Title: Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20111001
Title: Structure of the adenosine A(2A) receptor in complex with ZM241385 and the xanthines XAC and caffeine.
Journal: Structure (London, England : 1993) 20110907
Title: Biophysical mapping of the adenosine A2A receptor.
Journal: Journal of medicinal chemistry 20110714
Title: T-cell specific defect in expression of the NTPDase CD39 as a biomarker for lupus.
Journal: Cellular immunology 20110101
Title: Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions.
Journal: Molecular pharmacology 20100401
Title: Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands.
Journal: British journal of pharmacology 20100201
Title: Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Journal: Nature chemical biology 20091001
Title: Synthesis of hybrid analogues of caffeine and eudistomin D and its affinity for adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20090701
Title: N6-Cycloalkyl- and N6-bicycloalkyl-C5'(C2')-modified adenosine derivatives as high-affinity and selective agonists at the human A1 adenosine receptor with antinociceptive effects in mice.
Journal: Journal of medicinal chemistry 20090423
Title: Synthesis of eudistomin D analogues and its effects on adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20080401
Title: A pharmacological activator of AMP-activated protein kinase (AMPK) induces astrocyte stellation.
Journal: Brain research 20070907
Title: Synthesis of hybrid molecules of caffeine and eudistomin D and its effects on adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20070501
Title: Protective effect of adenosine and purine nucleos(t)ides against the death by hydrogen peroxide and glucose deprivation in rat primary astrocytes.
Journal: Neuroscience research 20050101
Title: [3H]OSIP339391, a selective, novel, and high affinity antagonist radioligand for adenosine A2B receptors.
Journal: Biochemical pharmacology 20040715
Title: Synthesis, molecular modeling studies, and pharmacological activity of selective A(1) receptor antagonists.
Journal: Journal of medicinal chemistry 20021024
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: Adenosine receptor-mediated control of in vitro release of pain-related neuropeptides from the rat spinal cord.
Journal: European journal of pharmacology 20020419
Title: Multiple dilator pathways in skeletal muscle contraction-induced arteriolar dilations.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20020401
Title: 1,8-disubstituted xanthine derivatives: synthesis of potent A2B-selective adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20020328
Title: Adenosine receptor antagonists and retinal neovascularization in vivo.
Journal: Investigative ophthalmology & visual science 20011201
Title: Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides.
Journal: Journal of medicinal chemistry 20011122
Title: [3H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors.
Journal: Biochemical pharmacology 20010315
Title: Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20010301
Title: Why are A(2B) receptors low-affinity adenosine receptors? Mutation of Asn273 to Tyr increases affinity of human A(2B) receptor for 2-(1-Hexynyl)adenosine.
Journal: Molecular pharmacology 20001201
Title: [(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.
Journal: Molecular pharmacology 20000501
Title: Anilide derivatives of an 8-phenylxanthine carboxylic congener are highly potent and selective antagonists at human A(2B) adenosine receptors.
Journal: Journal of medicinal chemistry 20000323
Title: Use of the triazolotriazine [3H]ZM 241385 as a radioligand at recombinant human A2B adenosine receptors.
Journal: Drug design and discovery 19991101
Title: Characterization of human A(2B) adenosine receptors: radioligand binding, western blotting, and coupling to G(q) in human embryonic kidney 293 cells and HMC-1 mast cells.
Journal: Molecular pharmacology 19991001
Title: Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 19980101
Title: Characterization of human A2A adenosine receptors with the antagonist radioligand [3H]-SCH 58261.
Journal: British journal of pharmacology 19970501
Title: Characterization of the human brain putative A2B adenosine receptor expressed in Chinese hamster ovary (CHO.A2B4) cells.
Journal: British journal of pharmacology 19961101
Title: Site-directed mutagenesis identifies residues involved in ligand recognition in the human A2a adenosine receptor.
Journal: The Journal of biological chemistry 19950609
Title: Species difference in the G protein selectivity of the human and bovine A1-adenosine receptor.
Journal: The Journal of biological chemistry 19941223
Title: Role of the second extracellular loop of adenosine receptors in agonist and antagonist binding. Analysis of chimeric A1/A3 adenosine receptors.
Journal: The Journal of biological chemistry 19941007
Title: Molecular cloning and characterization of the human A3 adenosine receptor.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19931101
Title: Potent convulsant actions of the adenosine receptor antagonist, xanthine amine congener (XAC).
Journal: Life sciences 19890101