Title: Initial testing of the CENP-E inhibitor GSK923295A by the pediatric preclinical testing program.
Journal: Pediatric blood & cancer 20120601
Title: First-time-in-human study of GSK923295, a novel antimitotic inhibitor of centromere-associated protein E (CENP-E), in patients with refractory cancer.
Journal: Cancer chemotherapy and pharmacology 20120301
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Title: Mayes PA, et al. Mitogen-activated protein kinase (MEK/ERK) inhibition sensitizes cancer cells to centromere-associated protein E (CENP-E) inhibition. Int J Cancer. 2013 Feb 1;132(3):E149-57.
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