Title: Discovery of (1R,2S)-2-{[(2,4-Dimethylpyrimidin-5-yl)oxy]methyl}-2-(3-fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropanecarboxamide (E2006): A Potent and Efficacious Oral Orexin Receptor Antagonist.
Journal: Journal of medicinal chemistry 20150611
Title: Discovery of (1R,2R)-N-(4-(6-isopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide, a potent and orally efficacious mGlu5 receptor negative allosteric modulator.
Journal: Bioorganic & medicinal chemistry letters 20130301
Title: Multi-component anion relay cascade of 1-acetylcyclopropanecarboxamides, aldehydes and acrylonitrile: access to biscyanoethylated furo[3,2-c]pyridinones.
Journal: Organic & biomolecular chemistry 20120621
Title: Highly asymmetric intramolecular cyclopropanation of acceptor-substituted diazoacetates by Co(II)-based metalloradical catalysis: iterative approach for development of new-generation catalysts.
Journal: Journal of the American Chemical Society 20111005
Title: Novel series of pyrrolotriazine analogs as highly potent pan-Aurora kinase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20110915
Title: Ursodeoxycholic acid amides as novel glucocorticoid receptor modulators.
Journal: Journal of medicinal chemistry 20110113
Title: Identification of a new biaryl scaffold generating potent renin inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20101001
Title: Synthesis, antifungal activities and 3D-QSAR study of N-(5-substituted-1,3,4-thiadiazol-2-yl)cyclopropanecarboxamides.
Journal: European journal of medicinal chemistry 20090701
Title: Synthesis and biological evaluation of cis-locked vinylogous combretastatin-A4 analogues: derivatives with a cyclopropyl-vinyl or a cyclopropyl-amide bridge.
Journal: Bioorganic & medicinal chemistry letters 20090301
Title: Potential energy scans and vibrational assignments of cyclopropanecarboxylic acid and cyclopropanecarboxamide.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20081215
Title: Effect of Maillard reacted peptides on human salt taste and the amiloride-insensitive salt taste receptor (TRPV1t).
Journal: Chemical senses 20080901
Title: Modifications of antiepileptic drugs for improved tolerability and efficacy.
Journal: Perspectives in medicinal chemistry 20080101
Title: Bradykinin B1 antagonists: biphenyl SAR studies in the cyclopropanecarboxamide series.
Journal: Bioorganic & medicinal chemistry letters 20070701
Title: Design, synthesis and melatoninergic potency of new N-acyl 8,9-dihydro-4-methoxy-7H-2-benzo[de]quinolinalkanamines.
Journal: Bioorganic chemistry 20070401
Title: High affinity electrophilic and photoactivatable covalent endocannabinoid probes for the CB1 receptor.
Journal: Journal of medicinal chemistry 20051006
Title: Convergent approach to (E)-alkene and cyclopropane peptide isosteres.
Journal: Organic letters 20050106
Title: Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56(Lck).
Journal: Bioorganic & medicinal chemistry letters 20031117
Title: Sequential elimination-cyclopropanation reactions promoted by samarium: highly diastereoselective synthesis of cyclopropylamides.
Journal: The Journal of organic chemistry 20030207
Title: Discovery and SAR of diarylsulfide cyclopropylamide LFA-1/ICAM-1 interaction antagonists.
Journal: Bioorganic & medicinal chemistry letters 20010423