Title: Selective fluorescent nonpeptidic antagonists for vasopressin V₂ GPCR: application to ligand screening and oligomerization assays.
Journal: Journal of medicinal chemistry 20121025
Title: V2 vasopressin receptor (V2R) mutations in partial nephrogenic diabetes insipidus highlight protean agonism of V2R antagonists.
Journal: The Journal of biological chemistry 20120113
Title: Vasopressin receptor antagonists and their role in clinical medicine.
Journal: Indian journal of endocrinology and metabolism 20120101
Title: [Hyponatremic hypervolemia in heart failure--the hot spot for vasopressin receptor antagonists?].
Journal: Wiadomosci lekarskie (Warsaw, Poland : 1960) 20120101
Title: Vasotocin- and mesotocin-induced increases in short-circuit current across tree frog skin.
Journal: Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20110201
Title: Clinical implication of the antidiuretic hormone (ADH) receptor antagonist mozavaptan hydrochloride in patients with ectopic ADH syndrome.
Journal: Japanese journal of clinical oncology 20110101
Title: [Vasopressin receptor antagonists: the vaptans].
Journal: Endocrinologia y nutricion : organo de la Sociedad Espanola de Endocrinologia y Nutricion 20100501
Title: Effects of arginine vasotocin and mesotocin on the activation and development of amiloride-blockable short-circuit current across larval, adult, and cultured larval bullfrog skins.
Journal: Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20100301
Title: Bumetanide-induced enlargement of the rat intrastrial space and effects of a vasopressin type 2 antagonist.
Journal: ORL; journal for oto-rhino-laryngology and its related specialties 20100101
Title: Time course changes of vasopressin-induced enlargement of the rat intrastrial space and the effects of a vasopressin type 2 antagonist.
Journal: Acta oto-laryngologica 20090701
Title: Normotensive sodium loading in conscious dogs: regulation of renin secretion during beta-receptor blockade.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20090201
Title: Role of vasopressin antagonists.
Journal: Clinical journal of the American Society of Nephrology : CJASN 20080701
Title: Effects of hypertonic stimuli and arginine vasotocin (AVT) on water absorption response in Japanese treefrog, Hyla japonica.
Journal: General and comparative endocrinology 20080601
Title: Effects of arginine vasotocin and vasopressin receptor antagonists on Na+ and Cl- transport in the isolated skin of two frog species, Hyla japonica and Rana nigromaculata.
Journal: General and comparative endocrinology 20080515
Title: Inhibitory effect of vasopressin receptor antagonist OPC-31260 on experimental brain oedema induced by global cerebral ischaemia.
Journal: Acta neurochirurgica 20080301
Title: Prevention of hypoxic brain oedema by the administration of vasopressin receptor antagonist OPC-31260.
Journal: Progress in brain research 20080101
Title: Vasopressin-induced nitric oxide production in rat inner medullary collecting duct is dependent on V2 receptor activation of the phosphoinositide pathway.
Journal: American journal of physiology. Renal physiology 20070801
Title: Biological half-life and organ distribution of [3H]8-arginine vasopressin following administration of vasopressin receptor antagonist OPC-31260.
Journal: Regulatory peptides 20070607
Title: Lithium effectively complements vasopressin V2 receptor antagonist in the treatment of hyponatraemia of SIADH rats.
Journal: Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 20070101
Title: Regulation of UT-A1-mediated transepithelial urea flux in MDCK cells.
Journal: American journal of physiology. Cell physiology 20061001
Title: Hyponatremia in cirrhosis: clinical features and management.
Journal: Gastroenterologie clinique et biologique 20061001
Title: Vasopressin antagonists as aquaretic agents for the treatment of hyponatremia.
Journal: The American journal of medicine 20060701
Title: Molecular analysis of impaired urinary diluting capacity in glucocorticoid deficiency.
Journal: American journal of physiology. Renal physiology 20060501
Title: Effects of long-term oral treatment with selective vasopressin V2 receptor antagonist (OPC-31260) on adriamycin-induced heart failure in rats.
Journal: International journal of cardiology 20060404
Title: [Renal action of vasopressin].
Journal: Nihon rinsho. Japanese journal of clinical medicine 20060201
Title: BSC1 inhibition complements effects of vasopressin V2 receptor antagonist on hyponatremia in SIADH rats.
Journal: Kidney international 20050501
Title: Effectiveness of vasopressin V2 receptor antagonists OPC-31260 and OPC-41061 on polycystic kidney disease development in the PCK rat.
Journal: Journal of the American Society of Nephrology : JASN 20050401
Title: 2,5-disubstituted 3,4-dihydro-2H-benzo[b][1,4]thiazepines as potent and selective V2 arginine vasopressin receptor antagonists.
Journal: Bioorganic & medicinal chemistry letters 20031117
Title: Therapeutic role of vasopressin receptor antagonism in patients with liver cirrhosis.
Journal: Clinical science (London, England : 1979) 20030701
Title: Gateways to clinical trials.
Journal: Methods and findings in experimental and clinical pharmacology 20030601
Title: Ameliorative effect of NC-1900, a new AVP4-9 analog, through vasopressin V1A receptor on scopolamine-induced impairments of spatial memory in the eight-arm radial maze.
Journal: Neuropharmacology 20030301
Title: Combined effects of vasopressin V2 receptor antagonist and loop diuretic in humans.
Journal: Clinical nephrology 20030301
Title: Vasopressin V(1) receptor-mediated activation of central sympatho-adrenomedullary outflow in rats.
Journal: European journal of pharmacology 20021213
Title: Adaptation to sustained high plasma vasopressin in water and electrolyte homeostasis in the rat transgenic for the metallothionein-vasopressin fusion gene.
Journal: The Journal of endocrinology 20020401
Title: Losartan treatment normalizes renal sodium and water handling in rats with mild congestive heart failure.
Journal: American journal of physiology. Renal physiology 20020201
Title: Role of sodium depletion in acute antidiuretic effect of bendroflumethiazide in rats with nephrogenic diabetes insipidus.
Journal: The Journal of pharmacology and experimental therapeutics 20011001
Title: Ameliorative effect of vasopressin-(4-9) through vasopressin V(1A) receptor on scopolamine-induced impairments of rat spatial memory in the eight-arm radial maze.
Journal: European journal of pharmacology 20010907
Title: Vascular and renal effects of vasopressin and its antagonists in conscious rats with chronic myocardial infarction; evidence for receptor shift.
Journal: European journal of pharmacology 20010706
Title: Pharmacological characterization of the human vasopressin receptor subtypes stably expressed in Chinese hamster ovary cells.
Journal: British journal of pharmacology 19981201
Title: 5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors.
Journal: Journal of medicinal chemistry 19980702
Title: The human V3 pituitary vasopressin receptor: ligand binding profile and density-dependent signaling pathways.
Journal: Endocrinology 19971001
Title: Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist.
Journal: The Journal of clinical investigation 19961215
Title: Characterization of a novel aquaretic agent, OPC-31260, as an orally effective, nonpeptide vasopressin V2 receptor antagonist.
Journal: British journal of pharmacology 19920401
Title: Yamamura Y, et al. Characterization of a novel aquaretic agent, OPC-31260, as an orally effective, nonpeptide vasopressin V2 receptor antagonist. Br J Pharmacol. 1992 Apr;105(4):787-91.
Title: Yamaguchi K, et al. Clinical implication of the antidiuretic hormone (ADH) receptor antagonist mozavaptan hydrochloride in patients with ectopic ADH syndrome. Jpn J Clin Oncol. 2011 Jan;41(1):148-52.
