispersions of ketoconazole with nicotinamide.
Journal: Chemical & pharmaceutical bulletin 20110101
Title: Overexpression of CYP3A4, but not of CYP2D6, promotes hypoxic response and cell growth of Hep3B cells.
Journal: Drug metabolism and pharmacokinetics 20110101
Title: Cushing syndrome due to ectopic adrenocorticotropic hormone secretion in a 3-year-old child.
Journal: Journal of pediatric endocrinology & metabolism : JPEM 20110101
Title: [Scedosporium apiospermum disseminated infection in a single lung transplant recipient].
Journal: Revista iberoamericana de micologia 20110101
Title: Effectiveness of chronic treatment with ketoconazole in a patient with diabetic Cushing's disease resistant to surgery.
Journal: Endokrynologia Polska 20110101
Title: Oral cavity eumycetoma.
Journal: Revista do Instituto de Medicina Tropical de Sao Paulo 20110101
Title: [Immunorehabilitation in patients with paecilomycosis-complicated echinococcosis and asthma].
Journal: Meditsinskaia parazitologiia i parazitarnye bolezni 20110101
Title: Trypanosoma cruzi epimastigotes are able to store and mobilize high amounts of cholesterol in reservosome lipid inclusions.
Journal: PloS one 20110101
Title: Nocardia transvalensis keratitis: an emerging pathology among travelers returning from Asia.
Journal: BMC infectious diseases 20110101
Title: Prevalence of exocrine pancreatic insufficiency in women with obesity syndrome: assessment by pancreatic fecal elastase 1.
Journal: ISRN gastroenterology 20110101
Title: Pneumocystis pneumonia during medicamentous treatment of Cushing's syndrome--a description of two cases.
Journal: Acta medica (Hradec Kralove) 20110101
Title: New aspects in the clinical course of pityriasis versicolor.
Journal: Anais brasileiros de dermatologia 20110101
Title: Oral antifungal therapy for chronic rhinosinusitis and its subtypes: a systematic review.
Journal: International forum of allergy & rhinology 20110101
Title: Pilot Study of 15 Patients Receiving a New Treatment Regimen for Androgenic Alopecia: The Effects of Atopy on AGA.
Journal: ISRN dermatology 20110101
Title: Prophylactic ketoconazole shampoo for tinea capitis in a high-risk pediatric population.
Journal: The journal of pediatric pharmacology and therapeutics : JPPT : the official journal of PPAG 20110101
Title: Optimization of a novel method based on solidification of floating organic droplet by high-performance liquid chromatography for evaluation of antifungal drugs in biological samples.
Journal: Talanta 20101215
Title: Structural interpretation in composite systems using powder X-ray diffraction: applications of error propagation to the pair distribution function.
Journal: Pharmaceutical research 20101201
Title: Metabolism and action of proteasome inhibitors in primary human hepatocytes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20101201
Title: A predictive ligand-based Bayesian model for human drug-induced liver injury.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20101201
Title: Characterisation of zuclopenthixol metabolism by in vitro and therapeutic drug monitoring studies.
Journal: Acta psychiatrica Scandinavica 20101201
Title: [Probable basidiobolomycosis in a Togolese rural young successfully treated with ketoconazole].
Journal: Bulletin de la Societe de pathologie exotique (1990) 20101201
Title: High performance liquid chromatographic assay for the simultaneous determination of midazolam and ketoconazole in plasma.
Journal: Journal of pharmaceutical and biomedical analysis 20101102
Title: Azole drugs trap cytochrome P450 EryK in alternative conformational states.
Journal: Biochemistry 20101102
Title: Pharmacokinetics and pharmacodynamics of docetaxel with or without ketoconazole modulation in chemonaive breast cancer patients.
Journal: Annals of oncology : official journal of the European Society for Medical Oncology 20101101
Title: Effects on plasma corticosterone levels and brain serotonin from interference with methamphetamine-induced corticosterone release in neonatal rats.
Journal: Stress (Amsterdam, Netherlands) 20101101
Title: Prediction of the intestinal first-pass metabolism of CYP3A substrates in humans using cynomolgus monkeys.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20101101
Title: Synthesis and biological evaluation of N-antipyrine-4-substituted amino-3-chloromaleimide derivatives.
Journal: European journal of medicinal chemistry 20101101
Title: Regulation of the hypoxic response in Candida albicans.
Journal: Eukaryotic cell 20101101
Title: Tumor necrosis factor alpha increases P-glycoprotein expression in a BME-UV in vitro model of mammary epithelial cells.
Journal: Biopharmaceutics & drug disposition 20101101
Title: Structure and mechanism of the complex between cytochrome P4503A4 and ritonavir.
Journal: Proceedings of the National Academy of Sciences of the United States of America 20101026
Title: Severe retention hyperkeratosis occurring with Susac syndrome.
Journal: Dermatology online journal 20101015
Title: Subcutaneous zygomycosis: report of 10 cases from two institutions in North India.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20101001
Title: Anticandidal effect of Ocimum sanctum essential oil and its synergy with fluconazole and ketoconazole.
Journal: Phytomedicine : international journal of phytotherapy and phytopharmacology 20101001
Title: Synthesis and CYP24A1 inhibitory activity of (E)-2-(2-substituted benzylidene)- and 2-(2-substituted benzyl)-6-methoxy-tetralones.
Journal: European journal of medicinal chemistry 20101001
Title: Synthesis and antifungal evaluation of novel triazole derivatives as inhibitors of cytochrome P450 14alpha-demethylase.
Journal: European journal of medicinal chemistry 20101001
Title: Biorelevant media to simulate fluids in the ascending colon of humans and their usefulness in predicting intracolonic drug solubility.
Journal: Pharmaceutical research 20101001
Title: Synthesis and antimicrobial activities of novel 1H-dibenzo[a,c]carbazoles from dehydroabietic acid.
Journal: European journal of medicinal chemistry 20101001
Title: Sources of variability in ketoconazole inhibition of human cytochrome P450 3A in vitro.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20101001
Title: Retrospective analysis of the consequences of acid suppressive therapy on ketoconazole efficacy in advanced castration-resistant prostate cancer.
Journal: The Annals of pharmacotherapy 20101001
Title: [Cardiac safety of cinitapride].
Journal: Gastroenterologia y hepatologia 20101001
Title: Presumptive Nocardia spp. infection in a dog treated with cyclosporin and ketoconazole.
Journal: New Zealand veterinary journal 20101001
Title: Comparative evaluation of ketoconazole-β-cyclodextrin systems prepared by coprecipitation and kneading.
Journal: Drug discoveries & therapeutics 20101001
Title: Synthesis and evaluation of anti-Toxoplasma gondii and antimicrobial activities of thiosemicarbazides, 4-thiazolidinones and 1,3,4-thiadiazoles.
Journal: European journal of medicinal chemistry 20100901
Title: A study of cytotoxicity of novel chlorokojic acid derivatives with their antimicrobial and antiviral activities.
Journal: European journal of medicinal chemistry 20100901
Title: CYP24A1 inhibition enhances the antitumor activity of calcitriol.
Journal: Endocrinology 20100901
Title: In vitro and in vivo metabolism of a novel cannabinoid-1 receptor inverse agonist, taranabant, in rats and monkeys.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20100901
Title: Synthesis and bioassay of aminosulfonyl-1,3,4-oxadiazoles and their interconversion to 1,3,4-thiadiazoles.
Journal: European journal of medicinal chemistry 20100901
Title: Synthesis and biochemical evaluation of a range of (4-substituted phenyl)sulfonate derivatives of 4-hydroxybenzyl imidazole-based compounds as potent inhibitors of 17alpha-hydroxylase/17,20-lyase (P45017alpha) derived from rat testicular microsomes.
Journal: Bioorganic & medicinal chemistry letters 20100901
Title: Effects of drug interactions on biotransformation and antiplatelet effect of clopidogrel in vitro.
Journal: British journal of pharmacology 20100901
Title: Primary cutaneous aspergillosis.
Journal: Acta dermato-venereologica 20100901
Title: [Metabolism of 3-cyanomethyl-4-methyl-DCK, a new anti-HIV candidate, in human intestinal microsomes].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20100901
Title: New antifungal peptides. Synthesis, bioassays and initial structure prediction by CD spectroscopy.
Journal: Bioorganic & medicinal chemistry letters 20100815
Title: Replacement of imidazolyl by pyridyl in biphenylmethylenes results in selective CYP17 and dual CYP17/CYP11B1 inhibitors for the treatment of prostate cancer.
Journal: Journal of medicinal chemistry 20100812
Title: Ketoconazole in the treatment of central serous chorioretinopathy: a pilot study.
Journal: Acta ophthalmologica 20100801
Title: The post-antifungal effect (PAFE) of amphotericin B, nystatin, ketoconazole and 5-fluorocytosine and its impact on the colonization traits of Candida glabrata.
Journal: Medical mycology 20100801
Title: Ketoconazole and rifampin significantly affect the pharmacokinetics, but not the safety or QTc interval, of casopitant, a neurokinin-1 receptor antagonist.
Journal: Journal of clinical pharmacology 20100801
Title: Infantile hypercalcemia and hypercalciuria: new insights into a vitamin D-dependent mechanism and response to ketoconazole treatment.
Journal: The Journal of pediatrics 20100801
Title: Antimicrobial activity and a SAR study of some novel benzimidazole derivatives bearing hydrazone moiety.
Journal: European journal of medicinal chemistry 20100801
Title: In vitro-in vivo extrapolation predicts drug-drug interactions arising from inhibition of codeine glucuronidation by dextropropoxyphene, fluconazole, ketoconazole, and methadone in humans.
Journal: The Journal of pharmacology and experimental therapeutics 20100801
Title: Advantages of human hepatocyte-derived transformants expressing a series of human cytochrome p450 isoforms for genotoxicity examination.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20100801
Title: Differential effects of ketoconazole and primaquine on the pharmacokinetics and tissue distribution of imatinib in mice.
Journal: Anti-cancer drugs 20100801
Title: A single-dose, crossover, placebo- and moxifloxacin-controlled study to assess the effects of neratinib (HKI-272) on cardiac repolarization in healthy adult subjects.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20100801
Title: Synthesis and CYP24A1 inhibitory activity of N-(2-(1H-imidazol-1-yl)-2-phenylethyl)arylamides.
Journal: Bioorganic & medicinal chemistry 20100715
Title: Isopropylidene substitution increases activity and selectivity of biphenylmethylene 4-pyridine type CYP17 inhibitors.
Journal: Journal of medicinal chemistry 20100708
Title: Synthesis of some N-alkyl substituted urea derivatives as antibacterial and antifungal agents.
Journal: European journal of medicinal chemistry 20100701
Title: Synthesis and bioassay of pyrrolyl oxazolines and thiazolines.
Journal: European journal of medicinal chemistry 20100701
Title: Androgen blockade for the treatment of high-flow priapism.
Journal: The journal of sexual medicine 20100701
Title: Enhancement of the drug susceptibility of a triclabendazole-resistant isolate of Fasciola hepatica using the metabolic inhibitor ketoconazole.
Journal: Parasitology research 20100701
Title: Cutaneous lymphoid hyperplasia associated with Leishmania panamensis infection.
Journal: Acta dermato-venereologica 20100701
Title: Validation of a differential in situ perfusion method with mesenteric blood sampling in rats for intestinal drug interaction profiling.
Journal: Biopharmaceutics & drug disposition 20100701
Title: [Ketoconazole antagonizes the immune and gonadotropic systems in the forced swimming test in male Wistar rats].
Journal: Canadian journal of physiology and pharmacology 20100701
Title: Conazoles.
Journal: Molecules (Basel, Switzerland) 20100609
Title: Effectiveness of cabergoline in monotherapy and combined with ketoconazole in the management of Cushing's disease.
Journal: Pituitary 20100601
Title: Naftifine-analogues as anti-Trypanosoma cruzi agents.
Journal: European journal of medicinal chemistry 20100601
Title: CYP3A4 catalytic activity is induced in confluent Huh7 hepatoma cells.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20100601
Title: Increases in discontinuous rib cartilage and fused carpal bone in rat fetuses exposed to the teratogens, busulfan, acetazolamide, vitamin A, and ketoconazole.
Journal: Human & experimental toxicology 20100601
Title: A phase I clinical study of high dose ketoconazole plus weekly docetaxel for metastatic castration resistant prostate cancer.
Journal: The Journal of urology 20100601
Title: The effects of CYP2D6 and CYP3A activities on the pharmacokinetics of immediate release oxycodone.
Journal: British journal of pharmacology 20100601
Title: Trichodermaketones A-D and 7-O-methylkoninginin D from the marine fungus Trichoderma koningii.
Journal: Journal of natural products 20100528
Title: Chemical epigenetics alters the secondary metabolite composition of guttate excreted by an atlantic-forest-soil-derived Penicillium citreonigrum.
Journal: Journal of natural products 20100528
Title: Second generation analogues of the cancer drug clinical candidate tipifarnib for anti-Chagas disease drug discovery.
Journal: Journal of medicinal chemistry 20100527
Title: Determination of commonly used azole antifungals in various waters and sewage sludge using ultra-high performance liquid chromatography-tandem mass spectrometry.
Journal: Journal of chromatography. A 20100521
Title: Pharmacophore modeling strategies for the development of novel nonsteroidal inhibitors of human aromatase (CYP19).
Journal: Bioorganic & medicinal chemistry letters 20100515
Title: Pasireotide alone or with cabergoline and ketoconazole in Cushing's disease.
Journal: The New England journal of medicine 20100513
Title: Activity of ketoconazole after taxane-based chemotherapy in castration-resistant prostate cancer.
Journal: BJU international 20100501
Title: Synthesis and the selective antifungal activity of 5,6,7,8-tetrahydroimidazo[1,2-a]pyridine derivatives.
Journal: European journal of medicinal chemistry 20100501
Title: Oral fingolimod for the treatment of relapsing-remitting multiple sclerosis.
Journal: Drugs of today (Barcelona, Spain : 1998) 20100501
Title: Sex differences in subacute toxicity and hepatic microsomal metabolism of triptolide in rats.
Journal: Toxicology 20100430
Title: Structural basis of human CYP51 inhibition by antifungal azoles.
Journal: Journal of molecular biology 20100409
Title: Probing possible egress channels for multiple ligands in human CYP3A4: a molecular modeling study.
Journal: Journal of molecular modeling 20100401
Title: Genotoxicity of a freshwater cyanotoxin, cylindrospermopsin, in two human cell lines: Caco-2 and HepaRG.
Journal: Environmental and molecular mutagenesis 20100401
Title: In vitro investigation of antifungal activity of allicin alone and in combination with azoles against Candida species.
Journal: Mycopathologia 20100401
Title: Testosterone hydroxylation in bovine liver: enzyme kinetic and inhibition study.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20100401
Title: Kinetics of removal of intravenous testosterone pulses in normal men.
Journal: European journal of endocrinology 20100401
Title: An eco-friendly synthesis and antimicrobial activities of dihydro-2H-benzo- and naphtho-1,3-oxazine derivatives.
Journal: European journal of medicinal chemistry 20100401
Title: In vitro and in vivo evaluation of oral tablet formulations prepared with ketoconazole and hydroxypropyl-beta-cyclodextrin.
Journal: Drug delivery 20100401
Title: Potent and selective inhibition of human cytochrome P450 3A4 by seco-pancratistatin structural analogs.
Journal: Bioorganic & medicinal chemistry letters 20100401
Title: Predictions of metabolic drug-drug interactions using physiologically based modelling: Two cytochrome P450 3A4 substrates coadministered with ketoconazole or verapamil.
Journal: Clinical pharmacokinetics 20100401
Title: Effects of ketoconazole on the biodistribution and metabolism of [11C]loperamide and [11C]N-desmethyl-loperamide in wild-type and P-gp knockout mice.
Journal: Nuclear medicine and biology 20100401
Title: [Malassezia folliculitis: 21 cases].
Journal: Annales de dermatologie et de venereologie 20100401
Title: Pyrenochaeta keratinophila sp. nov., isolated from an ocular infection in Spain.
Journal: Revista iberoamericana de micologia 20100331
Title: Phase I clinical trial of the CYP17 inhibitor abiraterone acetate demonstrating clinical activity in patients with castration-resistant prostate cancer who received prior ketoconazole therapy.
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20100320
Title: Phase 1 pharmacokinetic and drug-interaction study of dasatinib in patients with advanced solid tumors.
Journal: Cancer 20100315
Title: Response to azolic antifungal agents for treating feline sporotrichosis.
Journal: The Veterinary record 20100306
Title: Current concepts in systemic and topical therapy for superficial mycoses.
Journal: Clinics in dermatology 20100304
Title: Intralesional sodium stibogluconate alone or its combination with either intramuscular sodium stibogluconate or oral ketoconazole in the treatment of localized cutaneous leishmaniasis: a comparative study.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20100301
Title: Potent in vitro inhibition of CYP3A4 and P-glycoprotein by Rhodiola rosea.
Journal: Planta medica 20100301
Title: Synthesis, characterization and biocidal activity of new organotin complexes of 2-(3-oxocyclohex-1-enyl)benzoic acid.
Journal: European journal of medicinal chemistry 20100301
Title: Antimicrobial study of newly synthesized 6-substituted indolo[1,2-c]quinazolines.
Journal: European journal of medicinal chemistry 20100301
Title: Pulmonary toxicity and metabolic activation of dauricine in CD-1 mice.
Journal: The Journal of pharmacology and experimental therapeutics 20100301
Title: Composition optimization and stability testing of a parenteral antifungal solution based on a ternary solvent system.
Journal: AAPS PharmSciTech 20100301
Title: Comparative evaluation of ketoconazole tablet and topical ketoconazole 2% in orabase in treatment of Candida-infected denture stomatitis.
Journal: The journal of contemporary dental practice 20100301
Title: Effect of ketoconazole on the pharmacokinetics of udenafil in healthy Korean subjects.
Journal: British journal of clinical pharmacology 20100301
Title: Absorption barriers in the rat intestinal mucosa: 2. Application of physiologically based mathematical models to quantify mechanisms of drug permeation and metabolism.
Journal: Journal of pharmaceutical sciences 20100201
Title: Quantitative prediction and clinical observation of a CYP3A inhibitor-based drug-drug interactions with MLN3897, a potent C-C chemokine receptor-1 antagonist.
Journal: The Journal of pharmacology and experimental therapeutics 20100201
Title: Ketoconazole enantiomer for the treatment of diabetes mellitus.
Journal: Expert opinion on investigational drugs 20100201
Title: Use of antifungal agents for oral candidiasis: results of a national survey.
Journal: International journal of dental hygiene 20100201
Title: Sulfonamide-1,2,4-thiadiazole derivatives as antifungal and antibacterial agents: synthesis, biological evaluation, lipophilicity, and conformational studies.
Journal: Chemical & pharmaceutical bulletin 20100201
Title: The pharmacokinetics of ketoconazole and its effects on the pharmacokinetics of midazolam and fentanyl in dogs.
Journal: Journal of veterinary pharmacology and therapeutics 20100201
Title: Cutaneous malasseziasis: four case reports of atypical dermatitis and onychomycosis caused by Malassezia.
Journal: International journal of dermatology 20100201
Title: Adrenocorticotrophic hormone (ACTH) responsiveness to ghrelin increases after 6 months of ketoconazole use in patients with Cushing's disease: comparison with GH-releasing peptide-6 (GHRP-6).
Journal: Clinical endocrinology 20100101
Title: In young men, a moderate inhibition of testosterone synthesis capacity is only partly compensated by increased activity of the pituitary and the hypothalamus.
Journal: Clinical endocrinology 20100101
Title: Synergistic anti-candidal activity of tetrandrine on ketoconazole: an experimental study.
Journal: Planta medica 20100101
Title: Identification of the human cytochrome P450 enzymes involved in the two oxidative steps in the bioactivation of clopidogrel to its pharmacologically active metabolite.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20100101
Title: The application of in vitro technologies to study the metabolism of the androgenic/anabolic steroid stanozolol in the equine.
Journal: Steroids 20100101
Title: Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugs.
Journal: Bioorganic & medicinal chemistry 20100101
Title: Screening of antimycotics in Swedish sewage treatment plants--waters and sludge.
Journal: Water research 20100101
Title: CYP3A catalyses schizandrin biotransformation in human, minipig and rat liver microsomes.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20100101
Title: Candida albicans enhances experimental hepatic melanoma metastasis.
Journal: Clinical & experimental metastasis 20100101
Title: Esthesioneuroblastoma (Olfactory Neuroblastoma) with Ectopic ACTH Syndrome: a multidisciplinary case presentation from the Joan Karnell cancer center of Pennsylvania Hospital.
Journal: The oncologist 20100101
Title: Hormonal therapy for acne: why not as first line therapy? facts and controversies.
Journal: Clinics in dermatology 20100101
Title: [Acquired pigmented lesion of the foot].
Journal: Annales de dermatologie et de venereologie 20100101
Title: Everolimus versus azathioprine in a cyclosporine and ketoconazole-based immunosuppressive therapy in kidney transplant: 3-year follow-up of an open-label, prospective, cohort, comparative clinical trial.
Journal: Transplantation proceedings 20100101
Title: Effectiveness and cost of replacing a calcineurin inhibitor with sirolimus to slow the course of chronic kidney disease in renal allografts.
Journal: Transplantation proceedings 20100101
Title: [Echinococcosis complicated by paecilomycosis].
Journal: Meditsinskaia parazitologiia i parazitarnye bolezni 20100101
Title: Medical therapy of Cushing's disease: where are we now?
Journal: Frontiers of hormone research 20100101
Title: Diagnostic and therapeutic challenge in the management of a patient with ectopic adrenocorticotropin secretion.
Journal: Journal of endocrinological investigation 20100101
Title: The sensitivity and specificity of potassium hydroxide smear and fungal culture relative to clinical assessment in the evaluation of tinea pedis: a pooled analysis.
Journal: Dermatology research and practice 20100101
Title: Colletotrichum graminicola keratitis: first case report from India.
Journal: Indian journal of ophthalmology 20100101
Title: Management of diabetes mellitus in Cushing's syndrome.
Journal: Neuroendocrinology 20100101
Title: Management of dyslipidemia in Cushing's syndrome.
Journal: Neuroendocrinology 20100101
Title: Medical treatment of Cushing's syndrome: adrenal-blocking drugs and ketaconazole.
Journal: Neuroendocrinology 20100101
Title: Evaluation of terfenadine and ketoconazole-induced QT prolongation in conscious telemetered guinea pigs.
Journal: Pharmacological reports : PR 20100101
Title: High-performance thin-layer chromatographic determination of ketoconazole in pharmaceutical formulations.
Journal: Journal of cosmetic science 20100101
Title: A noninferiority clinical trial comparing fluconazole and ketoconazole in combination with cephalexin for the treatment of dogs with Malassezia dermatitis.
Journal: Veterinary therapeutics : research in applied veterinary medicine 20100101
Title: Sporothrix schenckii associated with armadillo hunting in Southern Brazil: epidemiological and antifungal susceptibility profiles.
Journal: Revista da Sociedade Brasileira de Medicina Tropical 20100101
Title: Use of granisetron transdermal system in the prevention of chemotherapy-induced nausea and vomiting: a review.
Journal: Cancer management and research 20100101
Title: Novel medical treatment of pituitary adrenocorticotropic hormone-dependent hypercortisolism: a case study.
Journal: Endocrine practice : official journal of the American College of Endocrinology and the American Association of Clinical Endocrinologists 20100101
Title: Childhood acute generalized exanthematous pustulosis induced by oral ketoconazole.
Journal: Acta dermatovenerologica Croatica : ADC 20100101
Title: Antioxidant and antimicrobial activity of some lichen species.
Journal: Mikrobiologiia 20100101
Title: [White piedra in a pediatric patient: a case report].
Journal: Revista iberoamericana de micologia 20091231
Title: Rapid LC-MS drug metabolite profiling using microsomal enzyme bioreactors in a parallel processing format.
Journal: Analytical chemistry 20091215
Title: Simultaneous determination of five systemic azoles in plasma by high-performance liquid chromatography with ultraviolet detection.
Journal: Journal of pharmaceutical and biomedical analysis 20091205
Title: Synergistic anticandidal activity of xanthorrhizol in combination with ketoconazole or amphotericin B.
Journal: FEMS yeast research 20091201
Title: Inhibition and stimulation of intestinal and hepatic CYP3A activity: studies in humanized CYP3A4 transgenic mice using triazolam.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20091201
Title: Side chain azasteroids and thiasteroids as sterol methyltransferase inhibitors in ergosterol biosynthesis.
Journal: Bioorganic & medicinal chemistry 20091201
Title: Synthesis and biological activities of new substituted thiazoline-quinoline derivatives.
Journal: Acta pharmaceutica (Zagreb, Croatia) 20091201
Title: Drugs in the medical treatment of Cushing's syndrome.
Journal: Expert opinion on emerging drugs 20091201
Title: The effects of ketoconazole and rifampicin on the pharmacokinetics of mirodenafil in healthy Korean male volunteers: an open-label, one-sequence, three-period, three-treatment crossover study.
Journal: Clinical therapeutics 20091201
Title: Rhabdomyomatous mesenchymal hamartoma: clinical overview and report of a case with spontaneous regression.
Journal: The West Indian medical journal 20091201
Title: Strategy of accelerated method development for high-throughput bioanalytical assays using ultra high-performance liquid chromatography coupled with mass spectrometry.
Journal: Analytical chemistry 20091115
Title: Phase II study of androgen synthesis inhibition with ketoconazole, hydrocortisone, and dutasteride in asymptomatic castration-resistant prostate cancer.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20091115
Title: Influence of quinidine, cimetidine, and ketoconazole on the enantioselective pharmacokinetics and metabolism of metoprolol in rats.
Journal: Chirality 20091101
Title: Synthesis of some novel pyrazolo[3,4-b]pyridine and pyrazolo[3,4-d]pyrimidine derivatives bearing 5,6-diphenyl-1,2,4-triazine moiety as potential antimicrobial agents.
Journal: European journal of medicinal chemistry 20091101
Title: Synthesis, antimicrobial and antioxidant activities of substituted pyrazoles, isoxazoles, pyrimidine and thioxopyrimidine derivatives.
Journal: European journal of medicinal chemistry 20091101
Title: Roles of different CYP enzymes in the formation of specific fluvastatin metabolites by human liver microsomes.
Journal: Basic & clinical pharmacology & toxicology 20091101
Title: Different effects of ketoconazole on the stereoselective first-pass metabolism of R/S-verapamil in the intestine and the liver: important for the mechanistic understanding of first-pass drug-drug interactions.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20091101
Title: Partial restoration of GH responsiveness to ghrelin in Cushing's disease after 6 months of ketoconazole treatment: comparison with GHRP-6 and GHRH.
Journal: European journal of endocrinology 20091101
Title: Synthesis, Raman, FT-IR, NMR spectroscopic characterization, antimicrobial activity, cytotoxicity and DNA binding of new mixed aza-oxo-thia macrocyclic compounds.
Journal: European journal of medicinal chemistry 20091101
Title: Evaluation of drug-polymer miscibility in amorphous solid dispersion systems.
Journal: Pharmaceutical research 20091101
Title: 5-Nitrofuranes and 5-nitrothiophenes with anti-Trypanosoma cruzi activity and ability to accumulate squalene.
Journal: Bioorganic & medicinal chemistry 20091101
Title: Deactivation of anti-cancer drug letrozole to a carbinol metabolite by polymorphic cytochrome P450 2A6 in human liver microsomes.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20091101
Title: In vitro antimalarial interactions between mefloquine and cytochrome P450 inhibitors.
Journal: Acta tropica 20091001
Title: Superficial distribution and identification of antifungal/antimicrobial agents on a modified tissue conditioner by SEM-EDS microanalysis: a preliminary study.
Journal: Journal of prosthodontics : official journal of the American College of Prosthodontists 20091001
Title: Ketoconazole-induced JNK phosphorylation and subsequent cell death via apoptosis in human osteosarcoma cells.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20091001
Title: Ketoconazole and prednisone to prevent recurrent ischemic priapism.
Journal: The Journal of urology 20091001
Title: Structure-activity studies on seco-pancratistatin analogs: potent inhibitors of human cytochrome P450 3A4.
Journal: Bioorganic & medicinal chemistry letters 20091001
Title: Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Journal: Nature chemical biology 20091001
Title: Biliary excretion of technetium-99m-sestamibi in wild-type dogs and in dogs with intrinsic (ABCB1-1Delta mutation) and extrinsic (ketoconazole treated) P-glycoprotein deficiency.
Journal: Journal of veterinary pharmacology and therapeutics 20091001
Title: Activity of dutasteride plus ketoconazole in castration-refractory prostate cancer after progression on ketoconazole alone.
Journal: Clinical genitourinary cancer 20091001
Title: In vitro and in vivo evaluation of the inhibition potential of risperidone toward clozapine biotransformation.
Journal: British journal of clinical pharmacology 20091001
Title: A novel class of highly potent multidrug resistance reversal agents: disubstituted adamantyl derivatives.
Journal: Bioorganic & medicinal chemistry letters 20090915
Title: Transfer of rolf S3-S4 linker to HERG eliminates activation gating but spares inactivation.
Journal: Biophysical journal 20090902
Title: The amino acid residues of transmembrane helix 5 of multidrug resistance protein CaCdr1p of Candida albicans are involved in substrate specificity and drug transport.
Journal: Biochimica et biophysica acta 20090901
Title: The arachidonic acid epoxygenase is a component of the signaling mechanisms responsible for VEGF-stimulated angiogenesis.
Journal: Archives of biochemistry and biophysics 20090901
Title: Prednisone reduces ketoconazole-induced skeletal defects in rat fetuses.
Journal: Archives of toxicology 20090901
Title: In vitro synergistic effects of antituberculous drugs plus antifungals against Coccidioides posadasii.
Journal: International journal of antimicrobial agents 20090901
Title: Infectious keratitis caused by Aspergillus tubingensis.
Journal: Cornea 20090901
Title: Aetiological treatment with itraconazole or ketoconazole in individuals with Trypanosoma cruzi/HIV co-infection.
Journal: Annals of tropical medicine and parasitology 20090901
Title: The effect on sotrastaurin pharmacokinetics of strong CYP3A inhibition by ketoconazole.
Journal: British journal of clinical pharmacology 20090901
Title: Inhibitory effects of ketoconazole, cimetidine and erythromycin on hepatic CYP3A activities in cats.
Journal: The Journal of veterinary medical science 20090901
Title: Synthesis and biochemical evaluation of a range of sulfonated derivatives of 4-hydroxybenzyl imidazole as highly potent inhibitors of rat testicular 17alpha-hydroxylase/17,20-lyase (P-450(17alpha)).
Journal: Bioorganic & medicinal chemistry letters 20090815
Title: Electron paramagnetic resonance method for the quantitative assay of ketoconazole in pharmaceutical preparations.
Journal: Analytical chemistry 20090815
Title: Differential effect of Shenmai injection, a herbal preparation, on the cytochrome P450 3A-mediated 1'-hydroxylation and 4-hydroxylation of midazolam.
Journal: Chemico-biological interactions 20090814
Title: Identification and chromosomal localization of one locus of Leishmania (L.) major related with resistance to itraconazole.
Journal: Parasitology research 20090801
Title: Spondylodiscitis due to an emergent fungal pathogen: Blastoschizomyces capitatus, a case report and review of the literature.
Journal: Rheumatology international 20090801
Title: Mono and bis-6-arylbenzimidazo[1,2-c]quinazolines: a new class of antimicrobial agents.
Journal: European journal of medicinal chemistry 20090801
Title: Synthesis and antimultidrug resistance evaluation of icariin and its derivatives.
Journal: Bioorganic & medicinal chemistry letters 20090801
Title: About the role of enantioselective selector-selectand interactions and the mobilities of diastereomeric associates in enantiomer separations using CE.
Journal: Electrophoresis 20090801
Title: Dermatomycosis in a pet inland bearded dragon (Pogona vitticeps) caused by a Chrysosporium species related to Nannizziopsis vriesii.
Journal: Veterinary dermatology 20090801
Title: Metabolism of loratadine and further characterization of its in vitro metabolites.
Journal: Drug metabolism letters 20090801
Title: Revisiting the metabolism of ketoconazole using accurate mass.
Journal: Drug metabolism letters 20090801
Title: Side chain flexibilities in the human ether-a-go-go related gene potassium channel (hERG) together with matched-pair binding studies suggest a new binding mode for channel blockers.
Journal: Journal of medicinal chemistry 20090723
Title: Hypokalemia, metabolic alkalosis, and hypertension in a lung cancer patient.
Journal: Kidney international 20090701
Title: Nonlinear stereoselective pharmacokinetics of ketoconazole in rat after administration of racemate.
Journal: Chirality 20090701
Title: In vitro inhibition of CYP3A4 by herbal remedies frequently used by cancer patients.
Journal: Phytotherapy research : PTR 20090701
Title: Novel CYP17 inhibitors: synthesis, biological evaluation, structure-activity relationships and modelling of methoxy- and hydroxy-substituted methyleneimidazolyl biphenyls.
Journal: European journal of medicinal chemistry 20090701
Title: Limited sampling strategy in rats to predict the inhibited activities of hepatic CYP3A.
Journal: Laboratory animals 20090701
Title: Steroidogenesis inhibitors alter but do not eliminate androgen synthesis mechanisms during progression to castration-resistance in LNCaP prostate xenografts.
Journal: The Journal of steroid biochemistry and molecular biology 20090701
Title: Regioselective synthesis and biological evaluation of bis(indolyl)methane derivatized 1,4-disubstituted 1,2,3-bistriazoles as anti-infective agents.
Journal: Bioorganic & medicinal chemistry letters 20090701
Title: Single-center experience with cyclosporine for treatment of idiopathic minimal change nephrotic syndrome in children.
Journal: Iranian journal of kidney diseases 20090701
Title: In vitro response of cutaneous mycosis fungal agents to the most widely used systemic antifungals in dermatology.
Journal: Anais brasileiros de dermatologia 20090701
Title: Drug-drug interaction prediction assessment.
Journal: Journal of biopharmaceutical statistics 20090701
Title: Cytotoxicity of ginkgolic acid in HepG2 cells and primary rat hepatocytes.
Journal: Toxicology letters 20090622
Title: Selective cytochrome P450 3A4 inhibitory activity of Amaryllidaceae alkaloids.
Journal: Bioorganic & medicinal chemistry letters 20090615
Title: An inhibition study of beauvericin on human and rat cytochrome P450 enzymes and its pharmacokinetics in rats.
Journal: Journal of enzyme inhibition and medicinal chemistry 20090601
Title: Neurocryptococcosis in a 10-year-old immunocompetent girl.
Journal: Acta neurochirurgica 20090601
Title: Evaluation of drug-drug interactions with fesoterodine.
Journal: European journal of clinical pharmacology 20090601
Title: CYP3A5*1/*3 genotype influences the blood concentration of tacrolimus in response to metabolic inhibition by ketoconazole.
Journal: Pharmacogenetics and genomics 20090601
Title: Effect of ketoconazole on the pharmacokinetic profile of ambrisentan.
Journal: Journal of clinical pharmacology 20090601
Title: Growth inhibitory action of ebselen on fluconazole-resistant Candida albicans: role of the plasma membrane H+-ATPase.
Journal: Microbial drug resistance (Larchmont, N.Y.) 20090601
Title: Bulky 1,4-benzoxazine derivatives with antifungal activity.
Journal: Bioorganic & medicinal chemistry 20090601
Title: Therapies for pediatric seborrheic dermatitis.
Journal: Pediatric annals 20090601
Title: Randomised controlled trial of the treatment of pastern dermatitis with a formulation containing kunzea oil.
Journal: The Veterinary record 20090516
Title: Synthesis and bioassay of a new class of heterocycles pyrrolyl oxadiazoles/thiadiazoles/triazoles.
Journal: European journal of medicinal chemistry 20090501
Title: Synthesis and anti-microbial screening of some Schiff bases of 3-amino-6,8-dibromo-2-phenylquinazolin-4(3H)-ones.
Journal: European journal of medicinal chemistry 20090501
Title: Synthesis, antimicrobial and cytotoxic activities of some 5-arylidene-4-thioxo-thiazolidine-2-ones.
Journal: European journal of medicinal chemistry 20090501
Title: Synthesis, antimicrobial evaluation and QSAR study of some 3-hydroxypyridine-4-one and 3-hydroxypyran-4-one derivatives.
Journal: European journal of medicinal chemistry 20090501
Title: Design, synthesis, and biological evaluation of novel triazole derivatives as inhibitors of cytochrome P450 14alpha-demethylase.
Journal: European journal of medicinal chemistry 20090501
Title: Electronic, Raman and FT-IR spectral investigations of the charge transfer interactions between ketoconazole and povidone drugs with iodine.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20090501
Title: Novel secondary hormonal therapy in advanced prostate cancer: an update.
Journal: Current opinion in urology 20090501
Title: Identification of quinone methide metabolites of dauricine in human liver microsomes and in rat bile.
Journal: Chemical research in toxicology 20090501
Title: Antimicrobial ambiguine isonitriles from the cyanobacterium Fischerella ambigua.
Journal: Journal of natural products 20090501
Title: Ketoconazole retains activity in patients with docetaxel-refractory prostate cancer.
Journal: Annals of oncology : official journal of the European Society for Medical Oncology 20090501
Title: New acyclic nucleosides analogues as potential analgesic, anti-inflammatory, anti-oxidant and anti-microbial derived from pyrimido[4,5-b]quinolines.
Journal: European journal of medicinal chemistry 20090401
Title: Contact allergy to ketoconazole cross-sensitive to miconazole.
Journal: Clinical and experimental dermatology 20090401
Title: In vitro activities of retigeric acid B alone and in combination with azole antifungal agents against Candida albicans.
Journal: Antimicrobial agents and chemotherapy 20090401
Title: Exploratory study on the clinical and mycological effectiveness of a herbal medicinal product from Solanum chrysotrichum in patients with Candida yeast-associated vaginal infection.
Journal: Planta medica 20090401
Title: Relative contributions of the Candida albicans ABC transporters Cdr1p and Cdr2p to clinical azole resistance.
Journal: Antimicrobial agents and chemotherapy 20090401
Title: Effect of different durations of ketoconazole dosing on the single-dose pharmacokinetics of midazolam: shortening the paradigm.
Journal: Journal of clinical pharmacology 20090401
Title: [Treatment of Cushing's disease with ketoconazole].
Journal: Anales de pediatria (Barcelona, Spain : 2003) 20090401
Title: In vitro metabolism and inhibitory effects of pranlukast in human liver microsomes.
Journal: Biological & pharmaceutical bulletin 20090401
Title: Effects of ketoconazole and carbamazepine on lapatinib pharmacokinetics in healthy subjects.
Journal: British journal of clinical pharmacology 20090401
Title: Ketoconazole allergy.
Journal: Clinics (Sao Paulo, Brazil) 20090401
Title: [Enzyme kinetics of ligustilide metabolism in rat liver microsomes].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20090401
Title: Direct antifungal susceptibility testing of positive Candida blood cultures by sensititre YeastOne.
Journal: The new microbiologica 20090401
Title: Steroidogenesis-disrupting compounds can be effectively studied for major fertility-related endpoints using in vitro cultured mouse follicles.
Journal: Toxicology letters 20090328
Title: Rational modification of a candidate cancer drug for use against Chagas disease.
Journal: Journal of medicinal chemistry 20090326
Title: Design, synthesis, and biological evaluation of novel 1-(1H-1,2,4-triazole-1-yl)-2-(2,4-difluorophenyl)-3-substituted benzylamino-2-propanols.
Journal: Bioorganic & medicinal chemistry letters 20090315
Title: Relation between lipophilicity of alkyl gallates and antifungal activity against yeasts and filamentous fungi.
Journal: Bioorganic & medicinal chemistry letters 20090315
Title: Modulation of the antifungal activity of new medicinal plant extracts active on Candida glabrata by the major transporters and regulators of the pleiotropic drug-resistance network in Saccharomyces cerevisiae.
Journal: Microbial drug resistance (Larchmont, N.Y.) 20090301
Title: Pharmacological interactions of anti-microbial agents in odontology.
Journal: Medicina oral, patologia oral y cirugia bucal 20090301
Title: Quantitative evaluation of pharmacokinetic inhibition of CYP3A substrates by ketoconazole: a simulation study.
Journal: Journal of clinical pharmacology 20090301
Title: The need for multiple doses of 400 mg ketoconazole as a precipitant inhibitor of a CYP3A substrate in an in vivo drug-drug interaction study.
Journal: Journal of clinical pharmacology 20090301
Title: A single-center, open-label, one-sequence study of dalcetrapib coadministered with ketoconazole, and an in vitro study of the S-methyl metabolite of dalcetrapib.
Journal: Clinical therapeutics 20090301
Title: Flexible structure of cytochrome P450: promiscuity of ligand binding in the CYP3A4 heme pocket.
Journal: Anticancer research 20090301
Title: Ketoconazole treatment for Cushing syndrome in McCune-Albright syndrome.
Journal: The Journal of pediatrics 20090301
Title: Aqueous solvent system for the solubilization of azole compounds.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20090215
Title: Rhinosporidiosis in a dog native to the UK.
Journal: The Veterinary record 20090214
Title: CYP1A1 induction and CYP3A4 inhibition by the fungicide imazalil in the human intestinal Caco-2 cells-comparison with other conazole pesticides.
Journal: Toxicology letters 20090210
Title: Clearance and clearance inhibition of the HIV-1 protease inhibitors ritonavir and saquinavir in sandwich-cultured rat hepatocytes and rat microsomes.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20090201
Title: Synthesis and antifungal activity of 1,2,3-triazole containing fluconazole analogues.
Journal: Bioorganic & medicinal chemistry letters 20090201
Title: Ketoconazole increases fingolimod blood levels in a drug interaction via CYP4F2 inhibition.
Journal: Journal of clinical pharmacology 20090201
Title: A new probabilistic rule for drug-dug interaction prediction.
Journal: Journal of pharmacokinetics and pharmacodynamics 20090201
Title: Inhibition of cytochrome P450 activity enhances the systemic availability of triclabendazole metabolites in sheep.
Journal: Journal of veterinary pharmacology and therapeutics 20090201
Title: Pharmacokinetic interaction between efavirenz and ketoconazole in rats.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20090201
Title: Effects of oral posaconazole on the pharmacokinetic properties of oral and intravenous midazolam: a phase I, randomized, open-label, crossover study in healthy volunteers.
Journal: Clinical therapeutics 20090201
Title: Clinical practice. Seborrheic dermatitis.
Journal: The New England journal of medicine 20090122
Title: Novel non-active site inhibitor of Cryptosporidium hominis TS-DHFR identified by a virtual screen.
Journal: Bioorganic & medicinal chemistry letters 20090115
Title: Synthesis, trypanocidal activity and docking studies of novel quinoxaline-N-acylhydrazones, designed as cruzain inhibitors candidates.
Journal: Bioorganic & medicinal chemistry 20090115
Title: Synthesis, Raman, FT-IR, NMR spectroscopic data and antimicrobial activity of mixed aza-oxo-thia macrocyclic compounds.
Journal: European journal of medicinal chemistry 20090101
Title: An open, randomized, prospective, comparative study of topical pimecrolimus 1% cream and topical ketoconazole 2% cream in the treatment of seborrheic dermatitis.
Journal: The Journal of dermatological treatment 20090101
Title: Decreased oral absorption of cyclosporine A after liver ischemia-reperfusion injury in rats: the contribution of CYP3A and P-glycoprotein to the first-pass metabolism in intestinal epithelial cells.
Journal: The Journal of pharmacology and experimental therapeutics 20090101
Title: Effect of oral ketoconazole on oral and intravenous pharmacokinetics of simvastatin and its acid in cynomolgus monkeys.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20090101
Title: Fungistatic effects of optical brightener 220 against Trichophyton tonsurans, Aspergillus fumigatus and Candida albicans.
Journal: The Journal of dermatological treatment 20090101
Title: Assessment of the CYP3A-mediated drug interaction potential of anacetrapib, a potent cholesteryl ester transfer protein (CETP) inhibitor, in healthy volunteers.
Journal: Journal of clinical pharmacology 20090101
Title: Inhibition of CYP3A4 expression by ketoconazole is mediated by the disruption of pregnane X receptor, steroid receptor coactivator-1, and hepatocyte nuclear factor 4alpha interaction.
Journal: Pharmacogenetics and genomics 20090101
Title: Etomidate infusion in the critical care setting for suppressing the acute phase of Cushing's syndrome.
Journal: Anesthesia and analgesia 20090101
Title: Glucocorticoid inhibition in the treatment of depression: can we think outside the endocrine hypothalamus?
Journal: Depression and anxiety 20090101
Title: A study to evaluate the efficacy and safety of oral fluconazole in the treatment of tinea versicolor.
Journal: Mymensingh medical journal : MMJ 20090101
Title: [Fungicidal activity of liranaftate against dermatophytes].
Journal: Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20090101
Title: In vitro susceptibility testing of dermatophytes isolated in Goiania, Brazil, against five antifungal agents by broth microdilution method.
Journal: Revista do Instituto de Medicina Tropical de Sao Paulo 20090101
Title: Alterations in growth and branching of Neurospora crassa caused by sub-inhibitory concentrations of antifungal agents.
Journal: Revista Argentina de microbiologia 20090101
Title: Tinea capitis due to Trichophyton soudanense in Chicago, Illinois: report of a case.
Journal: Pediatric dermatology 20090101
Title: Bioequivalence studies and sugar-based excipients effects on the properties of new generic ketoconazole tablets formulations and stability evaluation by using direct compression method.
Journal: Pharmaceutical development and technology 20090101
Title: High-throughput fluorescence assay of cytochrome P450 3A4.
Journal: Nature protocols 20090101
Title: Determination of ketoconazole in capsules by high-performance liquid chromatography and microbiological assay.
Journal: Journal of AOAC International 20090101
Title: Two-year experience with tacrolimus in renal transplantation after late conversion from cyclosporine therapy.
Journal: Transplantation proceedings 20090101
Title: Ketoconazole inhibits the growth and development of Ichthyophonus sp. (Mesomycetozoa) in vitro.
Journal: The Journal of eukaryotic microbiology 20090101
Title: [Guidelines for diagnosis and treatment of mucocutaneous candidiasis].
Journal: Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20090101
Title: Prediction of drug-drug interactions based on time-dependent inhibition from high throughput screening of cytochrome P450 3A4 inhibition.
Journal: Drug metabolism and pharmacokinetics 20090101
Title: Effect of the CYP3A inhibitor ketoconazole on the pharmacokinetics and pharmacodynamics of bortezomib in patients with advanced solid tumors: a prospective, multicenter, open-label, randomized, two-way crossover drug-drug interaction study.
Journal: Clinical therapeutics 20090101
Title: [Nizoral - an effective and affordable drug to treat vaginal candidiasis ].
Journal: Akusherstvo i ginekologiia 20090101
Title: In vivo active aldosterone synthase inhibitors with improved selectivity: lead optimization providing a series of pyridine substituted 3,4-dihydro-1H-quinolin-2-one derivatives.
Journal: Journal of medicinal chemistry 20081225
Title: Phase III trial of androgen ablation with or without three cycles of systemic chemotherapy for advanced prostate cancer.
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20081220
Title: Use of ketoconazole to treat dogs with pituitary-dependent hyperadrenocorticism: 48 cases (1994-2007).
Journal: Journal of the American Veterinary Medical Association 20081215
Title: Biopositive effects of low-dose UVB on epidermis: coordinate upregulation of antimicrobial peptides and permeability barrier reinforcement.
Journal: The Journal of investigative dermatology 20081201
Title: The combination of chemical and antibody inhibitors for superior P450 3A inhibition in reaction phenotyping studies.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20081201
Title: Effects of an ergosterol synthesis inhibitor on gene transcription of terpenoid biosynthesis in Blakeslea trispora.
Journal: Current microbiology 20081201
Title: Confirmation that cytochrome P450 2C8 (CYP2C8) plays a minor role in (S)-(+)- and (R)-(-)-ibuprofen hydroxylation in vitro.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20081201
Title: A double transgenic mouse model expressing human pregnane X receptor and cytochrome P450 3A4.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20081201
Title: Interindividual variation in relative CYP1A2/3A4 phenotype influences susceptibility of clozapine oxidation to cytochrome P450-specific inhibition in human hepatic microsomes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20081201
Title: Bone-targeted therapy: phase II study of strontium-89 in combination with alternating weekly chemohormonal therapies for patients with advanced androgen-independent prostate cancer.
Journal: American journal of clinical oncology 20081201
Title: Susceptibility to voriconazole, fluconazole, and ketoconazole of yeast isolated from patients with hematological malignancies.
Journal: Journal of chemotherapy (Florence, Italy) 20081201
Title: Presystemic elimination of budesonide in man when administered locally at different levels in the gut, with and without local inhibition by ketoconazole.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20081115
Title: Comparative efficacy and tolerability of Ketomousse (ketoconazole foam 1%) and ketoconazole cream 2% in the treatment of pityriasis versicolor: results of a prospective, multicentre, randomised study.
Journal: Mycoses 20081101
Title: Widespread, chronic, and fluconazole-resistant Trichophyton rubrum infection in an immunocompetent patient.
Journal: Mycoses 20081101
Title: Effect of commonly used herbicides on the virulence factor CDR1 in Candida albicans.
Journal: Environmental toxicology and chemistry 20081101
Title: Hypocortisolemic clamp unmasks jointly feedforward- and feedback-dependent control of overnight ACTH secretion.
Journal: European journal of endocrinology 20081101
Title: Effect of single and repeated doses of ketoconazole on the pharmacokinetics of roflumilast and roflumilast N-oxide.
Journal: Journal of clinical pharmacology 20081101
Title: Pharmacokinetics of the oral direct renin inhibitor aliskiren in combination with digoxin, atorvastatin, and ketoconazole in healthy subjects: the role of P-glycoprotein in the disposition of aliskiren.
Journal: Journal of clinical pharmacology 20081101
Title: Re: Oral ketoconazole for prevention of postoperative penile erection: a placebo controlled, randomized, double-blind trial: B. J. DeCastro, R. A. Costabile, L. P. McMann and A. C. Peterson. J Urol 2008; 179: 1930-1932.
Journal: The Journal of urology 20081101
Title: 1alpha,25-Dihydroxyvitamin D hydroxylase in adipocytes.
Journal: The Journal of steroid biochemistry and molecular biology 20081101
Title: Human CYP3A4-introduced HepG2 cells: in vitro screening system of new chemicals for the evaluation of CYP3A4-inhibiting activity.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20081101
Title: Monodictyochromes A and B, dimeric xanthone derivatives from the marine algicolous fungus Monodictys putredinis.
Journal: Journal of natural products 20081101
Title: In vitro CYP3A4 metabolism: inhibition by Echinacea purpurea and choice of substrate for the evaluation of herbal inhibition.
Journal: Basic & clinical pharmacology & toxicology 20081101
Title: Influence of quinidine, fluvoxamine, and ketoconazole on the enantioselective pharmacokinetics of citalopram in rats.
Journal: Canadian journal of physiology and pharmacology 20081101
Title: Histopathological effect of ketoconazole on rat placenta.
Journal: The Journal of veterinary medical science 20081101
Title: [Mixed vaginitis prevalence in Latin-American women, according to physician perception. Preference, effectiveness and security of clindamycin plus ketoconazole].
Journal: Ginecologia y obstetricia de Mexico 20081101
Title: Activation of the proopiomelanocortin gene with ketoconazole as a treatment for Parkinson's disease: a new hypothesis.
Journal: Annals of the New York Academy of Sciences 20081101
Title: Ketoconazole increases the plasma levels of ivermectin in sheep.
Journal: Veterinary parasitology 20081020
Title: Novel aldosterone synthase inhibitors with extended carbocyclic skeleton by a combined ligand-based and structure-based drug design approach.
Journal: Journal of medicinal chemistry 20081009
Title: Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Journal: Journal of medicinal chemistry 20081009
Title: Condensed bridgehead nitrogen heterocyclic system: synthesis and pharmacological activities of 1,2,4-triazolo-[3,4-b]-1,3,4-thiadiazole derivatives of ibuprofen and biphenyl-4-yloxy acetic acid.
Journal: European journal of medicinal chemistry 20081001
Title: Effect of coadministration of ketoconazole, a strong CYP3A4 inhibitor, on pharmacokinetics and tolerability of motesanib diphosphate (AMG 706) in patients with advanced solid tumors.
Journal: Investigational new drugs 20081001
Title: Maraviroc: in vitro assessment of drug-drug interaction potential.
Journal: British journal of clinical pharmacology 20081001
Title: Differential azole antifungal efficacies contrasted using a Saccharomyces cerevisiae strain humanized for sterol 14 alpha-demethylase at the homologous locus.
Journal: Antimicrobial agents and chemotherapy 20081001
Title: Inhibition of hERG channel trafficking: an under-explored mechanism for drug-induced QT prolongation.
Journal: ChemMedChem 20081001
Title: Management of recurrent and refractory Cushing disease.
Journal: Nature clinical practice. Endocrinology & metabolism 20081001
Title: Medical treatments for male and female pattern hair loss.
Journal: Journal of the American Academy of Dermatology 20081001
Title: Ocular pharmacokinetics of topically-applied ketoconazole solution containing hydroxypropyl beta-cyclodextrin to rabbits.
Journal: Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics 20081001
Title: Evidence for the mechanism of action of the antifungal phytolaccoside B isolated from Phytolacca tetramera Hauman.
Journal: Journal of natural products 20081001
Title: [Synergy between ajoene and ketoconazole in isolates of Microsporum canis. A preliminary study using fractional inhibitory concentration technique (FIC)].
Journal: Revista iberoamericana de micologia 20080930
Title: Screening of herbal constituents for aromatase inhibitory activity.
Journal: Bioorganic & medicinal chemistry 20080915
Title: Enamines as novel antibacterials and their structure-activity relationships.
Journal: European journal of medicinal chemistry 20080901
Title: Differential enzymatic reductions governing the differential hypoxia-selective cytotoxicities of phenazine 5,10-dioxides.
Journal: Chemical research in toxicology 20080901
Title: NO-donors. Part 17: Synthesis and antimicrobial activity of novel ketoconazole-NO-donor hybrid compounds.
Journal: Bioorganic & medicinal chemistry 20080901
Title: In vitro antifungal activity of polyfunctionalized 2-(hetero)arylquinolines prepared through imino Diels-Alder reactions.
Journal: Bioorganic & medicinal chemistry 20080901
Title: Steroidal saponins from the roots of Smilax aspera subsp. mauritanica.
Journal: Chemical & pharmaceutical bulletin 20080901
Title: Responses of the medaka HPG axis PCR array and reproduction to prochloraz and ketoconazole.
Journal: Environmental science & technology 20080901
Title: Comparison of the anti-inflammatory activities of imidazole antimycotics in relation to molecular structure.
Journal: Chemical biology & drug design 20080901
Title: Combined treatment with ketoconazole and cyproterone acetate in a boy with McCune-Albright syndrome and peripheral precocious puberty.
Journal: Journal of endocrinological investigation 20080901
Title: [A limited sampling strategy of phenotyping probe midazolam to predict inhibited activities of hepatic CYP3A in rats].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20080901
Title: Overcoming undesirable CYP1A2 inhibition of pyridylnaphthalene-type aldosterone synthase inhibitors: influence of heteroaryl derivatization on potency and selectivity.
Journal: Journal of medicinal chemistry 20080828
Title: Synthesis, biological evaluation, and molecular modeling of abiraterone analogues: novel CYP17 inhibitors for the treatment of prostate cancer.
Journal: Journal of medicinal chemistry 20080828
Title: Synthesis, biological evaluation, and molecular modeling studies of methylene imidazole substituted biaryls as inhibitors of human 17alpha-hydroxylase-17,20-lyase (CYP17)--part II: Core rigidification and influence of substituents at the methylene bridge.
Journal: Bioorganic & medicinal chemistry 20080815
Title: In situ dissolution testing using potentiometric sensors.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20080807
Title: Cushing's disease in dogs: cabergoline treatment.
Journal: Research in veterinary science 20080801
Title: Effects of ketoconazole and quinidine on pharmacokinetics of pactimibe and its plasma metabolite, R-125528, in humans.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20080801
Title: Pharmacokinetics of darunavir/ritonavir and ketoconazole following co-administration in HIV-healthy volunteers.
Journal: British journal of clinical pharmacology 20080801
Title: Adverse effects of ketoconazole in dogs--a retrospective study.
Journal: Veterinary dermatology 20080801
Title: Dysgonic strain of Microsporum canis pseudomycetoma in a Domestic Long-hair cat.
Journal: Australian veterinary journal 20080801
Title: What's your assessment? Pityrosporum folliculitis.
Journal: Dermatology nursing 20080801
Title: [Effect of ketoconazole on the activity of CYP4503A4 and CYP450 1A2 of hepatic microsomes in healthy adults].
Journal: Nan fang yi ke da xue xue bao = Journal of Southern Medical University 20080801
Title: Microsome biocolloids for rapid drug metabolism and inhibition assessment by LC-MS.
Journal: Drug metabolism letters 20080801
Title: A statistical methodology for drug-drug interaction surveillance.
Journal: Statistics in medicine 20080720
Title: Chemosensitization prevents tolerance of Aspergillus fumigatus to antimycotic drugs.
Journal: Biochemical and biophysical research communications 20080718
Title: New trypanocidal hybrid compounds from the association of hydrazone moieties and benzofuroxan heterocycle.
Journal: Bioorganic & medicinal chemistry 20080715
Title: Synthesis of novel ketoconazole derivatives as inhibitors of the human Pregnane X Receptor (PXR; NR1I2; also termed SXR, PAR).
Journal: Bioorganic & medicinal chemistry letters 20080715
Title: Expression of microsomal lanosterol 14alpha-demethylase (CYP51) in an engineered soluble monomeric form.
Journal: Biochemical and biophysical research communications 20080711
Title: 1-[(3-Aryloxy-3-aryl)propyl]-1H-imidazoles, new imidazoles with potent activity against Candida albicans and dermatophytes. Synthesis, structure-activity relationship, and molecular modeling studies.
Journal: Journal of medicinal chemistry 20080710
Title: A phase I study of docetaxel with ketoconazole modulation in patients with advanced cancers.
Journal: Cancer chemotherapy and pharmacology 20080701
Title: Synthesis and antimicrobial activities of 7-O-modified genistein derivatives.
Journal: European journal of medicinal chemistry 20080701
Title: Long-term treatment of familial male-limited precocious puberty (testotoxicosis) with cyproterone acetate or ketoconazole.
Journal: Clinical endocrinology 20080701
Title: Paecilomyces lilacinus olecranon bursitis in an immunocompromised host: case report and review.
Journal: Diagnostic microbiology and infectious disease 20080701
Title: Prediction of pharmacokinetic drug-drug interactions using human hepatocyte suspension in plasma and cytochrome P450 phenotypic data. II. In vitro-in vivo correlation with ketoconazole.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20080701
Title: Perturbation of gene expression and steroidogenesis with in vitro exposure of fathead minnow ovaries to ketoconazole.
Journal: Marine environmental research 20080701
Title: Potent in vitro antifungal activities of naturally occurring acetylenic acids.
Journal: Antimicrobial agents and chemotherapy 20080701
Title: Evaluation and treatment of oral candidiasis in HIV/AIDS patients in Enugu, Nigeria.
Journal: Oral and maxillofacial surgery 20080701
Title: Synthesis, biochemical evaluation and rationalisation of the inhibitory activity of a range of phenyl alkyl imidazole-based compounds as potent inhibitors of the enzyme complex 17alpha-hydroxylase/17,20-lyase (P450(17alpha)).
Journal: The Journal of steroid biochemistry and molecular biology 20080701
Title: Validation and application of Caco-2 assays for the in vitro evaluation of development candidate drugs as substrates or inhibitors of P-glycoprotein to support regulatory submissions.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20080701
Title: [Ketoconazole and clindamycin efficacy vs oral clindamycin in premature membranes rupture prevention].
Journal: Ginecologia y obstetricia de Mexico 20080701
Title: Biotypes, genotypes and ketoconazole susceptibility of Candida albicans isolates from a group of Thai AIDS patients.
Journal: The new microbiologica 20080701
Title: Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
Journal: Journal of medicinal chemistry 20080612
Title: Differential effects of ketoconazole on exposure to temsirolimus following intravenous infusion of temsirolimus.
Journal: British journal of cancer 20080603
Title: Malassezia folliculitis in China.
Journal: Mycopathologia 20080601
Title: In vitro antifungal susceptibility and molecular characterization of clinical isolates of Fusarium verticillioides (F. moniliforme) and Fusarium thapsinum.
Journal: Antimicrobial agents and chemotherapy 20080601
Title: Biweekly doxorubicin/ketoconazole as second-line treatment in docetaxel-resistant, hormone-refractory prostate cancer.
Journal: Urology 20080601
Title: Cutaneous hyalohyphomycosis caused by a Chrysosporium species related to Nannizziopsis vriesii in two green iguanas (Iguana iguana).
Journal: Medical mycology 20080601
Title: Synthesis and SAR studies of biaryloxy-substituted triazoles as antifungal agents.
Journal: Bioorganic & medicinal chemistry letters 20080601
Title: Safety profile and metabolic effects of 14 days of treatment with DIO-902: results of a phase IIa multicenter, randomized, double-blind, placebo-controlled, parallel-group trial in patients with type 2 diabetes mellitus.
Journal: Clinical therapeutics 20080601
Title: Application of micellar electrokinetic capillary chromatography for evaluation of inhibitory effects on cytochrome P450 reaction.
Journal: Journal of chromatography. A 20080502
Title: Synthesis and antimicrobial activity of novel sulfone-linked bis heterocycles.
Journal: European journal of medicinal chemistry 20080501
Title: An examination of the effect of intestinal first pass extraction on intestinal lymphatic transport of saquinavir in the rat.
Journal: Pharmaceutical research 20080501
Title: A stereospecific high-performance liquid chromatographic assay for the determination of ketoconazole enantiomers in rat plasma.
Journal: Biomedical chromatography : BMC 20080501
Title: Contribution of the N-glucuronidation pathway to the overall in vitro metabolic clearance of midazolam in humans.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20080501
Title: Application of CYP3A4 in vitro data to predict clinical drug-drug interactions; predictions of compounds as objects of interaction.
Journal: British journal of clinical pharmacology 20080501
Title: In vitro inhibition of CYP3A4 metabolism and P-glycoprotein-mediated transport by trade herbal products.
Journal: Basic & clinical pharmacology & toxicology 20080501
Title: Oral ketoconazole for prevention of postoperative penile erection: a placebo controlled, randomized, double-blind trial.
Journal: The Journal of urology 20080501
Title: Identification of the human cytochrome P450 enzymes involved in the in vitro biotransformation of lynestrenol and norethindrone.
Journal: The Journal of steroid biochemistry and molecular biology 20080501
Title: Chiral separations in sub- and supercritical fluid chromatography.
Journal: Journal of separation science 20080501
Title: Identification of human cytochrome P450 enzymes involved in the metabolism of IN-1130, a novel activin receptor-like kinase-5 (ALK5) inhibitor.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20080501
Title: Effects of ketoconazole on the pharmacokinetics and pharmacodynamics of morphine in healthy Greyhounds.
Journal: American journal of veterinary research 20080501
Title: The effect of ketoconazole on the pharmacokinetics and pharmacodynamics of ixabepilone: a first in class epothilone B analogue in late-phase clinical development.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20080501
Title: Selected endocrine disrupting compounds (vinclozolin, flutamide, ketoconazole and dicofol): effects on survival, occurrence of males, growth, molting and reproduction of Daphnia magna.
Journal: Environmental science and pollution research international 20080501
Title: Ketoconazole: a review of a workhorse antifungal molecule with a focus on new foam and gel formulations.
Journal: Drugs of today (Barcelona, Spain : 1998) 20080501
Title: Significance of isolation and drug susceptibility testing of non-Candida albicans species causing oropharyngeal candidiasis in HIV patients.
Journal: The Southeast Asian journal of tropical medicine and public health 20080501
Title: [Effect of polyoxyl ether analogous surfactants on the activity of cytochromes P450 3A in rats in vivo].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20080501
Title: Design, synthesis, and biological evaluation of (hydroxyphenyl)naphthalene and -quinoline derivatives: potent and selective nonsteroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 1 (17beta-HSD1) for the treatment of estrogen-dependent diseases.
Journal: Journal of medicinal chemistry 20080410
Title: New selective inhibitors of steroid 11beta-hydroxylation in the adrenal cortex. Synthesis and structure-activity relationship of potent etomidate analogues.
Journal: Journal of medicinal chemistry 20080410
Title: Spectroscopic and kinetic studies on the interaction of ketoconazole and povidone drugs with DDQ.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20080401
Title: Ketoconazole-induced testicular damage in rats reduced by Gentiana extract.
Journal: Experimental and toxicologic pathology : official journal of the Gesellschaft fur Toxikologische Pathologie 20080401
Title: [Management of hypercortisolism].
Journal: La Revue de medecine interne 20080401
Title: Unexpected emergence of acute hepatic injury in patients treated repeatedly with ketoconazole.
Journal: Journal of clinical gastroenterology 20080401
Title: Effects of CYP3A4 inhibitors on the pharmacokinetics of maraviroc in healthy volunteers.
Journal: British journal of clinical pharmacology 20080401
Title: 'Anti-cortisolic' treatment of warts.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20080401
Title: Combinatorial anti-Trichophyton effects of Ligusticum chuanxiong essential oil components with antibiotics.
Journal: Archives of pharmacal research 20080401
Title: Phaeohyphomycosis caused by Ulocladium species in a cat.
Journal: The Veterinary record 20080329
Title: Predominant role of 25OHD in the negative regulation of PTH expression: clinical relevance for hypovitaminosis D.
Journal: Life sciences 20080326
Title: Synthesis, crystal structure and antimicrobial activity of deoxybenzoin derivatives from genistein.
Journal: European journal of medicinal chemistry 20080301
Title: Inhibition of luteinizing hormone secretion by testosterone in men requires aromatization for its pituitary but not its hypothalamic effects: evidence from the tandem study of normal and gonadotropin-releasing hormone-deficient men.
Journal: The Journal of clinical endocrinology and metabolism 20080301
Title: Mixed inhibition of P450 3A4 as a chemoprotective mechanism against aflatoxin B1-induced cytotoxicity with cis-terpenones.
Journal: Chemical research in toxicology 20080301
Title: A novel ketoconazole bioadhesive effervescent tablet for vaginal delivery: design, in vitro and 'in vivo' evaluation.
Journal: International journal of pharmaceutics 20080227
Title: Synthesis, biological evaluation and molecular modelling studies of methyleneimidazole substituted biaryls as inhibitors of human 17alpha-hydroxylase-17,20-lyase (CYP17). Part I: Heterocyclic modifications of the core structure.
Journal: Bioorganic & medicinal chemistry 20080215
Title: Ethnoveterinary study for antidermatophytic activity of Piper betle, Alpinia galanga and Allium ascalonicum extracts in vitro.
Journal: Research in veterinary science 20080201
Title: Pharmacological evaluation of C-3 modified Betulinic acid derivatives with potent anticancer activity.
Journal: Investigational new drugs 20080201
Title: Antifungal canthin-6-one series accumulate in lipid droplets and affect fatty acid metabolism in Saccharomyces cerevisiae.
Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie 20080201
Title: Coexistence of hERG current block and disruption of protein trafficking in ketoconazole-induced long QT syndrome.
Journal: British journal of pharmacology 20080201
Title: Ketoconazole and the modulation of multidrug resistance-mediated transport in Caco-2 and MDCKII-MDR1 drug transport models.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20080201
Title: Ketoconazole, an antifungal imidazole, increases the sensitivity of rainbow trout to 17alpha-ethynylestradiol exposure.
Journal: Aquatic toxicology (Amsterdam, Netherlands) 20080131
Title: Antifungal and cytotoxic activities of some N-substituted aniline derivatives bearing a hetaryl fragment.
Journal: Bioorganic & medicinal chemistry 20080115
Title: [Prophylactic antifungal treatment in critically ill patients. A survey of a Cochrane review].
Journal: Ugeskrift for laeger 20080107
Title: New triazole and triazolothiadiazine derivatives as possible antimicrobial agents.
Journal: European journal of medicinal chemistry 20080101
Title: Ritonavir 100 mg does not cause QTc prolongation in healthy subjects: a possible role as CYP3A inhibitor in thorough QTc studies.
Journal: Clinical pharmacology and therapeutics 20080101
Title: Biochemical and functional evidence for the control of pain mechanisms by dehydroepiandrosterone endogenously synthesized in the spinal cord.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20080101
Title: Prediction of onset of crystallization from experimental relaxation times. II. Comparison between predicted and experimental onset times.
Journal: Journal of pharmaceutical sciences 20080101
Title: Pharmacokinetic interaction of ketoconazole and itraconazole with ciprofloxacin.
Journal: Biopharmaceutics & drug disposition 20080101
Title: Spectrofluorimetric study and detection of ketoconazole in the presence of beta-cyclodextrin.
Journal: Journal of fluorescence 20080101
Title: N-Phenyl and N-phenylalkyl-maleimides acting against Candida spp.: time-to-kill, stability, interaction with maleamic acids.
Journal: Bioorganic & medicinal chemistry 20080101
Title: Novel cholesterol biosynthesis inhibitors targeting human lanosterol 14alpha-demethylase (CYP51).
Journal: Bioorganic & medicinal chemistry 20080101
Title: The effects of CYP3A4 inhibition on erlotinib pharmacokinetics: computer-based simulation (SimCYP) predicts in vivo metabolic inhibition.
Journal: European journal of clinical pharmacology 20080101
Title: Synthesis, biological evaluation and molecular modelling studies of novel ACD- and ABD-ring steroidomimetics as inhibitors of CYP17.
Journal: Bioorganic & medicinal chemistry letters 20080101
Title: Activity of caspofungin and voriconazole against clinical isolates of Candida and other medically important yeasts by the CLSI M-44A disk diffusion method with Neo-Sensitabs tablets.
Journal: Chemotherapy 20080101
Title: Ketoconazole revisited: a preoperative or postoperative treatment in Cushing's disease.
Journal: European journal of endocrinology 20080101
Title: [Medical treatment for Cushing's syndrome].
Journal: Nihon rinsho. Japanese journal of clinical medicine 20080101
Title: [Ectopic Cushing's syndrome caused by a functioning pancreatic neuroendocrine tumour in a patient with von Hippel-Lindau disease].
Journal: Revista espanola de medicina nuclear 20080101
Title: Novel concepts in androgen receptor blockade.
Journal: Cancer journal (Sudbury, Mass.) 20080101
Title: [Itraconazole treatment in the suspension of pathological fungal colonization of the airway in patients with pulmonary tuberculosis].
Journal: Problemy tuberkuleza i boleznei legkikh 20080101
Title: Dermatophyte susceptibilities to antifungal azole agents tested in vitro by broth macro and microdilution methods.
Journal: Revista do Instituto de Medicina Tropical de Sao Paulo 20080101
Title: The effectiveness of retinoic acid treatment in bladder cancer: impact on recurrence, survival and TGFalpha and VEGF as end-point biomarkers.
Journal: Cancer biology & therapy 20080101
Title: Prevention of bladder cancer recurrence by retinoic acid-ketoconazole: a promising strategy?
Journal: Cancer biology & therapy 20080101
Title: Effect of coadministered ketoconazole, a strong cytochrome P450 3A4 enzyme inhibitor, on the pharmacokinetics of ciclesonide and its active metabolite desisobutyryl-ciclesonide.
Journal: Clinical pharmacokinetics 20080101
Title: The metabolism of amiodarone by various CYP isoenzymes of human and rat, and the inhibitory influence of ketoconazole.
Journal: Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques 20080101
Title: CYP2D6 is primarily responsible for the metabolism of clomiphene.
Journal: Drug metabolism and pharmacokinetics 20080101
Title: [Susceptibility to antifungal agents among Cryptococcus neoformans varieties isolated from patients at a university hospital].
Journal: Revista da Sociedade Brasileira de Medicina Tropical 20080101
Title: Reduction of fluconazole susceptibility of Candida albicans in APECED patients due to long-term use of ketoconazole and miconazole.
Journal: Scandinavian journal of infectious diseases 20080101
Title: [Mycetoma].
Journal: Annales de dermatologie et de venereologie 20080101
Title: Protothecosis as a cause of chronic diarrhoea in a dog.
Journal: Polish journal of veterinary sciences 20080101
Title: A novel approach to the prediction of drug-drug interactions in humans based on the serum incubation method.
Journal: Drug metabolism and pharmacokinetics 20080101
Title: A Bayesian meta-analysis on published sample mean and variance pharmacokinetic data with application to drug-drug interaction prediction.
Journal: Journal of biopharmaceutical statistics 20080101
Title: Diffuse cutaneous leishmaniasis: co-infection with human immunodeficiency virus (HIV).
Journal: Indian journal of dermatology, venereology and leprology 20080101
Title: Tinea nigra by Hortaea werneckii, a report of 22 cases from Mexico.
Journal: Studies in mycology 20080101
Title: [Modern approach to treatment of trophic ulcers of legs with perifocal varicose eczema, associated with mycotic infection].
Journal: Khirurgiia 20080101
Title: Evaluation of the relationship between androgenetic alopecia and demodex infestation.
Journal: Indian journal of dermatology 20080101
Title: [Resistance to azolic compounds in clinical Trichophyton spp. strains].
Journal: Revista iberoamericana de micologia 20071231
Title: Composition, enantiomeric distribution, and antimicrobial activity of Tanacetum argenteum subsp. flabellifolium essential oil.
Journal: Journal of pharmaceutical and biomedical analysis 20071221
Title: Induction of the NAD(P)H:quinone oxidoreductase 1 by ketoconazole and itraconazole: a mechanism of cancer chemoprotection.
Journal: Cancer letters 20071208
Title: Interactions of azole antifungal agents with the human breast cancer resistance protein (BCRP).
Journal: Journal of pharmaceutical sciences 20071201
Title: Identification of human liver cytochrome P450 enzymes involved in biotransformation of vicriviroc, a CCR5 receptor antagonist.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20071201
Title: Cyclic conversion of the novel Src kinase inhibitor [7-(2,6-dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-amine (TG100435) and Its N-oxide metabolite by flavin-containing monoxygenases and cytochrome P450 reductase.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20071201
Title: Effect of hydration on the permeation of ketoconazole through human nail plate in vitro.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20071201
Title: Phase II study of ketoconazole plus granulocyte-macrophage colony-stimulating factor for prostate cancer: effect of extent of disease on outcome.
Journal: The Journal of urology 20071201
Title: Cytochrome P3A4 inhibitors and other constituents of Fibraurea tinctoria.
Journal: Journal of natural products 20071201
Title: Bioactive polychlorinated bibenzyls from the liverwort Riccardia polyclada.
Journal: Journal of natural products 20071201
Title: Pharmacokinetic interaction between ketoconazole and praziquantel in healthy volunteers.
Journal: Journal of clinical pharmacy and therapeutics 20071201
Title: Nodular pulmonary histoplasmosis in Cushing's disease: a case report and literature review.
Journal: Tennessee medicine : journal of the Tennessee Medical Association 20071201
Title: Quantitative correlations among CYP3A sensitive substrates and inhibitors: literature analysis.
Journal: Current drug metabolism 20071201
Title: In vivo anti-Chagas vinylthio-, vinylsulfinyl-, and vinylsulfonylbenzofuroxan derivatives.
Journal: Journal of medicinal chemistry 20071129
Title: Induction of drought stress tolerance by ketoconazole in Catharanthus roseus is mediated by enhanced antioxidant potentials and secondary metabolite accumulation.
Journal: Colloids and surfaces. B, Biointerfaces 20071115
Title: Rational prescription of drugs within similar therapeutic or structural class for gastrointestinal disease treatment: drug metabolism and its related interactions.
Journal: World journal of gastroenterology 20071114
Title: Adaptive therapy for androgen-independent prostate cancer: a randomized selection trial of four regimens.
Journal: Journal of the National Cancer Institute 20071107
Title: Pharmacokinetic modulation of oral etoposide by ketoconazole in patients with advanced cancer.
Journal: Cancer chemotherapy and pharmacology 20071101
Title: The cytochrome p450 inhibitor ketoconazole potentiates 5-hydroxytryptamine-induced contraction in rat aorta.
Journal: The Journal of pharmacology and experimental therapeutics 20071101
Title: Use of isolated hepatocyte preparations for cytochrome P450 inhibition studies: comparison with microsomes for Ki determination.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20071101
Title: Synthesis and antifungal activities of novel 2-aminotetralin derivatives.
Journal: Journal of medicinal chemistry 20071101
Title: Cytotoxic doses of ketoconazole affect expression of a subset of hepatic genes.
Journal: Journal of toxicology and environmental health. Part A 20071101
Title: [Malassezia folliculitis: characteristics and therapeutic response in 26 patients].
Journal: Annales de dermatologie et de venereologie 20071101
Title: Formulation compatibility of myristyl nicotinate with drugs used to treat dermatological conditions involving an impaired skin barrier.
Journal: Drug development and industrial pharmacy 20071101
Title: Pharmacological management of Cushing's syndrome: an update.
Journal: Arquivos brasileiros de endocrinologia e metabologia 20071101
Title: 33-Year-old man with cough, fever, and weight loss.
Journal: Mayo Clinic proceedings 20071001
Title: Metabolism of tacrolimus (FK506) and recent topics in clinical pharmacokinetics.
Journal: Drug metabolism and pharmacokinetics 20071001
Title: A novel foam formulation of ketoconazole 2% for the treatment of seborrheic dermatitis on multiple body regions.
Journal: Journal of drugs in dermatology : JDD 20071001
Title: Efficacy of low-dose ketoconazole in hormone refractory prostate cancer patients at the National Cancer Centre and The Cancer Institute, Singapore.
Journal: Annals of the Academy of Medicine, Singapore 20071001
Title: The role of ketoconazole in seborrheic dermatitis.
Journal: Cutis 20071001
Title: Effect of one month ketoconazole treatment on GH, cortisol and ACTH release after ghrelin, GHRP-6 and GHRH administration in patients with Cushing's disease.
Journal: Arquivos brasileiros de endocrinologia e metabologia 20071001
Title: [Metabolic products and pathway of neferine in rat liver].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20071001
Title: Drug-drug interaction prediction: a Bayesian meta-analysis approach.
Journal: Statistics in medicine 20070910
Title: Influence of ketoconazole on the fecal and urinary disposition of docetaxel.
Journal: Cancer chemotherapy and pharmacology 20070901
Title: Diagnosis and treatment of ocular coccidioidomycosis in a female captive chimpanzee (Pan troglodytes): a case study.
Journal: Annals of the New York Academy of Sciences 20070901
Title: Synthesis of novel triazole derivatives as inhibitors of cytochrome P450 14alpha-demethylase (CYP51).
Journal: European journal of medicinal chemistry 20070901
Title: Azole therapy of clinical and experimental coccidioidomycosis.
Journal: Annals of the New York Academy of Sciences 20070901
Title: Ciclosporin use in multi-drug therapy for meningoencephalomyelitis of unknown aetiology in dogs.
Journal: The Journal of small animal practice 20070901
Title: Effects of endocrine disrupting chemicals on expression of phospholipid hydroperoxide glutathione peroxidase mRNA in rat testes.
Journal: Journal of veterinary science 20070901
Title: Restoration of hormonal action and muscle protein.
Journal: Critical care medicine 20070901
Title: Effective treatment for dermatophytoses of the foot: effect on restoration of depressed cell-mediated immunity.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20070901
Title: Candida interface keratitis after deep anterior lamellar keratoplasty: clinical, microbiologic, histopathologic, and confocal microscopic reports.
Journal: Cornea 20070901
Title: Ketoconazole in the treatment of chronic idiopathic central serous chorioretinopathy.
Journal: Retina (Philadelphia, Pa.) 20070901
Title: Development of an in vivo rat screen model to predict pharmacokinetic interactions of CYP3A4 substrates.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20070901
Title: Raman, FT-IR, NMR spectroscopic data and antimicrobial activity of bis[micro2-(benzimidazol-2-yl)-2-ethanethiolato-N,S,S-chloro-palladium(II)] dimer, [(micro2-CH2CH2NHNCC6H4)PdCl]2.C2H5OH complex.
Journal: European journal of medicinal chemistry 20070801
Title: Antiepileptic drugs affect neuronal androgen signaling via a cytochrome P450-dependent pathway.
Journal: The Journal of pharmacology and experimental therapeutics 20070801
Title: Transcription of key genes regulating gonadal steroidogenesis in control and ketoconazole- or vinclozolin-exposed fathead minnows.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20070801
Title: Combination of surgical avulsion and topical therapy for single nail onychomycosis: a randomized controlled trial.
Journal: The British journal of dermatology 20070801
Title: Activity of ketoconazole against Mycobacterium tuberculosis in vitro and in the mouse model.
Journal: Journal of medical microbiology 20070801
Title: Tinea capitis: no incision nor excision.
Journal: Journal of pediatric surgery 20070801
Title: Ketoconazole is inferior to ritonavir as an alternative booster for saquinavir in a once daily regimen in Thai HIV-1 infected patients.
Journal: AIDS (London, England) 20070731
Title: The prokinetic cinitapride has no clinically relevant pharmacokinetic interaction and effect on QT during coadministration with ketoconazole.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070701
Title: Eumycetoma presenting as a cerebellopontine angle mass lesion.
Journal: Clinical neurology and neurosurgery 20070701
Title: In vitro susceptibilities of 217 clinical isolates of zygomycetes to conventional and new antifungal agents.
Journal: Antimicrobial agents and chemotherapy 20070701
Title: Cytochrome P450-dependent metabolism of vitamin E isoforms is a critical determinant of their tissue concentrations in rats.
Journal: Lipids 20070701
Title: Identification and in vitro antifungal susceptibility testing of 200 clinical isolates of Candida spp. responsible for fingernail infections.
Journal: Mycopathologia 20070701
Title: Comparison between fluconazole and ketoconazole effectivity in the treatment of pityriasis versicolor.
Journal: Mycoses 20070701
Title: Oral paracoccidioidomycosis: a case without lung manifestations.
Journal: The journal of contemporary dental practice 20070701
Title: Melanin biosynthesis in Madurella mycetomatis and its effect on susceptibility to itraconazole and ketoconazole.
Journal: Microbes and infection 20070701
Title: Preparation, characterization, and scale-up of ketoconazole with enhanced dissolution and bioavailability.
Journal: Drug development and industrial pharmacy 20070701
Title: Tailored hormonal therapy in secretory adrenocortical cancer.
Journal: Annals of oncology : official journal of the European Society for Medical Oncology 20070701
Title: [Enzyme kinetics of schizandrin metabolism and sex differences in rat liver microsomes].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20070701
Title: Optimisation of hydrocortisone production by Curvularia lunata.
Journal: Applied biochemistry and biotechnology 20070701
Title: Comparison of fast liquid chromatography/tandem mass spectrometric methods for simultaneous determination of cladribine and clofarabine in mouse plasma.
Journal: Journal of pharmaceutical and biomedical analysis 20070628
Title: Discovery of novel indazole-linked triazoles as antifungal agents.
Journal: Bioorganic & medicinal chemistry letters 20070615
Title: Possible inhibitory mechanism of Curcuma drugs on CYP3A4 in 1alpha,25 dihydroxyvitamin D3 treated Caco-2 cells.
Journal: International journal of pharmaceutics 20070607
Title: Hepatitis and rhabdomyolysis in a patient with hormone refractory prostate cancer on ketoconazole and concurrent lovastatin therapy.
Journal: Investigational new drugs 20070601
Title: Pharmacological prevention of the deleterious effects of cardiopulmonary bypass.
Journal: Asian cardiovascular & thoracic annals 20070601
Title: A new ketoconazole topical gel formulation in seborrhoeic dermatitis: an updated review of the mechanism.
Journal: Expert opinion on pharmacotherapy 20070601
Title: Ketoconazole in the fathead minnow (Pimephales promelas): reproductive toxicity and biological compensation.
Journal: Environmental toxicology and chemistry 20070601
Title: Life-threatening Pneumocystis jiroveci pneumonia following treatment of severe Cushing's syndrome.
Journal: The Netherlands journal of medicine 20070601
Title: Non-interventional management of obstructive acute renal-failure in hormone-naïve prostate cancer.
Journal: The Canadian journal of urology 20070601
Title: Electrochemical reduction of sterol-14alpha-demethylase from Mycobacterium tuberculosis (CYP51b1).
Journal: Biochemistry. Biokhimiia 20070601
Title: Ketoconazole gel 2% in the treatment of moderate to severe seborrheic dermatitis.
Journal: Cutis 20070601
Title: [Mediastinal lymph nodes during the course of a metastatic prostate cancer].
Journal: Actas urologicas espanolas 20070601
Title: Schistosoma haematobium and urinary tract pathogens co-infections in a rural community of Edo State, Nigeria.
Journal: The Journal of communicable diseases 20070601
Title: A lesson for everyone in drug-drug interactions.
Journal: International journal of cardiology 20070516
Title: MgMfs1, a major facilitator superfamily transporter from the fungal wheat pathogen Mycosphaerella graminicola, is a strong protectant against natural toxic compounds and fungicides.
Journal: Fungal genetics and biology : FG & B 20070501
Title: Induction of cytochrome P450 1A1 by ketoconazole and itraconazole but not fluconazole in murine and human hepatoma cell lines.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20070501
Title: Sequential metabolism is responsible for diltiazem-induced time-dependent loss of CYP3A.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070501
Title: Antifungal susceptibility testing of Trichophyton rubrum by E-test.
Journal: Archives of dermatological research 20070501
Title: Effect of efavirenz on the pharmacokinetics of ketoconazole in HIV-infected patients.
Journal: European journal of clinical pharmacology 20070501
Title: Cytochrome P450 3A inhibition by ketoconazole affects prasugrel and clopidogrel pharmacokinetics and pharmacodynamics differently.
Journal: Clinical pharmacology and therapeutics 20070501
Title: Estimation of intragastric solubility of drugs: in what medium?
Journal: Pharmaceutical research 20070501
Title: Electrochemical properties of cytochroms P450 using nanostructured electrodes: direct electron transfer and electro catalysis.
Journal: Journal of inorganic biochemistry 20070501
Title: Lecythophora hoffmannii isolated from a case of canine osteomyelitis in Japan.
Journal: Medical mycology 20070501
Title: Flutrimazole shampoo 1% versus ketoconazole shampoo 2% in the treatment of pityriasis versicolor. A randomised double-blind comparative trial.
Journal: Mycoses 20070501
Title: Plasma pharmacokinetics and CYP3A12-dependent metabolism of c-kit inhibitor imatinib in dogs.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20070501
Title: Interventions for treating oral candidiasis for patients with cancer receiving treatment.
Journal: The Cochrane database of systematic reviews 20070418
Title: Activated pregnenolone X-receptor is a target for ketoconazole and its analogs.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20070415
Title: Antifungal treatment in sarcoidosis--a pilot intervention trial.
Journal: Respiratory medicine 20070401
Title: Characterization of hot-melt extruded drug delivery systems for onychomycosis.
Journal: European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V 20070401
Title: Synthesis and antimicrobial activities of Schiff bases derived from 5-chloro-salicylaldehyde.
Journal: European journal of medicinal chemistry 20070401
Title: Luteinizing hormone-induced caspase activation in rat preovulatory follicles is coupled to mitochondrial steroidogenesis.
Journal: Endocrinology 20070401
Title: Deacetylclivorine: a gender-selective metabolite of clivorine formed in female Sprague-Dawley rat liver microsomes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070401
Title: Second generation of 5-ethenylbenzofuroxan derivatives as inhibitors of Trypanosoma cruzi growth: synthesis, biological evaluation, and structure-activity relationships.
Journal: Bioorganic & medicinal chemistry 20070401
Title: Synthesis of DL-standishinal and its related compounds for the studies on structure-activity relationship of inhibitory activity against aromatase.
Journal: Bioorganic & medicinal chemistry 20070401
Title: In vitro activity of an ear rinse containing tromethamine, EDTA, benzyl alcohol and 0.1% ketoconazole on Malassezia organisms from dogs with otitis externa.
Journal: Veterinary dermatology 20070401
Title: Adrenal androgen levels as predictors of outcome in prostate cancer patients treated with ketoconazole plus antiandrogen withdrawal: results from a cancer and leukemia group B study.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20070401
Title: Pharmacokinetic modelling of pentoxifylline and lisofylline after oral and intravenous administration in mice.
Journal: The Journal of pharmacy and pharmacology 20070401
Title: [Lithium gluconate 8% in the treatment of seborrheic dermatitis].
Journal: Annales de dermatologie et de venereologie 20070401
Title: Inhibitory or scavenging action of ketoconazole and ciclopiroxolamine against reactive oxygen species released by primed inflammatory cells.
Journal: The British journal of dermatology 20070401
Title: Effect of ion suppression on judgment of enzyme inhibition and avoidance of error by utilizing a stable isotope-labeled probe substrate: example of CYP3A4 inhibition with [13C4,15N] labeled midazolam as a substrate.
Journal: Drug metabolism and pharmacokinetics 20070401
Title: [Cushing syndrome].
Journal: Revue de l'infirmiere 20070401
Title: [Effectiveness of the treatment plan for androgenetic alopecia].
Journal: Georgian medical news 20070401
Title: Eumycetoma pedis due to Exophiala jeanselmei.
Journal: Indian journal of medical microbiology 20070401
Title: The development of a cocktail CYP2B6, CYP2C8, and CYP3A5 inhibition assay and a preliminary assessment of utility in a drug discovery setting.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070301
Title: Effect of oral ketoconazole on intestinal first-pass effect of midazolam and fexofenadine in cynomolgus monkeys.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070301
Title: Three-dimensional quantitative structure-activity relationship analysis of human CYP51 inhibitors.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070301
Title: Antifungal activities of azole agents against the Malassezia species.
Journal: International journal of antimicrobial agents 20070301
Title: Development of quantitative real-time PCR assays for fathead minnow (Pimephales promelas) gonadotropin beta subunit mRNAs to support endocrine disruptor research.
Journal: Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20070301
Title: Potential cancer chemopreventive in vitro activities of monomeric xanthone derivatives from the marine algicolous fungus Monodictys putredinis.
Journal: Journal of natural products 20070301
Title: Potentiating effects of nonactive/active vitamin D analogues and ketoconazole in parathyroid cells.
Journal: Clinical endocrinology 20070301
Title: Metronidazole 0.75% gel vs. ketoconazole 2% cream in the treatment of facial seborrheic dermatitis: a randomized, double-blind study.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20070301
Title: Clinical inquiries. What's the best treatment for cradle cap?
Journal: The Journal of family practice 20070301
Title: Antiplasmodial interactions between artemisinin and triclosan or ketoconazole combinations against blood stages of Plasmodium falciparum in vitro.
Journal: The American journal of tropical medicine and hygiene 20070301
Title: Report of an imported cutaneous disseminated case of paracoccidioidomycosis.
Journal: Revista iberoamericana de micologia 20070301
Title: Hyperadrenocorticism: treating dogs.
Journal: Compendium (Yardley, PA) 20070301
Title: CP-154,526, a CRF type-1 receptor antagonist, attenuates the cue-and methamphetamine-induced reinstatement of extinguished methamphetamine-seeking behavior in rats.
Journal: Psychopharmacology 20070201
Title: Evidence of Oatp and Mdr1 in cryopreserved rat hepatocytes.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20070201
Title: Synthesis, characterization and antimicrobial activity of Fe(II), Zn(II), Cd(II) and Hg(II) complexes with 2,6-bis(benzimidazol-2-yl) pyridine ligand.
Journal: European journal of medicinal chemistry 20070201
Title: Inhibition of CYP3A4 and CYP3A5 catalyzed metabolism of alprazolam and quinine by ketoconazole as racemate and four different enantiomers.
Journal: European journal of clinical pharmacology 20070201
Title: Transporter-mediated drug interactions: clinical implications and in vitro assessment.
Journal: Expert opinion on drug metabolism & toxicology 20070201
Title: [A text-book case of tropical facial elephantiasis].
Journal: Revue de stomatologie et de chirurgie maxillo-faciale 20070201
Title: Concentrations of mycophenolic acid and glucuronide metabolites under concomitant therapy with cyclosporine or tacrolimus.
Journal: Therapeutic drug monitoring 20070201
Title: [Oral isolates of Saccharomyces in patients with oral fungal infection and their susceptibility to antifungal drugs].
Journal: Hua xi kou qiang yi xue za zhi = Huaxi kouqiang yixue zazhi = West China journal of stomatology 20070201
Title: [Acanthamoeba keratitis: about the first two Tunisian cases].
Journal: Bulletin de la Societe de pathologie exotique (1990) 20070201
Title: [Cutaneous sporotricosis in a Malagasy patient].
Journal: Medecine tropicale : revue du Corps de sante colonial 20070201
Title: Determination of antifungal activity of polyenzyme preparation Candidaseb using in vitro methods.
Journal: Hindustan antibiotics bulletin 20070201
Title: Inhibition of drug metabolism by blocking the activation of nuclear receptors by ketoconazole.
Journal: Oncogene 20070111
Title: Effects of three cytochrome P450 inhibitors, ketoconazole, fluconazole, and paroxetine, on the pharmacokinetics of lasofoxifene.
Journal: British journal of clinical pharmacology 20070101
Title: Reversal of androgenetic alopecia by topical ketoconzole: relevance of anti-androgenic activity.
Journal: Journal of dermatological science 20070101
Title: A novel model for the prediction of drug-drug interactions in humans based on in vitro cytochrome p450 phenotypic data.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20070101
Title: Synthesis and antifungal activity of (Z)-5-arylidenerhodanines.
Journal: Bioorganic & medicinal chemistry 20070101
Title: Design of endoperoxides with anti-Candida activity.
Journal: Bioorganic & medicinal chemistry 20070101
Title: Molecular evidence and functional expression of multidrug resistance associated protein (MRP) in rabbit corneal epithelial cells.
Journal: Experimental eye research 20070101
Title: Antimicrobial effectiveness of ketoconazole against metronidazole-resistant Helicobacter pylori isolates from Iranian dyspeptic patients.
Journal: The Journal of antimicrobial chemotherapy 20070101
Title: The stereoselective metabolism of halofantrine to desbutylhalofantrine in the rat: evidence of tissue-specific enantioselectivity in microsomal metabolism.
Journal: Chirality 20070101
Title: CYP3A4 mediated in vitro metabolism of vinflunine in human liver microsomes.
Journal: Acta pharmacologica Sinica 20070101
Title: 1H NMR monitoring of the canine metabolic profile after oral administration of xenobiotics using multivariate statistics.
Journal: Molecular pharmaceutics 20070101
Title: Value of colposcopy in the diagnosis of candidiasis in patients with vulvodynia.
Journal: The Journal of reproductive medicine 20070101
Title: Simultaneous determination of docetaxel and ketoconazole in rat plasma by liquid chromatography/electrospray ionization tandem mass spectrometry.
Journal: Rapid communications in mass spectrometry : RCM 20070101
Title: Comparison of different perrmeation enhancers on topical ketoconazole formulations.
Journal: Arzneimittel-Forschung 20070101
Title: Human intestinal P-glycoprotein activity estimated by the model substrate digoxin.
Journal: Scandinavian journal of clinical and laboratory investigation 20070101
Title: Ketoconazole therapy: an efficacious alternative to achieve eucortisolism in patients with Cushing's syndrome.
Journal: Medicina 20070101
Title: Antiviral and antimicrobial profiles of selected isoquinoline alkaloids from Fumaria and Corydalis species.
Journal: Zeitschrift fur Naturforschung. C, Journal of biosciences 20070101
Title: Abdominal wall mycetoma presented as obstructed incisional hernia of cesarean section in eastern Sudan.
Journal: Infectious diseases in obstetrics and gynecology 20070101
Title: Significant prostate-specific antigen (PSA) response to low-dose ketoconazole in a patient with non-metastatic androgen-independent prostate cancer (AIPC) and a review of the literature.
Journal: American journal of therapeutics 20070101
Title: Pharmacokinetics of cinacalcet hydrochloride when administered with ketoconazole.
Journal: Clinical pharmacokinetics 20070101
Title: Clinical efficacies of shampoos containing ciclopirox olamine (1.5%) and ketoconazole (2.0%) in the treatment of seborrhoeic dermatitis.
Journal: The Journal of dermatological treatment 20070101
Title: Simultaneous ectopic adrenocorticotropic hormone syndrome and adrenal metastasis of a medullary thyroid carcinoma causing paraneoplastic Cushing's syndrome.
Journal: International seminars in surgical oncology : ISSO 20070101
Title: Extina foam (2%).
Journal: Skinmed 20070101
Title: Multiple oral dosing of ketoconazole increases dog exposure to ivermectin.
Journal: Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques 20070101
Title: Ketoconazole-evoked [Ca2+]i rises and non-Ca2+-triggered cell death in rabbit corneal epithelial cells (SIRC).
Journal: Journal of receptor and signal transduction research 20070101
Title: [Quo vadis, hypophysis? Some news and prospects].
Journal: Vnitrni lekarstvi 20070101
Title: Localized cutaneous leishmaniasis in South India: successful treatment with ketoconazole.
Journal: Indian journal of dermatology, venereology and leprology 20070101
Title: CYP3A4 and pregnane X receptor humanized mice.
Journal: Journal of biochemical and molecular toxicology 20070101
Title: [The 50th Anniversary Educational Symposium of the Japanese Society for Medical Mycology: Dermatomycoses caused by Malassezia].
Journal: Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20070101
Title: Effect of hypercortisolism control on high blood pressure in Cushing's syndrome.
Journal: Medicina 20070101
Title: Identification of CYP3A4 as the primary cytochrome P450 responsible for the metabolism of tandospirone by human liver microsomes.
Journal: European journal of drug metabolism and pharmacokinetics 20070101
Title: In vitro release--in vivo microbiological and toxicological studies on ketoconazole lipid granules.
Journal: Pharmaceutical development and technology 20070101
Title: Identification of CYP3A4 as the primary cytochrome P450 responsible for the metabolism of tandospirone by human liver microsomes.
Journal: European journal of drug metabolism and pharmacokinetics 20070101
Title: In vitro antifungal activity of 2-(4-substituted phenyl)-3(2H)-isothiazolones.
Journal: Folia microbiologica 20070101
Title: Pregnenolone and dexamethasone, modulators of cytochrome P450-3A, not increase but reduce urinary alpha-CEHC excretion in rats.
Journal: BioFactors (Oxford, England) 20070101
Title: Seborrhoeic dermatitis.
Journal: BMJ clinical evidence 20070101
Title: Treatment algorithm in hormone-resistant prostate cancer: Practical guidelines.
Journal: Indian journal of urology : IJU : journal of the Urological Society of India 20070101
Title: Repeated 28-day oral toxicity study of ketoconazole in rats based on the draft protocol for the 'Enhanced OECD Test Guideline No. 407' to detect endocrine effects.
Journal: Archives of toxicology 20061201
Title: The role of P-glycoprotein in the bioactivation of raloxifene.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20061201
Title: Drug-metabolizing enzyme inhibition by ketoconazole does not reduce interindividual variability of CYP3A activity as measured by oral midazolam.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20061201
Title: Antifungal susceptibilities of the species of the Pseudallescheria boydii complex.
Journal: Antimicrobial agents and chemotherapy 20061201
Title: Antifolates as antimycotics? Connection between the folic acid cycle and the ergosterol biosynthesis pathway in Candida albicans.
Journal: International journal of antimicrobial agents 20061201
Title: Cytochrome P450-dependent metabolism of midazolam in hepatic microsomes from chickens, turkeys, pheasant and bobwhite quail.
Journal: Journal of veterinary pharmacology and therapeutics 20061201
Title: White piedra in children.
Journal: Journal of the American Academy of Dermatology 20061201
Title: In vitro antifungal efficacy of ciclopirox olamine alone and associated with zinc pyrithione compared to ketoconazole against Malassezia globosa and Malassezia restricta reference strains.
Journal: Mycopathologia 20061201
Title: Mechanisms of venoocclusive disease resulting from the combination of cyclophosphamide and roxithromycin.
Journal: Therapeutic drug monitoring 20061201
Title: Preoperative immunosuppressive therapy and surgery as a treatment for anal furunculosis.
Journal: Veterinary surgery : VS 20061201
Title: Bioactive oligostilbenoids from the stem bark of Hopea exalata.
Journal: Journal of natural products 20061201
Title: Evaluation of the effects of hydrophilic organic solvents on CYP3A-mediated drug-drug interaction in vitro.
Journal: Human & experimental toxicology 20061201
Title: [Study on metabolism of tetramethylpyrazine in system of rat liver microsomes].
Journal: Zhongguo Zhong yao za zhi = Zhongguo zhongyao zazhi = China journal of Chinese materia medica 20061201
Title: [Canine lymphadenitis caused by Cryptococcus neoformans. First case in Chile].
Journal: Revista iberoamericana de micologia 20061201
Title: Common pharmacophores for uncharged human ether-a-go-go-related gene (hERG) blockers.
Journal: Journal of medicinal chemistry 20061116
Title: Human adrenocarcinoma (H295R) cells for rapid in vitro determination of effects on steroidogenesis: hormone production.
Journal: Toxicology and applied pharmacology 20061115
Title: The H295R system for evaluation of endocrine-disrupting effects.
Journal: Ecotoxicology and environmental safety 20061101
Title: Effectiveness and tolerability of a standardized extract from Ageratina pichinchensis on patients with tinea pedis: an explorative pilot study controlled with ketoconazole.
Journal: Planta medica 20061101
Title: In vitro methods for antifungal susceptibility testing of Trichophyton spp.
Journal: Mycological research 20061101
Title: Otomycosis: clinical features and treatment implications.
Journal: Otolaryngology--head and neck surgery : official journal of American Academy of Otolaryngology-Head and Neck Surgery 20061101
Title: OPC-67683, a nitro-dihydro-imidazooxazole derivative with promising action against tuberculosis in vitro and in mice.
Journal: PLoS medicine 20061101
Title: Inhibition of the enzymatic activity of heme oxygenases by azole-based antifungal drugs.
Journal: The Journal of pharmacology and experimental therapeutics 20061001
Title: Characterization of the rhesus monkey CYP3A64 enzyme: species comparisons of CYP3A substrate specificity and kinetics using baculovirus-expressed recombinant enzymes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20061001
Title: Metabolism of endosulfan-alpha by human liver microsomes and its utility as a simultaneous in vitro probe for CYP2B6 and CYP3A4.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20061001
Title: Influence of tartaric acid on the bioadhesion and mechanical properties of hot-melt extruded hydroxypropyl cellulose films for the human nail.
Journal: Drug development and industrial pharmacy 20061001
Title: Decision support tool to individualize cyclosporine dose in stable, long-term heart transplant recipients receiving metabolic inhibitors: overcoming limitations of cyclosporine C2 monitoring.
Journal: The Journal of heart and lung transplantation : the official publication of the International Society for Heart Transplantation 20061001
Title: In-vitro susceptibility testing by agar dilution method to determine the minimum inhibitory concentrations of amphotericin B, fluconazole and ketoconazole against ocular fungal isolates.
Journal: Indian journal of medical microbiology 20061001
Title: A fission yeast-based test system for the determination of IC50 values of anti-prostate tumor drugs acting on CYP21.
Journal: Journal of enzyme inhibition and medicinal chemistry 20061001
Title: Evidence for cytochrome P450 3A expression and catalytic activity in rat blood lymphocytes.
Journal: Life sciences 20060927
Title: Synthesis, biochemical evaluation and rationalisation of the inhibitory activity of a range of 4-substituted phenyl alkyl imidazole-based inhibitors of the enzyme complex 17alpha-hydroxylase/17,20-lyase (P450(17alpha)).
Journal: Bioorganic & medicinal chemistry letters 20060915
Title: Retinoic acid as a novel medical therapy for Cushing's disease in dogs.
Journal: Endocrinology 20060901
Title: Response to low-dose ketoconazole and subsequent dose escalation to high-dose ketoconazole in patients with androgen-independent prostate cancer.
Journal: Cancer 20060901
Title: Disopyramide: although potentially life-threatening in the setting of long QT, could it be life-saving in short QT syndrome?
Journal: Journal of molecular and cellular cardiology 20060901
Title: Metabolism and metabolic inhibition of gambogic acid in rat liver microsomes.
Journal: Acta pharmacologica Sinica 20060901
Title: Metabolic activation of pradefovir by CYP3A4 and its potential as an inhibitor or inducer.
Journal: Antimicrobial agents and chemotherapy 20060901
Title: RAT CYP3A and CYP2B1/2 were not associated with nevirapine-induced hepatotoxicity.
Journal: Methods and findings in experimental and clinical pharmacology 20060901
Title: Intervention at the level of the neuroendocrine-immune axis and postoperative pneumonia rate in long-term alcoholics.
Journal: American journal of respiratory and critical care medicine 20060815
Title: Suppressive effects of antimycotics on tumor necrosis factor-alpha-induced CCL27, CCL2, and CCL5 production in human keratinocytes.
Journal: Biochemical pharmacology 20060814
Title: The use of a fluorescence-based oxygen uptake assay in the analysis of cytotoxicity.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20060801
Title: Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: design, synthesis, and microbiological evaluation.
Journal: Bioorganic & medicinal chemistry 20060801
Title: Inhibition of UDP-glucuronosyltransferase 2b7-catalyzed morphine glucuronidation by ketoconazole: dual mechanisms involving a novel noncompetitive mode.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060801
Title: Activating mutations in the luteinizing hormone receptor gene: a human model of non-follicle-stimulating hormone-dependent inhibin production and germ cell maturation.
Journal: The Journal of clinical endocrinology and metabolism 20060801
Title: Synthesis and biochemical evaluation of a range of potent benzyl imidazole-based compounds as potential inhibitors of the enzyme complex 17alpha-hydroxylase/17,20-lyase (P450(17alpha)).
Journal: Bioorganic & medicinal chemistry letters 20060801
Title: Use of omeprazole sulfone in a single plasma sample as a probe for CYP3A4.
Journal: European journal of clinical pharmacology 20060801
Title: Secondary hormonal manipulations in prostate cancer.
Journal: Hematology/oncology clinics of North America 20060801
Title: Transporter-mediated intestinal absorption of fexofenadine in rats.
Journal: Drug metabolism and pharmacokinetics 20060801
Title: Cushing's paraneoplastic syndrome as first manifestation of an adenocarcinoma of unknown origin.
Journal: Clinical & translational oncology : official publication of the Federation of Spanish Oncology Societies and of the National Cancer Institute of Mexico 20060801
Title: Optimization and validation of a high-performance liquid chromatographic method with UV detection for the determination of ketoconazole in canine plasma.
Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20060724
Title: Enhancement of DMNQ-induced hepatocyte toxicity by cytochrome P450 inhibition.
Journal: Toxicology and applied pharmacology 20060715
Title: Clinical results of topical fluconazole for the treatment of filamentous fungal keratitis.
Journal: Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie 20060701
Title: Stereoselective metabolism of endosulfan by human liver microsomes and human cytochrome P450 isoforms.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060701
Title: Quinacrine is mainly metabolized to mono-desethyl quinacrine by CYP3A4/5 and its brain accumulation is limited by P-glycoprotein.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060701
Title: Expression, purification, and characterization of mouse CYP2d22.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060701
Title: Ketoconazole and miconazole are antagonists of the human glucocorticoid receptor: consequences on the expression and function of the constitutive androstane receptor and the pregnane X receptor.
Journal: Molecular pharmacology 20060701
Title: Stochastic prediction of CYP3A-mediated inhibition of midazolam clearance by ketoconazole.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060701
Title: Influence of high-dose ketoconazole on the pharmacokinetics of docetaxel.
Journal: Cancer biology & therapy 20060701
Title: In vitro susceptibilities of Malaysian clinical isolates of Cryptococcus neoformans var. grubii and Cryptococcus gattii to five antifungal drugs.
Journal: Mycoses 20060701
Title: Predictive power of an in vitro system to assess drug interactions of an antimuscarinic medication: a comparison of in vitro and in vivo drug-drug interaction studies of trospium chloride with digoxin.
Journal: Journal of clinical pharmacology 20060701
Title: Pharmacokinetic effect of ketoconazole on solifenacin in healthy volunteers.
Journal: Basic & clinical pharmacology & toxicology 20060701
Title: Phytochemistry and antifungal properties of the newly discovered tree Pleodendron costaricense.
Journal: Journal of natural products 20060701
Title: Chronic mucocutaneous candidiasis associated with malignant thymoma and systemic lupus erythematosus with hypergammaglobulinemia: a case report and literature review.
Journal: Cutis 20060701
Title: Interaction between ketoconazole and domperidone and the risk of QT prolongation--important safety information.
Journal: South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde 20060701
Title: Pharmacokinetic interaction between ketoconazole and SPP301 in healthy volunteers.
Journal: International journal of clinical pharmacology and therapeutics 20060701
Title: Biotransformation of fluticasone: in vitro characterization.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060601
Title: Comparison of mouse and rat cytochrome P450-mediated metabolism in liver and intestine.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060601
Title: Phase II study of mitoxantrone and ketoconazole for hormone-refractory prostate cancer.
Journal: Cancer 20060601
Title: In vitro antifungal activities of Allium cepa, Allium sativum and ketoconazole against some pathogenic yeasts and dermatophytes.
Journal: Fitoterapia 20060601
Title: Man versus machine: is there an optimal method for QT measurements in thorough QT studies?
Journal: Journal of clinical pharmacology 20060601
Title: Cytoskeleton reassembly in cardiomyocytes infected by Trypanosoma cruzi is triggered by treatment with ergosterol biosynthesis inhibitors.
Journal: International journal of antimicrobial agents 20060601
Title: Canine intestinal contents vs. simulated media for the assessment of solubility of two weak bases in the human small intestinal contents.
Journal: Pharmaceutical research 20060601
Title: Antifungal effects of the volatile oils from Allium plants against Trichophyton species and synergism of the oils with ketoconazole.
Journal: Phytomedicine : international journal of phytotherapy and phytopharmacology 20060601
Title: Ketoconazole as a secondary hormonal intervention in advanced prostate cancer.
Journal: Clinical journal of oncology nursing 20060601
Title: Polymorphic behaviour of Compritol888 ATO as bulk lipid and as SLN and NLC.
Journal: Journal of microencapsulation 20060601
Title: Fungal toenail infections.
Journal: Clinical evidence 20060601
Title: Surface plasmon resonance analysis of antifungal azoles binding to CYP3A4 with kinetic resolution of multiple binding orientations.
Journal: Biochemistry 20060523
Title: Identification and quantitation of cis-ketoconazole impurity by capillary zone electrophoresis-mass spectrometry.
Journal: Journal of chromatography. A 20060505
Title: alpha(2)-Adrenergic receptors activate MAPK and Akt through a pathway involving arachidonic acid metabolism by cytochrome P450-dependent epoxygenase, matrix metalloproteinase activation and subtype-specific transactivation of EGFR.
Journal: Cellular signalling 20060501
Title: Lack of effect of ketoconazole-mediated CYP3A inhibition on sorafenib clinical pharmacokinetics.
Journal: Cancer chemotherapy and pharmacology 20060501
Title: Metabolism and effect of para-toluene-sulfonamide on rat liver microsomal cytochrome P450 from in vivo and in vitro studies.
Journal: Acta pharmacologica Sinica 20060501
Title: The use of SLN and NLC as topical particulate carriers for imidazole antifungal agents.
Journal: Die Pharmazie 20060501
Title: [Skin infection with Fusarium in an immunocompetent patient].
Journal: Actas dermo-sifiliograficas 20060501
Title: [Three cases of cutaneous blastomycosis].
Journal: Medecine et maladies infectieuses 20060501
Title: Structure-based optimization of azole antifungal agents by CoMFA, CoMSIA, and molecular docking.
Journal: Journal of medicinal chemistry 20060420
Title: Drugs for treating paracoccidioidomycosis.
Journal: The Cochrane database of systematic reviews 20060419
Title: Synthesis and evaluation of heteroaryl-substituted dihydronaphthalenes and indenes: potent and selective inhibitors of aldosterone synthase (CYP11B2) for the treatment of congestive heart failure and myocardial fibrosis.
Journal: Journal of medicinal chemistry 20060406
Title: Inhibition of the HERG K+ channel by the antifungal drug ketoconazole depends on channel gating and involves the S6 residue F656.
Journal: FEBS letters 20060403
Title: Development, validation and utility of an in vitro technique for assessment of potential clinical drug-drug interactions involving P-glycoprotein.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20060401
Title: In vitro and in vivo inhibitory effect of stiripentol on clobazam metabolism.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060401
Title: Interactions of two major metabolites of prasugrel, a thienopyridine antiplatelet agent, with the cytochromes P450.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060401
Title: Identification of human liver cytochrome P450 enzymes responsible for the metabolism of lonafarnib (Sarasar).
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060401
Title: Antifungal agents for preventing fungal infections in non-neutropenic critically ill and surgical patients: systematic review and meta-analysis of randomized clinical trials.
Journal: The Journal of antimicrobial chemotherapy 20060401
Title: Formation of 4'-carboxyl acid metabolite of imrecoxib by rat liver microsomes.
Journal: Acta pharmacologica Sinica 20060401
Title: Long term control of hypercortisolism with fluconazole: case report and in vitro studies.
Journal: European journal of endocrinology 20060401
Title: In vitro efficacy of a buffered chelating solution as an antimicrobial potentiator for antifungal drugs against fungal pathogens obtained from horses with mycotic keratitis.
Journal: American journal of veterinary research 20060401
Title: Ketoconazole renders poor CYP3A phenotype status with midazolam as probe drug.
Journal: Therapeutic drug monitoring 20060401
Title: Acanthamoeba keratitis in a 5-year-old boy without a history of contact lens usage.
Journal: Cornea 20060401
Title: Aureobasidium pullulans keratitis.
Journal: Clinical & experimental ophthalmology 20060401
Title: [The effect of propyl gallate on the activity of various antifungal drugs against filamentous fungi in vitro].
Journal: [Zhonghua yan ke za zhi] Chinese journal of ophthalmology 20060401
Title: The vitamin D prodrugs 1alpha(OH)D2, 1alpha(OH)D3 and BCI-210 suppress PTH secretion by bovine parathyroid cells.
Journal: Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 20060301
Title: Coxiella burnetii inhabits a cholesterol-rich vacuole and influences cellular cholesterol metabolism.
Journal: Cellular microbiology 20060301
Title: Inhibition of Vitamin D3 metabolism enhances VDR signalling in androgen-independent prostate cancer cells.
Journal: The Journal of steroid biochemistry and molecular biology 20060301
Title: [Penicilliosis in Laos].
Journal: Presse medicale (Paris, France : 1983) 20060301
Title: Novel endoperoxides: synthesis and activity against Candida species.
Journal: Bioorganic & medicinal chemistry letters 20060215
Title: Partial structures of ketoconazole as modulators of the large conductance calcium-activated potassium channel (BK(Ca)).
Journal: Bioorganic & medicinal chemistry letters 20060215
Title: Griseofulvin and ketoconazole solubilization by bile salts studied using fluorescence spectroscopy.
Journal: Colloids and surfaces. B, Biointerfaces 20060201
Title: Clinical evolution of paracoccidioidomycosis in 38 children and teenagers.
Journal: Mycopathologia 20060201
Title: Use of capecitabine after renal allograft transplantation in dog erythrocyte antigen-matched dogs.
Journal: Veterinary surgery : VS 20060201
Title: CYP3A4 activity in four different animal species liver microsomes using 7-benzyloxyquinoline and HPLC/spectrofluorometric determination.
Journal: Journal of pharmaceutical and biomedical analysis 20060123
Title: Development of a fluorescence-based assay for screening of modulators of human organic anion transporter 1B3 (OATP1B3).
Journal: European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V 20060101
Title: Dysmorphogenic effects of some fungicides derived from the imidazole on rat embryos cultured in vitro.
Journal: Reproductive toxicology (Elmsford, N.Y.) 20060101
Title: Determination of the enzyme(s) involved in the metabolism of amiodarone in liver and intestine of rat: the contribution of cytochrome P450 3A isoforms.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20060101
Title: Intestinal and hepatic CYP3A4 catalyze hydroxylation of 1alpha,25-dihydroxyvitamin D(3): implications for drug-induced osteomalacia.
Journal: Molecular pharmacology 20060101
Title: An unusual presentation of malassezia dermatosis.
Journal: Dermatology (Basel, Switzerland) 20060101
Title: Hyperkeratotic head and neck Malassezia dermatosis.
Journal: Dermatology (Basel, Switzerland) 20060101
Title: Impact of the cyclosporine-ketoconazole interaction in children with steroid-dependent idiopathic nephrotic syndrome.
Journal: European journal of clinical pharmacology 20060101
Title: Effects of cytochrome P450 3A modulators ketoconazole and carbamazepine on quetiapine pharmacokinetics.
Journal: British journal of clinical pharmacology 20060101
Title: Bioavailability of two oral formulations of loratadine 20 mg with concomitant ketoconazole: an open-label, randomized, two-period crossover comparison in healthy Mexican adult volunteers.
Journal: Clinical therapeutics 20060101
Title: Effect of drug utilization reviews on the quality of in-hospital prescribing: a quasi-experimental study.
Journal: BMC health services research 20060101
Title: Recurrent vulvovaginal candidiasis.
Journal: Missouri medicine 20060101
Title: Carney complex (CNC).
Journal: Orphanet journal of rare diseases 20060101
Title: Malassezia and seborrheic dermatitis: etiology and treatment.
Journal: Journal of cosmetic science 20060101
Title: Ketoconazole-tacrolimus coadministration in kidney transplant recipients: two-year results of a prospective randomized study.
Journal: American journal of nephrology 20060101
Title: In vitro studies on quetiapine metabolism using the substrate depletion approach with focus on drug-drug interactions.
Journal: Drug metabolism and drug interactions 20060101
Title: Efficacy and safety of a new once-daily topical ketoconazole 2% gel in the treatment of seborrheic dermatitis: a phase III trial.
Journal: Journal of drugs in dermatology : JDD 20060101
Title: In vitro activity of R126638 and ketoconazole against Malassezia species.
Journal: Acta dermato-venereologica 20060101
Title: Clinical features and diagnosis of 42 travellers with cutaneous leishmaniasis.
Journal: Travel medicine and infectious disease 20060101
Title: [Effect of steroid biosynthesis modificators on the progesterone biotransformation by a recombinant yeasts expressing cytochrome P450c17].
Journal: Biomeditsinskaia khimiia 20060101
Title: Xolegel (ketoconazole, 2%).
Journal: Skinmed 20060101
Title: [Drug-related problems in a patient with Cushing's disease].
Journal: Farmacia hospitalaria : organo oficial de expresion cientifica de la Sociedad Espanola de Farmacia Hospitalaria 20060101
Title: Mycetoma : a review.
Journal: American journal of clinical dermatology 20060101
Title: Clinical efficacy of a new ciclopiroxolamine/zinc pyrithione shampoo in scalp seborrheic dermatitis treatment.
Journal: European journal of dermatology : EJD 20060101
Title: Effect of ketoconazole and rifampicin on the pharmacokinetics of ranitidine in healthy human volunteers: a possible role of P-glycoprotein.
Journal: Drug metabolism and drug interactions 20060101
Title: Effect of ketoconazole on the pharmacokinetics of ornidazole--a possible role of p-glycoprotein and CYP3A.
Journal: Drug metabolism and drug interactions 20060101
Title: [Laboratory evolutive aspects of children under paracoccidioidomycosis treatment].
Journal: Revista da Sociedade Brasileira de Medicina Tropical 20060101
Title: Co-administration of ketoconazole and tacrolimus therapy: a transplanted rat model.
Journal: International urology and nephrology 20060101
Title: [Relative bioavailability and bioequivalence of the antimycotics ketoconazole and fluconazole].
Journal: Antibiotiki i khimioterapiia = Antibiotics and chemoterapy [sic] 20060101
Title: In vitro susceptibility of oral Candida to seven antifungal agents.
Journal: Oral microbiology and immunology 20051201
Title: Significant differences in the disposition of cyclic prodrugs of opioid peptides in rats and guinea pigs following IV administration.
Journal: Journal of pharmaceutical sciences 20051201
Title: Bioactive small molecules reveal antagonism between the integrated stress response and sterol-regulated gene expression.
Journal: Cell metabolism 20051201
Title: Evaluation and treatment of Cushing's syndrome.
Journal: The American journal of medicine 20051201
Title: A comparison of hair quality and cosmetic acceptance following the use of two anti-dandruff shampoos.
Journal: The journal of investigative dermatology. Symposium proceedings 20051201
Title: Effects of beta-thujaplicin on anti-Malassezia pachydermatis remedy for canine otitis externa.
Journal: The Journal of veterinary medical science 20051201
Title: Ketoconazole induced torsades de pointes without concomitant use of QT interval-prolonging drug.
Journal: Journal of cardiovascular electrophysiology 20051201
Title: Fungal nail infections.
Journal: Clinical evidence 20051201
Title: Candidiasis (vulvovaginal).
Journal: Clinical evidence 20051201
Title: Novel tetralone-derived retinoic acid metabolism blocking agents: synthesis and in vitro evaluation with liver microsomal and MCF-7 CYP26A1 cell assays.
Journal: Journal of medicinal chemistry 20051117
Title: Characterization of rat small intestinal and colon precision-cut slices as an in vitro system for drug metabolism and induction studies.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20051101
Title: Uncommon clinical presentations of cutaneous leishmaniasis in Sudan.
Journal: Transactions of the Royal Society of Tropical Medicine and Hygiene 20051101
Title: Upregulation of sterol C14-demethylase expression in Trypanosoma cruzi treated with sterol biosynthesis inhibitors.
Journal: Molecular and biochemical parasitology 20051101
Title: Effect of azole antifungals ketoconazole and fluconazole on the pharmacokinetics of dexloxiglumide.
Journal: British journal of clinical pharmacology 20051101
Title: The effect of calcium chelating or binding agents on Candida albicans.
Journal: Oral surgery, oral medicine, oral pathology, oral radiology, and endodontics 20051101
Title: Clinical status of agents being developed for leishmaniasis.
Journal: Expert opinion on investigational drugs 20051101
Title: Extraction, hemisynthesis, and synthesis of canthin-6-one analogues. Evaluation of their antifungal activities.
Journal: Journal of natural products 20051101
Title: An overview of antifungal drugs and their use for treatment of deep and superficial mycoses in animals.
Journal: Clinical techniques in small animal practice 20051101
Title: [Metabolic kinetics of MN9202 in Beagle dog liver microsomes].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20051101
Title: Increase of the LC-MS/MS sensitivity and detection limits using on-line sample preparation with large volume plasma injection.
Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20051025
Title: Characterization of human cytochrome P450 isoenzymes involved in the metabolism of vinorelbine.
Journal: Fundamental & clinical pharmacology 20051001
Title: [Drug-drug interaction of antifungal drugs].
Journal: Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20051001
Title: The effects of inhibiting cytochrome P450 3A, p-glycoprotein, and gastric acid secretion on the oral bioavailability of methadone in dogs.
Journal: Journal of veterinary pharmacology and therapeutics 20051001
Title: Enantiomeric separation of ketoconazole and terconazole antifungals by electrokinetic chromatography: Rapid quantitative analysis of ketoconazole in pharmaceutical formulations.
Journal: Electrophoresis 20051001
Title: The role of ketoconazole in the prevention of ovarian hyperstimulation syndrome in patients with polycystic ovary syndrome during assisted reproductive technology cycles.
Journal: Saudi medical journal 20051001
Title: Effects of ketoconazole on glucuronidation by UDP-glucuronosyltransferase enzymes.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20050915
Title: [Determination of antidangdruff agent salicylic acid, zinc pyrithione, octopirox, climbazole and ketoconazole in shampoo by high performance liquid chromatography].
Journal: Wei sheng yan jiu = Journal of hygiene research 20050901
Title: Increased expression and hotspot mutations of the multidrug efflux transporter, CDR1 in azole-resistant Candida albicans isolates from vaginitis patients.
Journal: FEMS microbiology letters 20050815
Title: Metabolism of the alpha,beta-unsaturated ketones, chalcone and trans-4-phenyl-3-buten-2-one, by rat liver microsomes and estrogenic activity of the metabolites.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20050801
Title: The advantages of the Ussing chamber in drug absorption studies.
Journal: Journal of biomolecular screening 20050801
Title: 2-O-(2-hydroxybutyl)-beta-cyclodextrin as a chiral selector for the capillary electrophoretic separation of chiral drugs.
Journal: Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20050801
Title: DNA fingerprinting pattern and susceptibility to antifungal drugs in Cryptococcus neoformans variety grubii isolates from Barcelona city and rural environmental samples.
Journal: Mycopathologia 20050801
Title: Identification of OATP1B3 as a high-affinity hepatocellular transporter of paclitaxel.
Journal: Cancer biology & therapy 20050801
Title: Ketobemidone is a substrate for cytochrome P4502C9 and 3A4, but not for P-glycoprotein.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20050801
Title: SLN and NLC for topical delivery of ketoconazole.
Journal: Journal of microencapsulation 20050801
Title: [3H]linopirdine binding to rat brain membranes is not relevant for M-channel interaction.
Journal: European journal of pharmacology 20050725
Title: Development and application of a new on-line SPE system combined with LC-MS/MS detection for high throughput direct analysis of pharmaceutical compounds in plasma.
Journal: Journal of chromatography. A 20050708
Title: Effect of several compounds on biliary excretion of paclitaxel and its metabolites in guinea-pigs.
Journal: Anti-cancer drugs 20050701
Title: Dimemorfan N-demethylation by mouse liver microsomal cytochrome P450 enzymes.
Journal: Life sciences 20050701
Title: Alanine scanning of transmembrane helix 11 of Cdr1p ABC antifungal efflux pump of Candida albicans: identification of amino acid residues critical for drug efflux.
Journal: The Journal of antimicrobial chemotherapy 20050701
Title: A novel foam vehicle for delivery of topical corticosteroids.
Journal: Journal of the American Academy of Dermatology 20050701
Title: Rate-limiting biotransformation of triamterene is mediated by CYP1A2.
Journal: International journal of clinical pharmacology and therapeutics 20050701
Title: Fusarium solani breast abscess.
Journal: Indian journal of medical microbiology 20050701
Title: [In vitro activity of ketoconazole, itraconazole and terbinafine against Malassezia strains isolated from neonates].
Journal: Mikrobiyoloji bulteni 20050701
Title: Characterization of testosterone 11 beta-hydroxylation catalyzed by human liver microsomal cytochromes P450.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20050601
Title: Long-term outcome for men with androgen independent prostate cancer treated with ketoconazole and hydrocortisone.
Journal: The Journal of urology 20050601
Title: Ketoconazole increases plasma concentrations of antimalarial mefloquine in healthy human volunteers.
Journal: Journal of clinical pharmacy and therapeutics 20050601
Title: The effect of ketoconazole on the pharmacokinetics of a selective alpha 1A-adrenoceptor antagonist.
Journal: Journal of clinical pharmacology 20050601
Title: Genome-wide expression profiling of the response to azole, polyene, echinocandin, and pyrimidine antifungal agents in Candida albicans.
Journal: Antimicrobial agents and chemotherapy 20050601
Title: Comparison of the clinical efficacy of oral terbinafine and ketoconazole combined with cephalexin in the treatment of Malassezia dermatitis in dogs--a pilot study.
Journal: Veterinary dermatology 20050601
Title: [Abdominal zygomycosis in a bitch due to Absidia corymbifera].
Journal: Revista iberoamericana de micologia 20050601
Title: Effect of 2-(4-aminophenylmethyl)-6-hydroxy-3, 4-dihydronaphthalen-1(2H)-one on all-trans and 13-cis-retinoic acid levels in plasma quantified by high perfomance liquid chromatography coupled to tandem mass spectrometry.
Journal: Journal of enzyme inhibition and medicinal chemistry 20050601
Title: [Allergic fungal sinusitis and allergic broncho-pulmonary aspergillosis: a fortuitous association or a nosological rhino-bronchial entity?].
Journal: Revue des maladies respiratoires 20050601
Title: [Comparison of efficacy of combination of ketokonazol 400 mg + clindamycin 100 mg with ketokonazol 800 mg + clindamycin 100 mg in the treatment of vaginitis due to Candida and bacterial vaginosis].
Journal: Ginecologia y obstetricia de Mexico 20050601
Title: Lack of cataleptogenic potentiation with non-imidazole H3 receptor antagonists reveals potential drug-drug interactions between imidazole-based H3 receptor antagonists and antipsychotic drugs.
Journal: Brain research 20050531
Title: Selective inhibition of dog hepatic CYP2B11 and CYP3A12.
Journal: The Journal of pharmacology and experimental therapeutics 20050501
Title: Intestinal metabolism of PAH: in vitro demonstration and study of its impact on PAH transfer through the intestinal epithelium.
Journal: Environmental research 20050501
Title: Anti-proliferative synergy of lysophospholipid analogues and ketoconazole against Trypanosoma cruzi (Kinetoplastida: Trypanosomatidae): cellular and ultrastructural analysis.
Journal: The Journal of antimicrobial chemotherapy 20050501
Title: Blood concentrations of everolimus are markedly increased by ketoconazole.
Journal: Journal of clinical pharmacology 20050501
Title: Comparison of in vitro activities of antifungal drugs and ethanolic extract of propolis against Trichophyton rubrum and T. mentagrophytes by using a microdilution assay.
Journal: Mycoses 20050501
Title: Separation study of cadmium as CdI4(2-) through a bulk liquid membrane containing ketoconazole and oleic acid.
Journal: Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20050501
Title: Effect of solubilizing and microemulsifying excipients in polyethylene glycol 6000 solid dispersion on enhanced dissolution and bioavailability of ketoconazole.
Journal: Archives of pharmacal research 20050501
Title: Mefloquine resistance reversal action of ketoconazole - a cytochrome P450 inhibitor, against mefloquine-resistant malaria.
Journal: Parasitology 20050501
Title: Slime production and proteinase activity of Candida species isolated from blood samples and the comparison of these activities with minimum inhibitory concentration values of antifungal agents.
Journal: Memorias do Instituto Oswaldo Cruz 20050501
Title: Cloning and heterologous expression of the NADPH cytochrome P450 oxidoreductase genes from an industrial dicarboxylic acid-producing Candida tropicalis.
Journal: Yeast (Chichester, England) 20050430
Title: Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: synthesis, in vitro biological activity, pharmacokinetics, and antitumor activity in the LAPC4 human prostate cancer xenograft model.
Journal: Journal of medicinal chemistry 20050421
Title: Enhancement of nifedipine-induced gingival overgrowth by concomitant ketoconazole in rats.
Journal: Pharmacology 20050401
Title: Xenobiotics and the glucocorticoid receptor: additive antagonistic effects on tyrosine aminotransferase activity in rat hepatoma cells.
Journal: Basic & clinical pharmacology & toxicology 20050401
Title: Studies to investigate the pharmacokinetic interactions between ranolazine and ketoconazole, diltiazem, or simvastatin during combined administration in healthy subjects.
Journal: Journal of clinical pharmacology 20050401
Title: Transient band-like keratopathy after treatment for seborrheic dermatitis.
Journal: Cornea 20050401
Title: A study of the in vitro interaction between lidocaine and premedications using human liver microsomes.
Journal: Journal of clinical pharmacy and therapeutics 20050401
Title: Topical application of ketoconazole stimulates hair growth in C3H/HeN mice.
Journal: The Journal of dermatology 20050401
Title: Hepatotoxicity associated with cyclosporine monitoring using C2 recommendations in adults renal recipients receiving ketoconazole.
Journal: Transplantation proceedings 20050401
Title: Assessment of the hepatic and intestinal first-pass metabolism of midazolam in a CYP3A drug-drug interaction model rats.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20050401
Title: Oxidative stress mediates drug-induced hepatotoxicity in rats: a possible role of DNA fragmentation.
Journal: Toxicology 20050330
Title: Synthesis and evaluation of imidazolylmethylenetetrahydronaphthalenes and imidazolylmethyleneindanes: potent inhibitors of aldosterone synthase.
Journal: Journal of medicinal chemistry 20050324
Title: Microbiological assay of ketoconazole in shampoo.
Journal: International journal of pharmaceutics 20050323
Title: Synthesis and evaluation of (pyridylmethylene)tetrahydronaphthalenes/-indanes and structurally modified derivatives: potent and selective inhibitors of aldosterone synthase.
Journal: Journal of medicinal chemistry 20050310
Title: Metabolism of alfentanil by cytochrome p4503a (cyp3a) enzymes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20050301
Title: Experimentally induced androgen depletion accentuates ethnicity-related contrasts in luteinizing hormone secretion in asian and caucasian men.
Journal: The Journal of clinical endocrinology and metabolism 20050301
Title: Characterization of human cytochrome P450 enzymes involved in the in vitro metabolism of perospirone.
Journal: Biopharmaceutics & drug disposition 20050301
Title: Refractory anaphylactic shock associated with ketoconazole treatment.
Journal: The Annals of pharmacotherapy 20050301
Title: A randomized, phase II trial of ketoconazole plus alendronate versus ketoconazole alone in patients with androgen independent prostate cancer and bone metastases.
Journal: The Journal of urology 20050301
Title: Population-based case-control study of oral ketoconazole treatment for birth outcomes.
Journal: Congenital anomalies 20050301
Title: Pityriasis versicolor alba.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20050301
Title: Co-administration of ketoconazole with H1-antagonists ebastine and loratadine in healthy subjects: pharmacokinetic and pharmacodynamic effects.
Journal: British journal of clinical pharmacology 20050301
Title: Seborrheic dermatitis. The link between facial rash and neurologic disease.
Journal: Postgraduate medicine 20050301
Title: Effect of ketoconazole on the pharmacokinetics and safety of telithromycin and clarithromycin in older subjects with renal impairment.
Journal: International journal of clinical pharmacology and therapeutics 20050301
Title: Pharmacological management of paracoccidioidomycosis.
Journal: Expert opinion on pharmacotherapy 20050301
Title: Molecular design of two sterol 14alpha-demethylase homology models and their interactions with the azole antifungals ketoconazole and bifonazole.
Journal: Journal of computer-aided molecular design 20050301
Title: A simultaneous assessment of CYP3A4 metabolism and induction in the DPX-2 cell line.
Journal: The AAPS journal 20050301
Title: CYP3A4 is a vitamin D-24- and 25-hydroxylase: analysis of structure function by site-directed mutagenesis.
Journal: The Journal of clinical endocrinology and metabolism 20050201
Title: In vivo effects of cyclosporin A and ketoconazole on the pharmacokinetics of representative substrates for P-glycoprotein and cytochrome P450 (CYP) 3A in rats.
Journal: Biological & pharmaceutical bulletin 20050201
Title: [Metabolism of bicyclol in rat and human liver microsomes in vitro].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20050201
Title: Role of ketoconazole in renal transplant recipients.
Journal: Transplantation 20050127
Title: Antifungal and insect antifeedant 2-phenylethanol esters from the liverwort Balantiopsis cancellata from Chile.
Journal: Journal of agricultural and food chemistry 20050126
Title: Age and testosterone feedback jointly control the dose-dependent actions of gonadotropin-releasing hormone in healthy men.
Journal: The Journal of clinical endocrinology and metabolism 20050101
Title: Adult height after ketoconazole treatment in patients with familial male-limited precocious puberty.
Journal: The Journal of clinical endocrinology and metabolism 20050101
Title: A phase I study of estramustine, weekly docetaxel, and carboplatin chemotherapy in patients with hormone-refractory prostate cancer.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20050101
Title: Potent CYP3A4 inhibitory constituents of Piper cubeba.
Journal: Journal of natural products 20050101
Title: Corneofungimetry bioassay on Malassezia spp. under ketoconazole and desonide influences.
Journal: Skin pharmacology and physiology 20050101
Title: Determination of the absolute configuration and solution conformation of the antifungal agents ketoconazole, itraconazole, and miconazole with vibrational circular dichroism.
Journal: Chirality 20050101
Title: Co-administration of cyclosporine and ketoconazole in children with minimal change nephrotic syndrome.
Journal: Nephron. Clinical practice 20050101
Title: [Entomophthoramycosis (zygomycosis) caused by Conidiobolus coronatus in Mato Grosso (Brazil): case report].
Journal: Revista da Sociedade Brasileira de Medicina Tropical 20050101
Title: Phaeohyphomycosis in Korea.
Journal: Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20050101
Title: Clinical treatment of corneal infection due to Fonsecaea pedrosoi--case report.
Journal: Arquivos brasileiros de oftalmologia 20050101
Title: Estimation of potency of HERG channel blockers: impact of voltage protocol and temperature.
Journal: Journal of pharmacological and toxicological methods 20050101
Title: Antifungal susceptibilities of dermatophytic agents isolated from clinical specimens.
Journal: European journal of dermatology : EJD 20050101
Title: Case report of subcutaneous entomophthoromycosis with retroperitoneal invasion.
Journal: Revista da Sociedade Brasileira de Medicina Tropical 20050101
Title: Efficient short-term control of hypercortisolaemia by low-dose etomidate in severe paediatric Cushing's disease.
Journal: Hormone research 20050101
Title: Trichophyton tonsurans associated tinea corporis infection with the development of Majocchi's granuloma in a renal transplant patient.
Journal: Journal of drugs in dermatology : JDD 20050101
Title: Co-administration of ketoconazole and tacrolimus therapy: a transplanted rat model.
Journal: International urology and nephrology 20050101
Title: An evaluation of high-doses ketoconazole with hydrocortisone substitution in hormone-refractory prostate cancer.
Journal: Acta chirurgica Iugoslavica 20050101
Title: [Effect of tofisopam on CYP3A4 enzyme activity on human recombinant 3A4 supersome].
Journal: Acta pharmaceutica Hungarica 20050101
Title: [Successful treatment of a case of extense verrucous chromoblastomychosis with surgical exeresis associated with the use of ketoconazole].
Journal: Revista cubana de medicina tropical 20050101
Title: Novel retinoic acid metabolism blocking agents endowed with multiple biological activities are efficient growth inhibitors of human breast and prostate cancer cells in vitro and a human breast tumor xenograft in nude mice.
Journal: Journal of medicinal chemistry 20041230
Title: Potent, selective and low-calcemic inhibitors of CYP24 hydroxylase: 24-sulfoximine analogues of the hormone 1alpha,25-dihydroxyvitamin D(3).
Journal: Journal of medicinal chemistry 20041230
Title: In vitro metabolism of carbofuran by human, mouse, and rat cytochrome P450 and interactions with chlorpyrifos, testosterone, and estradiol.
Journal: Chemico-biological interactions 20041207
Title: Identification and characterization of potent CYP3A4 inhibitors in Schisandra fruit extract.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20041201
Title: Influence of ketoconazole on azimilide pharmacokinetics in healthy subjects.
Journal: British journal of clinical pharmacology 20041201
Title: Synergistic interaction between ketoconazole and several antidepressant drugs with allopregnanolone treatments in ovariectomized Wistar rats forced to swim.
Journal: Progress in neuro-psychopharmacology & biological psychiatry 20041201
Title: In vitro antifungal activity of sertaconazole compared with nine other drugs against 250 clinical isolates of dermatophytes and Scopulariopsis brevicaulis.
Journal: Chemotherapy 20041201
Title: Combination therapy of once-weekly fluconazole (100, 150, or 300 mg) with topical application of ketoconazole cream in the treatment of onychomycosis.
Journal: Japanese journal of infectious diseases 20041201
Title: Clinicopathologic features of an unusual outbreak of cryptococcosis in dogs, cats, ferrets, and a bird: 38 cases (January to July 2003).
Journal: Journal of the American Veterinary Medical Association 20041201
Title: Effect of various cytochrome P450 3A and P-glycoprotein modulators on the biliary clearance of bromosulphaphthalein in male wistar rats.
Journal: Die Pharmazie 20041201
Title: Synthesis and antileishmanial activity of 3-imidazolylalkylindoles. Part I.
Journal: Journal of enzyme inhibition and medicinal chemistry 20041201
Title: Gamma-tocotrienol metabolism and antiproliferative effect in prostate cancer cells.
Journal: Annals of the New York Academy of Sciences 20041201
Title: Seborrhoeic dermatitis.
Journal: Clinical evidence 20041201
Title: Synthesis and CYP24 inhibitory activity of 2-substituted-3,4-dihydro-2H-naphthalen-1-one (tetralone) derivatives.
Journal: Bioorganic & medicinal chemistry letters 20041115
Title: Tumor apoptosis induced by ruthenium(II)-ketoconazole is enhanced in nonsusceptible carcinoma by monoclonal antibody to EGF receptor.
Journal: International journal of cancer 20041110
Title: A phase I trial of pharmacokinetic modulation of carboxyamidotriazole (CAI) with ketoconazole in patients with advanced cancer.
Journal: Cancer chemotherapy and pharmacology 20041101
Title: Effects of acute and chronic ketoconazole administration on hypothalamo--pituitary--adrenal axis activity and brain corticotropin-releasing hormone.
Journal: Psychoneuroendocrinology 20041101
Title: (2S,3R)-2-aminododecan-3-ol, a new antifungal agent from the ascidian Clavelina oblonga.
Journal: Journal of natural products 20041101
Title: Vulvovaginal candidiasis in children and adolescents with type 1 diabetes mellitus.
Journal: Journal of pediatric endocrinology & metabolism : JPEM 20041101
Title: [Treatment for seborrheic dermatitis].
Journal: Annales de dermatologie et de venereologie 20041101
Title: Pharmacokinetic interaction between ketoconazole and imatinib mesylate (Glivec) in healthy subjects.
Journal: Cancer chemotherapy and pharmacology 20041001
Title: Stress-restress evokes sustained iNOS activity and altered GABA levels and NMDA receptors in rat hippocampus.
Journal: Psychopharmacology 20041001
Title: Effect of ketoconazole on the pharmacokinetics of rosiglitazone in healthy subjects.
Journal: British journal of clinical pharmacology 20041001
Title: The systemic treatment of onychomycosis.
Journal: Clinics in podiatric medicine and surgery 20041001
Title: Pathogenesis of allergic bronchopulmonary aspergillosis and an evidence-based review of azoles in treatment.
Journal: Respiratory medicine 20041001
Title: Multiple oral dosing of ketoconazole influences pharmacokinetics of quinidine after intravenous and oral administration in beagle dogs.
Journal: Journal of veterinary pharmacology and therapeutics 20041001
Title: Comparative evaluation of Sensititre YeastOne vs. the NCCLS M27A protocol and E-test for antifungal susceptibility testing of yeasts.
Journal: Mycoses 20041001
Title: Anti-Candida effects of estragole in combination with ketoconazole or amphotericin B.
Journal: Phytotherapy research : PTR 20041001
Title: Influence of human nail etching for the assessment of topical onychomycosis therapies.
Journal: International journal of pharmaceutics 20040910
Title: Concomitant administration of cyclosporine and ketoconazole in idiopathic nephrotic syndrome.
Journal: Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 20040901
Title: Co-administration of cyclosporine and ketoconazole in idiopathic childhood nephrosis.
Journal: Pediatric nephrology (Berlin, Germany) 20040901
Title: CYP2B6, CYP3A4, and CYP2C19 are responsible for the in vitro N-demethylation of meperidine in human liver microsomes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040901
Title: Identification of an N-methyl-4-phenylpyridinium-like metabolite of the antidiarrheal agent loperamide in human liver microsomes: underlying reason(s) for the lack of neurotoxicity despite the bioactivation event.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040901
Title: In vitro metabolism of MK-0767 [(+/-)-5-[(2,4-dioxothiazolidin-5-yl)methyl]-2-methoxy-N-[[(4-trifluoromethyl) phenyl]methyl]benzamide], a peroxisome proliferator-activated receptor alpha/gamma agonist. I. Role of cytochrome P450, methyltransferases, flavin monooxygenases, and esterases.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040901
Title: Effect of cytochrome P450 inhibitors (diethyl dithiocarbamate, ketoconazole and grapefruit juice) on the pharmacokinetics of all-trans-retinoic acid.
Journal: Farmaco (Societa chimica italiana : 1989) 20040901
Title: Comparative study of 2% ketoconazole cream and 1% hydrocortisone cream in the treatment of infantile seborrheic dermatitis.
Journal: Journal of the Medical Association of Thailand = Chotmaihet thangphaet 20040901
Title: Use of oral ketoconazole to prevent postoperative erections following penile surgery.
Journal: International journal of impotence research 20040801
Title: Interaction of triazolam and ketoconazole in P-glycoprotein-deficient mice.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040801
Title: Concurrent Fusarium chlamydosporum and Microsphaeropsis arundinis infections in a cat.
Journal: Journal of feline medicine and surgery 20040801
Title: Ketoconazole, a cytochrome P450 3A4 inhibitor, markedly increases concentrations of levo-acetyl-alpha-methadol in opioid-naive individuals.
Journal: Clinical pharmacology and therapeutics 20040801
Title: Paranasal sinus aspergillosis: its categorization to develop a treatment protocol.
Journal: Mycoses 20040801
Title: Invasion of epithelial mammalian cells by Paracoccidioides brasiliensis leads to cytoskeletal rearrangement and apoptosis of the host cell.
Journal: Microbes and infection 20040801
Title: Specific interactions of steroids, arylhydrocarbons and flavonoids with progesterone receptors from the cytosol of the fungus Rhizopus nigricans.
Journal: The Journal of steroid biochemistry and molecular biology 20040801
Title: Imidazole analogues of fluoxetine, a novel class of anti-Candida agents.
Journal: Journal of medicinal chemistry 20040729
Title: Computer-assisted design of selective imidazole inhibitors for cytochrome p450 enzymes.
Journal: Journal of medicinal chemistry 20040701
Title: Bioequivalence evaluation of two brands of ketoconazole tablets (Onofin-K and Nizoral) in a healthy female Mexican population.
Journal: Biopharmaceutics & drug disposition 20040701
Title: Sesquiterpenes and flavonol glycosides from Zingiber aromaticum and their CYP3A4 and CYP2D6 inhibitory activities.
Journal: Journal of natural products 20040701
Title: Ketoconazole, an antifungal agent, protects against adiposity induced by a cafeteria diet.
Journal: Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme 20040701
Title: Improved outcome of zygomycosis in patients with hematological diseases?
Journal: Leukemia & lymphoma 20040701
Title: Prescribing practices for seborrheic dermatitis vary with the physician's specialty: implications for clinical practice.
Journal: The Journal of dermatological treatment 20040701
Title: Antifungal chalcones and new caffeic acid esters from Zuccagnia punctata acting against soybean infecting fungi.
Journal: Journal of agricultural and food chemistry 20040602
Title: Co-administration of ketoconazole to tacrolimus-treated kidney transplant recipients: a prospective randomized study.
Journal: Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 20040601
Title: Oral administration of a low dose of midazolam (75 microg) as an in vivo probe for CYP3A activity.
Journal: European journal of clinical pharmacology 20040601
Title: Susceptibility of sequential Fonsecaea pedrosoi isolates from chromoblastomycosis patients to antifungal agents.
Journal: Mycoses 20040601
Title: Lipid raft polarization contributes to hyphal growth in Candida albicans.
Journal: Eukaryotic cell 20040601
Title: Chromoblastomycosis caused by Rhinocladiella aquaspersa.
Journal: Medical mycology 20040601
Title: Antifungal susceptibility of 50 Candida isolates from invasive mycoses in Chile.
Journal: Medical mycology 20040601
Title: Human cytochrome P450: metabolism of testosterone by CYP3A4 and inhibition by ketoconazole.
Journal: Current protocols in toxicology 20040601
Title: A prospective, randomized study of coadministration of ketoconazole and cyclosporine a in kidney transplant recipients: ten-year follow-up.
Journal: Transplantation 20040515
Title: An evaluation of intermediate-dose ketoconazole in hormone refractory prostate cancer.
Journal: European urology 20040501
Title: The use of a cyclosporin-ketoconazole combination: making renal transplantation affordable in developing countries.
Journal: European journal of clinical pharmacology 20040501
Title: Effect of cytochrome P450 3A4 inhibition on the pharmacokinetics of docetaxel.
Journal: Clinical pharmacology and therapeutics 20040501
Title: Comparison of capillary zone electrophoresis and high performance liquid chromatography methods for quantitative determination of ketoconazole in drug formulations.
Journal: Farmaco (Societa chimica italiana : 1989) 20040501
Title: Pharmacologic management of pattern hair loss.
Journal: Facial plastic surgery clinics of North America 20040501
Title: Efficacy of combined cyclosporine A and ketoconazole treatment of anal furunculosis.
Journal: The Journal of small animal practice 20040501
Title: Multicentric lymphoma in a dog after cyclosporine therapy.
Journal: The Journal of small animal practice 20040501
Title: Effects of the antifungal imidazole ketoconazole on CYP1A and CYP3A in rainbow trout and killifish.
Journal: Environmental toxicology and chemistry 20040501
Title: Model for the drug-drug interaction responsible for CYP3A enzyme inhibition. I: evaluation of cynomolgus monkeys as surrogates for humans.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20040501
Title: Model for the drug-drug interaction responsible for CYP3A enzyme inhibition. II: establishment and evaluation of dexamethasone-pretreated female rats.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20040501
Title: Identification and relative contributions of human cytochrome P450 isoforms involved in the metabolism of glibenclamide and lansoprazole: evaluation of an approach based on the in vitro substrate disappearance rate.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20040501
Title: Role of CYP3A enzymes in the biotransformation of triazolam in rat liver.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20040501
Title: Cyclosporine and low-dose ketoconazole in renal transplant recipients: a single-center experience.
Journal: Transplantation 20040415
Title: In vitro metabolism of fipronil by human and rat cytochrome P450 and its interactions with testosterone and diazepam.
Journal: Chemico-biological interactions 20040415
Title: The use of the novel substrate-heme complex approach in the derivation of a representation of the active site of the enzyme complex 17alpha-hydroxylase and 17,20-lyase.
Journal: Biochemical and biophysical research communications 20040409
Title: Comparison of prediction methods for in vivo clearance of (S,S)-3-[3-(methylsulfonyl)phenyl]-1-propylpiperidine hydrochloride, a dopamine D2 receptor antagonist, in humans.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040401
Title: Quantitative contribution of CYP2D6 and CYP3A to oxycodone metabolism in human liver and intestinal microsomes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040401
Title: Prevalence of Candida dubliniensis among germ tube-positive yeasts recovered from the respiratory specimens in HIV-negative patients.
Journal: Mycoses 20040401
Title: Prostate cancer metastasis to supraclavicular lymph node.
Journal: Clinical advances in hematology & oncology : H&O 20040401
Title: Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.
Journal: Biochemical and biophysical research communications 20040319
Title: Antiandrogen withdrawal alone or in combination with ketoconazole in androgen-independent prostate cancer patients: a phase III trial (CALGB 9583).
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20040315
Title: History of the development of azole derivatives.
Journal: Clinical microbiology and infection : the official publication of the European Society of Clinical Microbiology and Infectious Diseases 20040301
Title: [Ketoconazole in the prevention of acute delirium episodes].
Journal: Revista brasileira de psiquiatria (Sao Paulo, Brazil : 1999) 20040301
Title: Solubilizing poorly soluble antimycotic agents by emulsification via a solvent-free process.
Journal: AAPS PharmSciTech 20040301
Title: Chronic mucocutaneous candidiasis: a case report.
Journal: Journal of the Indian Society of Pedodontics and Preventive Dentistry 20040301
Title: Role of multiple drug resistance protein 1 in neutral but not acidic glycosphingolipid biosynthesis.
Journal: The Journal of biological chemistry 20040227
Title: Sirolimus and ketoconazole co-prescription in renal transplant recipients.
Journal: Transplantation 20040215
Title: Synthesis and antifungal activities of phenylenedithioureas.
Journal: Bioorganic & medicinal chemistry letters 20040209
Title: Enantioselectivity of inhibition of cytochrome P450 3A4 (CYP3A4) by ketoconazole: Testosterone and methadone as substrates.
Journal: Chirality 20040201
Title: Comparative efficacy of topical therapy with a slow-release mucoadhesive buccal tablet containing miconazole nitrate versus systemic therapy with ketoconazole in HIV-positive patients with oropharyngeal candidiasis.
Journal: Journal of acquired immune deficiency syndromes (1999) 20040201
Title: Development of an in vivo preclinical screen model to estimate absorption and first-pass hepatic extraction of xenobiotics. II. Use of ketoconazole to identify P-glycoprotein/CYP3A-limited bioavailability in the monkey.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040201
Title: Efficacy of a new ketoconazole bioadhesive vaginal tablet on Candida albicans.
Journal: Farmaco (Societa chimica italiana : 1989) 20040201
Title: [Modern antimycotics. What the treating physician needs to know].
Journal: Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete 20040201
Title: Role of phenobarbital-inducible cytochrome P450s as a source of active oxygen species in DNA-oxidation.
Journal: Cancer letters 20040120
Title: Synthesis of galactopyranosyl amino alcohols as a new class of antitubercular and antifungal agents.
Journal: Bioorganic & medicinal chemistry letters 20040119
Title: Highly selective inhibition of human CYP3Aa in vitro by azamulin and evidence that inhibition is irreversible.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20040101
Title: Ketocazole as an adjunct to finasteride in the treatment of androgenetic alopecia in men.
Journal: Medical hypotheses 20040101
Title: High-throughput screening for the assessment of time-dependent inhibitions of new drug candidates on recombinant CYP2D6 and CYP3A4 using a single concentration method.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20040101
Title: Interventions for treating oral candidiasis for patients with cancer receiving treatment.
Journal: The Cochrane database of systematic reviews 20040101
Title: Drug-drug interactions evaluated by a highly active reconstituted native human cytochrome P4503A4 and human NADPH-cytochrome P450 reductase system.
Journal: Arzneimittel-Forschung 20040101
Title: The role of cytochrome-P450 inhibitors in the prevention of hepatotoxicity after paracetamol overdose in rats.
Journal: Human & experimental toxicology 20040101
Title: Oral paracoccidioidomycosis or squamous cell carcinoma?
Journal: General dentistry 20040101
Title: Antimycotics: why are they effective in the treatment of seborrheic dermatitis?
Journal: Dermatology (Basel, Switzerland) 20040101
Title: Effect of concomitant administration of cyclosporine and ketoconazole in children with focal segmental glomerulosclerosis.
Journal: American journal of nephrology 20040101
Title: In vitro fungitoxic activity of Larrea divaricata cav. extracts.
Journal: Letters in applied microbiology 20040101
Title: Azoles for allergic bronchopulmonary aspergillosis associated with asthma.
Journal: The Cochrane database of systematic reviews 20040101
Title: In vitro antifungal susceptibility of Candida spp. isolates from patients with chronic periodontitis and from control patients.
Journal: Brazilian oral research 20040101
Title: In vitro susceptibility of Candida species isolated from cancer patients to some antifungal agents.
Journal: Drug metabolism and drug interactions 20040101
Title: [Determination of biological activity of hydrogel preparations based on ketoconazole and clotrimazole].
Journal: Antibiotiki i khimioterapiia = Antibiotics and chemoterapy [sic] 20040101
Title: Resistance reversal action of ketoconazole against mefloquine resistance of Plasmodium yoelii nigeriensis.
Journal: Experimental parasitology 20040101
Title: Determination of pharmaceutical compounds in skin by imaging matrix-assisted laser desorption/ionisation mass spectrometry.
Journal: Rapid communications in mass spectrometry : RCM 20040101
Title: Antifungal effects of herbal essential oils alone and in combination with ketoconazole against Trichophyton spp.
Journal: Journal of applied microbiology 20040101
Title: Etest for assessing the susceptibility of filamentous fungi.
Journal: Acta microbiologica et immunologica Hungarica 20040101
Title: Metastatic hepatic carcinoid associated with ectopic ACTH syndrome, resistant to octreotide and ketoconazole therapy.
Journal: Annals of Saudi medicine 20040101
Title: In vitro activities of transition metal derivatives of ketoconazole and clotrimazole against a wild type strain of Saccharomyces cerevisiae in absence or presence of human neutrophils.
Journal: Arzneimittel-Forschung 20040101
Title: Management of androgen-independent prostate cancer.
Journal: Cancer control : journal of the Moffitt Cancer Center 20040101
Title: Spontaneous remission of Cushing's disease after disappearance of a microadenoma attached to the pituitary stalk.
Journal: Pituitary 20040101
Title: [Prophylaxis of fungal infection in patients with hematologic neoplasms and severe neutropenia after high-dose chemotherapy].
Journal: Antibiotiki i khimioterapiia = Antibiotics and chemoterapy [sic] 20040101
Title: Cushing's disease and pregnancy.
Journal: Pituitary 20040101
Title: [Current possibilities of using antimyocotic drugs in the treatment of various skin disorders].
Journal: Wiadomosci parazytologiczne 20040101
Title: The influence of ketoconazole on the activity of asparagine protease produced by Candida strains.
Journal: Research communications in molecular pathology and pharmacology 20040101
Title: Microbial transformation of (-)-carvone.
Journal: Zeitschrift fur Naturforschung. C, Journal of biosciences 20040101
Title: Phase 3 randomized trial evaluating second-line hormonal therapy versus docetaxel-estramustine combination chemotherapy on progression-free survival in asymptomatic patients with a rising prostate-specific antigen level after hormonal therapy for prostate cancer: an Eastern Cooperative Oncology Group (E1899), Intergroup/Clinical Trials Support Unit study.
Journal: Urology 20031229
Title: QT and RR intervals in conscious and anesthetized guinea pigs with highly varying RR intervals and given QTc-lengthening test articles.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20031201
Title: Experimental evaluation of antifungal and antiseptic agents against Rhodotorula spp.
Journal: Mycoses 20031201
Title: Trypanocidal constituents in plants 2.xanthones from the stem bark of Garcinia subelliptica.
Journal: Biological & pharmaceutical bulletin 20031201
Title: Acute lung injury in 2003.
Journal: Acta pharmacologica Sinica 20031201
Title: Successful treatment of dandruff with 1.5% ciclopirox olamine shampoo in Korea.
Journal: The Journal of dermatological treatment 20031201
Title: Multiple mechanisms account for variation in base-line sensitivity to azole fungicides in field isolates of Mycosphaerella graminicola.
Journal: Pest management science 20031201
Title: Liver cirrhosis developed after ketoconazole-induced acute hepatic injury.
Journal: Journal of gastroenterology and hepatology 20031201
Title: Clofibrate, a peroxisome-proliferator, enhances reverse cholesterol transport through cytochrome P450 activation and oxysterol generation.
Journal: The Tohoku journal of experimental medicine 20031201
Title: New triterpene glycosides from the stems of Anomospermum grandifolium.
Journal: Journal of natural products 20031201
Title: Identification of the human cytochrome P450s responsible for the in vitro metabolism of a leukotriene B4 receptor antagonist, CP-195,543.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20031201
Title: Emerging systemic pharmacologic approaches in acute respiratory distress syndrome.
Journal: Respiratory care clinics of North America 20031201
Title: Cutaneous blastomycosis presenting as non-healing ulcer and responding to oral ketoconazole.
Journal: Dermatology online journal 20031201
Title: Clinical strategies in the management of biochemical recurrence after radical prostatectomy.
Journal: Clinical prostate cancer 20031201
Title: Candidiasis (vulvovaginal).
Journal: Clinical evidence 20031201
Title: Stripping voltammetric and polarographic techniques for the determination of anti-fungal ketoconazole on the mercury electrode.
Journal: Journal of pharmaceutical and biomedical analysis 20031124
Title: Threshold for antiproliferative and proapoptotic activity of ttaxol in HepG2 cells expressing human CYP3A4: effect of P-glycoprotein transporters.
Journal: Pharmacology 20031101
Title: Pharmacokinetic and pharmacodynamic interactions of oral midazolam with ketoconazole, fluoxetine, fluvoxamine, and nefazodone.
Journal: Journal of clinical pharmacology 20031101
Title: Docetaxel and ketoconazole in advanced hormone-refractory prostate carcinoma: a phase I and pharmacokinetic study.
Journal: Cancer 20031101
Title: Fungal infection of sutureless self-sealing incision for cataract surgery.
Journal: Ophthalmology 20031101
Title: A double-blind, randomized, placebo-controlled study to assess the efficacy of ketoconazole for reducing the risk of ovarian hyperstimulation syndrome.
Journal: Fertility and sterility 20031101
Title: Ketoconazole alters cyclosporine pharmacokinetic profile and may predispose to acute rejection.
Journal: Transplantation proceedings 20031101
Title: Unintentional rechallenge resulting in a causative relationship between ketoconazole and acute liver injury.
Journal: International journal of clinical practice 20031101
Title: Identification and prediction of promiscuous aggregating inhibitors among known drugs.
Journal: Journal of medicinal chemistry 20031009
Title: Ketoconazole-induced neurologic sequelae.
Journal: Veterinary and human toxicology 20031001
Title: Ketoconazole and lopinavir/ritonavir coadministration: boosting beyond boosting.
Journal: AIDS research and human retroviruses 20031001
Title: Antifungal pharmacotherapy for neonatal candidiasis.
Journal: Seminars in perinatology 20031001
Title: Fungal dermatitis with olanzapine in schizophrenia.
Journal: Canadian journal of psychiatry. Revue canadienne de psychiatrie 20031001
Title: Clotrimazole, ketoconazole, and clodinafop-propargyl inhibit the in vitro growth of Babesia bigemina and Babesia bovis (Phylum Apicomplexa).
Journal: Parasitology 20031001
Title: Lem3p is essential for the uptake and potency of alkylphosphocholine drugs, edelfosine and miltefosine.
Journal: The Journal of biological chemistry 20030919
Title: Genome-wide expression profiling of the response to polyene, pyrimidine, azole, and echinocandin antifungal agents in Saccharomyces cerevisiae.
Journal: The Journal of biological chemistry 20030912
Title: Effect of ketoconazole on venlafaxine plasma concentrations in extensive and poor metabolisers of debrisoquine.
Journal: European journal of clinical pharmacology 20030901
Title: The effect of ketoconazole and diltiazem on oestrogen metabolism in postmenopausal women after single dose oestradiol treatment.
Journal: British journal of clinical pharmacology 20030901
Title: Application of compartmental modeling to an examination of in vitro intestinal permeability data: assessing the impact of tissue uptake, P-glycoprotein, and CYP3A.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030901
Title: Metabolism and elimination of quinine in healthy volunteers.
Journal: European journal of clinical pharmacology 20030901
Title: Antileishmanial activities of dihydrochalcones from piper elongatum and synthetic related compounds. Structural requirements for activity.
Journal: Bioorganic & medicinal chemistry 20030901
Title: Long-term results of treatment in patients with ACTH-secreting pituitary macroadenomas.
Journal: European journal of endocrinology 20030901
Title: Disseminated paracoccidioidomycosis: correlation between clinical and in vitro resistance to ketoconazole and trimethoprim sulphamethoxazole.
Journal: Mycoses 20030901
Title: A red rash on the face.
Journal: The Journal of family practice 20030901
Title: Gastric function in the elderly: effects on absorption of ketoconazole.
Journal: Journal of clinical pharmacology 20030901
Title: Limited utility of cyclosporine C2 monitoring in heart transplant recipients receiving ketoconazole.
Journal: Transplantation proceedings 20030901
Title: Effect of antifungal drugs on pathogenic Naegleria spp isolated from natural water sources.
Journal: Journal of the Medical Association of Thailand = Chotmaihet thangphaet 20030901
Title: Fluorine substitution can block CYP3A4 metabolism-dependent inhibition: identification of (S)-N-[1-(4-fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an orally bioavailable KCNQ2 opener devoid of CYP3A4 metabolism-dependent inhibition.
Journal: Journal of medicinal chemistry 20030828
Title: [Therapeutic safety of antimycotics in the treatment of systemic fungal infections].
Journal: Orvosi hetilap 20030824
Title: Prediction of hERG potassium channel affinity by traditional and hologram qSAR methods.
Journal: Bioorganic & medicinal chemistry letters 20030818
Title: Substituent effect on the reductive N-dearylation of 3-(indol-1-yl)-1,2-benzisoxazoles by rat liver microsomes.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030801
Title: Quantitative determination of some pharmaceutical piperazine derivatives through complexation with iron(III) chloride.
Journal: Farmaco (Societa chimica italiana : 1989) 20030801
Title: Hepatotoxicity and toxicokinetics of ketoconazole in rabbits.
Journal: Acta pharmacologica Sinica 20030801
Title: In vitro susceptibility testing of ciclopirox, terbinafine, ketoconazole and itraconazole against dermatophytes and nondermatophytes, and in vitro evaluation of combination antifungal activity.
Journal: The British journal of dermatology 20030801
Title: Activities of therapeutic agents against Naegleria fowleri in vitro and in a mouse model of primary amebic meningoencephalitis.
Journal: The Journal of parasitology 20030801
Title: Selectivities of human cytochrome P450 inhibitors toward rat P450 isoforms: study with cDNA-expressed systems of the rat.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030701
Title: In vitro metabolism of midazolam, triazolam, nifedipine, and testosterone by human liver microsomes and recombinant cytochromes p450: role of cyp3a4 and cyp3a5.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030701
Title: Cyclosporin C(2) and C(0) concentration monitoring in stable, long-term heart transplant recipients receiving metabolic inhibitors.
Journal: The Journal of heart and lung transplantation : the official publication of the International Society for Heart Transplantation 20030701
Title: The use of oral antifungal agents to treat onychomycosis.
Journal: Dermatologic clinics 20030701
Title: Evaluation of different calorimetric methods to determine the glass transition temperature and molecular mobility below T(g) for amorphous drugs.
Journal: International journal of pharmaceutics 20030618
Title: Involvement of CYP3A4, CYP2C8, and CYP2D6 in the metabolism of (R)- and (S)-methadone in vitro.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030601
Title: Comparative efficacies of oral ketoconazole and terbinafine for reducing Malassezia population sizes on the skin of Basset Hounds.
Journal: Veterinary dermatology 20030601
Title: Variations in color.
Journal: The Journal of family practice 20030601
Title: Gender differences in microsomal metabolic activation of hepatotoxic clivorine in rat.
Journal: Chemical research in toxicology 20030601
Title: Influence of drugs interacting with CYP3A4 on the pharmacokinetics, pharmacodynamics, and safety of the prandial glucose regulator repaglinide.
Journal: Journal of clinical pharmacology 20030601
Title: Antifungal compounds from Zanthoxylum chiloperone var. angustifolium.
Journal: Phytotherapy research : PTR 20030601
Title: Coadministration of tacrolimus and ketoconazole in renal transplant recipients: cost analysis and review of metabolic effects.
Journal: Transplantation proceedings 20030601
Title: Lithium gluconate 8% vs ketoconazole 2% in the treatment of seborrhoeic dermatitis: a multicentre, randomized study.
Journal: The British journal of dermatology 20030601
Title: Clotrimazole, ketoconazole, and clodinafop-propargyl as potent growth inhibitors of equine Babesia parasites during in vitro culture.
Journal: The Journal of parasitology 20030601
Title: Candidiasis (vulvovaginal).
Journal: Clinical evidence 20030601
Title: Identification of the cytochrome P450 enzymes involved in the N-oxidation of voriconazole.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030501
Title: Expression of the human CYP3A4 gene in the small intestine of transgenic mice: in vitro metabolism and pharmacokinetics of midazolam.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20030501
Title: Quinine 3-hydroxylation as a biomarker reaction for the activity of CYP3A4 in man.
Journal: European journal of clinical pharmacology 20030501
Title: Anti-Aspergillus activities of plant essential oils and their combination effects with ketoconazole or amphotericin B.
Journal: Archives of pharmacal research 20030501
Title: Effectiveness and tolerability of a standardized phytodrug derived from Solanum chrysotrichum on Tinea pedis: a controlled and randomized clinical trial.
Journal: Planta medica 20030501
Title: Modulatory effect of cAMP on fungal ergosterol level and inhibitory activity of azole drugs.
Journal: Canadian journal of microbiology 20030501
Title: Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery.
Journal: Journal of medicinal chemistry 20030424
Title: Validation of an HPLC method on short columns to assay ketoconazole and formaldehyde in shampoo.
Journal: Journal of pharmaceutical and biomedical analysis 20030424
Title: Production of progesterone from de novo-synthesized cholesterol in cumulus cells and its physiological role during meiotic resumption of porcine oocytes.
Journal: Biology of reproduction 20030401
Title: Demonstration of UVB-induced synthesis of 1 alpha,25-dihydroxyvitamin D3 (calcitriol) in human skin by microdialysis.
Journal: Archives of dermatological research 20030401
Title: Interaction between ketoconazole and almotriptan in healthy volunteers.
Journal: Journal of clinical pharmacology 20030401
Title: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites.
Journal: Pharmaceutical research 20030401
Title: Differential metabolism of midazolam in mouse liver and intestine microsomes: a comparison of cytochrome P450 activity and expression.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20030401
Title: Hepatotoxicity of ketoconazole in Sprague-Dawley rats: glutathione depletion, flavin-containing monooxygenases-mediated bioactivation and hepatic covalent binding.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20030401
Title: Effects of novel 17alpha-hydroxylase/C17, 20-lyase (P450 17, CYP 17) inhibitors on androgen biosynthesis in vitro and in vivo.
Journal: The Journal of steroid biochemistry and molecular biology 20030401
Title: High-content profiling of drug-drug interactions: cellular targets involved in the modulation of microtubule drug action by the antifungal ketoconazole.
Journal: Journal of biomolecular screening 20030401
Title: Retinoic acid metabolism inhibition by 3-azolylmethyl-1H-indoles and 2, 3 or 5-(alpha-azolylbenzyl)-1H-indoles.
Journal: Journal of enzyme inhibition and medicinal chemistry 20030401
Title: Prednisone metabolism in recipients of kidney or liver transplants and in lung recipients receiving ketoconazole.
Journal: Transplantation 20030327
Title: Enhancement of moxidectin bioavailability in lamb by a natural flavonoid: quercetin.
Journal: Veterinary parasitology 20030325
Title: Randomized, multicenter, phase II trial of two multicomponent regimens in androgen-independent prostate cancer.
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20030301
Title: Metabolism and metabolic inhibition of cilnidipine in human liver microsomes.
Journal: Acta pharmacologica Sinica 20030301
Title: Apparent mechanism-based inhibition of human CYP3A in-vitro by lopinavir.
Journal: The Journal of pharmacy and pharmacology 20030301
Title: [Nosocomial urinary infection due to Trichosporon asahii. First two cases in Chile].
Journal: Revista iberoamericana de micologia 20030301
Title: [Post traumatic subcutaneous mycosis due to Fusarium solani].
Journal: Revista iberoamericana de micologia 20030301
Title: Terbinafine effectiveness in ketoconazole-resistant mucocutaneous candidasis in polyglandular autoimmune syndrome type 1.
Journal: The Journal of the Association of Physicians of India 20030301
Title: Roles of human liver cytochrome P450 3A4 and 1A2 enzymes in the oxidation of myristicin.
Journal: Toxicology letters 20030203
Title: Rhabdomyolysis from cytochrome p-450 interaction of ketoconazole and simvastatin in prostate cancer.
Journal: The Journal of urology 20030201
Title: A murine model of coccidioidal meningitis.
Journal: The Journal of infectious diseases 20030201
Title: The effect of ketoconazole on the in vivo intestinal permeability of fexofenadine using a regional perfusion technique.
Journal: British journal of clinical pharmacology 20030201
Title: Steroid synthesis inhibition with ketoconazole and its effect upon the regulation of the hypothalamus-pituitary-adrenal system in healthy humans.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20030201
Title: Efficacy and safety of low-dose ketoconazole (50 mg) to reduce the cost of cyclosporine in renal allograft recipients.
Journal: Transplantation proceedings 20030201
Title: Antifungal agents of use in animal health--chemical, biochemical and pharmacological aspects.
Journal: Journal of veterinary pharmacology and therapeutics 20030201
Title: Coccidiomycosis in a dog.
Journal: The Canadian veterinary journal = La revue veterinaire canadienne 20030201
Title: [How to manage seborrheic dermatitis].
Journal: Revue medicale de Liege 20030201
Title: Identification of novel enzyme-prodrug combinations for use in cytochrome P450-based gene therapy for cancer.
Journal: Archives of biochemistry and biophysics 20030101
Title: Oxidative activation of acylguanidine prodrugs: intestinal presystemic activation in rats limits absorption and can be inhibited by co-administration of ketoconazole.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20030101
Title: Lack of effect of ketoconazole on the pharmacokinetics of rosuvastatin in healthy subjects.
Journal: British journal of clinical pharmacology 20030101
Title: Antifungal activity of the essential oil of Agastache rugosa Kuntze and its synergism with ketoconazole.
Journal: Letters in applied microbiology 20030101
Title: A case of infantile acne due to pityrosporum.
Journal: Pediatric dermatology 20030101
Title: [Conjunctival infection due to penicillium SP].
Journal: Archivos de la Sociedad Espanola de Oftalmologia 20030101
Title: [Molecular biological analysis of Tinea faciei caused by a clinically anomalous strain of Trichophyton mentagrophytes].
Journal: Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20030101
Title: The effect of granisetron on in vitro metabolism of paclitaxel and docetaxel.
Journal: Cancer journal (Sudbury, Mass.) 20030101
Title: Seborrheic dermatitis today, gone tomorrow? The link between the biocene and treatment.
Journal: Dermatology (Basel, Switzerland) 20030101
Title: Randomized, open-labeled, non-inferiority study between ciclopiroxolamine 1% cream and ketoconazole 2% foaming gel in mild to moderate facial seborrheic dermatitis.
Journal: Dermatology (Basel, Switzerland) 20030101
Title: Ketoconazole in the treatment of prostate cancer.
Journal: Clinical journal of oncology nursing 20030101
Title: Treatment of cutaneous leishmaniasis with ketoconazole cream.
Journal: The Journal of dermatological treatment 20030101
Title: Framing the future of antifungals in atopic dermatitis.
Journal: Dermatology (Basel, Switzerland) 20030101
Title: Tolerance to antidepressant treatment may be overcome by ketoconazole. Report of two cases.
Journal: Journal of psychiatric research 20030101
Title: Azoles for allergic bronchopulmonary aspergillosis associated with asthma.
Journal: The Cochrane database of systematic reviews 20030101
Title: [Madura foot (mycetoma)].
Journal: Vestnik khirurgii imeni I. I. Grekova 20030101
Title: [Finger agenesis after in utero exposure to ketoconazole: a case report].
Journal: Therapie 20030101
Title: Ketoconazole foam--connetics: connetics ketoconazole foam.
Journal: Drugs in R&D 20030101
Title: In vitro drug-drug interactions with perospirone and concomitantly administered drugs in human liver microsomes.
Journal: European journal of drug metabolism and pharmacokinetics 20030101
Title: [Vaginal candidiasis--treatment protocols using miconazole and fluconazole].
Journal: Akusherstvo i ginekologiia 20030101
Title: Oral manifestations of paracoccidioidomycosis. Report of 21 cases from Argentina.
Journal: Mycoses 20030101
Title: Fungal peritonitis in 15 patients on continuous ambulatory peritoneal dialysis (CAPD).
Journal: Mycoses 20030101
Title: Synthesis, in vitro/in vivo antifungal evaluation and structure-activity relationship study of 3(2H)-pyridazinones.
Journal: Arzneimittel-Forschung 20030101
Title: Occurrence of dermatomycoses and in-vitro therapeutic efficacy of three antifungal drugs on the growth of Epidermophyton floccosum.
Journal: Mycopathologia 20030101
Title: [Investigation of quantitative and species composition and antifungal drug susceptibility of yeasts isolated from patients with generalized periodontitis complicated by candidosis].
Journal: Mikrobiolohichnyi zhurnal (Kiev, Ukraine : 1993) 20030101
Title: [Madura's foot (mycetoma)].
Journal: Chirurgia (Bucharest, Romania : 1990) 20030101
Title: Medical treatment of hyperadrenocorticism in the dog.
Journal: Australian veterinary journal 20030101
Title: Protective effect of ketoconazole against experimentally induced gastric ulcers in rats.
Journal: Research communications in molecular pathology and pharmacology 20030101
Title: [In vitro sensitivity of Histoplasma capsulatum var. capsulatum to amphotericin B, ketoconazole, itroconazole and fluconazole].
Journal: Revista cubana de medicina tropical 20030101
Title: Separation of antifungal chiral drugs by SFC and HPLC: a comparative study.
Journal: Journal of biochemical and biophysical methods 20021231
Title: Pharmacophore model of drugs involved in P-glycoprotein multidrug resistance: explanation of structural variety (hypothesis).
Journal: Journal of medicinal chemistry 20021219
Title: Mathematical modelling of antifungal action.
Journal: Mycoses 20021201
Title: [Observations on the efficacy of Botai ointment in treating dermatosis common among armed forces receiving at-sea training].
Journal: Di 1 jun yi da xue xue bao = Academic journal of the first medical college of PLA 20021201
Title: Application of semisimultaneous midazolam administration for hepatic and intestinal cytochrome P450 3A phenotyping.
Journal: Clinical pharmacology and therapeutics 20021201
Title: Prevalence and antifungal susceptibilities of yeast isolates during one year at a university hospital in Turkey.
Journal: Journal of chemotherapy (Florence, Italy) 20021201
Title: Inhibition of the microsomal metabolism of 1,8-cineole in the common brushtail possum (Trichosurus vulpecula) by terpenes and other chemicals.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20021201
Title: National Cancer Institute intramural approach to advanced prostate cancer.
Journal: Clinical prostate cancer 20021201
Title: Triiodide ion and alizarin red S as two new reagents for the determination of clotrimazole and ketoconazole.
Journal: Journal of pharmaceutical and biomedical analysis 20021107
Title: Paracoccidioidomycosis: report of 2 cases mimicking squamous cell carcinoma.
Journal: Oral surgery, oral medicine, oral pathology, oral radiology, and endodontics 20021101
Title: Pharmacokinetics and electrocardiographic pharmacodynamics of artemether-lumefantrine (Riamet) with concomitant administration of ketoconazole in healthy subjects.
Journal: British journal of clinical pharmacology 20021101
Title: Chromatographic determination of clotrimazole, ketoconazole and fluconazole in pharmaceutical formulations.
Journal: Farmaco (Societa chimica italiana : 1989) 20021101
Title: Corticosteroids and pregnancy.
Journal: Seminars in reproductive medicine 20021101
Title: Synthesis of novel water soluble benzylazolium prodrugs of lipophilic azole antifungals.
Journal: Bioorganic & medicinal chemistry letters 20021007
Title: Sirolimus oral absorption in rats is increased by ketoconazole but is not affected by D-alpha-tocopheryl poly(ethylene glycol 1000) succinate.
Journal: The Journal of pharmacology and experimental therapeutics 20021001
Title: Interaction of cytochrome P450 3A inhibitors with P-glycoprotein.
Journal: The Journal of pharmacology and experimental therapeutics 20021001
Title: Preclinical activity of ketoconazole in combination with calcitriol or the vitamin D analogue EB 1089 in prostate cancer cells.
Journal: The Journal of urology 20021001
Title: Efficacy of ozonized sunflower oil in the treatment of tinea pedis.
Journal: Mycoses 20021001
Title: Vulvovaginal candidiasis.
Journal: BMJ (Clinical research ed.) 20020914
Title: Expression of paclitaxel-inactivating CYP3A activity in human colorectal cancer: implications for drug therapy.
Journal: British journal of cancer 20020909
Title: Putative role of the orphan nuclear receptor SXR (steroid and xenobiotic receptor) in the mechanism of CYP3A4 inhibition by xenobiotics.
Journal: The Journal of biological chemistry 20020906
Title: Macrophage plasma membrane cholesterol contributes to Brucella abortus infection of mice.
Journal: Infection and immunity 20020901
Title: In vitro, pharmacokinetic, and pharmacodynamic interactions of ketoconazole and midazolam in the rat.
Journal: The Journal of pharmacology and experimental therapeutics 20020901
Title: Characterization of quinidine 3-hydroxylation as a probe for the CYP 3A enzyme using a novel capillary electrophoresis technique.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20020901
Title: Evaluation of a 15-day screening assay using intact male rats for identifying steroid biosynthesis inhibitors and thyroid modulators.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20020901
Title: Ketoconazole suppresses interleukin-4 plus anti-CD40-induced IgE class switching in surface IgE negative B cells from patients with atopic dermatitis.
Journal: The Journal of investigative dermatology 20020901
Title: Azole susceptibility patterns and genetic relationship among oral Candida strains isolated in the era of highly active antiretroviral therapy.
Journal: Journal of acquired immune deficiency syndromes (1999) 20020901
Title: Design, synthesis, and biological evaluation of aryloxyethyl thiocyanate derivatives against Trypanosoma cruzi.
Journal: Journal of medicinal chemistry 20020829
Title: Low dose ketoconazole with replacement doses of hydrocortisone in patients with progressive androgen independent prostate cancer.
Journal: The Journal of urology 20020801
Title: Corneal ulcer caused by the new fungal species Sarcopodium oculorum.
Journal: Journal of clinical microbiology 20020801
Title: Ketoconazole potentiates the antitumor effects of nocodazole: In vivo therapy for human tumor xenografts in nude mice.
Journal: Molecular carcinogenesis 20020801
Title: In vivo measurement of human skin absorption of topically applied substances by a photoacoustic technique.
Journal: Physiological measurement 20020801
Title: Comparative efficacy of various treatment regimens for androgenetic alopecia in men.
Journal: The Journal of dermatology 20020801
Title: Randomized trial with itraconazole, ketoconazole and sulfadiazine in paracoccidioidomycosis.
Journal: Medical mycology 20020801
Title: Role of ketoconazole treatment in urinary-free cortisol-to-cortisone and tetrahydrocortisol-to-tetrahydrocortisone ratios in nonectopic Cushing's syndrome.
Journal: Endocrine 20020801
Title: Modulation of irinotecan metabolism by ketoconazole.
Journal: Journal of clinical oncology : official journal of the American Society of Clinical Oncology 20020715
Title: Determination of ketoconazole in human plasma by high-performance liquid chromatography-tandem mass spectrometry.
Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20020705
Title: HPLC-MS/MS analysis of the products generated from all-trans-retinoic acid using recombinant human CYP26A.
Journal: Journal of lipid research 20020701
Title: Application of modeling and simulation to integrate clinical pharmacology knowledge across a new drug application.
Journal: International journal of clinical pharmacology and therapeutics 20020701
Title: Ketoconazole and kids.
Journal: Postgraduate medicine 20020701
Title: [Tinea].
Journal: Archives de pediatrie : organe officiel de la Societe francaise de pediatrie 20020701
Title: Ketoconazole suppresses prostaglandin E(2)-induced cyclooxygenase-2 expression in human epidermoid carcinoma A-431 cells.
Journal: The Journal of investigative dermatology 20020701
Title: Protothecal colitis in a German shepherd dog.
Journal: Australian veterinary journal 20020701
Title: Double-blind antiglucocorticoid treatment in schizophrenia and schizoaffective disorder: a pilot study.
Journal: The world journal of biological psychiatry : the official journal of the World Federation of Societies of Biological Psychiatry 20020701
Title: Antifungal agents. 10. New derivatives of 1-[(aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-candida activity, and quantitative structure-analysis relationship studies.
Journal: Journal of medicinal chemistry 20020620
Title: New regulators of drug sensitivity in the family of yeast zinc cluster proteins.
Journal: The Journal of biological chemistry 20020614
Title: Cutaneous candidiasis in a dog caused by Candida guilliermondii.
Journal: The Veterinary record 20020608
Title: Simultaneous determination of ketoconazole and formaldehyde in a shampoo: liquid chromatography method development and validation.
Journal: Journal of chromatography. A 20020607
Title: Expression profiling in squamous carcinoma cells reveals pleiotropic effects of vitamin D3 analog EB1089 signaling on cell proliferation, differentiation, and immune system regulation.
Journal: Molecular endocrinology (Baltimore, Md.) 20020601
Title: Single- and multiple-dose pharmacokinetics of bosentan and its interaction with ketoconazole.
Journal: British journal of clinical pharmacology 20020601
Title: Oral treatments for toenail onychomycosis: a systematic review.
Journal: Archives of dermatology 20020601
Title: A randomised, single-blind, single-centre clinical trial to evaluate comparative clinical efficacy of shampoos containing ciclopirox olamine (1.5%) and salicylic acid (3%), or ketoconazole (2%, Nizoral) for the treatment of dandruff/seborrhoeic dermatitis.
Journal: The Journal of dermatological treatment 20020601
Title: Fluconazole versus ketoconazole in the treatment of tinea versicolor.
Journal: The Journal of dermatological treatment 20020601
Title: In vitro characterization of the inhibitory effects of ketoconazole on metabolic activities of cytochrome P-450 in canine hepatic microsomes.
Journal: American journal of veterinary research 20020601
Title: 7-Benzyloxyquinoline oxidation by P450eryF A245T: finding of a new fluorescent substrate probe.
Journal: Chemical research in toxicology 20020601
Title: Effects of ketoconazole on progesterone and cAMP production in MA-10 mouse Leydig tumor cells.
Journal: Biological & pharmaceutical bulletin 20020601
Title: [Intranasal rhinosporidiosis: presentation of the 1st case seen in the Congo].
Journal: Bulletin de la Societe de pathologie exotique (1990) 20020601
Title: Chronic administration of verapamil, ketoconazole and carbamazepine: impact on immunological parameters.
Journal: International journal of pharmaceutics 20020515
Title: Three-dimensional quantitative structure-activity relationships of inhibitors of P-glycoprotein.
Journal: Molecular pharmacology 20020501
Title: Potential role for the hypothalamo-pituitary-adrenal axis in the conditioned reinforcer-induced reinstatement of extinguished cocaine seeking in rats.
Journal: Psychopharmacology 20020501
Title: Oral FK 506 blood levels are elevated in pig short bowel model: further investigations with co-administration of an intestinal CYP3A4 inhibitor.
Journal: Transplantation proceedings 20020501
Title: [Candida infection of the skin and mucous membranes still a topic. Administering azoles with clinical understanding].
Journal: MMW Fortschritte der Medizin 20020409
Title: Effects of 3-MeSO2-DDE and some CYP inhibitors on glucocorticoid steroidogenesis in the H295R human adrenocortical carcinoma cell line.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20020401
Title: Human CYP3A4 and the metabolism of nefazodone and hydroxynefazodone by human liver microsomes and heterologously expressed enzymes.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20020401
Title: Ketoconazole increases cocaine and opioid use in methadone maintained patients.
Journal: Drug and alcohol dependence 20020401
Title: In vitro inhibition of pimozide N-dealkylation by selective serotonin reuptake inhibitors and azithromycin.
Journal: Journal of clinical psychopharmacology 20020401
Title: Antimicrobial activities of a new schizozygane indoline alkaloid from Schizozygia coffaeoides and the revised structure of isoschizogaline.
Journal: Journal of natural products 20020401
Title: Black-dot tinea capitis. Patchy hair loss is common in pediatric patients.
Journal: Postgraduate medicine 20020401
Title: Clinical comparison of the efficacy and tolerability of once daily Canesten with twice daily Nizoral (clotrimazole 1% cream vs. ketoconazole 2% cream) during a 28-day topical treatment of interdigital tinea pedis.
Journal: Mycoses 20020401
Title: Case report. Nattrassia mangiferae endophthalmitis.
Journal: Mycoses 20020401
Title: Chronic mucocutaneous candidiasis.
Journal: JAAPA : official journal of the American Academy of Physician Assistants 20020401
Title: Cyclosporin and ketoconazole interaction for treatment of perianal fistulas in the dog.
Journal: Australian veterinary journal 20020401
Title: Superficial mycosis superimposing on isolated lichen planus of the lip: a case report and review of the literature.
Journal: Cutis 20020401
Title: [Identification and antifungal susceptibility of Candida spp isolated from invasive mycoses. Influence of growth inhibition percentage to determine minimal inhibitory concentration].
Journal: Revista medica de Chile 20020401
Title: Cyclosporine and ketoconazole for the treatment of perianal fistulas in dogs.
Journal: Journal of the American Veterinary Medical Association 20020401
Title: Simple high-performance liquid chromatography method for the simultaneous determination of ketoconazole and piperine in rat plasma and hepatocyte culture.
Journal: Journal of chromatography. A 20020308
Title: Effect of antifungal azoles on the heme detoxification system of malarial parasite.
Journal: Journal of biochemistry 20020301
Title: Effect of oral ketoconazole on first-pass effect of nifedipine after oral administration in dogs.
Journal: Journal of pharmaceutical sciences 20020301
Title: Minimal effect of ketoconazole on cyclosporine (SangCyA) oral absorption and first-pass metabolism in rats: evidence of a significant vehicle effect on SangCyA absorption.
Journal: Biopharmaceutics & drug disposition 20020301
Title: Multicenter Brazilian study of oral Candida species isolated from AIDS patients.
Journal: Memorias do Instituto Oswaldo Cruz 20020301
Title: Cytochrome P450 enzymes contributing to demethylation of maprotiline in man.
Journal: Pharmacology & toxicology 20020301
Title: Identification of the human P450 enzymes involved in the in vitro metabolism of the synthetic steroidal hormones Org 4060 and Org 30659.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20020201
Title: Infectious keratitis in orthokeratology.
Journal: Clinical & experimental ophthalmology 20020201
Title: Ring substituted 3-phenyl-1-(2-pyrazinyl)-2-propen-1-ones as potential photosynthesis-inhibiting, antifungal and antimycobacterial agents.
Journal: Farmaco (Societa chimica italiana : 1989) 20020201
Title: Effect of multiple dosing of ketoconazole on pharmacokinetics of midazolam, a cytochrome P-450 3A substrate in beagle dogs.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20020101
Title: Peppermint oil enhances cyclosporine oral bioavailability in rats: comparison with D-alpha-tocopheryl poly(ethylene glycol 1000) succinate (TPGS) and ketoconazole.
Journal: Journal of pharmaceutical sciences 20020101
Title: CYP3A4-mediated hepatic metabolism of the HIV-1 protease inhibitor saquinavir in vitro.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20020101
Title: Interventions for treating oral candidiasis for patients with cancer receiving treatment.
Journal: The Cochrane database of systematic reviews 20020101
Title: Comparison of two methods for antifungal susceptibility testing of Trichophyton rubrum.
Journal: European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology 20020101
Title: Mycetoma caused by Fusarium solani with osteolytic lesions on the hand: case report.
Journal: Mycopathologia 20020101
Title: A unique case of bladder mycetoma.
Journal: Tropical doctor 20020101
Title: Pathology case of the month. Chronic leg ulcer in a missionary worker. Cutaneous leishmaniasis.
Journal: The Journal of the Louisiana State Medical Society : official organ of the Louisiana State Medical Society 20020101
Title: Ectopic ACTH-syndrome due to a thymic carcinoid tumor.
Journal: Acta clinica Belgica 20020101
Title: More economical use of cyclosporine through combination drug therapy.
Journal: Journal of the American Animal Hospital Association 20020101
Title: Sustained release bioadhesive effervescent ketoconazole microcapsules tabletted for vaginal delivery.
Journal: Journal of microencapsulation 20020101
Title: Post-antifungal effect and effects of sub-MIC concentrations on previously treated Candida spp.: influence of exposure time and concentration.
Journal: Scandinavian journal of infectious diseases 20020101
Title: Euclidean and fractal computer-assisted corneofungimetry: a comparison of 2% ketoconazole and 1% terbinafine topical formulations.
Journal: Dermatology (Basel, Switzerland) 20020101
Title: A case of confluent and reticulated papillomatosis responsive to ketoconazole cream.
Journal: Nihon Ishinkin Gakkai zasshi = Japanese journal of medical mycology 20020101
Title: A double-blind placebo-controlled study of ketoconazole + desonide gel combination in the treatment of facial seborrheic dermatitis.
Journal: Dermatology (Basel, Switzerland) 20020101
Title: Efficacy and skin tolerability of Saliker in the treatment of dandruff.
Journal: European journal of dermatology : EJD 20020101
Title: Antifungal topical therapy in oral chronic candidosis. A comparative study.
Journal: Medicina oral : organo oficial de la Sociedad Espanola de Medicina Oral y de la Academia Iberoamericana de Patologia y Medicina Bucal 20020101
Title: Desloratadine has no clinically relevant electrocardiographic or pharmacodynamic interactions with ketoconazole.
Journal: Clinical pharmacokinetics 20020101
Title: Ketoconazole potentiates terfenadine-induced apoptosis in human Hep G2 cells through inhibition of cytochrome p450 3A4 activity.
Journal: Journal of cellular biochemistry 20020101
Title: Atopic dermatitis with mononuclear phagocytic activity deficiency.
Journal: Allergologia et immunopathologia 20020101
Title: A multicenter randomized trial of ketoconazole 2% and zinc pyrithione 1% shampoos in severe dandruff and seborrheic dermatitis.
Journal: Skin pharmacology and applied skin physiology 20020101
Title: Efficacy and skin tolerability of saliker in the treatment of dandruff.
Journal: European journal of dermatology : EJD 20020101
Title: Low dose ketoconazole therapy and thyroid functions in rats.
Journal: Acta medica (Hradec Kralove) 20020101
Title: The preventive effect of ketoconazole on experimental metastasis from a human pancreatic carcinoma may be related to its effect on prostaglandin synthesis.
Journal: International journal of gastrointestinal cancer 20020101
Title: Invitro drug sensitivity of Trichophyton species against griseofulvin and ketoconazole.
Journal: Hindustan antibiotics bulletin 20020101
Title: Ectopic adrenocorticotropic hormone syndrome caused by metastatic carcinoma of the prostate: therapeutic response to ketoconazole.
Journal: Endocrine practice : official journal of the American College of Endocrinology and the American Association of Clinical Endocrinologists 20020101
Title: Toward a novel metal-based chemotherapy against tropical diseases. 6. Synthesis and characterization of new copper(II) and gold(I) clotrimazole and ketoconazole complexes and evaluation of their activity against Trypanosoma cruzi.
Journal: Inorganic chemistry 20011231
Title: Fatal aplastic anemia during treatment with ketoconazole.
Journal: The American journal of medicine 20011215
Title: No evidence of oxidant events in amphotericin B cytotoxicity versus L. infantum promastigotes.
Journal: Parasite (Paris, France) 20011201
Title: Novel steroidal pyrimidyl inhibitors of P450 17 (17 alpha-hydroxylase/C17-20-lyase).
Journal: Archiv der Pharmazie 20011201
Title: Effects of ketoconazole on oestrus cycle and convulsant action of pentylenetetrazol in mice.
Journal: Pharmacology & toxicology 20011201
Title: Diazinon is activated by CYP2C19 in human liver.
Journal: Toxicology and applied pharmacology 20011115
Title: Enhanced antifungal activity of ketoconazole by Euphorbia characias latex against Candida albicans.
Journal: Journal of ethnopharmacology 20011101
Title: Quantitative liquid chromatography/mass spectrometry/mass spectrometry warfarin assay for in vitro cytochrome P450 studies.
Journal: Analytical biochemistry 20011101
Title: Importance of inhibin B in the regulation of FSH secretion in the human male.
Journal: The Journal of clinical endocrinology and metabolism 20011101
Title: Effects of azoles on human acute myelogenous leukemia blasts and T lymphocytes derived from acute leukemia patients with chemotherapy-induced cytopenia.
Journal: International immunopharmacology 20011101
Title: Improved responsiveness of PCOS patients to clomiphene after CYP17a inhibitor.
Journal: Journal of assisted reproduction and genetics 20011101
Title: Gene amplification in amphotericin B-resistant Leishmania tarentolae.
Journal: Experimental parasitology 20011101
Title: Relative contribution of CYP3A to amitriptyline clearance in humans: in vitro and in vivo studies.
Journal: Journal of clinical pharmacology 20011001
Title: A clinical case of canine mycotic pneumonia.
Journal: Journal of veterinary medicine. A, Physiology, pathology, clinical medicine 20011001
Title: Comparative efficacy of ketoconazole and fluconazole in the treatment of pityriasis versicolor: a one year follow-up study.
Journal: The Journal of dermatology 20011001
Title: Ketoconazole and Flutamide in the treatment of disseminated intravascular clotting from prostate cancer: a case report and review.
Journal: Journal of the Medical Association of Thailand = Chotmaihet thangphaet 20011001
Title: Effect of pharmacotechnical design on the in vitro interaction of ketoconazole tablets with non-systemic antacids.
Journal: International journal of pharmaceutics 20010911
Title: [Spondylodiscitis due to Histoplasma duboisii. Report of two cases and review of the literature].
Journal: Neuro-Chirurgie 20010901
Title: 7-Deoxyloganin 7-hydroxylase in Lonicera japonica cell cultures.
Journal: Phytochemistry 20010901
Title: Post-antifungal effect of polyene, azole and DNA-analogue agents against oral Candida albicans and Candida tropicalis isolates in HIV disease.
Journal: Journal of oral pathology & medicine : official publication of the International Association of Oral Pathologists and the American Academy of Oral Pathology 20010901
Title: A simple algorithm for designing group sequential clinical trials.
Journal: Biometrics 20010901
Title: Lack of effect of reboxetine on cardiac repolarization.
Journal: Clinical pharmacology and therapeutics 20010901
Title: Medical treatment of canine pituitary-dependent hyperadrenocorticism (Cushing's disease).
Journal: The Veterinary clinics of North America. Small animal practice 20010901
Title: Severe respiratory failure secondary to Cushing's myopathy.
Journal: Journal of endocrinological investigation 20010901
Title: Oral histoplasmosis.
Journal: The Journal of the Association of Physicians of India 20010901
Title: Comparative study of the efficacy of oral ketoconazole with intra-lesional meglumine antimoniate (Glucantime) for the treatment of cutaneous leishmaniasis.
Journal: The Journal of dermatological treatment 20010901
Title: Pulmonary candidiasis caused by Candida albicans in a Greek tortoise (Testudo graeca) and treatment with intrapulmonary amphotericin B.
Journal: Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians 20010901
Title: Cyclosporin immunosuppression of sheep: pharmacokinetics and allograft survival.
Journal: Veterinary immunology and immunopathology 20010830
Title: Primary culture system of adrenocortical cells from dogs to evaluate direct effects of chemicals on steroidogenesis.
Journal: Toxicology 20010828
Title: 3-Phenyl-5-acyloxymethyl-2H,5H-furan-2-ones: synthesis and biological activity of a novel group of potential antifungal drugs.
Journal: Journal of medicinal chemistry 20010816
Title: Ketoconazole-induced conformational changes in the active site of cytochrome P450eryF.
Journal: Journal of molecular biology 20010803
Title: State-dependent block of rabbit vascular smooth muscle delayed rectifier and Kv1.5 channels by inhibitors of cytochrome P450-dependent enzymes.
Journal: The Journal of pharmacology and experimental therapeutics 20010801
Title: Rationale for combination ketoconazole/ vitamin D treatment of prostate cancer.
Journal: Urology 20010801
Title: Modulation of the cytochrome P450-mediated metabolism of ifosfamide by ketoconazole and rifampin.
Journal: Clinical pharmacology and therapeutics 20010801
Title: A systematic review of the effectiveness of antifungal drugs for the prevention and treatment of oropharyngeal candidiasis in HIV-positive patients.
Journal: Oral surgery, oral medicine, oral pathology, oral radiology, and endodontics 20010801
Title: Application of capillary zone electrophoresis with off-line solid-phase extraction to in vitro metabolism studies of antifungals.
Journal: Electrophoresis 20010801
Title: Ketoconazole suppresses food restriction-induced increases in heroin self-administration in rats: sex differences.
Journal: Experimental and clinical psychopharmacology 20010801
Title: Characterization of amorphous ketoconazole using modulated temperature differential scanning calorimetry.
Journal: Journal of pharmaceutical sciences 20010801
Title: Arthroderma benhamiae infection in a rabbit.
Journal: The Journal of veterinary medical science 20010801
Title: [Modern local therapy of foot mycoses in servicemen].
Journal: Voenno-meditsinskii zhurnal 20010801
Title: Adsorptive behavior and electrochemical determination of the anti-fungal agent ketoconazole.
Journal: Fresenius' journal of analytical chemistry 20010801
Title: Uptake of Malassezia furfur by human dermal fibroblasts: effect of ketoconazole and cytoskeleton inhibitors.
Journal: Archives of dermatological research 20010801
Title: Heterogeneity in antifungal susceptibility of clones of Candida albicans isolated on single and sequential visits from a HIV-infected southern Chinese cohort.
Journal: Journal of oral pathology & medicine : official publication of the International Association of Oral Pathologists and the American Academy of Oral Pathology 20010701
Title: Effect of an extract of the root of Scutellaria baicalensis and its flavonoids on aflatoxin B1 oxidizing cytochrome P450 enzymes.
Journal: Planta medica 20010701
Title: Ca(2+) transport into an intracellular acidic compartment of Candida parapsilosis.
Journal: FEBS letters 20010629
Title: Application to drug-food interactions of living cells as in vitro model expressing cytochrome P450 activity: enzyme inhibition by lemon juice.
Journal: Talanta 20010621
Title: Oropharyngeal candidiasis in patients with human immunodeficiency virus: correlation of clinical outcome with in vitro resistance, serum azole levels, and immunosuppression.
Journal: Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20010601
Title: Arachidonic acid directly activates members of the mitogen-activated protein kinase superfamily in rabbit proximal tubule cells.
Journal: Kidney international 20010601
Title: Aromatization mediates testosterone's short-term feedback restraint of 24-hour endogenously driven and acute exogenous gonadotropin-releasing hormone-stimulated luteinizing hormone and follicle-stimulating hormone secretion in young men.
Journal: The Journal of clinical endocrinology and metabolism 20010601
Title: Photo quiz. Congenital cutaneous candidiasis.
Journal: Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20010601
Title: Successful treatment of Acanthamoeba meningitis with combination oral antimicrobials.
Journal: The Pediatric infectious disease journal 20010601
Title: Systemic ketoconazole is an effective treatment of atopic dermatitis with IgE-mediated hypersensitivity to yeasts.
Journal: Allergy 20010601
Title: Temporary remission of disseminated paecilomycosis in a German shepherd dog treated with ketoconazole.
Journal: Journal of the South African Veterinary Association 20010601
Title: [In vitro antifungal susceptibility of dematiaceous filamentous fungi using the E-test].
Journal: Revista espanola de quimioterapia : publicacion oficial de la Sociedad Espanola de Quimioterapia 20010601
Title: The effect of gut metabolism on tacrolimus bioavailability in renal transplant recipients.
Journal: Transplantation 20010515
Title: Mechanism of action of anti-proliferative lysophospholipid analogues against the protozoan parasite Trypanosoma cruzi: potentiation of in vitro activity by the sterol biosynthesis inhibitor ketoconazole.
Journal: The Journal of antimicrobial chemotherapy 20010501
Title: Effect of inoculum form on in vitro antifungal susceptibilities of Aspergillus spp.
Journal: The Journal of antimicrobial chemotherapy 20010501
Title: Low salivary cortisol levels and aggressive behavior.
Journal: Archives of general psychiatry 20010501
Title: The interaction of saquinavir (soft gelatin capsule) with ketoconazole, erythromycin and rifampicin: comparison of the effect in healthy volunteers and in HIV-infected patients.
Journal: European journal of clinical pharmacology 20010501
Title: Metabolism of amiodarone (Part III): identification of rabbit cytochrome P450 isoforms involved in the hydroxylation of mono-N-desethylamiodarone.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20010501
Title: [Endemic mycotic infections].
Journal: La Revue du praticien 20010415
Title: Liquid chromatographic determination of ketoconazole, a potent inhibitor of CYP3A4-mediated metabolism.
Journal: Journal of chromatography. B, Biomedical sciences and applications 20010405
Title: Evaluation of the male pubertal onset assay to detect testosterone and steroid biosynthesis inhibitors in CD rats.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20010401
Title: Application of the relative activity factor approach in scaling from heterologously expressed cytochromes p450 to human liver microsomes: studies on amitriptyline as a model substrate.
Journal: The Journal of pharmacology and experimental therapeutics 20010401
Title: Hypokalemia, metabolic alkalosis, and hypertension: Cushing's syndrome in a patient with metastatic prostate adenocarcinoma.
Journal: American journal of kidney diseases : the official journal of the National Kidney Foundation 20010401
Title: Pharmacokinetics of cyclosporine in heart transplant recipients receiving metabolic inhibitors.
Journal: The Journal of heart and lung transplantation : the official publication of the International Society for Heart Transplantation 20010401
Title: Interaction of two novel 14-epivitamin D3 analogs with vitamin D3 receptor-retinoid X receptor heterodimers on vitamin D3 responsive elements.
Journal: Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research 20010401
Title: Successful treatment of visceral leishmaniasis with allopurinol plus ketoconazole in an infant who developed pancreatitis caused by meglumine antimoniate.
Journal: The Pediatric infectious disease journal 20010401
Title: Ranitidine-related Stevens-Johnson syndrome in patients with severe liver diseases: a report of two cases.
Journal: Journal of gastroenterology and hepatology 20010401
Title: Preparation and physical characterization of alginate microparticles using air atomization method.
Journal: Drug development and industrial pharmacy 20010401
Title: Hard palate perforation: an unusual finding in paracoccidioidomycosis.
Journal: International journal of dermatology 20010401
Title: Drug sensitivity of Candida yeast isolated from patients with allergic diseases.
Journal: Bulletin of experimental biology and medicine 20010401
Title: Treatments for common superficial fungal infections.
Journal: Dermatology nursing 20010401
Title: Coadministration of ketoconazole and cyclosporine for kidney transplant recipients: long-term follow-up and study of metabolic consequences.
Journal: American journal of kidney diseases : the official journal of the National Kidney Foundation 20010301
Title: Clinical inquiries. What is the best oral antifungal medication for tinea capitis?
Journal: The Journal of family practice 20010301
Title: A new class of nonsteroidal aromatase inhibitors: design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17 alpha-hydroxylase/C17,20-lyase.
Journal: Journal of medicinal chemistry 20010301
Title: Treatment for coccidioidomycosis in pregnancy?
Journal: Postgraduate medicine 20010301
Title: Fatal liver failure due to ketoconazole treatment of a girl with Cushing's syndrome.
Journal: Journal of pediatric endocrinology & metabolism : JPEM 20010301
Title: [Ocular parasitoses and mycoses: cases diagnosed in the Central University Hospital of Sfax between 1996 and 1999].
Journal: Bulletin de la Societe de pathologie exotique (1990) 20010301
Title: Effects of ketoconazole on the acquisition of intravenous cocaine self-administration under different feeding conditions in rats.
Journal: Psychopharmacology 20010301
Title: Emedastine-ketoconazole: pharmacokinetic and pharmacodynamic interactions in healthy volunteers.
Journal: International journal of clinical pharmacology and therapeutics 20010301
Title: In vitro/in vivo scaling of alprazolam metabolism by CYP3A4 and CYP3A5 in humans.
Journal: Biopharmaceutics & drug disposition 20010301
Title: Aminoglutethimide, a steroidogenesis inhibitor, abolishes hormonal induction of ornithine decarboxylase in steroidogenic tissues: evidence for its role as cAMP-dependent protein kinase inhibitor.
Journal: Biochemical and biophysical research communications 20010216
Title: Muting of androgen negative feedback unveils impoverished gonadotropin-releasing hormone/luteinizing hormone secretory reactivity in healthy older men.
Journal: The Journal of clinical endocrinology and metabolism 20010201
Title: CYP3A4 is the major CYP isoform mediating the in vitro hydroxylation and demethylation of flunitrazepam.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20010201
Title: Modulation of P450 CYP3A4-dependent metabolism by P-glycoprotein: implications for P450 phenotyping.
Journal: The Journal of pharmacology and experimental therapeutics 20010201
Title: A novel sequence element is involved in the transcriptional regulation of expression of the ERG1 (squalene epoxidase) gene in Saccharomyces cerevisiae.
Journal: European journal of biochemistry 20010201
Title: Lack of effect of a single dose of ketoconazole on the pharmacokinetics of citalopram.
Journal: Pharmacotherapy 20010201
Title: Determination of minumum inhibitory concentrations of Candida species isolated from vaginal swab specimens by using broth macrodilution and E-test.
Journal: Journal of chemotherapy (Florence, Italy) 20010201
Title: Effect of ketoconazole, itraconazole and fluconazole on the gastrointestinal colonization of mice by Candida albicans.
Journal: Journal of chemotherapy (Florence, Italy) 20010201
Title: Ketoconazole in bipolar patients with depressive symptoms: a case series and literature review.
Journal: Bipolar disorders 20010201
Title: Species difference in stereoselective involvement of CYP3A in the mono-N-dealkylation of disopyramide.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20010201
Title: Indications for the involvement of a CYP3A-like iso-enzyme in the metabolism of chlorobornane (Toxaphene) congeners in seals from inhibition studies with liver microsomes.
Journal: Aquatic toxicology (Amsterdam, Netherlands) 20010101
Title: Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20010101
Title: Meiosis-activating sterol and the maturation of isolated mouse oocytes.
Journal: Biology of reproduction 20010101
Title: The combination of oral amphotericin B with azoles prevents the emergence of resistant Candida species in neutropenic patients.
Journal: British journal of haematology 20010101
Title: Studies on the metabolism of troglitazone to reactive intermediates in vitro and in vivo. Evidence for novel biotransformation pathways involving quinone methide formation and thiazolidinedione ring scission.
Journal: Chemical research in toxicology 20010101
Title: Endogenous lipoid pneumonia associated with undifferentiated connective tissue disease (UCTD).
Journal: Medical science monitor : international medical journal of experimental and clinical research 20010101
Title: [The yeast fungus Malassezia: pathogen, pathogenesis and therapy].
Journal: Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete 20010101
Title: Differential regulation of gonadotropin secretion by testosterone in the human male: absence of a negative feedback effect of testosterone on follicle-stimulating hormone secretion.
Journal: The Journal of clinical endocrinology and metabolism 20010101
Title: Effect of ketoconazole 1% and 2% shampoos on severe dandruff and seborrhoeic dermatitis: clinical, squamometric and mycological assessments.
Journal: Dermatology (Basel, Switzerland) 20010101
Title: Investigation of ketoconazole copper(II) and cobalt(II) complexes and their spectrophotometric applications.
Journal: Journal of AOAC International 20010101
Title: Ketoconazole and pulmonary failure after esophagectomy: a prospective clinical trial.
Journal: Diseases of the esophagus : official journal of the International Society for Diseases of the Esophagus 20010101
Title: [Antifungal susceptibility of emerging yeast pathogens].
Journal: Enfermedades infecciosas y microbiologia clinica 20010101
Title: Systemic ketoconazole for yeast allergic patients with atopic dermatitis.
Journal: Journal of the European Academy of Dermatology and Venereology : JEADV 20010101
Title: A novel extractionless hplc fluorescence method for the determination of glyburide in the human plasma: application to a bioequivalence study.
Journal: Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques 20010101
Title: Guess what! Tinea capitis by Trichophyton schöenleinii.
Journal: European journal of dermatology : EJD 20010101
Title: A preliminary study on the feasibility of an automated blood-sampling system in conjunction with liquid chromatography/mass spectrometry.
Journal: Rapid communications in mass spectrometry : RCM 20010101
Title: Azoles for allergic bronchopulmonary aspergillosis associated with asthma.
Journal: The Cochrane database of systematic reviews 20010101
Title: Case report. Disseminated tinea of the verrucous type due to epidermophyton floccosum.
Journal: Mycoses 20010101
Title: A plea to bridge the gap between antifungals and the management of onychomycosis.
Journal: American journal of clinical dermatology 20010101
Title: [Apropos of 'Onychomycoses caused by non-dermatophytic filamentous fungi in Cádiz'].
Journal: Enfermedades infecciosas y microbiologia clinica 20010101
Title: [Antitoxic properties of hepazan--a novel inducer of microsomal enzyme system].
Journal: Eksperimental'naia i klinicheskaia farmakologiia 20010101
Title: [Acanthamoeba lesions of the cornea].
Journal: Vestnik oftalmologii 20010101
Title: Successful treatment of CAPD peritonitis caused by rhodotorula mucilaginosa.
Journal: Peritoneal dialysis international : journal of the International Society for Peritoneal Dialysis 20010101
Title: Lack of CYP3A4 inhibition by grapefruit juice and ketoconazole upon clozapine administration in vivo.
Journal: Drug metabolism and drug interactions 20010101
Title: [Vulvovaginal candidiasis in childhood--diagnostic and therapeutic results].
Journal: Akusherstvo i ginekologiia 20010101
Title: Recovery of bone mineral density after surgical cure, but not by ketoconazole treatment, in Cushing's syndrome.
Journal: Osteoporosis international : a journal established as result of cooperation between the European Foundation for Osteoporosis and the National Osteoporosis Foundation of the USA 20010101
Title: [Vaginal candidiasis: etiology and sensitivity profile to antifungal agents in clinical use].
Journal: Revista Argentina de microbiologia 20010101
Title: Drug susceptibility testing of Malassezia furfur strains to antifungal agents.
Journal: Folia medica 20010101
Title: [The sensitivity to ketoconazole of Candida strains isolated from the digestive tract ontocenoses in children].
Journal: Wiadomosci parazytologiczne 20010101
Title: Antiandrogenic effects of novel androgen synthesis inhibitors on hormone-dependent prostate cancer.
Journal: Cancer research 20001201
Title: Lipoproteins regulate expression of the steroidogenic acute regulatory protein (StAR) in mouse adrenocortical cells.
Journal: The Journal of biological chemistry 20001124
Title: The involvement of flavin-containing monooxygenase but not CYP3A4 in metabolism of itopride hydrochloride, a gastroprokinetic agent: comparison with cisapride and mosapride citrate.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20001001
Title: Identification of cytochrome P4503A as the major subfamily responsible for the metabolism of roquinimex in man.
Journal: Xenobiotica; the fate of foreign compounds in biological systems 20000901
Title: 3-Phenyl-5-methyl-2H,5H-furan-2-ones: tuning antifungal activity by varying substituents on the phenyl ring.
Journal: Bioorganic & medicinal chemistry letters 20000821
Title: Comparison of three different in vitro mutation assays used for the investigation of cytochrome P450-mediated mutagenicity of nitro-polycyclic aromatic hydrocarbons.
Journal: Mutation research 20000323
Title: Modulation by drugs of human hepatic sodium-dependent bile acid transporter (sodium taurocholate cotransporting polypeptide) activity.
Journal: The Journal of pharmacology and experimental therapeutics 19991201
Title: Cushing's syndrome in pregnancy treated by ketoconazole: case report and review of the literature.
Journal: Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology 19990601
Title: In vitro susceptibilities of clinical yeast isolates to the new antifungal eberconazole compared with their susceptibilities to clotrimazole and ketoconazole.
Journal: Antimicrobial agents and chemotherapy 19990501
Title: Interplay between CYP3A-mediated metabolism and polarized efflux of terfenadine and its metabolites in intestinal epithelial Caco-2 (TC7) cell monolayers.
Journal: Pharmaceutical research 19990501
Title: Cytochrome P450 3A4 in vivo ketoconazole competitive inhibition: determination of Ki and dangers associated with high clearance drugs in general.
Journal: Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques 19990101
Title: Ketoconazole reduces low dose cocaine self-administration in rats.
Journal: Drug and alcohol dependence 19981201
Title: Characterization of the cloned human intermediate-conductance Ca2+-activated K+ channel.
Journal: The American journal of physiology 19980901
Title: Synergy of nitric oxide and azoles against Candida species in vitro.
Journal: Antimicrobial agents and chemotherapy 19980901
Title: Blockade of HERG and Kv1.5 by ketoconazole.
Journal: The Journal of pharmacology and experimental therapeutics 19980801
Title: Trazodone is metabolized to m-chlorophenylpiperazine by CYP3A4 from human sources.
Journal: Drug metabolism and disposition: the biological fate of chemicals 19980601
Title: Kinetic characterization and identification of the enzymes responsible for the hepatic biotransformation of adinazolam and N-desmethyladinazolam in man.
Journal: The Journal of pharmacy and pharmacology 19980301
Title: Reduction of oxysterol levels up-regulates HMG-CoA reductase activity in rat liver.
Journal: Atherosclerosis 19970601
Title: Selective biotransformation of the human immunodeficiency virus protease inhibitor saquinavir by human small-intestinal cytochrome P4503A4: potential contribution to high first-pass metabolism.
Journal: Drug metabolism and disposition: the biological fate of chemicals 19970201
Title: Combined use of astemizole and ketoconazole resulting in torsade de pointes.
Journal: Journal of the Formosan Medical Association = Taiwan yi zhi 19970201
Title: Hepatic injury during ketoconazole therapy in patients with onychomycosis: a controlled cohort study.
Journal: Hepatology (Baltimore, Md.) 19970101
Title: In vitro synergistic activity of ketoconazole with valproic acid against Candida species.
Journal: Arzneimittel-Forschung 19960901
Title: Human reductive halothane metabolism in vitro is catalyzed by cytochrome P450 2A6 and 3A4.
Journal: Drug metabolism and disposition: the biological fate of chemicals 19960901
Title: Paranoid delusions caused by ketoconazole.
Journal: International journal of dermatology 19960101
Title: Treatment of New World cutaneous and mucosal leishmaniases.
Journal: Clinics in dermatology 19960101
Title: Antifungal agents. 9. 3-Aryl-4-[alpha-(1H-imidazol-1-yl)arylmethyl]pyrroles: a new class of potent anti-Candida agents.
Journal: Journal of medicinal chemistry 19951013
Title: In vitro susceptibility of filamentous fungi to itraconazole.
Journal: Indian journal of pathology & microbiology 19951001
Title: Synthesis and antifungal activity of new azole derivatives containing an N-acylmorpholine ring.
Journal: Journal of medicinal chemistry 19950929
Title: Mechanism for species-specific induction of Leydig cell tumors in rats by lansoprazole.
Journal: Fundamental and applied toxicology : official journal of the Society of Toxicology 19950701
Title: Novel steroidal inhibitors of human cytochrome P45017 alpha (17 alpha-hydroxylase-C17,20-lyase): potential agents for the treatment of prostatic cancer.
Journal: Journal of medicinal chemistry 19950623
Title: In vitro activity of D0870 compared with those of other azoles against fluconazole-resistant Candida spp.
Journal: Antimicrobial agents and chemotherapy 19950401
Title: Selectivity of isoprenoid-containing imidazole antifungal compounds for sterol 14-demethylase P450 (P450(14)DM) and 7-ethoxycoumarin O-deethylase P450 of rat liver microsomes.
Journal: Biochemical pharmacology 19941018
Title: Hypersensitivity to ketoconazole.
Journal: Annals of allergy 19941001
Title: Pneumocystis carinii is resistant to imidazole antifungal agents.
Journal: Antimicrobial agents and chemotherapy 19940801
Title: Derivatives of a novel cyclopeptolide. 1. Synthesis, antifungal activity, and structure-activity relationships.
Journal: Journal of medicinal chemistry 19940624
Title: Selective inhibition of mammalian lanosterol 14 alpha-demethylase by RS-21607 in vitro and in vivo.
Journal: Biochemistry 19940419
Title: Antimicrobial and antitumoral activities of 6-allyl-5,6-dihydro-5-hydroxypyran-2-one, a lactone produced by a new Drechslera species.
Journal: Die Pharmazie 19940401
Title: Ro 09-1470 is a selective inhibitor of P-450 lanosterol C-14 demethylase of fungi.
Journal: Antimicrobial agents and chemotherapy 19931201
Title: Effects of the combination of ketoconazole and calmodulin inhibitors against Candida albicans in vitro. Short communication.
Journal: Arzneimittel-Forschung 19930901
Title: Antifungal agents. VI. In vitro antifungal activities of halobenzoyl esters of cis- and trans-[2-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-ylmethyl)-1,3- dioxolan-4-yl]carbinols.
Journal: Farmaco (Societa chimica italiana : 1989) 19930801
Title: Synthesis and structure-activity relationships of phenyl-substituted benzylamine antimycotics: a novel benzylbenzylamine antifungal agent for systemic treatment.
Journal: Journal of medicinal chemistry 19930723
Title: Selective inhibition of mammalian lanosterol 14 alpha-demethylase: a possible strategy for cholesterol lowering.
Journal: Journal of medicinal chemistry 19930723
Title: Effects of the combination of ketoconazole and calcium channel antagonists against Candida albicans in vitro.
Journal: Arzneimittel-Forschung 19930701
Title: Ventricular fibrillation secondary to itraconazole induced hypokalaemia.
Journal: The Journal of infection 19930501
Title: Ketoconazole induced papilledema.
Journal: Acta ophthalmologica 19930401
Title: Torsades de pointes after terfenadine-itraconazole interaction.
Journal: BMJ (Clinical research ed.) 19930116
Title: Erythromycin and ketoconazole (Nizoral) associated with terfenadine (Seldane)-induced ventricular arrhythmias.
Journal: General dentistry 19930101
Title: Evidence for CYP3A-mediated N-deethylation of amiodarone in human liver microsomal fractions.
Journal: Drug metabolism and disposition: the biological fate of chemicals 19930101
Title: [Treatment with terfenadine and ketoconazole or itraconazole can cause torsades de pointes ventricular tachycardia].
Journal: Duodecim; laaketieteellinen aikakauskirja 19930101
Title: Drug-induced gynecomastia.
Journal: Pharmacotherapy 19930101
Title: Antifungal activity of meridine, a natural product from the marine sponge Corticium sp.
Journal: Journal of natural products 19921101
Title: Antibacterial and antifungal agents. XV. Synthesis and antifungal activity of structural analogues of bifonazole and ketoconazole.
Journal: Archiv der Pharmazie 19921101
Title: Stereoisomers of ketoconazole: preparation and biological activity.
Journal: Journal of medicinal chemistry 19920724
Title: Reduction of chromium(VI) to chromium(V) by rat liver cytosolic and microsomal fractions: is DT-diaphorase involved?
Journal: Carcinogenesis 19920701
Title: Torsades de Pointes after treatment with terfenadine and ketoconazole.
Journal: European heart journal 19920701
Title: Comparative study of six antifungal treatments in an experimental model of murine cryptococcosis.
Journal: European journal of epidemiology 19920501
Title: Uroporphyrinogen oxidation catalyzed by reconstituted cytochrome P450IA2.
Journal: Archives of biochemistry and biophysics 19920501
Title: In vitro activity of cloconazole, sulconazole, butoconazole, isoconazole, fenticonazole, and five other antifungal agents against clinical isolates of Candida albicans and Candida spp.
Journal: Mycopathologia 19920401
Title: The mechanism of bioactivation and antigen formation of amodiaquine in the rat.
Journal: Biochemical pharmacology 19920401
Title: Placebo-controlled clinical trial of sodium stibogluconate (Pentostam) versus ketoconazole for treating cutaneous leishmaniasis in Guatemala.
Journal: The Journal of infectious diseases 19920301
Title: Acute renal failure after liver transplantation in patients treated with cyclosporine.
Journal: Transplantation proceedings 19920201
Title: Ketoconazole and high-dose methylprednisolone predisposing to cyclosporine-induced seizures: report of 3 cases.
Journal: Acta haematologica 19920101
Title: Synthesis, specificity, and antifungal activity of inhibitors of the Candida albicans delta 24-sterol methyltransferase.
Journal: Journal of medicinal chemistry 19920101
Title: Myopathy associated with ketoconazole treatment.
Journal: American journal of diseases of children (1960) 19910901
Title: Ketoconazole-induced fulminant hepatitis necessitating liver transplantation.
Journal: Journal of the American Academy of Dermatology 19910801
Title: Drug induced suicidal ideation.
Journal: The Israel journal of psychiatry and related sciences 19910101
Title: Torsades de pointes occurring in association with terfenadine use.
Journal: JAMA 19901205
Title: Effects of pentamidine alone and in combination with ketoconazole or itraconazole on the growth of Candida albicans.
Journal: Antimicrobial agents and chemotherapy 19901201
Title: Massive hepatic enlargement with fatty change associated with ketoconazole.
Journal: DICP : the annals of pharmacotherapy 19901201
Title: Cyclosporine and itraconazole interaction in heart and lung transplant recipients.
Journal: Annals of internal medicine 19900815
Title: Efficacy of ketoconazole against Leishmania braziliensis panamensis cutaneous leishmaniasis.
Journal: The American journal of medicine 19900801
Title: Arterial hypertension as a complication of prolonged ketoconazole treatment.
Journal: Journal of hypertension. Supplement : official journal of the International Society of Hypertension 19891201
Title: Adverse psychiatric reaction to ketoconazole.
Journal: The American journal of psychiatry 19890701
Title: Neurologic complications of ketoconazole therapy for advanced prostatic cancer.
Journal: Urology 19890601
Title: [Toxic hepatitis caused by ketoconazole: a report of 4 cases].
Journal: Revista paulista de medicina 19890101
Title: Studies on antifungal agents. 23. Novel substituted 3,5-diphenyl-3-(1H-imidazol-1-ylmethyl)- 2-alkylisoxazolidine derivatives.
Journal: Journal of medicinal chemistry 19881001
Title: In-vivo effects of itraconazole on hepatic mixed-function oxidase.
Journal: The Journal of antimicrobial chemotherapy 19880201
Title: Prolonged jaundice following ketoconazole-induced hepatic injury.
Journal: Digestive diseases and sciences 19880201
Title: [Cholestatic hepatitis caused by ketoconazole].
Journal: Annales de gastroenterologie et d'hepatologie 19880101
Title: Itraconazole and cyclosporin nephrotoxicity.
Journal: Lancet (London, England) 19871017
Title: Hypertension during high-dose ketoconazole treatment: a probable mineralocorticosteroid effect.
Journal: Lancet (London, England) 19870912
Title: Antifungal activity of the allylamine derivative terbinafine in vitro.
Journal: Antimicrobial agents and chemotherapy 19870901
Title: Lysosomotropic agents. 7. Broad-spectrum antifungal activity of lysosomotropic detergents.
Journal: Journal of medicinal chemistry 19870801
Title: Synthesis and oral antifungal activity of novel azolylpropanolones and related compounds.
Journal: Journal of medicinal chemistry 19870601
Title: Immune hemolytic anemia associated with ketoconazole therapy.
Journal: Clinical pharmacy 19870601
Title: Hepatic reactions associated with ketoconazole in the United Kingdom.
Journal: British medical journal (Clinical research ed.) 19870214
Title: Ketoconazole-induced hepatitis: a case with a definite cause-effect relationship.
Journal: Liver 19870201
Title: [Hepatic lesions induced by drugs. Report of 26 cases].
Journal: Acta gastroenterologica Latinoamericana 19870101
Title: Activity of SM-4470, a new imidazole derivative, against experimental fungal infections.
Journal: Antimicrobial agents and chemotherapy 19860901
Title: In vitro activity of ketoconazole against herpes simplex virus.
Journal: Antimicrobial agents and chemotherapy 19860801
Title: Ketoconazole-associated hepatic injury. A clinicopathological study of 55 cases.
Journal: Journal of hepatology 19860101
Title: Experimental cyclosporine nephrotoxicity: risk of concomitant chemotherapy.
Journal: Clinical nephrology 19860101
Title: Ketoconazole-induced fulminant hepatitis.
Journal: Gut 19850601
Title: Activity of UK-49,858, a bis-triazole derivative, against experimental infections with Candida albicans and Trichophyton mentagrophytes.
Journal: Antimicrobial agents and chemotherapy 19850501
Title: Treatment of canine blastomycosis with amphotericin B and ketoconazole.
Journal: Journal of the American Veterinary Medical Association 19840515
Title: Hepatic injury associated with ketoconazole therapy. Analysis of 33 cases.
Journal: Gastroenterology 19840301
Title: Toxic hepatitis following ketoconazole treatment.
Journal: Scandinavian journal of infectious diseases 19840101
Title: [Ketoconazole-induced hepatitis. Case report].
Journal: Zeitschrift fur Gastroenterologie 19831201
Title: [Toxic hepatitis caused by ketoconazole].
Journal: Nederlands tijdschrift voor geneeskunde 19830618
Title: Synthesis of (E)-1-(5-chlorothien-2-yl)-2-(1H-imidazol-1-yl)ethanone 2,6-dichlorophenylhydrazone hydrochloride, a novel, orally active antifungal agent.
Journal: Journal of medicinal chemistry 19830301
Title: [Toxic hepatitis caused by ketoconazole (Nizoral)].
Journal: Nederlands tijdschrift voor geneeskunde 19830219
Title: 3',5'-cyclic adenosine monophosphate response element binding protein up-regulated cytochrome P450 lanosterol 14alpha-demethylase expression involved in follicle-stimulating hormone-induced mouse oocyte maturation.
Journal: Molecular endocrinology (Baltimore, Md.)