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Title: Highly regioselective synthesis of polysubstituted tetrahydroquinolines by an iodine-induced tandem cyclization reaction from propargylic alcohols and amines.
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Title: Oxygen and temperature sensitivity of blue to green to yellow light-emitting Pt(II) complexes.
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Title: Subtle structural changes in tetrahydroquinolines, a new class of nonsteroidal selective androgen receptor modulators, induce different functions.
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Title: An asymmetric organocatalytic Povarov reaction with 2-hydroxystyrenes.
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Title: The asymmetric synthesis of CF3- or -CF2-substituted tetrahydroquinolines by employing a chiral phosphoric acid as catalyst.
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Title: Asymmetric synthesis of 2-alkyl-substituted tetrahydroquinolines by an enantioselective aza-Michael reaction.
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Title: Cyclocondensation of amino-propargyl silanes.
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Title: Catalytic asymmetric synthesis of chromenes and tetrahydroquinolines via sequential allylic alkylation and intramolecular Heck coupling.
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Title: Highly enantioselective assembly of functionalized tetrahydroquinolines with creation of an all-carbon quaternary center.
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Title: 1,2,3,4-tetrahydroquinoline-based selective human neuronal nitric oxide synthase (nNOS) inhibitors: lead optimization studies resulting in the identification of N-(1-(2-(methylamino)ethyl)-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-carboximidamide as a preclinical development candidate.
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Title: Ocular pharmacokinetics of a novel tetrahydroquinoline analog in rabbit: compartmental analysis and PK-PD evaluation.
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Title: The novel non-steroidal selective androgen receptor modulator S-101479 has additive effects with bisphosphonate, selective estrogen receptor modulator, and parathyroid hormone on the bones of osteoporotic female rats.
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Title: Efficient synthesis and free-radical scavenging capacity of new 2,4-substituted tetrahydroquinolines prepared via BiCl₃-catalyzed three-component Povarov reaction, using N-vinylamides.
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Title: 2-Oxo-N-aryl-1,2,3,4-tetrahydroquinoline-6-sulfonamides as activators of the tumor cell specific M2 isoform of pyruvate kinase.
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Title: Chiral phosphoric acid-catalyzed enantioselective three-component Povarov reaction using enecarbamates as dienophiles: highly diastereo- and enantioselective synthesis of substituted 4-aminotetrahydroquinolines.
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Title: 1-Benzoyl-3-[3-cyano-8-methyl-4-(1-methyl-1H-pyrrol-2-yl)-5,6,7,8-tetra-hydro-quinolin-2-yl]thio-urea.
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Title: Design, synthesis, and biological evaluation of 3,4-dihydroquinolin-2(1H)-one and 1,2,3,4-tetrahydroquinoline-based selective human neuronal nitric oxide synthase (nNOS) inhibitors.
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Title: FeCl3-mediated synthesis of polysubstituted tetrahydroquinolines via domino Mannich/Friedel-Crafts reactions of aldehydes and amines.
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Title: Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs).
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Title: Highly enantioselective synthesis of tetrahydroquinolines via cobalt(II)-catalyzed tandem 1,5-hydride transfer/cyclization.
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Title: Scandium(III) zeolites as new heterogeneous catalysts: [4+2]cyclocondensation of in situ generated aryl imines with alkenes.
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Title: Tetrahydroquinoline glucocorticoid receptor agonists: discovery of a 3-hydroxyl for improving receptor selectivity.
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Title: (3S)-2-Benzyl-3-carb-oxy-1,2,3,4-tetra-hydro-isoquinolinium chloride monohydrate.
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Title: Functional importance of tyrosine 294 and the catalytic selectivity for the bis-Fe(IV) state of MauG revealed by replacement of this axial heme ligand with histidine .
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Title: InCl3-catalyzed allylic Friedel-Crafts reactions toward the stereocontrolled synthesis of 1,2,3,4-tetrahydroquinolines.
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Title: Comparison of the activity of non-steroidal ecdysone agonists between dipteran and lepidopteran insects, using cell-based EcR reporter assays.
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Title: Synthesis, testing and structure-activity studies on a library of 5-HT₄ ligands.
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Title: Quinoline-based compounds as modulators of HIV transcription through NF-kappaB and Sp1 inhibition.
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Title: Enantioselective organocatalytic C-H bond functionalization via tandem 1,5-hydride transfer/ring closure: asymmetric synthesis of tetrahydroquinolines.
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Title: 5,8-Dimeth-oxy-2-phenyl-1,4-dihydro-quinoline-3-carbonitrile.
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Title: A small-molecule oxocarbazate inhibitor of human cathepsin L blocks severe acute respiratory syndrome and ebola pseudotype virus infection into human embryonic kidney 293T cells.
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Title: Quinaphos and Dihydro-Quinaphos phosphine-phosphoramidite ligands for asymmetric hydrogenation.
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Title: Palladium-catalyzed ring-expansion reaction of indoles with alkynes: from indoles to tetrahydroquinoline derivatives under mild reaction conditions.
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Title: Asymmetric three-component inverse electron-demand aza-Diels-Alder reaction: efficient synthesis of ring-fused tetrahydroquinolines.
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Title: Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs.
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Title: Assessment of species specificity of moulting accelerating compounds in Lepidoptera: comparison of activity between Bombyx mori and Spodoptera littoralis by in vitro reporter and in vivo toxicity assays.
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Title: Discovering some novel tetrahydroquinoline derivatives bearing the biologically active sulfonamide moiety as a new class of antitumor agents.
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Title: Diverse effects on mitochondrial and nuclear functions elicited by drugs and genetic knockdowns in bloodstream stage Trypanosoma brucei.
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Title: Iridium-catalyzed, silyl-directed borylation of nitrogen-containing heterocycles.
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Title: Diphosphine-catalyzed mixed double-Michael reaction: a unified synthesis of indolines, dihydropyrrolopyridines, benzimidazolines, tetrahydroquinolines, tetrahydroisoquinolines, dihydrobenzo-1,4-oxazines, and dihydrobenzo-3,1-oxazines.
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Title: Novel tetrahydrochinoline derived CETP inhibitors.
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Title: Zn(OTf)2-catalyzed reactions of ethenetricarboxylates with 2-aminobenzaldehydes leading to tetrahydroquinoline derivatives.
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Title: Efficient entry into 2-substituted tetrahydroquinoline systems through alkylative ring expansion: stereoselective formal synthesis of (+/-)-martinellic acid.
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Title: Easy access to isoquinolines and tetrahydroquinolines from ketoximes and alkynes via rhodium-catalyzed C-H bond activation.
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Title: Tetrahydroquinoline derivatives as CRTH2 antagonists.
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Title: N,1-Bis(4-chloro-2-methyl-benz-yl)-3-methyl-2-oxo-1,2,3,4-tetra-hydro-quinoline-3-carboxamide.
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Title: Tetrahydroquinoline sulfonamides as vasopressin 1b receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20091101
Title: Design, synthesis and anticancer evaluation of novel tetrahydroquinoline derivatives containing sulfonamide moiety.
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Title: Substituted tetrahydroquinolines as potent allosteric inhibitors of reverse transcriptase and its key mutants.
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Title: Gold-catalyzed intramolecular allylic amination of 2-tosylaminophenylprop-1-en-3-ols. A concise synthesis of (+/-)-angustureine.
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Title: Improved asymmetric synthesis of 3,4-dihydro-2-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-5-[3-(trifluoromethoxy)phenyl]-alpha-(trifluoromethyl)-1(2H)-quinolineethanol, a potent cholesteryl ester transfer protein inhibitor.
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Title: Design and synthesis of potent inhibitors of cholesteryl ester transfer protein (CETP) exploiting a 1,2,3,4-tetrahydroquinoline platform.
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Title: Self-assembly of hydrogensquarates: crystal structures and properties.
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Title: Substituted 1,2,3,4-tetrahydroquinolin-6-yloxypropanes as beta3-adrenergic receptor agonists: design, synthesis, biological evaluation and pharmacophore modeling.
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Title: Lewis acid or Brønsted acid catalyzed reactions of vinylidene cyclopropanes with activated carbon-nitrogen, nitrogen-nitrogen, and iodine-nitrogen double-bond-containing compounds.
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Title: Synthesis and biotransformation of tetrahydroquinoline by Mortierella isabelina.
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Title: QSAR study on tetrahydroquinoline analogues as plasmodium protein farnesyltransferase inhibitors: a comparison of rationales of malarial and mammalian enzyme inhibitory activities for selectivity.
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Title: Air-stable and phosphine-free iridium catalysts for highly enantioselective hydrogenation of quinoline derivatives.
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Title: Bis(1,2,3,4-tetra-hydro-quinolin-6-yl)methane.
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Title: Ruthenium-catalyzed enantioselective carbon-carbon bond forming reaction via allenylidene-ene process: synthetic approach to chiral heterocycles such as chromane, thiochromane, and 1,2,3,4-tetrahydroquinoline derivatives.
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Title: Natural products as an inspiration in the diversity-oriented synthesis of bioactive compound libraries.
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Title: Synthesis and characterization of 5,6,7,8-tetrahydroquinoline C5a receptor antagonists.
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Title: Suzuki-Miyaura approach to JNJ-26076713, an orally active tetrahydroquinoline-containing alphaVbeta3/alphaVbeta5 integrin antagonist. enantioselective synthesis and stereochemical studies.
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Title: Strictosidine synthase: mechanism of a Pictet-Spengler catalyzing enzyme.
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Title: Selective androgen receptor modulators in preclinical and clinical development.
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Title: Effect of ecdysone receptor gene switch ligands on endogenous gene expression in 293 cells.
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Title: Design, synthesis, and evaluation of tetrahydroquinoline and pyrrolidine sulfonamide carbamates as gamma-secretase inhibitors.
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Title: Cobaltpolyoxometalate-catalyzed cyclization of glucal with aryl amines: Synthesis of 2,4-disubstituted tetrahydroquinolines.
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Title: Lewis acid catalyzed reaction of arylvinylidenecyclopropanes with ethyl (arylimino)acetates: a facile synthetic protocol for pyrrolidine and 1,2,3,4-tetrahydroquinoline derivatives.
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Title: Resistance mutations at the lipid substrate binding site of Plasmodium falciparum protein farnesyltransferase.
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Title: Chiral tetrahydroquinoline derivatives as potent anti-hyperalgesic agents in animal models of sustained inflammation and chronic neuropathic pain.
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Title: Moexipril and left ventricular hypertrophy.
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Title: Tetrahydroquinoline sulfonamides as gamma-secretase inhibitors.
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Title: Heteroarotinoids with anti-cancer activity against ovarian cancer cells.
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Title: Metabolic aromatization of N-alkyl-1,2,3,4-tetrahydroquinoline substructures to quinolinium by human liver microsomes and horseradish peroxidase.
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Title: Microwave-assisted, solid-phase synthesis of a chiral 1,2,3,4-tetrahydro-quinoline library.
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Title: Synthesis and stereochemical investigations of novel nitrogen-containing 13alpha-estrone derivatives.
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Title: Synthesis and SAR of novel histamine H3 receptor antagonists.
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Title: Homoleptic rare earth dipyridylamides [Ln2(N(NC5H4)2)6], Ln = Ce, Nd, Sm, Ho, Er, Tm, Yb, and Sc: metal oxidation by the amine melt and in 1,2,3,4-tetrahydroquinoline with the focus of different metal activation by amalgams, liquid ammonia, and microwaves.
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Title: Structure-activity relationships of a series of tariquidar analogs as multidrug resistance modulators.
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Title: Adding pharmacogenomics to the development of new marine-derived anticancer agents.
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Title: Synthesis, spectral studies and in vitro assessment for antiamoebic activity of new cyclooctadiene ruthenium(II) complexes with 5-nitrothiophene-2-carboxaldehyde thiosemicarbazones.
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Title: First QSAR report on FSH receptor antagonistic activity: quantitative investigations on physico-chemical and structural features among 6-amino-4-phenyltetrahydroquinoline derivatives.
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Title: Identification of photoproducts of hexahydroquinoline derivatives by GC-EI-MS and HPLC-ESI-MS.
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Title: Protein farnesyltransferase inhibitors exhibit potent antimalarial activity.
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Title: Resistance to a protein farnesyltransferase inhibitor in Plasmodium falciparum.
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Title: Asymmetric synthesis of novel tetrahydroquinoline derivatives with a sugar building block and their bioactivities.
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Title: Structure-property relationship in py-hexahydrocinchonidine diastereomers: ab initio and NMR study.
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Title: Synthesis of novel steroid-tetrahydroquinoline hybrid molecules and D-homosteroids by intramolecular cyclization reactions.
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Title: Intramolecular arylation reactions of alkenes: a flexible approach to chromans and tetrahydroquinoline derivatives.
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Title: A solid-phase, library synthesis of natural-product-like derivatives from an enantiomerically pure tetrahydroquinoline scaffold.
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Title: Helquinoline, a new tetrahydroquinoline antibiotic from Janibacter limosus Hel 1+.
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Title: A solution- and solid-phase approach to tetrahydroquinoline-derived polycyclics having a 10-membered ring.
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Title: Solution- and solid-phase synthesis of natural product-like tetrahydroquinoline-based polycyclics having a medium size ring.
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Title: The effect of remote chirality on the antibacterial activity of indolinyl, tetrahydroquinolyl and dihydrobenzoxazinyl oxazolidinones.
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Title: Enantiomerically pure tetrahydroquinoline derivatives as in vivo potent antagonists of the glycine binding site associated to the NMDA receptor.
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Title: 1,4-benzothiazine analogues and apoptosis: structure-activity relationship.
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Title: Synthesis and SAR of cis-1-benzoyl-1,2,3,4-tetrahydroquinoline ligands for control of gene expression in ecdysone responsive systems.
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