[1]Locationinpatent:experimentalpartSutherlin,DanielP.;Sampath,Deepak;Berry,Megan;Castanedo,Georgette;Chang,Zhigang;Chuckowree,Irina;Dotson,Jenna;Folkes,Adrian;Friedman,Lori;Goldsmith,Richard;Heffron,Tim;Lee,Leslie;Lesnick,John;Lewis,Cristina;Mathieu,Simon;Nonomiya,Jim;Olivero,Alan;Pang,Jodie;Prior,WeiWei;Salphati,Laurent;Sideris,Steve;Tian,Qingping;Tsui,Vickie;Wan,NanChi;Wang,Shumei;Wiesmann,Christian;Wong,Susan;Zhu,Bing-Yan[JournalofMedicinalChemistry,2010,vol.53,#3,p.1086-1097]
[1]Locationinpatent:experimentalpartSutherlin,DanielP.;Sampath,Deepak;Berry,Megan;Castanedo,Georgette;Chang,Zhigang;Chuckowree,Irina;Dotson,Jenna;Folkes,Adrian;Friedman,Lori;Goldsmith,Richard;Heffron,Tim;Lee,Leslie;Lesnick,John;Lewis,Cristina;Mathieu,Simon;Nonomiya,Jim;Olivero,Alan;Pang,Jodie;Prior,WeiWei;Salphati,Laurent;Sideris,Steve;Tian,Qingping;Tsui,Vickie;Wan,NanChi;Wang,Shumei;Wiesmann,Christian;Wong,Susan;Zhu,Bing-Yan[JournalofMedicinalChemistry,2010,vol.53,#3,p.1086-1097]
Title: Rational design of phosphoinositide 3-kinase α inhibitors that exhibit selectivity over the phosphoinositide 3-kinase β isoform.
Journal: Journal of medicinal chemistry 20111124
Title: Discovery of (thienopyrimidin-2-yl)aminopyrimidines as potent, selective, and orally available pan-PI3-kinase and dual pan-PI3-kinase/mTOR inhibitors for the treatment of cancer.
Journal: Journal of medicinal chemistry 20100211
Title: Sutherlin DP, et al. Discovery of (thienopyrimidin-2-yl)aminopyrimidines as potent, selective, and orally available pan-PI3-kinase and dual pan-PI3-kinase/mTOR inhibitors for the treatment of cancer. J Med Chem. 2010 Feb 11;53(3):1086-97.
