Title: Synthesis of some new benzisothiazolone and benzenesulfonamide derivatives of biological interest starting from saccharin sodium.
Journal: Archiv der Pharmazie 20131001
Title: Amide derivatives of benzene-sulfonanilide, pharmaceutical composition thereof and method for cancer treatment using the same (US20120095092).
Journal: Expert opinion on therapeutic patents 20121001
Title: Eight isostructural 4,4'-disubstituted N-phenylbenzenesulfonamides.
Journal: Acta crystallographica. Section C, Crystal structure communications 20121001
Title: Benzenesulfonamide attenuates monocrotaline-induced pulmonary arterial hypertension in a rat model.
Journal: European journal of pharmacology 20120905
Title: Virtual screening leads to the discovery of novel non-nucleotide P2Y₁ receptor antagonists.
Journal: Bioorganic & medicinal chemistry 20120901
Title: Placing supercritical fluid chromatography one step ahead of reversed-phase high performance liquid chromatography in the achiral purification arena: a hydrophilic interaction chromatography cross-linked diol chemistry as a new generic stationary phase.
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Title: Magnetic levitation as a platform for competitive protein-ligand binding assays.
Journal: Analytical chemistry 20120717
Title: FT-IR, FT-Raman and computational study of (E)-N-carbamimidoyl-4-((4-methoxybenzylidene)amino)benzenesulfonamide.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20120615
Title: Sulfonamide bearing oligonucleotides: simple synthesis and efficient RNA recognition.
Journal: Bioorganic & medicinal chemistry 20120615
Title: The novel endocrine disruptor tolylfluanid impairs insulin signaling in primary rodent and human adipocytes through a reduction in insulin receptor substrate-1 levels.
Journal: Biochimica et biophysica acta 20120601
Title: Research on the structure-surface adsorptive activity relationships of triazolyl glycolipid derivatives for mild steel in HCl.
Journal: Carbohydrate research 20120601
Title: Design of [(2-pyrimidinylthio)acetyl]benzenesulfonamides as inhibitors of human carbonic anhydrases.
Journal: European journal of medicinal chemistry 20120501
Title: N-(3-Methyl-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20120501
Title: N-(3-Nitro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20120501
Title: Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal: Journal of medicinal chemistry 20120412
Title: Discovery of novel 2-N-aryl-substituted benzenesulfonamidoacetamides: orally bioavailable tubulin polymerization inhibitors with marked antitumor activities.
Journal: ChemMedChem 20120401
Title: (3aR*,6S*,7aR*)-7a-Chloro-6-methyl-2-(4-methyl-phenyl-sulfon-yl)-2,3,3a,6,7,7a-hexa-hydro-3a,6-ep-oxy-1H-isoindole.
Journal: Acta crystallographica. Section E, Structure reports online 20120401
Title: Identification of novel kynurenine production-inhibiting benzenesulfonamide derivatives in cancer cells.
Journal: Biochemical and biophysical research communications 20120316
Title: Inhibitory effects of azole-type fungicides on interleukin-17 gene expression via retinoic acid receptor-related orphan receptors α and γ.
Journal: Toxicology and applied pharmacology 20120315
Title: Synthesis and evaluation of anticancer activity of some novel 6-aryl-2-(p-sulfamylphenyl)-pyridazin-3(2H)-ones.
Journal: European journal of medicinal chemistry 20120301
Title: 4-{(4Z)-4-[(2Z)-3-(4-Fluoro-anilino)-1-hy-droxy-but-2-en-1-yl-idene]-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl}-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20120301
Title: Selective precipitation and purification of monovalent proteins using oligovalent ligands and ammonium sulfate.
Journal: Bioconjugate chemistry 20120215
Title: Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives.
Journal: Bioorganic & medicinal chemistry letters 20120201
Title: N-Ethyl-N-(4-methyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20120201
Title: 2-(N-Cyclo-hexyl-carbamo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20120201
Title: Dependence of avidity on linker length for a bivalent ligand-bivalent receptor model system.
Journal: Journal of the American Chemical Society 20120111
Title: 5-HT₂c receptor selectivity and structure-activity relationship of N-methyl-N-(1-methylpiperidin-4-yl)benzenesulfonamide analogs.
Journal: Bioorganic & medicinal chemistry letters 20120101
Title: Hydroxybenzothiazoles as new nonsteroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1).
Journal: PloS one 20120101
Title: Novel 4-(4-substituted-thiazol-2-ylamino)-N-(pyridin-2-yl)-benzenesulfonamides as cytotoxic and radiosensitizing agents.
Journal: Archives of pharmacal research 20120101
Title: Synthesis, in-vitro anticancer screening and radiosensitizing evaluation of some new N-(quinoxalin-2-yl)benzenesulfonamide derivatives.
Journal: Arzneimittel-Forschung 20120101
Title: Regulation of expression of citrate synthase by the retinoic acid receptor-related orphan receptor α (RORα).
Journal: PloS one 20120101
Title: FH535 potentiation of cigarette smoke condensate cytotoxicity is associated with changes in β-catenin and EGR-1 signaling.
Journal: International journal of toxicology 20120101
Title: Label-free detection of protein binding with multisine SPR microchips.
Journal: Lab on a chip 20111221
Title: Estimation of analyte concentration by surface plasmon resonance-based biosensing using parameter identification techniques.
Journal: Analytical biochemistry 20111215
Title: FT-IR, FT-Raman and quantum chemical calculations of (E)-N-carbamimidoyl-4-((3,4-dimethoxybenzylidene) amino) benzenesulfonamide.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20111215
Title: Radiosynthesis of three [11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumors.
Journal: Bioorganic & medicinal chemistry letters 20111201
Title: Synthesis and biological evaluation of some new 2-pyrazolines bearing benzene sulfonamide moiety as potential anti-inflammatory and anti-cancer agents.
Journal: European journal of medicinal chemistry 20111201
Title: Synthesis, in vitro anticancer screening and radiosensitizing evaluation of some new 4-[3-(substituted)thioureido]-N-(quinoxalin-2-yl)-benzenesulfonamide derivatives.
Journal: Acta pharmaceutica (Zagreb, Croatia) 20111201
Title: Synthesis and acrosin inhibitory activity of substituted 4-amino-N-(diaminomethylene) benzenesulfonamide derivatives.
Journal: Bioorganic & medicinal chemistry letters 20111115
Title: A double prodrug system for colon targeting of benzenesulfonamide COX-2 inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20111115
Title: Rhodium-catalyzed annulation of N-benzoylsulfonamide with isocyanide through C-H activation.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20111104
Title: Substituted phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonamides as antimitotics. Antiproliferative, antiangiogenic and antitumoral activity, and quantitative structure-activity relationships.
Journal: European journal of medicinal chemistry 20111101
Title: 2,4-Dichloro-N-(3,5-dimethyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20111101
Title: 4-Chloro-N-(3,4-dichloro-phen-yl)-2-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20111101
Title: Identification of novel small molecule inhibitors of 4-diphosphocytidyl-2-C-methyl-D-erythritol (CDP-ME) kinase of Gram-negative bacteria.
Journal: Bioorganic & medicinal chemistry 20111001
Title: Design and synthesis of new N-(5-trifluoromethyl)-1H-1,2,4-triazol-3-yl benzenesulfonamides as possible antimalarial prototypes.
Journal: Molecules (Basel, Switzerland) 20110920
Title: Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against human α- and bacterial/fungal β-carbonic anhydrases.
Journal: Bioorganic & medicinal chemistry letters 20110915
Title: Fluoroalkyl and alkyl chains have similar hydrophobicities in binding to the 'hydrophobic wall' of carbonic anhydrase.
Journal: Journal of the American Chemical Society 20110907
Title: Synthesis and in vivo evaluation of [O-methyl-11C] N-[3,5-dichloro-2-(methoxy)phenyl]-4-(methoxy)-3-(1-piperazinyl)benzenesulfonamide as an imaging probe for 5-HT6 receptors.
Journal: Bioorganic & medicinal chemistry 20110901
Title: N-(2,6-Dimethyl-phen-yl)-2,4-dimethyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110901
Title: 1-Benzyl-2,5-diphenyl-3-tosylimidazol-idin-4-one.
Journal: Acta crystallographica. Section E, Structure reports online 20110901
Title: 4-(3-Methyl-5-phenyl-1H-pyrazol-1-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110901
Title: 4-(3,7-Dimethyl-4-oxo-4,5-dihydro-isoxazolo[4,5-d]pyridazin-5-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110901
Title: 4-(5-Oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110901
Title: 4-(3-Methyl-4,5-dihydro-1H-benzo[g]indazol-1-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110901
Title: Using covalent dimers of human carbonic anhydrase II to model bivalency in immunoglobulins.
Journal: Journal of the American Chemical Society 20110803
Title: Potassium N-bromo-2-methyl-benzene-sulfonamidate sesquihydrate.
Journal: Acta crystallographica. Section E, Structure reports online 20110801
Title: 2-(4-Chloro-phen-yl)-5-(cyclo-hex-1-en-1-yl)-3-(4-methyl-phenyl-sulfon-yl)-1-phenyl-imidazolidin-4-one.
Journal: Acta crystallographica. Section E, Structure reports online 20110801
Title: 4-Chloro-N-(3,5-dimethyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110801
Title: Systematic errors in isothermal titration calorimetry: concentrations and baselines.
Journal: Analytical biochemistry 20110715
Title: Synthesis of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide as anticancer and anti-inflammatory agents.
Journal: Bioorganic & medicinal chemistry letters 20110715
Title: Potassium N,2-dichloro-benzene-sulfonamidate sesquihydrate.
Journal: Acta crystallographica. Section E, Structure reports online 20110701
Title: Potassium N,4-dichloro-benzene-sulfonamidate monohydrate.
Journal: Acta crystallographica. Section E, Structure reports online 20110701
Title: Potassium N-bromo-4-chloro-benzene-sulfonamidate monohydrate.
Journal: Acta crystallographica. Section E, Structure reports online 20110701
Title: Amino-caprolactam γ-secretase inhibitors showing potential for the treatment of Alzheimer's disease.
Journal: Bioorganic & medicinal chemistry letters 20110615
Title: Conformational variability of different sulfonamide inhibitors with thienyl-acetamido moieties attributes to differential binding in the active site of cytosolic human carbonic anhydrase isoforms.
Journal: Bioorganic & medicinal chemistry 20110615
Title: Crossing borders to bind proteins--a new concept in protein recognition based on the conjugation of small organic molecules or short peptides to polypeptides from a designed set.
Journal: Analytical and bioanalytical chemistry 20110601
Title: Ethyl 3-[2-(3,4-dimeth-oxy-benz-yl)-1-phenyl-sulfonyl-1H-indol-3-yl]acrylate chloro-form hemisolvate.
Journal: Acta crystallographica. Section E, Structure reports online 20110601
Title: A novel COX-2 inhibitor pyrazole derivative proven effective as an anti-inflammatory and analgesic drug.
Journal: Basic & clinical pharmacology & toxicology 20110401
Title: Synthesis and biological evaluation of some 4-functionalized-pyrazoles as antimicrobial agents.
Journal: European journal of medicinal chemistry 20110401
Title: 2-(4-Chloro-phen-yl)-1,5-diphenyl-3-tosyl-imidazolidin-4-one.
Journal: Acta crystallographica. Section E, Structure reports online 20110401
Title: 4-Chloro-N-(4-nitro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110401
Title: 2-Methyl-N-(4-nitro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110401
Title: 2-Chloro-N-(4-nitro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110401
Title: Studies of tricyclic piperazine/piperidine furnished molecules as novel integrin αvβ3/αIIbβ3 dual antagonists using 3D-QSAR and molecular docking.
Journal: Journal of molecular graphics & modelling 20110201
Title: N-(4-Meth-oxy-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110201
Title: Molecular structure and vibrational investigation of benzenesulfonic acid methyl ester using DFT (LSDA, B3LYP, B3PW91 and MPW1PW91) theory calculations.
Journal: Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20110101
Title: Synthesis and in vitro anticancer evaluation of some novel hexahydroquinoline derivatives having a benzenesulfonamide moiety.
Journal: European journal of medicinal chemistry 20110101
Title: Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures (II).
Journal: Bioorganic & medicinal chemistry letters 20110101
Title: Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20110101
Title: 4-Chloro-N-(2,3-dichloro-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110101
Title: N-(2,5-Dichloro-phen-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110101
Title: 2,4-Dimethyl-N-(4-methyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20110101
Title: Induction of SCEs and DNA fragmentation in bovine peripheral lymphocytes by in vitro exposure to tolylfluanid-based fungicide.
Journal: Genetics and molecular biology 20110101
Title: Copper and its complexes in medicine: a biochemical approach.
Journal: Molecular biology international 20110101
Title: Virtual screening of 2,3-disubstituted-4(3H)-quinazolinones possessing benzenesulfonamide moiety for COX-2 inhibitor.
Journal: Bioinformation 20110101
Title: Inhibition of influenza A virus (H1N1) fusion by benzenesulfonamide derivatives targeting viral hemagglutinin.
Journal: PloS one 20110101
Title: Selective elution of target protein from affinity resins by a simple reductant with a thiol group.
Journal: Bioorganic & medicinal chemistry letters 20101215
Title: 4- and 6-(p-Sulphamoylphenyl)androstenediones: Studies of aromatase inhibitor-based oestrone sulphatase inhibition.
Journal: Steroids 20101201
Title: Design and synthesis of an androgen receptor pure antagonist (CH5137291) for the treatment of castration-resistant prostate cancer.
Journal: Bioorganic & medicinal chemistry 20101201
Title: N-(2,3-Dichloro-phen-yl)-2,4-dimethyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20101201
Title: N-(2,6-Dichloro-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20101201
Title: N-(2,3-Dichloro-phen-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20101201
Title: N-(2,3-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20101201
Title: 5,6,7,8-Tetrahydropyrido[4,3-d]pyrimidines as novel class of potent and highly selective CaMKII inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20101115
Title: A diverse series of substituted benzenesulfonamides as aldose reductase inhibitors with antioxidant activity: design, synthesis, and in vitro activity.
Journal: Journal of medicinal chemistry 20101111
Title: 4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.
Journal: Bioorganic & medicinal chemistry 20101101
Title: Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIII.
Journal: Bioorganic & medicinal chemistry 20101101
Title: Free-solution interaction assay of carbonic anhydrase to its inhibitors using back-scattering interferometry.
Journal: Electrophoresis 20101101
Title: N-(5-Chloro-2-meth-oxy-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20101101
Title: 4-[(2-Hy-droxy-benzyl-idene)amino]-N-(5-methyl-isoxazol-3-yl)benzene-sulfonamide: a monoclinic polymorph.
Journal: Acta crystallographica. Section E, Structure reports online 20101001
Title: Synthesis of anti-microtubule N-(2-Arylindol-7-yl)benzenesulfonamide derivatives and their antitumor mechanisms.
Journal: ChemMedChem 20100903
Title: Discovery of pyrrole-indoline-2-ones as Aurora kinase inhibitors with a different inhibition profile.
Journal: Journal of medicinal chemistry 20100826
Title: Identification of N-(2-(azepan-1-yl)-2-phenylethyl)-benzenesulfonamides as novel inhibitors of GlyT1.
Journal: Bioorganic & medicinal chemistry letters 20100815
Title: 2-Methyl-N-(2-methyl-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100801
Title: N-(4-Chloro-benzo-yl)-2-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100801
Title: Cell adhesion to unnatural ligands mediated by a bifunctional protein.
Journal: Journal of the American Chemical Society 20100721
Title: Pteridine-sulfonamide conjugates as dual inhibitors of carbonic anhydrases and dihydrofolate reductase with potential antitumor activity.
Journal: Bioorganic & medicinal chemistry 20100715
Title: Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigations.
Journal: Bioorganic & medicinal chemistry 20100715
Title: Synthesis of quinazolines from N-(2-nitrophenylsulfonyl)iminodiacetate and alpha-(2-nitrophenylsulfonyl)amino ketones via 2H-indazole 1-oxides.
Journal: The Journal of organic chemistry 20100702
Title: Synthesis and in vitro anticancer screening of some novel 4-[2-amino-3-cyano-4-substituted-5,6,7,8-tetrahydroquinolin-1-(4H)-yl]benzenesulfonamides.
Journal: European journal of medicinal chemistry 20100701
Title: 2,4-Dichloro-N-(3-methyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100701
Title: 2,4-Dichloro-N-(3-chloro-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100701
Title: N-(4-Methyl-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100701
Title: New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20100615
Title: A rationale for the activity profile of benzenesulfonamide derivatives as cyclooxygenase (COX) inhibitors.
Journal: European journal of medicinal chemistry 20100601
Title: 4-Chloro-N-(3,4-dimethyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100601
Title: N-(Phenyl-sulfon-yl)acetamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100601
Title: 2-Chloro-N-(3-chloro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100601
Title: 2-Chloro-N-(4-methyl-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100601
Title: Correlation analyses on binding affinity of substituted benzenesulfonamides with carbonic anhydrase using ab initio MO calculations on their complex structures.
Journal: Journal of chemical information and modeling 20100524
Title: 3D-QSAR study of benzene sulfonamide analogs as carbonic anhydrase II inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20100515
Title: Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: structure-based drug design, synthesis, and biological evaluation.
Journal: Bioorganic & medicinal chemistry 20100501
Title: 17,18-Dibromo-8-methyl-4,12-ditosyl-3,4,5,6,7,8,9,10,11,12,13,14-dodeca-hydro-2H-benzo[b][1,4,7,11,15]dioxatriaza-cyclo-hepta-decine.
Journal: Acta crystallographica. Section E, Structure reports online 20100501
Title: N-Phenyl-N-(prop-2-en-1-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100501
Title: N-(4-Hydroxy-phen-yl)benzene-sulfon-amide.
Journal: Acta crystallographica. Section E, Structure reports online 20100501
Title: N-(3,5-Dichloro-phen-yl)-2,4-dimethyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100501
Title: N-(2,6-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100501
Title: catena-Poly[neodymium(III)-bis-[μ-N-(dimorpholinophosphor-yl)benzene-sulfonamidato]-sodium(I)-bis-[μ-N-(dimorpholinophosphor-yl)benzene-sulfonamidato]].
Journal: Acta crystallographica. Section E, Structure reports online 20100401
Title: N-Cyclo-hexyl-4-meth-yl-N-propyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100401
Title: 2-Methyl-N-(4-methyl-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100401
Title: 2,4-Dimethyl-N-(3-methyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100401
Title: Recognition and binding of a helix-loop-helix peptide to carbonic anhydrase occurs via partly folded intermediate structures.
Journal: Biophysical journal 20100203
Title: N-(2-Chloro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100201
Title: N-(4-Chloro-benzo-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100201
Title: 2-Methyl-N-(3-methyl-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100201
Title: cis-N-(2-Hydroxy-cyclo-hexyl)-p-toluene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100201
Title: Computational study of the interactions between guanine derivatives and cyclin-dependent kinase 2 (CDK2) by CoMFA and QM/MM.
Journal: Journal of chemical information and modeling 20100101
Title: Synthesis and biological activities of some novel triazoloquinazolines and triazinoquinazolines containing benzenesulfonamide moieties.
Journal: Arzneimittel-Forschung 20100101
Title: Tamsulosin-induced severe hypotension during general anesthesia: a case report.
Journal: Journal of medical case reports 20100101
Title: Pharmacophore elucidation and molecular docking studies on 5-phenyl-1-(3-pyridyl)-1h-1,2,4-triazole-3-carboxylic acid derivatives as COX-2 inhibitors.
Journal: Scientia pharmaceutica 20100101
Title: [Synthesis and investigation on antidiabetic activity of 4-(1-aryl-3-oxo-5-phenylpentylamino) benzenesulfonamide].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20100101
Title: N-Cyclo-hexyl-N-ethyl-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100101
Title: N,N'-Bis(phenyl-sulfon-yl)succinamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100101
Title: N,N'-Bis(phenyl-sulfon-yl)maleamide.
Journal: Acta crystallographica. Section E, Structure reports online 20100101
Title: Environmentally sensitive fluorescent sensors based on synthetic peptides.
Journal: Sensors (Basel, Switzerland) 20100101
Title: Radiolabelling of proteins with fluorine-18 via click chemistry.
Journal: Chemical communications (Cambridge, England) 20091228
Title: Thermodynamic optimisation in drug discovery: a case study using carbonic anhydrase inhibitors.
Journal: ChemMedChem 20091201
Title: N-Benzyl-N-cyclo-hexyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: 4-Benzene-sulfonamido-benzoic acid.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: N-Cyclo-hexyl-N-(prop-2-en-1-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: N-Benzyl-N-cyclo-hexyl-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: N-(4-Chloro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: N-Cyclo-hexyl-N-propyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: 4-Methyl-N-(2-methyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091201
Title: Discovery and optimization of novel 4-[(aminocarbonyl)amino]-N-[4-(2-aminoethyl)phenyl]benzenesulfonamide ghrelin receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20091101
Title: In vivo and in vitro anti-leishmanial activities of 4-nitro-N-pyrimidin- and N-pyrazin-2-ylbenzenesulfonamides, and N2-(4-nitrophenyl)-N1-propylglycinamide.
Journal: Bioorganic & medicinal chemistry 20091101
Title: 2,2-Dimethyl-N-(phenyl-sulfon-yl)acetamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091101
Title: N-(3-Chloro-benzo-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091101
Title: N-(2,5-Dimethyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091101
Title: N-Cyclohexyl-N-methylbenzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091101
Title: Theoretical characterization of substrate access/exit channels in the human cytochrome P450 3A4 enzyme: involvement of phenylalanine residues in the gating mechanism.
Journal: The journal of physical chemistry. B 20091001
Title: N-Benzo-ylbenzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20091001
Title: Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20090901
Title: 2-Chloro-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090901
Title: N-(2-Formyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090901
Title: N-(2-Acetyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090901
Title: o-Toluene-sulfonamide: a redetermination.
Journal: Acta crystallographica. Section E, Structure reports online 20090901
Title: 4-[(Z)-(2-Eth-oxy-4-oxochroman-3-yl-idene)methyl-amino]benzene-sulfonamide monohydrate.
Journal: Acta crystallographica. Section E, Structure reports online 20090801
Title: 2,4-Dichloro-N-(3,4-dichloro-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090801
Title: In vitro pharmacological characterization of a novel allosteric modulator of alpha 7 neuronal acetylcholine receptor, 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), exhibiting unique pharmacological profile.
Journal: The Journal of pharmacology and experimental therapeutics 20090701
Title: Hybrid molecules between benzenesulfonamides and active antimicrobial benzo[d]isothiazol-3-ones.
Journal: European journal of medicinal chemistry 20090601
Title: Toward the development of metal-based synthetic nucleases: DNA binding and oxidative DNA cleavage of a mixed copper(II) complex with N-(9H-purin-6-yl)benzenesulfonamide and 1,10-phenantroline. Antitumor activity in human Caco-2 cells and Jurkat T lymphocytes. Evaluation of p53 and Bcl-2 proteins in the apoptotic mechanism.
Journal: Journal of inorganic biochemistry 20090601
Title: Sodium N-chloro-2-methyl-benzene-sulfonamidate sesquihydrate.
Journal: Acta crystallographica. Section E, Structure reports online 20090601
Title: 4-Methyl-N-phenyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090601
Title: Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor.
Journal: Journal of medicinal chemistry 20090528
Title: Investigation of the fate of sulfonamides downgradient of a decommissioned sewage farm near Berlin, Germany.
Journal: Journal of contaminant hydrology 20090512
Title: Ligand-directed tosyl chemistry for protein labeling in vivo.
Journal: Nature chemical biology 20090501
Title: Synthesis and biological evaluation of novel pyrazoles and pyrazolo[3,4-d]pyrimidines incorporating a benzenesulfonamide moiety.
Journal: Archiv der Pharmazie 20090401
Title: N-(3,4-Dimethyl-phen-yl)-4-methyl-benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090401
Title: Addition reactions of chloro- or iodomethyllithium to imines. Synthesis of enantiopure aziridines and beta-chloroamines.
Journal: The Journal of organic chemistry 20090320
Title: Synthesis and biological evaluation of sulfonylurea and thiourea derivatives substituted with benzenesulfonamide groups as potential hypoglycemic agents.
Journal: Bioorganic & medicinal chemistry letters 20090315
Title: Improvement of monolithic solid material by utilization of spacer for identification of the target using affinity resins.
Journal: Bioorganic & medicinal chemistry letters 20090301
Title: Carbonic anhydrase inhibitors: two-prong versus mono-prong inhibitors of isoforms I, II, IX, and XII exemplified by photochromic cis-1,2-alpha-dithienylethene derivatives.
Journal: Bioorganic & medicinal chemistry letters 20090301
Title: Ethyl 2-[N-(2-Formyl-phen-yl)benzene-sulfonamido]acetate.
Journal: Acta crystallographica. Section E, Structure reports online 20090301
Title: A novel class of allosteric modulators of AMPA/Kainate receptors.
Journal: Bioorganic & medicinal chemistry letters 20090215
Title: Synthesis and biological evaluation of benzenesulfonamide-substituted 4-(6-alkylpyridin-2-yl)-5-(quinoxalin-6-yl)imidazoles as transforming growth factor-beta type 1 receptor kinase inhibitors.
Journal: European journal of medicinal chemistry 20090201
Title: Synthesis of some pyrazolyl benzenesulfonamide derivatives as dual anti-inflammatory antimicrobial agents.
Journal: Journal of enzyme inhibition and medicinal chemistry 20090201
Title: N-(2,3-Dimethyl-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20090201
Title: Cryptophane xenon-129 nuclear magnetic resonance biosensors targeting human carbonic anhydrase.
Journal: Journal of the American Chemical Society 20090121
Title: Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide.
Journal: Bioorganic & medicinal chemistry letters 20090101
Title: Label-free determination of protein-ligand binding constants using mass spectrometry and validation using surface plasmon resonance and isothermal titration calorimetry.
Journal: Journal of molecular recognition : JMR 20090101
Title: Synthesis and Antiviral Studies of Novel N-Sulphonamidomethyl piperazinyl Fluoroquinolones.
Journal: Indian journal of pharmaceutical sciences 20090101
Title: Dual inhibitors of matrix metalloproteinases and carbonic anhydrases: iminodiacetyl-based hydroxamate-benzenesulfonamide conjugates.
Journal: Journal of medicinal chemistry 20081225
Title: Synthesis of biologically active N-methyl derivatives of amidines and cyclized five-membered products of amidines with oxalyl chloride.
Journal: European journal of medicinal chemistry 20081201
Title: Recent improvements in the development of A(2B) adenosine receptor agonists.
Journal: Purinergic signalling 20081201
Title: Effect of the oral absorption of benzenesulfonanilide-type cyclooxygenase-1 inhibitors on analgesic action and gastric ulcer formation.
Journal: Journal of pharmaceutical sciences 20081201
Title: N-(3,5-Dichloro-phen-yl)benzene-sulfonamide.
Journal: Acta crystallographica. Section E, Structure reports online 20081101
Title: External pH influences the transcriptional profile of the carbonic anhydrase, CAH-4b in Caenorhabditis elegans.
Journal: Molecular and biochemical parasitology 20081001
Title: Tetra-aquabis-(2-sulfamoylbenzoato)manganese(II).
Journal: Acta crystallographica. Section E, Structure reports online 20081001
Title: Residual ligand entropy in the binding of p-substituted benzenesulfonamide ligands to bovine carbonic anhydrase II.
Journal: Journal of the American Chemical Society 20080917
Title: Chromofluorescent indicator for intracellular Zn2+/Hg2+ dynamic exchange.
Journal: Organic letters 20080904
Title: Photophysical and complexation properties of benzenesulfonamide derivatives with different donor and acceptor moieties.
Journal: Journal of fluorescence 20080901
Title: Tetramethylcyclopropyl analogue of the leading antiepileptic drug, valproic acid: evaluation of the teratogenic effects of its amide derivatives in NMRI mice.
Journal: Birth defects research. Part A, Clinical and molecular teratology 20080901
Title: Chemometrical examination of active parameters and interactions in flow injection-capillary electrophoresis.
Journal: Electrophoresis 20080901
Title: Inhibition of human mitochondrial carbonic anhydrases VA and VB with para-(4-phenyltriazole-1-yl)-benzenesulfonamide derivatives.
Journal: Bioorganic & medicinal chemistry letters 20080815
Title: 2,2,2-Trimethyl-N-(phenyl-sulfon-yl)-acetamide.
Journal: Acta crystallographica. Section E, Structure reports online 20080801
Title: 2,2-Dichloro-N-(phenyl-sulfon-yl)-acetamide.
Journal: Acta crystallographica. Section E, Structure reports online 20080801
Title: Affinity-labeling-based introduction of a reactive handle for natural protein modification.
Journal: Chemistry, an Asian journal 20080707
Title: Carbonic anhydrase inhibitors: design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes.
Journal: Bioorganic & medicinal chemistry letters 20080615
Title: Exploration of physicochemical properties and molecular modelling studies of 2-sulfonyl-phenyl-3-phenyl-indole analogs as cyclooxygenase-2 inhibitors.
Journal: European journal of medicinal chemistry 20080601
Title: Similar sulfonamides with different crystal structures: sulfasymazine and sulfatriazine.
Journal: Acta crystallographica. Section C, Crystal structure communications 20080601
Title: Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20080501
Title: 2-[N-(X-chlorophenyl)carbamoyl]benzenesulfonamide (with X = 2 and 4).
Journal: Acta crystallographica. Section C, Crystal structure communications 20080501
Title: Functional human 5-HT6 receptor assay for high throughput screening of chemical ligands and binding proteins.
Journal: Combinatorial chemistry & high throughput screening 20080501
Title: Behaviour and biodegradation of sulfonamides (p-TSA, o-TSA, BSA) during drinking water treatment.
Journal: Chemosphere 20080401
Title: Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry 20080401
Title: Design and synthesis of N-(3,5-difluoro-4-hydroxyphenyl)benzenesulfonamides as aldose reductase inhibitors.
Journal: Bioorganic & medicinal chemistry 20080401
Title: Electrophysiological characterization of a novel Kv channel blocker N,N'-[oxybis(2,1-ethanediyloxy-2,1-ethanediyl) ]bis(4-methyl)-benzenesulfonamide found in virtual screening.
Journal: Acta pharmacologica Sinica 20080401
Title: Ethyl 2-(bromo-meth-yl)-5-meth-oxy-1-phenyl-sulfonyl-1H-indole-3-carboxyl-ate.
Journal: Acta crystallographica. Section E, Structure reports online 20080401
Title: Identification and significance of sulphonamides (p-TSA, o-TSA, BSA) in an urban water cycle (Berlin, Germany).
Journal: Water research 20080301
Title: Selective COX-2 inhibitors. Part 2: synthesis and biological evaluation of 4-benzylideneamino- and 4-phenyliminomethyl-benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry 20080301
Title: Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes.
Journal: Purinergic signalling 20080301
Title: Synthesis and cyclooxygenase inhibitory activities of linear 1-(methanesulfonylphenyl or benzenesulfonamido)-2-(pyridyl)acetylene regioisomers.
Journal: Bioorganic & medicinal chemistry 20080215
Title: Benzenesulfonamide indole inhibitors of cytosolic phospholipase A2alpha: optimization of in vitro potency and rat pharmacokinetics for oral efficacy.
Journal: Bioorganic & medicinal chemistry 20080201
Title: Metal-based sulfonamides: their preparation, characterization and in-vitro antibacterial, antifungal & cytotoxic properties. X-ray structure of 4-[(2-hydroxybenzylidene) amino] benzenesulfonamide.
Journal: Journal of enzyme inhibition and medicinal chemistry 20080201
Title: Ethyl 2-[(phenyl-sulfan-yl)meth-yl]-1-(phenyl-sulfon-yl)-1H-indole-3-carboxyl-ate.
Journal: Acta crystallographica. Section E, Structure reports online 20080201
Title: (2-Methyl-1-phenyl-sulfonyl-1H-indol-3-yl)methanol.
Journal: Acta crystallographica. Section E, Structure reports online 20080201
Title: Carbonic anhydrase inhibitors: copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII.
Journal: Bioorganic & medicinal chemistry letters 20080115
Title: New celecoxib derivatives as anti-inflammatory agents.
Journal: Journal of medicinal chemistry 20080110
Title: Identification of N-(quinolin-8-yl)benzenesulfonamides as agents capable of down-regulating NFkappaB activity within two separate high-throughput screens of NFkappaB activation.
Journal: Bioorganic & medicinal chemistry letters 20080101
Title: An efficient solvent-free synthesis of benzoxanthenes catalyzed by BSA or O-TSA.
Journal: Preparative biochemistry & biotechnology 20080101
Title: Antimicrobial activity of some sulfonamide derivatives on clinical isolates of Staphylococus aureus.
Journal: Annals of clinical microbiology and antimicrobials 20080101
Title: Binding modes of two novel non-nucleoside reverse transcriptase inhibitors, YM-215389 and YM-228855, to HIV type-1 reverse transcriptase.
Journal: Antiviral chemistry & chemotherapy 20080101
Title: Small molecule inhibitors of integrin alpha2beta1.
Journal: Journal of medicinal chemistry 20071101
Title: A remarkable accelerating effect of Ag-salt on intramolecular cyclization of o-(1-alkynyl)benzenesulfonamides.
Journal: The Journal of organic chemistry 20071026
Title: A strategy for designing 'multi-prong' enzyme inhibitors by incorporating selective ligands to the liposomal surface.
Journal: Chemical communications (Cambridge, England) 20070828
Title: Design, synthesis and pharmacological evaluation of 4-[2-alkylthio-5(4)-(4-substitutedphenyl)imidazole-4(5)yl]benzenesulfonamides as selective COX-2 inhibitors.
Journal: Acta pharmacologica Sinica 20070801
Title: Quantitative determination of three sulfonamides in environmental water samples using liquid chromatography coupled to electrospray tandem mass spectrometry.
Journal: Journal of chromatography. A 20070720
Title: Structure-based design of 2-arylamino-4-cyclohexylmethoxy-5-nitroso-6-aminopyrimidine inhibitors of cyclin-dependent kinase 2.
Journal: Organic & biomolecular chemistry 20070521
Title: Structural analysis of charge discrimination in the binding of inhibitors to human carbonic anhydrases I and II.
Journal: Journal of the American Chemical Society 20070502
Title: Pharmacophoric 2-hydroxyalkyl benzenesulfonamide: a single-step synthesis from benzenesulfonamide via hemiaminal.
Journal: European journal of medicinal chemistry 20070401
Title: Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties.
Journal: Bioorganic & medicinal chemistry letters 20070315
Title: Synthesis and in vivo evaluation of [18F]-4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide as a PET imaging probe for COX-2 expression.
Journal: Bioorganic & medicinal chemistry 20070215
Title: Dependence of effective molarity on linker length for an intramolecular protein-ligand system.
Journal: Journal of the American Chemical Society 20070207
Title: Thermodynamic parameters for the association of fluorinated benzenesulfonamides with bovine carbonic anhydrase II.
Journal: Chemistry, an Asian journal 20070108
Title: Strategies for controlled placement of nanoscale building blocks.
Journal: Nanoscale research letters 20070101
Title: Discovery of HIV-1 protease inhibitors with picomolar affinities incorporating N-aryl-oxazolidinone-5-carboxamides as novel P2 ligands.
Journal: Journal of medicinal chemistry 20061214
Title: Thiol-mediated anchoring of ligands to self-assembled monolayers for studies of biospecific interactions.
Journal: Langmuir : the ACS journal of surfaces and colloids 20061121
Title: Synthesis and in vitro antitumor evaluation of some indeno[1,2-c]pyrazol(in)es substituted with sulfonamide, sulfonylurea(-thiourea) pharmacophores, and some derived thiazole ring systems.
Journal: Bioorganic & medicinal chemistry 20061001
Title: Intracellular inhibition of carboxylesterases by benzil: modulation of CPT-11 cytotoxicity.
Journal: Molecular cancer therapeutics 20060901
Title: Binding of sulfonyl-containing arylalkylamines at human 5-HT6 serotonin receptors.
Journal: Journal of medicinal chemistry 20060824
Title: Urotensin-II blockade with SB-611812 attenuates cardiac dysfunction in a rat model of coronary artery ligation.
Journal: Journal of molecular and cellular cardiology 20060801
Title: Sorption-desorption of flucarbazone and propoxycarbazone and their benzenesulfonamide and triazolinone metabolites in two soils.
Journal: Pest management science 20060701
Title: Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori.
Journal: Bioorganic & medicinal chemistry letters 20060415
Title: Molecular structure and conformations of benzenesulfonamide: gas electron diffraction and quantum chemical calculations.
Journal: The Journal of organic chemistry 20060414
Title: Benzoxazole benzenesulfonamides are novel allosteric inhibitors of fructose-1,6-bisphosphatase with a distinct binding mode.
Journal: Bioorganic & medicinal chemistry letters 20060401
Title: Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.
Journal: Journal of medicinal chemistry 20060323
Title: Ultrahigh resolution crystal structures of human carbonic anhydrases I and II complexed with 'two-prong' inhibitors reveal the molecular basis of high affinity.
Journal: Journal of the American Chemical Society 20060308
Title: Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II 'selective' inhibitor celecoxib.
Journal: Bioorganic & medicinal chemistry letters 20060115
Title: Downregulation of survivin expression and concomitant induction of apoptosis by celecoxib and its non-cyclooxygenase-2-inhibitory analog, dimethyl-celecoxib (DMC), in tumor cells in vitro and in vivo.
Journal: Molecular cancer 20060101
Title: Short communication inhibitory activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene)amino]-N-(4,6-dimethylpyrimidin-2-yl) benzenesulphonamide and its derivatives against orthopoxvirus replication in vitro.
Journal: Antiviral chemistry & chemotherapy 20060101
Title: CC 05, a novel anti-inflammatory compound, exerts its effect by inhibition of cyclooxygenase-2 activity.
Journal: European journal of pharmacology 20050927
Title: QSAR analysis of thiazole benzenesulfonamide substituted 3-pyridylethanolamines as beta3-adrenergic receptor agonist.
Journal: Bioorganic & medicinal chemistry letters 20050615
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes.
Journal: Bioorganic & medicinal chemistry letters 20050615
Title: Synthesis and biological evaluation of 3,4-diphenyl-1,2,5-oxadiazole-2-oxides and 3,4-diphenyl-1,2,5-oxadiazoles as potential hybrid COX-2 inhibitor/nitric oxide donor agents.
Journal: Bioorganic & medicinal chemistry 20050415
Title: Design, synthesis, and biological evaluation of N-acetyl-2-carboxybenzenesulfonamides: a novel class of cyclooxygenase-2 (COX-2) inhibitors.
Journal: Bioorganic & medicinal chemistry 20050401
Title: Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II.
Journal: Bioorganic & medicinal chemistry letters 20050401
Title: Benzenesulfonamide analogs of fluoroquinolones. Antibacterial activity and QSAR studies.
Journal: European journal of medicinal chemistry 20050401
Title: Discovery and selection of TMC114, a next generation HIV-1 protease inhibitor.
Journal: Journal of medicinal chemistry 20050324
Title: Spacer-based selectivity in the binding of 'two-prong' ligands to recombinant human carbonic anhydrase I.
Journal: Biochemistry 20050308
Title: Studies of non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: synthesis and structure-activity relationships of 2-cyano and 2-hydroxy thiazolidenebenzenesulfonamide derivatives.
Journal: Bioorganic & medicinal chemistry 20050215
Title: QSAR studies on benzene sulfonamide carbonic anhydrase inhibitors: need of hydrophobic parameter for topological modeling of binding constants of sulfonamides to human CA-II.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Novel use of chemical shift in NMR as molecular descriptor: a first report on modeling carbonic anhydrase inhibitory activity and related parameters.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Characterization of beta3-adrenergic receptor: determination of pharmacophore and 3D QSAR model for beta3 adrenergic receptor agonism.
Journal: Journal of computer-aided molecular design 20050201
Title: Predictive flip regression: a technique for QSAR of derivatives of symmetric molecules.
Journal: Journal of chemical information and modeling 20050101
Title: In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II.
Journal: Angewandte Chemie (International ed. in English) 20041217
Title: Studies of nonnucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Design and synthesis of thiazolidenebenzenesulfonamides.
Journal: Bioorganic & medicinal chemistry 20041201
Title: Pharmacomodulation of a sulfamide 5-HT6 receptor ligand.
Journal: Journal of enzyme inhibition and medicinal chemistry 20041201
Title: Topological modeling of lipophilicity, diuretic activity, and carbonic inhibition activity of benzene sulfonamides: a molecular connectivity approach.
Journal: Bioorganic & medicinal chemistry letters 20041115
Title: Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives.
Journal: Bioorganic & medicinal chemistry letters 20041115
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.
Journal: Bioorganic & medicinal chemistry letters 20041101
Title: Two-prong inhibitors for human carbonic anhydrase II.
Journal: Journal of the American Chemical Society 20041020
Title: Novel synthesis of 3,4-diarylisoxazole analogues of valdecoxib: reversal cyclooxygenase-2 selectivity by sulfonamide group removal.
Journal: Journal of medicinal chemistry 20040923
Title: Protein surface-assisted enhancement in the binding affinity of an inhibitor for recombinant human carbonic anhydrase-II.
Journal: Journal of the American Chemical Society 20040908
Title: Synthesis and antiviral activity of P1' arylsulfonamide azacyclic urea HIV protease inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20040802
Title: Synthesis, antiviral, and anti-HIV-1 integrase activities of 3-aroyl-1,1-dioxo-1,4,2-benzodithiazines.
Journal: Bioorganic & medicinal chemistry 20040701
Title: Rewiring cell adhesion.
Journal: Journal of the American Chemical Society 20040602
Title: A versatile polypeptide platform for integrated recognition and reporting: affinity arrays for protein-ligand interaction analysis.
Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20040517
Title: New heteroarylbenzenesulphonamides as matrix metalloproteinase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20040308
Title: Abeta aggregation inhibitors. Part 1: Synthesis and biological activity of phenylazo benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20040308
Title: QSAR study on benzenesulphonamide carbonic anhydrase inhibitors: topological approach using Balaban index.
Journal: Bioorganic & medicinal chemistry 20040215
Title: Polar substitutions in the benzenesulfonamide ring of celecoxib afford a potent 1,5-diarylpyrazole class of COX-2 inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20040119
Title: Application of CoMFA and CoMSIA 3D-QSAR and docking studies in optimization of mercaptobenzenesulfonamides as HIV-1 integrase inhibitors.
Journal: Journal of medicinal chemistry 20040115
Title: QSAR study using topological indices for inhibition of carbonic anhydrase II by sulfanilamides and Schiff bases.
Journal: Molecular diversity 20040101
Title: Synthesis and cyclooxygenase-2 inhibiting property of 1,5-diarylpyrazoles with substituted benzenesulfonamide moiety as pharmacophore: Preparation of sodium salt for injectable formulation.
Journal: Journal of medicinal chemistry 20030911
Title: Sorption-desorption of two 'aged' sulfonylaminocarbonyltriazolinone herbicide metabolites in soil.
Journal: Journal of agricultural and food chemistry 20030604
Title: Synthesis of 1-(6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)semi-carbazides and their transformation into 4-chloro-2-mercapto-N-(4,5-dihydro-5-oxo-4-phenyl-1H-1,2,4-triazol-3-yl)benzenesulfonamides as potential anticancer and anti-HIV agents.
Journal: Farmaco (Societa chimica italiana : 1989) 20030601
Title: Valdecoxib-induced toxic epidermal necrolysis in a patient allergic to sulfa drugs.
Journal: Pharmacotherapy 20030401
Title: Tripodal ligand incorporating dual fluorescent ionophore: a coordinative control of photoinduced electron transfer.
Journal: Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology 20030301
Title: Synthesis of heteroaromatic analogues of (2-aryl-1-cyclopentenyl-1-alkylidene)-(arylmethyloxy)amine COX-2 inhibitors: effects on the inhibitory activity of the replacement of the cyclopentene central core with pyrazole, thiophene or isoxazole ring.
Journal: European journal of medicinal chemistry 20030201
Title: Using cyclooxygenase-2 inhibitors as molecular platforms to develop a new class of apoptosis-inducing agents.
Journal: Journal of the National Cancer Institute 20021204
Title: Diversity in the oxidation of substrates by cytochrome P450 2D6: lack of an obligatory role of aspartate 301-substrate electrostatic bonding.
Journal: Biochemistry 20020910
Title: An excretion balance and pharmacokinetic study of the novel anticancer agent E7070 in cancer patients.
Journal: Anti-cancer drugs 20020901
Title: The pharmacokinetics of a thiazole benzenesulfonamide beta 3-adrenergic receptor agonist and its analogs in rats, dogs, and monkeys: improving oral bioavailability.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20020701
Title: Metabolism of a thiazole benzenesulfonamide derivative, a potent and elective agonist of the human beta3-adrenergic receptor, in rats: identification of a novel isethionic acid conjugate.
Journal: Drug metabolism and disposition: the biological fate of chemicals 20020701
Title: Effects of soil pH and soil water content on prosulfuron dissipation.
Journal: Journal of agricultural and food chemistry 20020522
Title: Enantiomeric separation of a thiazolbenzenesulfonamide compound using packed-column subcritical fluid chromatography.
Journal: Chirality 20020515
Title: Synthesis of unsymmetrical aroyl acyl imides by aminocarbonylation of aryl bromides.
Journal: The Journal of organic chemistry 20020125
Title: Rational determination of transfer free energies of small drugs across the water-oil interface.
Journal: Journal of medicinal chemistry 20020103
Title: Synthesis, characterization and antifungal activities of some benzenesulphonylamino acid derivatives.
Journal: Bollettino chimico farmaceutico 20020101
Title: Synthesis and anti-HIV activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene) amino]-N(4,6-dimethyl-2-pyrimidinyl)-benzene sulfonamide and its derivatives.
Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20011201
Title: Comparative study of new benzenesulphonamide fluoroquinolones structurally related to ciprofloxacin against selected ciprofloxacin-susceptible and -resistant Gram-positive cocci.
Journal: The Journal of antimicrobial chemotherapy 20011101
Title: Subtle differences in dissociation rates of interactions between destabilized human carbonic anhydrase II mutants and immobilized benzenesulfonamide inhibitors probed by a surface plasmon resonance biosensor.
Journal: Analytical biochemistry 20010915
Title: Two isomorphous benzenesulfonamide crystal structures determined by intermolecular C-H...O, C-H...pi and C-H...Cl interactions.
Journal: Acta crystallographica. Section C, Crystal structure communications 20010901
Title: Synthesis of optically active N-(2-pyridyloxiran-2-ylmethyl) benzenesulfonamide derivatives and their herbicidal activity.
Journal: Bioscience, biotechnology, and biochemistry 20010701
Title: Ethenesulfonamide derivatives, a novel class of orally active endothelin-A receptor antagonists.
Journal: Chemical & pharmaceutical bulletin 20010501
Title: QSAR of antineoplastics IV: Hansch analysis of N-(7-indolyl)benzenesulfonamides against KB human nasopharynx carcinoma, colon 38 murine adenocarcinoma and P388 murine leukemia cell lines.
Journal: Drug design and discovery 20010101
Title: QSAR of antineoplastics V: Exploration of receptor interaction sites of antitumor N-(7-indolyl)benzenesulfonamides targeting GI phase using electrotopological state atom index.
Journal: Drug design and discovery 20010101
Title: Design and synthesis of benzoic acid derivatives as influenza neuraminidase inhibitors using structure-based drug design.
Journal: Journal of medicinal chemistry 19971205
