Title: Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
Journal: Bioorganic & medicinal chemistry 20121115
Title: Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Journal: Bioorganic & medicinal chemistry letters 20101101
Title: Synthesis and anticancer activity of chromone-based analogs of lavendustin A.
Journal: European journal of medicinal chemistry 20100901
Title: A rapid synthesis of lavendustin-mimetic small molecules by click fragment assembly.
Journal: Bioorganic & medicinal chemistry letters 20100701
Title: Brain-derived neurotrophic factor controls cannabinoid CB1 receptor function in the striatum.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20100616
Title: Genistein directly inhibits native and recombinant NMDA receptors.
Journal: Neuropharmacology 20100601
Title: Modulation of AMPA excitatory postsynaptic currents in the spinal cord dorsal horn neurons by insulin.
Journal: Neuroscience 20100310
Title: Protein tyrosine kinase involvement in learning-produced changes in Hermissenda type B photoreceptors.
Journal: Journal of neurophysiology 20091201
Title: Tyrosine kinase-independent inhibition by genistein on spermatogenic T-type calcium channels attenuates mouse sperm motility and acrosome reaction.
Journal: Cell calcium 20090201
Title: Structure-activity relationship studies on a novel class of antiproliferative agents derived from Lavendustin A. Part I: Ring A modifications.
Journal: Bioorganic & medicinal chemistry 20080815
Title: Influence of the tyrosine kinase inhibitors STI571 (Glivec), lavendustin A and genistein on human mast cell line (HMC-1(560)) activation.
Journal: Journal of cellular biochemistry 20080301
Title: A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Journal: Proceedings of the National Academy of Sciences of the United States of America 20071218
Title: Effects of monocarboxylic acid-derived Cl- channel blockers on depolarization-activated potassium currents in rat ventricular myocytes.
Journal: Experimental physiology 20070501
Title: Synthesis and anticancer activity of lavendustin A derivatives containing arylethenylchromone substituents.
Journal: European journal of medicinal chemistry 20060801
Title: Cytotoxicity of organic compounds against ovarian cancer cells: a quantitative structure-activity relationship study.
Journal: Molecular pharmaceutics 20060101
Title: Phytoestrogen action in Leydig cells of Biłgoraj ganders (Anser anser).
Journal: Reproductive biology 20060101
Title: Tyrosine phosphorylation of the N-methyl-D-aspartate receptor is enhanced in synaptic membrane fractions of the adult rat hippocampus.
Journal: Brain research. Molecular brain research 20051207
Title: Regulatory and necrotic volume increase in boar spermatozoa.
Journal: Journal of cellular physiology 20050801
Title: Protective effect of a protein kinase inhibitor on cellular injury induced by cephaloridine in the porcine kidney cell line LLC-PK(1).
Journal: The Journal of toxicological sciences 20050801
Title: IP3 production in the hypersensitive response of lemon seedlings against Alternaria alternata involves active protein tyrosine kinases but not a G-protein.
Journal: Biological research 20050101
Title: 4-Anilinoquinazolines with Lavendustin A subunit as inhibitors of epidermal growth factor receptor tyrosine kinase: syntheses, chemical and pharmacological properties.
Journal: European journal of medicinal chemistry 20041201
Title: A unique mechanism for cyclic adenosine 3',5'-monophosphate-induced increase of 32-kDa tyrosine-phosphorylated protein in boar spermatozoa.
Journal: Molecular reproduction and development 20041001
Title: Activation of phospholipase D induced by hydrogen peroxide in suspension-cultured rice cells.
Journal: Plant & cell physiology 20040901
Title: Correlation between semaphorin3A-induced facilitation of axonal transport and local activation of a translation initiation factor eukaryotic translation initiation factor 4E.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20040707
Title: Ceramide inhibits L-type calcium channel currents in GH3 cells.
Journal: Molecular and cellular endocrinology 20040415
Title: Evidence that activation of Src family kinase is not required for fertilization-associated [Ca2+]i oscillations in mouse eggs.
Journal: Reproduction (Cambridge, England) 20040401
Title: Lavendustin A enhances axon elongation in VHL gene-transfected neural stem cells.
Journal: Neuroreport 20040322
Title: Role of tyrosine kinase in desflurane-induced preconditioning.
Journal: Anesthesiology 20040301
Title: The efficacy of tyrosine kinase inhibitors on human pancreatic cancer cell lines.
Journal: The Journal of surgical research 20031201
Title: Involvement of spinal tyrosine kinase in inflammatory and N-methyl-D-aspartate-induced hyperalgesia in rats.
Journal: European journal of pharmacology 20030516
Title: Synthesis, anticancer activity, and inhibition of tubulin polymerization by conformationally restricted analogues of lavendustin A.
Journal: Journal of medicinal chemistry 20030424
Title: Evidence for a role of protein tyrosine kinases in cell death induced by gp120 in CHP100 neuroblastoma cells.
Journal: Toxicology letters 20030404
Title: Intracellular signaling involved in macrophage adhesion and FBGC formation as mediated by ligand-substrate interaction.
Journal: Journal of biomedical materials research 20021215
Title: Synthesis and investigation of conformationally restricted analogues of lavendustin A as cytotoxic inhibitors of tubulin polymerization.
Journal: Journal of medicinal chemistry 20021010
Title: Neonatal exposure to genistein induces estrogen receptor (ER)alpha expression and multioocyte follicles in the maturing mouse ovary: evidence for ERbeta-mediated and nonestrogenic actions.
Journal: Biology of reproduction 20021001
Title: Genistein inhibits cardiac L-type Ca(2+) channel activity by a tyrosine kinase-independent mechanism.
Journal: Molecular pharmacology 20020901
Title: Role of Src protein tyrosine kinases in late preconditioning against myocardial infarction.
Journal: American journal of physiology. Heart and circulatory physiology 20020801
Title: Identification of myo-inositol 1,2-cyclic monophosphate by electrospray tandem mass spectrometry, a major constituent of EGF-stimulated phosphoinositide turnover in MDA 468 cells.
Journal: Experimental cell research 20020715
Title: Direct inhibition of the cloned Kv1.5 channel by AG-1478, a tyrosine kinase inhibitor.
Journal: American journal of physiology. Cell physiology 20020601
Title: Regulation of an ERG K+ current by Src tyrosine kinase.
Journal: The Journal of biological chemistry 20020419
Title: Phosphorylation of the salivary Na(+)-K(+)-2Cl(-) cotransporter.
Journal: American journal of physiology. Cell physiology 20020401
Title: Acute and chronic effects of genistein, tyrphostin and lavendustin A on steroid synthesis in luteinized human granulosa cells.
Journal: Human reproduction (Oxford, England) 20020301
Title: Trophic factor-induced excitatory synaptogenesis involves postsynaptic modulation of nicotinic acetylcholine receptors.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20020115
Title: Stimulation of cardiac glucose transport by inhibitors of oxidative phosphorylation.
Journal: Life sciences 20011005
Title: Stabilization of supersaturated solutions of a lipophilic drug for dermal delivery.
Journal: International journal of pharmaceutics 20010814
Title: Activation of the phosphatidylinositol 3-kinase-Akt/protein kinase B signaling pathway in arachidonic acid-stimulated human myeloid and endothelial cells: involvement of the ErbB receptor family.
Journal: The Journal of biological chemistry 20010720
Title: Modulation of excitability in Aplysia tail sensory neurons by tyrosine kinases.
Journal: Journal of neurophysiology 20010601
Title: Activation of store-operated Ca2+ entry in RBL cells without the contribution of protein kinases.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20010601
Title: Protein tyrosine kinase inhibitors alter human dopamine transporter activity in Xenopus oocytes.
Journal: The Journal of pharmacology and experimental therapeutics 20010301
Title: PC12 cells utilize the homophilic binding site of L1 for cell-cell adhesion but L1-alphavbeta3 interaction for neurite outgrowth.
Journal: Journal of neurochemistry 20010301
Title: Thapsigargin inhibits angiogenesis in the rat isolated aorta: studies on the role of intracellular calcium pools.
Journal: Cardiovascular research 20010216
Title: Design, synthesis, and biological evaluation of a series of lavendustin A analogues that inhibit EGFR and Syk tyrosine kinases, as well as tubulin polymerization.
Journal: Journal of medicinal chemistry 20010201
Title: Direct inhibition of the hexose transporter GLUT1 by tyrosine kinase inhibitors.
Journal: Biochemistry 20010123
Title: Study of cytoskeletal changes induced by okadaic acid in BE(2)-M17 cells by means of a quantitative fluorimetric microplate assay.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20010101
Title: Signal transduction-mediated activation of the aryl hydrocarbon receptor in rat hepatoma H4IIE cells.
Journal: The Journal of biological chemistry 19971212
Title: Identification of a second region upstream of the mouse heme oxygenase-1 gene that functions as a basal level and inducer-dependent transcription enhancer.
Journal: The Journal of biological chemistry 19950519
Title: Effect of various protein kinase inhibitors on the induction of milk protein gene expression by prolactin.
Journal: Molecular and cellular endocrinology 19930301
Title: Onoda T, et al. Isolation of a novel tyrosine kinase inhibitor, lavendustin A, from Streptomyces griseolavendus. J Nat Prod. 1989 Nov-Dec;52(6):1252-7.
Title: Hu DE, et al. Suppression of VEGF-induced angiogenesis by the protein tyrosine kinase inhibitor, lavendustin A. Br J Pharmacol. 1995 Jan;114(2):262-8.
Title: Gubellini P, et al. Endogenous neurotrophins are required for the induction of GABAergic long-term potentiation in the neonatal rat hippocampus. J Neurosci. 2005 Jun 15;25(24):5796-802.