Title: Inhibitory effects of benzodiazepines on the adenosine A(2B) receptor mediated secretion of interleukin-8 in human mast cells.
Journal: European journal of pharmacology 20130130
Title: Design, synthesis and structure-activity relationships of novel benzoxazolone derivatives as 18 kDa translocator protein (TSPO) ligands.
Journal: Bioorganic & medicinal chemistry 20120915
Title: Synaptic and nonsynaptic mitochondria demonstrate a different degree of calcium-induced mitochondrial dysfunction.
Journal: Life sciences 20120522
Title: Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
Journal: Journal of medicinal chemistry 20120510
Title: The role of 18 kDa mitochondrial translocator protein (TSPO) in programmed cell death, and effects of steroids on TSPO expression.
Journal: Current molecular medicine 20120501
Title: Translocator protein (TSPO) in breast cancer.
Journal: Current molecular medicine 20120501
Title: LXR and TSPO as new therapeutic targets to increase the levels of neuroactive steroids in the central nervous system of diabetic animals.
Journal: Neurochemistry international 20120501
Title: Actions of translocator protein ligands on neutrophil adhesion and motility induced by G-protein coupled receptor signaling.
Journal: Biochemical and biophysical research communications 20120113
Title: The translocator protein (peripheral benzodiazepine receptor) mediates rat-selective activation of the mitochondrial permeability transition by norbormide.
Journal: Biochimica et biophysica acta 20111201
Title: Improvement of cerebral metabolism mediated by Ro5-4864 is associated with relief of intracranial pressure and mitochondrial protective effect in experimental brain injury.
Journal: Pharmaceutical research 20111101
Title: Dynamic modulation of Ca2+ sparks by mitochondrial oscillations in isolated guinea pig cardiomyocytes under oxidative stress.
Journal: Journal of molecular and cellular cardiology 20111101
Title: Biophysical properties and functional consequences of reactive oxygen species (ROS)-induced ROS release in intact myocardium.
Journal: The Journal of physiology 20111101
Title: Tertiary amides with a five-membered heteroaromatic ring as new probes for the translocator protein.
Journal: European journal of medicinal chemistry 20110901
Title: Erythrocyte peripheral type benzodiazepine receptor/voltage-dependent anion channels are upregulated by Plasmodium falciparum.
Journal: Blood 20110825
Title: Translocator protein (18 kDa)/peripheral benzodiazepine receptor specific ligands induce microglia functions consistent with an activated state.
Journal: Glia 20110201
Title: Evaluation of novel N1-methyl-2-phenylindol-3-ylglyoxylamides as a new chemotype of 18 kDa translocator protein-selective ligand suitable for the development of positron emission tomography radioligands.
Journal: Journal of medicinal chemistry 20110113
Title: 4'-chlorodiazepam--agonist of peripheral benzodiazepine receptors as a protecting factor in IL-1 induced deregulation of collagen biosynthesis in cultured human chondrocytes.
Journal: European journal of pharmacology 20101125
Title: Peripheral benzodiazepine receptor ligand Ro5-4864 inhibits isoprenaline-induced cardiac hypertrophy in rats.
Journal: European journal of pharmacology 20101010
Title: Overexpression of translocator protein in inflammatory bowel disease: potential diagnostic and treatment value.
Journal: Inflammatory bowel diseases 20100901
Title: Antiproliferative effect of peripheral benzodiazepine receptor antagonist PK11195 in rat mammary tumor cells.
Journal: Molecular and cellular biochemistry 20100701
Title: Novel irreversible fluorescent probes targeting the 18 kDa translocator protein: synthesis and biological characterization.
Journal: Journal of medicinal chemistry 20100527
Title: 4'-Chlorodiazepam, a translocator protein (18 kDa) antagonist, improves cardiac functional recovery during postischemia reperfusion in rats.
Journal: Experimental biology and medicine (Maywood, N.J.) 20100401
Title: Suppressive effect of diazepam on IFN-gamma production by human T cells.
Journal: International immunopharmacology 20100301
Title: Translocator protein (18 kDa) mediates the pro-growth effects of diazepam on Ehrlich tumor cells in vivo.
Journal: European journal of pharmacology 20100125
Title: Reversal of propoxur-induced impairment of memory and oxidative stress by 4'-chlorodiazepam in rats.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20100101
Title: Neuroprotective effects of a ligand of translocator protein-18 kDa (Ro5-4864) in experimental diabetic neuropathy.
Journal: Neuroscience 20091201
Title: Allosteric modulation by benzodiazepines of GABA-gated chloride channels of an identified insect motor neurone.
Journal: Invertebrate neuroscience : IN 20091101
Title: Spinal translocator protein (TSPO) modulates pain behavior in rats with CFA-induced monoarthritis.
Journal: Brain research 20090825
Title: The translocator protein (18 kDa): central nervous system disease and drug design.
Journal: Journal of medicinal chemistry 20090212
Title: Neuroprotective effect of Ro5-4864 following brain injury.
Journal: Experimental neurology 20081201
Title: Effects of Vinpocetine on mitochondrial function and neuroprotection in primary cortical neurons.
Journal: Neurochemistry international 20081201
Title: Anxiolytic-like effects of N,N-dialkyl-2-phenylindol-3-ylglyoxylamides by modulation of translocator protein promoting neurosteroid biosynthesis.
Journal: Journal of medicinal chemistry 20080925
Title: Effects of 4'-chlorodiazepam on cellular excitation-contraction coupling and ischaemia-reperfusion injury in rabbit heart.
Journal: Cardiovascular research 20080701
Title: Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor.
Journal: Bioorganic & medicinal chemistry 20080601
Title: Control of peripheral benzodiazepine receptor-mediated breast cancer in rats by soy protein.
Journal: Molecular carcinogenesis 20080401
Title: Ro5-4864 promotes neonatal motor neuron survival and nerve regeneration in adult rats.
Journal: The European journal of neuroscience 20080201
Title: Steroidogenesis in BeWo cells: role of protein kinase A and benzodiazepines.
Journal: The international journal of biochemistry & cell biology 20080101
Title: Ligands of the mitochondrial 18 kDa translocator protein attenuate apoptosis of human glioblastoma cells exposed to erucylphosphohomocholine.
Journal: Cellular oncology : the official journal of the International Society for Cellular Oncology 20080101
Title: The scale-free dynamics of eukaryotic cells.
Journal: PloS one 20080101
Title: The potential anticancer agent PK11195 induces apoptosis irrespective of p53 and ATM status in chronic lymphocytic leukemia cells.
Journal: Haematologica 20071201
Title: Peripheral benzodiazepine receptor-induced myocardial protection is mediated by inhibition of mitochondrial membrane permeabilization.
Journal: The Journal of pharmacology and experimental therapeutics 20071001
Title: Intracellular cholesterol changes induced by translocator protein (18 kDa) TSPO/PBR ligands.
Journal: Neuropharmacology 20070801
Title: Sequential opening of mitochondrial ion channels as a function of glutathione redox thiol status.
Journal: The Journal of biological chemistry 20070727
Title: The peripheral-type benzodiazepine receptor is involved in control of Ca2+-induced permeability transition pore opening in rat brain mitochondria.
Journal: Cell calcium 20070701
Title: Characterization of two classes of benzodiazepine binding sites in Schistosoma mansoni.
Journal: Parasitology 20070701
Title: Novel 1,4-benzodiazepine derivatives with antiproliferative properties on tumor cell lines.
Journal: Bioorganic & medicinal chemistry letters 20070501
Title: Inhibition of the mitochondrial F1F0-ATPase by ligands of the peripheral benzodiazepine receptor.
Journal: Bioorganic & medicinal chemistry letters 20070315
Title: [Peripheral benzodiazepine receptor agonist Ro5-4864 inhibits mitochondrial permeability transition in rat heart].
Journal: Sheng li xue bao : [Acta physiologica Sinica] 20070225
Title: New fluorescent 2-phenylindolglyoxylamide derivatives as probes targeting the peripheral-type benzodiazepine receptor: design, synthesis, and biological evaluation.
Journal: Journal of medicinal chemistry 20070125
Title: A novel conjugable translocator protein ligand labeled with a fluorescence dye for in vitro imaging.
Journal: Bioconjugate chemistry 20070101
Title: Channel-like functions of the 18-kDa translocator protein (TSPO): regulation of apoptosis and steroidogenesis as part of the host-defense response.
Journal: Current pharmaceutical design 20070101
Title: Effects of peripheral-type benzodiazepine receptor ligands on Ehrlich tumor cell proliferation.
Journal: European journal of pharmacology 20061121
Title: Discovery of antiglioma activity of biaryl 1,2,3,4-tetrahydroisoquinoline derivatives and conformationally flexible analogues.
Journal: Journal of medicinal chemistry 20060921
Title: The peripheral-type benzodiazepine receptor and the cardiovascular system. Implications for drug development.
Journal: Pharmacology & therapeutics 20060601
Title: 5-aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors.
Journal: Die Pharmazie 20060601
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Increased expression of peripheral benzodiazepine receptor (PBR) in dimethylbenz[a]anthracene-induced mammary tumors in rats.
Journal: Glycoconjugate journal 20060501
Title: Implication of glucocorticoid in anti-inflammatory effects of Ro5-4864 in mouse pleurisy induced by carrageenan.
Journal: Life sciences 20060313
Title: Peripheral benzodiazepine receptor: characterization in human T-lymphoma Jurkat cells.
Journal: Molecular pharmacology 20060101
Title: PK11195 potently sensitizes to apoptosis induction independently from the peripheral benzodiazepin receptor.
Journal: Oncogene 20051117
Title: Ro5-4864, a synthetic ligand of peripheral benzodiazepine receptor, reduces aging-associated myelin degeneration in the sciatic nerve of male rats.
Journal: Mechanisms of ageing and development 20051101
Title: Role of the peripheral benzodiazepine receptor in sensory neuron regeneration.
Journal: Molecular and cellular neurosciences 20051001
Title: Modulation of cholinephosphotransferase activity in breast cancer cell lines by Ro5-4864, a peripheral benzodiazepine receptor agonist.
Journal: Biochemical and biophysical research communications 20050722
Title: Ro5-4864, a peripheral benzodiazepine receptor ligand, reduces reactive gliosis and protects hippocampal hilar neurons from kainic acid excitotoxicity.
Journal: Journal of neuroscience research 20050401
Title: Peripheral benzodiazepine receptor (PBR) ligand cytotoxicity unrelated to PBR expression.
Journal: Biochemical pharmacology 20050301
Title: Benzodiazepine receptor-dependent modulation of neutrophil (PMN) free amino- and alpha-keto acid profiles or immune functions.
Journal: Amino acids 20050201
Title: Evidence in favour of a role for peripheral-type benzodiazepine receptor ligands in amplification of neuronal apoptosis.
Journal: Apoptosis : an international journal on programmed cell death 20050101
Title: Nootropic nefiracetam inhibits proconvulsant action of peripheral-type benzodiazepines in epileptic mutant EL mice.
Journal: Annals of the New York Academy of Sciences 20041001
Title: Monitoring drug-induced neurodegeneration by imaging of peripheral benzodiazepine receptors.
Journal: Annals of the New York Academy of Sciences 20041001
Title: Peripheral type benzodiazepine receptor in human parathyroid glands: up-regulation in adenoma.
Journal: Journal of endocrinological investigation 20041001
Title: The role of peripheral benzodiazepine receptors on the function and survival of isolated human pancreatic islets.
Journal: European journal of endocrinology 20040801
Title: Peripheral benzodiazepine receptor ligands: mitochondrial transmembrane potential depolarization and apoptosis induction in rat C6 glioma cells.
Journal: Biochemical pharmacology 20040701
Title: Functional characterization and expression of PBR in rat gastric mucosa: stimulation of chloride secretion by PBR ligands.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20040601
Title: Antinociceptive effects of peripheral benzodiazepine receptors.
Journal: Pharmacology 20040401
Title: N,N-dialkyl-2-phenylindol-3-ylglyoxylamides. A new class of potent and selective ligands at the peripheral benzodiazepine receptor.
Journal: Journal of medicinal chemistry 20040325
Title: Involvement of steroids in anti-inflammatory effects of peripheral benzodiazepine receptor ligands.
Journal: Life sciences 20040130
Title: Peripheral benzodiazepine receptors in potatoes (Solanum tuberosum).
Journal: Biochemical and biophysical research communications 20040102
Title: Effects of peripheral benzodiazepine receptor ligands on proliferation and differentiation of human mesenchymal stem cells.
Journal: Journal of cellular physiology 20040101
Title: Benzodiazepine binding to mitochondrial membranes of the amoeba Acanthamoeba castellanii and the yeast Saccharomyces cerevisiae.
Journal: Acta biochimica Polonica 20040101
Title: Effects of acute and long-term diazepam administrations on neutrophil activity: a flow cytometric study.
Journal: European journal of pharmacology 20031008
Title: Structure activity studies of a novel cytotoxic benzodiazepine.
Journal: Bioorganic & medicinal chemistry letters 20031006
Title: Ligands of the peripheral benzodiazepine receptor have therapeutic effects in pneumopathies in vivo.
Journal: Immunology letters 20030908
Title: Anticholinergic and antiglutamatergic agents protect against soman-induced brain damage and cognitive dysfunction.
Journal: Toxicological sciences : an official journal of the Society of Toxicology 20030901
Title: Antidepressant-like effect of Ro5-4864, a peripheral-type benzodiazepine receptor ligand, in forced swimming test.
Journal: European journal of pharmacology 20030613
Title: Comparison of two PBR ligands with classical antiinflammatory drugs in LPS-induced arthritis in rats.
Journal: Life sciences 20030425
Title: Benzodiazepine-induced protein tyrosine nitration in rat astrocytes.
Journal: Hepatology (Baltimore, Md.) 20030201
Title: Peripheral benzodiazepine receptors: on mice and human brain imaging.
Journal: Journal of neurochemistry 20030201
Title: Mitochondrial benzodiazepine receptors regulate oxygen homeostasis in the early mouse embryo.
Journal: Reproductive toxicology (Elmsford, N.Y.) 20030101
Title: Effects on free radical generation by ligands of the peripheral benzodiazepine receptor in cultured neural cells.
Journal: Journal of neurochemistry 20021201
Title: Identification of a peptide antagonist to the peripheral-type benzodiazepine receptor that inhibits hormone-stimulated leydig cell steroid formation.
Journal: The Journal of pharmacology and experimental therapeutics 20021101
Title: Involvement of the peripheral benzodiazepine receptor in the development of rheumatoid arthritis in Mrl/lpr mice.
Journal: European journal of pharmacology 20020927
Title: Modulation of tamoxifen-induced apoptosis by peripheral benzodiazepine receptor ligands in breast cancer cells.
Journal: Biochemical pharmacology 20020701
Title: Platelet-activating factor induces permeability transition and cytochrome c release in isolated brain mitochondria.
Journal: Journal of neuroscience research 20020701
Title: Peripheral benzodiazepine receptor ligands reverse apoptosis resistance of cancer cells in vitro and in vivo.
Journal: Cancer research 20020301
Title: Binding and neuropharmacological profile of zaleplon, a novel nonbenzodiazepine sedative/hypnotic.
Journal: European journal of pharmacology 20020102
Title: Peripheral benzodiazepine binding sites/receptors (PBRs) have been localized to rat central and peripheral endocrine tissues.
Journal: Journal of andrology 20020101
Title: Binding of [3H]CB 34, a selective ligand for peripheral benzodiazepine receptors, to rat brain membranes.
Journal: European journal of pharmacology 20011207
Title: Specific ligands of the peripheral benzodiazepine receptor induce apoptosis and cell cycle arrest in human colorectal cancer cells.
Journal: British journal of cancer 20011101
Title: Nutritional parameters modify muricidal behavior of male Wistar rats: preventive effects of amino acids and 4' Cl diazepam.
Journal: Life sciences 20011026
Title: 2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands.
Journal: Bioorganic & medicinal chemistry 20011001
Title: Diazepam inhibits HIV-1 Tat-induced migration of human microglia.
Journal: Journal of neurovirology 20011001
Title: Effect of midazolam on interleukin-6 mRNA expression in human peripheral blood mononuclear cells in the absence of lipopolysaccharide.
Journal: Cytokine 20010921
Title: Structural and functional study of reconstituted peripheral benzodiazepine receptor.
Journal: Biochemical and biophysical research communications 20010608
Title: Inverse agonist binding of peripheral benzodiazepine receptors in anxiety disorder.
Journal: European archives of psychiatry and clinical neuroscience 20010601
Title: Reduction of acute inflammation in rats by diazepam: role of peripheral benzodiazepine receptors and corticosterone.
Journal: Immunopharmacology and immunotoxicology 20010501
Title: Expression of the peripheral-type benzodiazepine receptor and apoptosis induction in hepatic stellate cells.
Journal: Gastroenterology 20010401
Title: Peripheral-type benzodiazepine receptor ligands: mitochondrial permeability transition induction in rat cardiac tissue.
Journal: Biochemical pharmacology 20010315
Title: The influence of the antidepressant pirlindole and its dehydro-derivative on the activity of monoamine oxidase A and GABAA receptor binding.
Journal: Journal of neural transmission. Supplementum 19980101
Title: Diazepam-mediated inhibition of human immunodeficiency virus type 1 expression in human brain cells.
Journal: Antimicrobial agents and chemotherapy 19971101
Title: Mitochondrial diazepam-binding inhibitor receptor complex agonists antagonize dizocilpine amnesia: putative role for allopregnanolone.
Journal: The Journal of pharmacology and experimental therapeutics 19940701
Title: Anticonvulsant activity of delta-HCH, calcium channel blockers and calmodulin antagonists in seizures induced by lindane and other convulsant drugs.
Journal: Brain research 19930917
Title: Toxicokinetics of Ro 5-4864, lindane and picrotoxin compared.
Journal: Pharmacology, biochemistry, and behavior 19910201
Title: Isolation and characterization of a rat brain triakontatetraneuropeptide, a posttranslational product of diazepam binding inhibitor: specific action at the Ro 5-4864 recognition site.
Journal: Journal of neurochemistry 19891001
Title: 'Central' and 'peripheral' benzodiazepines and kinetics of lindane-induced toxicity.
Journal: Pharmacology, biochemistry, and behavior 19890201
Title: Coincidence of seizure susceptibility to caffeine and to the benzodiazepine inverse agonist, DMCM, in SWR and CBA inbred mice.
Journal: Pharmacology, biochemistry, and behavior 19870201
