Title: Effects of single swim stress on changes in TRPV1-mediated plasticity in the amygdala.
Journal: Behavioural brain research 20130101
Title: Functional interactions between NMDA receptors and TRPV1 in trigeminal sensory neurons mediate mechanical hyperalgesia in the rat masseter muscle.
Journal: Pain 20120701
Title: Structure-activity relationships of vanilloid receptor agonists for arteriolar TRPV1.
Journal: British journal of pharmacology 20120301
Title: Resolving TRPV1- and TNF-α-mediated spinal cord synaptic plasticity and inflammatory pain with neuroprotectin D1.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20111019
Title: The antinociceptive potency of N-arachidonoyl-dopamine (NADA) and its interaction with endomorphin-1 at the spinal level.
Journal: Pharmacology, biochemistry, and behavior 20111001
Title: Role of TRPV1 in nociception and edema induced by monosodium urate crystals in rats.
Journal: Pain 20110801
Title: TRPM3 is a nociceptor channel involved in the detection of noxious heat.
Journal: Neuron 20110512
Title: TRPV1-antagonist AMG9810 promotes mouse skin tumorigenesis through EGFR/Akt signaling.
Journal: Carcinogenesis 20110501
Title: Synergistic role of TRPV1 and TRPA1 in pancreatic pain and inflammation.
Journal: Gastroenterology 20110401
Title: Effect of transient receptor potential vanilloid 1 (TRPV1) receptor antagonist compounds SB705498, BCTC and AMG9810 in rat models of thermal hyperalgesia measured with an increasing-temperature water bath.
Journal: European journal of pharmacology 20100901
Title: The involvement of the transient receptor potential A1 (TRPA1) in the maintenance of mechanical and cold hyperalgesia in persistent inflammation.
Journal: Pain 20100301
Title: Comparison of the peripheral mediator background of heat injury- and plantar incision-induced drop of the noxious heat threshold in the rat.
Journal: Life sciences 20100213
Title: Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
Journal: The Journal of pharmacology and experimental therapeutics 20100201
Title: Activation of TRPV1 and TRPA1 leads to muscle nociception and mechanical hyperalgesia.
Journal: Pain 20090801
Title: Differential effects of transient receptor vanilloid one (TRPV1) antagonists in acid-induced excitation of esophageal vagal afferent fibers of rats.
Journal: Neuroscience 20090630
Title: Effect of increasing temperature on TRPV1-mediated responses in isolated rat pulmonary sensory neurons.
Journal: American journal of physiology. Lung cellular and molecular physiology 20080301
Title: The role of TRPV1 in different subtypes of dorsal root ganglion neurons in rat chronic inflammatory nociception induced by complete Freund's adjuvant.
Journal: Molecular pain 20080101
Title: Three-dimensional quantitative structure-activity relationships and activity predictions of human TRPV1 channel antagonists: comparative molecular field analysis and comparative molecular similarity index analysis of cinnamides.
Journal: Journal of medicinal chemistry 20071115
Title: Novel vanilloid receptor-1 antagonists: 1. Conformationally restricted analogues of trans-cinnamides.
Journal: Journal of medicinal chemistry 20070726
Title: The potential of transient receptor potential vanilloid type 1 channel modulators for the treatment of pain.
Journal: Journal of medicinal chemistry 20070531
Title: Arvanil, anandamide and N-arachidonoyl-dopamine (NADA) inhibit emesis through cannabinoid CB1 and vanilloid TRPV1 receptors in the ferret.
Journal: The European journal of neuroscience 20070501
Title: Antihyperalgesic effects of vanilloid-1 and bradykinin-1 receptor antagonists following spinal cord injury in rats.
Journal: Journal of neurosurgery. Spine 20070501
Title: The vanilloid receptor TRPV1 is tonically activated in vivo and involved in body temperature regulation.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20070328
Title: Thermal sensitivity of isolated vagal pulmonary sensory neurons: role of transient receptor potential vanilloid receptors.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20060901
Title: AMG 9810 [(E)-3-(4-t-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)acrylamide], a novel vanilloid receptor 1 (TRPV1) antagonist with antihyperalgesic properties.
Journal: The Journal of pharmacology and experimental therapeutics 20050401
Title: Discovery of potent, orally available vanilloid receptor-1 antagonists. Structure-activity relationship of N-aryl cinnamides.
Journal: Journal of medicinal chemistry 20050113
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: D-glucose-6-phosphate dehydrogenase (Entner-Doudoroff enzyme) from Pseudomonas fluorescens. Purification, properties and regulation.
Journal: European journal of biochemistry 19751115
Title: Gavva NR, et al. AMG9810 [(E)-3-(4-t-butylphenyl)-N-(2,3-dihydrobenzo[b,4 dioxin-6-yl)acrylamide, a novel vanilloid receptor 1 (TRPV1) antagonist with antihyperalgesic properties. J Pharmacol Exp Ther. 2005 Apr;313(1):474-84.
Title: Li S, et al. TRPV1-antagonist AMG9810 promotes mouse skin tumorigenesis through EGFR/Akt signaling. Carcinogenesis. 2011 May;32(5):779-85.
