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Title: Dual fluorescent HPMA copolymers for passive tumor targeting with pH-sensitive drug release: synthesis and characterization of distribution and tumor accumulation in mice by noninvasive multispectral optical imaging.
Journal: Biomacromolecules 20120312
Title: Biological activity of anti-CD20 multivalent HPMA copolymer-Fab' conjugates.
Journal: Biomacromolecules 20120312
Title: Treatment of prostate carcinoma with (galectin-3)-targeted HPMA copolymer-(G3-C12)-5-Fluorouracil conjugates.
Journal: Biomaterials 20120301
Title: Multifunctional pH-disintegrable micellar nanoparticles of asymmetrically functionalized β-cyclodextrin-based star copolymer covalently conjugated with doxorubicin and DOTA-Gd moieties.
Journal: Biomaterials 20120301
Title: Synthesis and in vitro anti-tumor activity of novel HPMA copolymer-drug conjugates with potential cell surface targeting property for carcinoma cells.
Journal: European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V 20120201
Title: Selective inhibitory effect of HPMA copolymer-cyclopamine conjugate on prostate cancer stem cells.
Journal: Biomaterials 20120201
Title: Enhancing the therapeutic efficacy of adenovirus in combination with biomaterials.
Journal: Biomaterials 20120201
Title: Synthesis and characterization of biodegradable and thermosensitive polymeric micelles with covalently bound doxorubicin-glucuronide prodrug via click chemistry.
Journal: Bioconjugate chemistry 20111221
Title: Biodegradable star HPMA polymer-drug conjugates: Biodegradability, distribution and anti-tumor efficacy.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20110925
Title: Conformational consequences of cooperative binding of a coiled-coil peptide motif to poly(N-(2-hydroxypropyl) methacrylamide) HPMA copolymers.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20110730
Title: Modifying the body distribution of HPMA-based copolymers by molecular weight and aggregate formation.
Journal: Biomacromolecules 20110711
Title: HPMA based amphiphilic copolymers mediate central nervous effects of domperidone.
Journal: Macromolecular rapid communications 20110518
Title: Effect of film thickness on the antifouling performance of poly(hydroxy-functional methacrylates) grafted surfaces.
Journal: Langmuir : the ACS journal of surfaces and colloids 20110419
Title: Biodegradable star HPMA polymer conjugates of doxorubicin for passive tumor targeting.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20110418
Title: Coupling to polymeric scaffolds stabilizes biofunctional peptides for intracellular applications.
Journal: Molecular pharmacology 20110401
Title: Light induced drug delivery into cancer cells.
Journal: Biomaterials 20110201
Title: Comparative biodistribution of PAMAM dendrimers and HPMA copolymers in ovarian-tumor-bearing mice.
Journal: Biomacromolecules 20110110
Title: Immobilization of chloroperoxidase onto highly hydrophilic polyethylene chains via bio-conjugation: catalytic properties and stabilities.
Journal: Bioresource technology 20110101
Title: Sphingosine-1-phosphate promotes the differentiation of human umbilical cord mesenchymal stem cells into cardiomyocytes under the designated culturing conditions.
Journal: Journal of biomedical science 20110101
Title: Achieving highly effective nonfouling performance for surface-grafted poly(HPMA) via atom-transfer radical polymerization.
Journal: Langmuir : the ACS journal of surfaces and colloids 20101116
Title: HPMA-RGD hydrogels seeded with mesenchymal stem cells improve functional outcome in chronic spinal cord injury.
Journal: Stem cells and development 20101001
Title: Synthesis and in vitro evaluation of defined HPMA folate conjugates: influence of aggregation on folate receptor (FR) mediated cellular uptake.
Journal: Biomacromolecules 20100913
Title: HPMA copolymer conjugates of paclitaxel and docetaxel with pH-controlled drug release.
Journal: Molecular pharmaceutics 20100802
Title: Synthesis, characterization and enhanced photoconductivity from a mesoporous titania on dye doping.
Journal: Analytica chimica acta 20100726
Title: Functional diversification of AGAMOUS lineage genes in regulating tomato flower and fruit development.
Journal: Journal of experimental botany 20100601
Title: Langmuir-Blodgett films of biocompatible poly(HPMA)-block-poly(lauryl methacrylate) and poly(HPMA)-random-poly(lauryl methacrylate): influence of polymer structure on membrane formation and stability.
Journal: Langmuir : the ACS journal of surfaces and colloids 20100420
Title: Water-soluble polymer-drug conjugates for combination chemotherapy against visceral leishmaniasis.
Journal: Bioorganic & medicinal chemistry 20100401
Title: Chemical conjugation of cowpea mosaic viruses with reactive HPMA-based polymers.
Journal: Journal of biomaterials science. Polymer edition 20100101
Title: Development of a macromolecular prodrug for the treatment of inflammatory arthritis: mechanisms involved in arthrotropism and sustained therapeutic efficacy.
Journal: Arthritis research & therapy 20100101
Title: HPMA copolymer conjugates with reduced anti-CD20 antibody for cell-specific drug targeting. I. Synthesis and in vitro evaluation of binding efficacy and cytostatic activity.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20091116
Title: Hyperbranched polyamidoamines containing beta-cyclodextrin for controlled release of chlorambucil.
Journal: Macromolecular bioscience 20091110
Title: Antitumor efficacy of colon-specific HPMA copolymer/9-aminocamptothecin conjugates in mice bearing human-colon carcinoma xenografts.
Journal: Macromolecular bioscience 20091110
Title: Synthesis and bioactivity of poly(HPMA)-lysozyme conjugates: the use of novel thiazolidine-2-thione coupling chemistry.
Journal: Organic & biomolecular chemistry 20090907
Title: Nortriptyline for smoking cessation: release and human skin diffusion from patches.
Journal: International journal of pharmaceutics 20090813
Title: Evaluation of pharmacokinetics of bioreducible gene delivery vectors by real-time PCR.
Journal: Pharmaceutical research 20090701
Title: HPMA-based polymer conjugates with drug combination.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20090628
Title: N-(2-hydroxypropyl)methacrylamide-amphotericin B (HPMA-AmB) copolymer conjugates as antileishmanial agents.
Journal: International journal of antimicrobial agents 20090501
Title: Cetuximab retargeting of adenovirus via the epidermal growth factor receptor for treatment of intraperitoneal ovarian cancer.
Journal: Human gene therapy 20090301
Title: Self-assembling diblock copolymers of poly[N-(2-hydroxypropyl)methacrylamide] and a beta-sheet peptide.
Journal: Macromolecular bioscience 20090109
Title: Biorecognition and subcellular trafficking of HPMA copolymer-anti-PSMA antibody conjugates by prostate cancer cells.
Journal: Molecular pharmaceutics 20090101
Title: Synthesis and evaluation of a well-defined HPMA copolymer-dexamethasone conjugate for effective treatment of rheumatoid arthritis.
Journal: Pharmaceutical research 20081201
Title: Feasibility of using a bone-targeted, macromolecular delivery system coupled with prostaglandin E(1) to promote bone formation in aged, estrogen-deficient rats.
Journal: Pharmaceutical research 20081201
Title: One-pot conversion of RAFT-generated multifunctional block copolymers of HPMA to doxorubicin conjugated acid- and reductant-sensitive crosslinked micelles.
Journal: Biomacromolecules 20081101
Title: From defined reactive diblock copolymers to functional HPMA-based self-assembled nanoaggregates.
Journal: Biomacromolecules 20081101
Title: HPMA copolymer-doxorubicin-gadolinium conjugates: synthesis, characterization, and in vitro evaluation.
Journal: Macromolecular bioscience 20080811
Title: Synthesis and biological evaluation of disulfide-linked HPMA copolymer-mesochlorin e6 conjugates.
Journal: Macromolecular bioscience 20080513
Title: New HPMA copolymer-based drug carriers with covalently bound hydrophobic substituents for solid tumour targeting.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20080421
Title: Doxorubicin release is not a prerequisite for the in vitro cytotoxicity of HPMA-based pharmaceuticals: in vitro effect of extra drug-free GlyPheLeuGly sequences.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20080421
Title: Enhanced antitumor activity of combinations of free and HPMA copolymer-bound drugs.
Journal: International journal of pharmaceutics 20080303
Title: Dynamic light scattering study of self-assembly of HPMA hybrid graft copolymers.
Journal: Biomacromolecules 20080201
Title: Pharmacokinetic modeling of absorption behavior of 9-aminocamptothecin (9-AC) released from colon-specific HPMA copolymer-9-AC conjugate in rats.
Journal: Pharmaceutical research 20080101
Title: Biodegradable, cationic methacrylamide-based polymers for gene delivery to ovarian cancer cells in mice.
Journal: Molecular pharmaceutics 20080101
Title: Campylobacter jejuni survives within epithelial cells by avoiding delivery to lysosomes.
Journal: PLoS pathogens 20080101
Title: Stability in plasmas of various species of HPMA copolymer-PGE1 conjugates.
Journal: Pharmaceutical research 20071201
Title: [Pilot study of a cell membrane like biomimetic drug-eluting coronary stent].
Journal: Sheng wu yi xue gong cheng xue za zhi = Journal of biomedical engineering = Shengwu yixue gongchengxue zazhi 20070601
Title: Effect of radiotherapy and hyperthermia on the tumor accumulation of HPMA copolymer-based drug delivery systems.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20070226
Title: Biodistribution and pharmacokinetics of colon-specific HPMA copolymer--9-aminocamptothecin conjugate in mice.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20070212
Title: Designing polymer conjugates as lysosomotropic nanomedicines.
Journal: Biochemical Society transactions 20070201
Title: Novel dexamethasone-HPMA copolymer conjugate and its potential application in treatment of rheumatoid arthritis.
Journal: Arthritis research & therapy 20070101
Title: Affinity separation of immunoglobulin G subclasses on dye attached poly(hydroxypropyl methacrylate) beads.
Journal: International journal of biological macromolecules 20061115
Title: Properties of HPMA copolymer-doxorubicin conjugates with pH-controlled activation: effect of polymer chain modification.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20060928
Title: Polymeric conjugates of mono- and bi-cyclic alphaVbeta3 binding peptides for tumor targeting.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20060828
Title: Enhancement of ethyl propionate synthesis by poly (AAc-co-HPMA-cl-MBAm)-immobilized Pseudomonas aeruginosa MTCC-4713, exposed to Hg2+ and NH4+ ions.
Journal: Acta microbiologica et immunologica Hungarica 20060601
Title: Hybrid hydrogels self-assembled from HPMA copolymers containing peptide grafts.
Journal: Macromolecular bioscience 20060314
Title: Colon-specific 9-aminocamptothecin-HPMA copolymer conjugates containing a 1,6-elimination spacer.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20060110
Title: Polymer-peptide conjugates for angiogenesis targeted tumor radiotherapy.
Journal: Nuclear medicine and biology 20060101
Title: Macrophage targeted N-(2-hydroxypropyl)methacrylamide conjugates for magnetic resonance imaging.
Journal: Molecular pharmaceutics 20060101
Title: Effect of physicochemical modification on the biodistribution and tumor accumulation of HPMA copolymers.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20051210
Title: Ultrasound-enhanced transfection activity of HPMA-stabilized DNA polyplexes with prolonged plasma circulation.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20050902
Title: Targeting tumor angiogenesis: comparison of peptide and polymer-peptide conjugates.
Journal: Journal of nuclear medicine : official publication, Society of Nuclear Medicine 20050901
Title: Induction of systemic antitumour resistance with targeted polymers.
Journal: Scandinavian journal of immunology 20050701
Title: Polymer therapeutics designed for a combination therapy of hormone-dependent cancer.
Journal: Angewandte Chemie (International ed. in English) 20050627
Title: Water-soluble polymers for targeted drug delivery to human squamous carcinoma of head and neck.
Journal: Journal of drug targeting 20050401
Title: Intracellular targeting of polymer-bound drugs for cancer chemotherapy.
Journal: Advanced drug delivery reviews 20050227
Title: Improved preservation of X-gal reaction product for electron microscopy using hydroxypropyl methacrylate.
Journal: Neuroscience letters 20050201
Title: Oligopeptides as targeting structures in cancer theraPY.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20050103
Title: Final report of the safety assessment of methacrylate ester monomers used in nail enhancement products.
Journal: International journal of toxicology 20050101
Title: Vitamin-mediated targeting as a potential mechanism to increase drug uptake by tumours.
Journal: Journal of inorganic biochemistry 20041001
Title: The arthrotropism of macromolecules in adjuvant-induced arthritis rat model: a preliminary study.
Journal: Pharmaceutical research 20041001
Title: Aggregation properties of a HPMA-camptothecin copolymer in isotonic solutions.
Journal: Biophysical chemistry 20040801
Title: The effect of the processing and formulation parameters on the size of nanoparticles based on block copolymers of poly(ethylene glycol) and poly(N-isopropylacrylamide) with and without hydrolytically sensitive groups.
Journal: Biomaterials 20040501
Title: Targeting angiogenesis with a conjugate of HPMA copolymer and TNP-470.
Journal: Nature medicine 20040301
Title: Polymer-conjugated bovine pancreatic and seminal ribonucleases inhibit growth of human tumors in nude mice.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20040220
Title: Polymer therapeutics - Sixth International Symposium: from laboratory to clinical practice.
Journal: IDrugs : the investigational drugs journal 20040201
Title: A novel crosslinkable polymer as drug-loaded coating for biomedical device.
Journal: Journal of materials science. Materials in medicine 20040201
Title: Prevention of gliotic scar formation by NeuroGel allows partial endogenous repair of transected cat spinal cord.
Journal: Journal of neuroscience research 20040115
Title: HPMA copolymer-1,5-diazaanthraquinone conjugates as novel anticancer therapeutics.
Journal: Journal of drug targeting 20040101
Title: Starlike vs. classic macromolecular prodrugs: two different antibody-targeted HPMA copolymers of doxorubicin studied in vitro and in vivo as potential anticancer drugs.
Journal: Pharmaceutical research 20031001
Title: [Synthesis and characterization of biomacromolecular conjugates for magnetic resonance imaging].
Journal: Sheng wu yi xue gong cheng xue za zhi = Journal of biomedical engineering = Shengwu yixue gongchengxue zazhi 20030901
Title: Cytostatic and immunomobilizing activities of polymer-bound drugs: experimental and first clinical data.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20030828
Title: Subcellular trafficking of HPMA copolymer-Tat conjugates in human ovarian carcinoma cells.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20030828
Title: Mechanisms of cytotoxicity in human ovarian carcinoma cells exposed to free Mce6 or HPMA copolymer-Mce6 conjugates.
Journal: Photochemistry and photobiology 20030601
Title: Correlation of subcellular compartmentalization of HPMA copolymer-Mce6 conjugates with chemotherapeutic activity in human ovarian carcinoma cells.
Journal: Pharmaceutical research 20030501
Title: HPMA copolymers with pH-controlled release of doxorubicin: in vitro cytotoxicity and in vivo antitumor activity.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20030221
Title: Tat-conjugated synthetic macromolecules facilitate cytoplasmic drug delivery to human ovarian carcinoma cells.
Journal: Bioconjugate chemistry 20030101
Title: HPMA copolymer delivery of chemotherapy and photodynamic therapy in ovarian cancer.
Journal: Advances in experimental medicine and biology 20030101
Title: PDEPT: polymer-directed enzyme prodrug therapy. 2. HPMA copolymer-beta-lactamase and HPMA copolymer-C-Dox as a model combination.
Journal: Bioconjugate chemistry 20030101
Title: Polyacetal-doxorubicin conjugates designed for pH-dependent degradation.
Journal: Bioconjugate chemistry 20030101
Title: HPMA copolymers platinates containing dicarboxylato ligands. Preparation, characterisation and in vitro and in vivo evaluation.
Journal: Journal of drug targeting 20021101
Title: Synthesis of hydroxypropyl methacrylate/polysaccharide graft copolymers as matrices for controlled release tablets.
Journal: Drug development and industrial pharmacy 20021001
Title: Immunomodulating activities of soluble synthetic polymer-bound drugs.
Journal: Advanced drug delivery reviews 20020913
Title: Synthesis and characterization of a catalytic antibody-HPMA copolymer-Conjugate as a tool for tumor selective prodrug activation.
Journal: Bioorganic & medicinal chemistry 20020901
Title: The role of galactose, lactose, and galactose valency in the biorecognition of N-(2-hydroxypropyl)methacrylamide copolymers by human colon adenocarcinoma cells.
Journal: Pharmaceutical research 20020801
Title: HPMA-hydrogels containing cytostatic drugs. Kinetics of the drug release and in vivo efficacy.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20020517
Title: Targeted delivery of doxorubicin by HPMA copolymer-hyaluronan bioconjugates.
Journal: Pharmaceutical research 20020401
Title: In vitro and in vivo effect of HPMA copolymer-bound doxorubicin targeted to transferrin receptor of B-cell lymphoma 38C13.
Journal: Journal of drug targeting 20020201
Title: Acquired and specific immunological mechanisms co-responsible for efficacy of polymer-bound drugs.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20020117
Title: Design of novel bioconjugates for targeted drug delivery.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20020117
Title: Star structure of antibody-targeted HPMA copolymer-bound doxorubicin: a novel type of polymeric conjugate for targeted drug delivery with potent antitumor effect.
Journal: Bioconjugate chemistry 20020101
Title: Antisense oligonucleotides delivered to the lysosome escape and actively inhibit the hepatitis B virus.
Journal: Bioconjugate chemistry 20020101
Title: Use of hydrophilic hydroxypropyl methacrylate/ethylene glycol methacrylate packing material in size-exclusion chromatography.
Journal: Journal of AOAC International 20020101
Title: N-(2-hydroxypropyl)methacrylamide (HPMA) copolymers for targeted delivery of 8-aminoquinoline antileishmanial drugs.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20011213
Title: Biorecognizable HPMA copolymer-drug conjugates for colon-specific delivery of 9-aminocamptothecin.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010810
Title: Polymer-drug conjugates, PDEPT and PELT: basic principles for design and transfer from the laboratory to clinic.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: Synthesis and characterization of HPMA copolymer-aminopropylgeldanamycin conjugates.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: Doxorubicin bound to a HPMA copolymer carrier through hydrazone bond is effective also in a cancer cell line with a limited content of lysosomes.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: Combination chemotherapy and photodynamic therapy of targetable N-(2-hydroxypropyl)methacrylamide copolymer-doxorubicin/mesochlorin e(6)-OV-TL 16 antibody immunoconjugates.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: Preparation and biological evaluation of polymerizable antibody Fab' fragment targeted polymeric drug delivery system.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: The effects of subcellular localization of N-(2-hydroxypropyl)methacrylamide copolymer-Mce(6) conjugates in a human ovarian carcinoma.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: Water-soluble HPMA copolymer-wortmannin conjugate retains phosphoinositide 3-kinase inhibitory activity in vitro and in vivo.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: Potential of lectin-N-(2-hydroxypropyl)methacrylamide copolymer-drug conjugates for the treatment of pre-cancerous conditions.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010706
Title: New HPMA copolymers containing doxorubicin bound via pH-sensitive linkage: synthesis and preliminary in vitro and in vivo biological properties.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010518
Title: Preliminary evaluation of caspases-dependent apoptosis signaling pathways of free and HPMA copolymer-bound doxorubicin in human ovarian carcinoma cells.
Journal: Journal of controlled release : official journal of the Controlled Release Society 20010428
Title: Phase I clinical and pharmacokinetic study of PNU166945, a novel water-soluble polymer-conjugated prodrug of paclitaxel.
Journal: Anti-cancer drugs 20010401
Title: The influence of a colonic microbiota on HPMA copolymer lectin conjugates binding in rodent intestine.
Journal: Journal of drug targeting 20010401
Title: Polymer-coated adenovirus permits efficient retargeting and evades neutralising antibodies.
Journal: Gene therapy 20010301
Title: [Study of 'living' radical polymerization by FTIR in situ].
Journal: Guang pu xue yu guang pu fen xi = Guang pu 20010201
Title: The effect of two hydrophilic monomers on the water uptake of a heterocyclic methacrylate system.
Journal: Biomaterials 20010101
Title: Crosslinkable coatings from phosphorylcholine-based polymers.
Journal: Biomaterials 20010101
Title: Modification of cyclosporin A and conjugation of its derivative to HPMA copolymers.
Journal: Bioconjugate chemistry 20010101
Title: Synthetic macromolecular drug carriers: biodistribution of poly[(N-2-hydroxypropyl)methacrylamide] copolymers and their accumulation in solid rat tumors.
Journal: PDA journal of pharmaceutical science and technology 20010101
Title: N-(2-hydroxypropyl)methacrylamide copolymer-6-(3-aminopropyl)-ellipticine conjugates. Synthesis, in vitro, and preliminary in vivo evaluation.
Journal: Bioconjugate chemistry 20010101
Title: Enhanced biorecognition and internalization of HPMA copolymers containing multiple or multivalent carbohydrate side-chains by human hepatocarcinoma cells.
Journal: Bioconjugate chemistry 20010101