Title: Primary amino acid derivatives: substitution of the 4'-N'-benzylamide site in (R)-N'-benzyl 2-amino-3-methylbutanamide, (R)-N'-benzyl 2-amino-3,3-dimethylbutanamide, and (R)-N'-benzyl 2-amino-3-methoxypropionamide provides potent anticonvulsants with pain-attenuating properties.
Journal: Journal of medicinal chemistry 20111013
Title: Primary amino acid derivatives: compounds with anticonvulsant and neuropathic pain protection activities.
Journal: Journal of medicinal chemistry 20110714
Title: 1,2-Diamines as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1).
Journal: Bioorganic & medicinal chemistry letters 20091201