Title: Identification of potent Yes1 kinase inhibitors using a library screening approach.
Journal: Bioorganic & medicinal chemistry letters 20130801
Title: Serotonin-induced brain glycogenolysis in rainbow trout (Oncorhynchus mykiss).
Journal: The Journal of experimental biology 20120901
Title: Diverse effects of 5-HT2C receptor blocking agents on c-Fos expression in the rat basal ganglia.
Journal: European journal of pharmacology 20120815
Title: Paroxetine-induced reduction of sexual incentive motivation in female rats is not modified by 5-HT1B or 5-HT2C antagonists.
Journal: Psychopharmacology 20120301
Title: A novel mechanism for regulating hepatic glycogen synthesis involving serotonin and cyclin-dependent kinase-5.
Journal: Diabetes 20120101
Title: SB 206553, a putative 5-HT2C inverse agonist, attenuates methamphetamine-seeking in rats.
Journal: BMC neuroscience 20120101
Title: Discovery and development of α7 nicotinic acetylcholine receptor modulators.
Journal: Journal of medicinal chemistry 20111208
Title: Pulmonary vascular effects of serotonin and selective serotonin reuptake inhibitors in the late-gestation ovine fetus.
Journal: American journal of physiology. Lung cellular and molecular physiology 20111201
Title: Participation of cyclooxygenase pathway in the vasoconstriction induced by 5-HT in the in situ autoperfused kidney of long-term diabetic rats.
Journal: European journal of pharmacology 20110520
Title: Blockade of 5-HT(2A) and/or 5-HT(2C) receptors modulates sevoflurane-induced immobility.
Journal: Journal of anesthesia 20110401
Title: Serotonin 2A and 2B receptor-induced phrenic motor facilitation: differential requirement for spinal NADPH oxidase activity.
Journal: Neuroscience 20110331
Title: Serotonin receptor 5-HT2B mediates serotonin-induced mechanical hyperalgesia.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20110126
Title: Differences between human wild-type and C23S variant 5-HT2C receptors in inverse agonist-induced resensitization.
Journal: Pharmacological reports : PR 20110101
Title: Locomotion after spinal cord injury depends on constitutive activity in serotonin receptors.
Journal: Journal of neurophysiology 20101201
Title: Development, validation, and use of quantitative structure-activity relationship models of 5-hydroxytryptamine (2B) receptor ligands to identify novel receptor binders and putative valvulopathic compounds among common drugs.
Journal: Journal of medicinal chemistry 20101111
Title: Constitutive activity of serotonin 2C receptors at G protein-independent signaling: modulation by RNA editing and antidepressants.
Journal: Molecular pharmacology 20101101
Title: The central serotonin 2B receptor: a new pharmacological target to modulate the mesoaccumbens dopaminergic pathway activity.
Journal: Journal of neurochemistry 20100901
Title: The serotonin 2C receptor potently modulates the head-twitch response in mice induced by a phenethylamine hallucinogen.
Journal: Psychopharmacology 20100401
Title: Acquisition session length modulates consolidation effects produced by 5-HT2C ligands in a mouse autoshaping-operant procedure.
Journal: Behavioural pharmacology 20100301
Title: 5-HT2A receptor antagonists improve motor impairments in the MPTP mouse model of Parkinson's disease.
Journal: Neuropharmacology 20100101
Title: Mining biologically-active molecules for inhibitors of fatty acid amide hydrolase (FAAH): identification of phenmedipham and amperozide as FAAH inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20091201
Title: In vivo evidence that constitutive activity of serotonin2C receptors in the medial prefrontal cortex participates in the control of dopamine release in the rat nucleus accumbens: differential effects of inverse agonist versus antagonist.
Journal: Journal of neurochemistry 20091001
Title: Overexpression of 5-HT2C receptors in forebrain leads to elevated anxiety and hypoactivity.
Journal: The European journal of neuroscience 20090701
Title: Old and new pharmacology: positive allosteric modulation of the alpha7 nicotinic acetylcholine receptor by the 5-hydroxytryptamine(2B/C) receptor antagonist SB-206553 (3,5-dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b']di pyrrole-1(2H)-carboxamide).
Journal: The Journal of pharmacology and experimental therapeutics 20090301
Title: Modulation of striatal dopamine release by 5-HT2A and 5-HT2C receptor antagonists: [11C]raclopride PET studies in the rat.
Journal: Psychopharmacology 20081101
Title: Ontogeny of serotonin and serotonin2A receptors in rat auditory cortex.
Journal: Hearing research 20081001
Title: 5HT2 receptor activation facilitates P2X receptor mediated excitatory neurotransmission to cardiac vagal neurons in the nucleus ambiguus.
Journal: Neuropharmacology 20080601
Title: Inverse agonist and neutral antagonist actions of antidepressants at recombinant and native 5-hydroxytryptamine2C receptors: differential modulation of cell surface expression and signal transduction.
Journal: Molecular pharmacology 20080301
Title: Identification of a key amino acid of the human 5-HT(2B) serotonin receptor important for sarpogrelate binding.
Journal: Journal of pharmacological sciences 20070701
Title: WAY-163909 [(7bR,10aR)-1,2,3,4,8,9,10,10a-octahydro-7bH-cyclopenta-[b][1,4]diazepino[6,7,1hi]indole]: A novel 5-hydroxytryptamine 2C receptor-selective agonist with preclinical antipsychotic-like activity.
Journal: The Journal of pharmacology and experimental therapeutics 20070101
Title: Role of the 5-HT2C receptor in improving weight-supported stepping in adult rats spinalized as neonates.
Journal: Brain research 20060927
Title: 5-HT receptor subtypes involved in the anxiogenic-like action and associated Fos response of acute fluoxetine treatment in rats.
Journal: Psychopharmacology 20060401
Title: Clozapine and haloperidol differentially alter the constitutive activity of central serotonin2C receptors in vivo.
Journal: Biological psychiatry 20060315
Title: Role of 5-HT2A and 5-HT2C/B receptors in the acute effects of 3,4-methylenedioxymethamphetamine (MDMA) on striatal single-unit activity and locomotion in freely moving rats.
Journal: Psychopharmacology 20051001
Title: Behavioral tolerance to lysergic acid diethylamide is associated with reduced serotonin-2A receptor signaling in rat cortex.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050901
Title: Anxiolytic-like effect of milnacipran in the four-plate test in mice: mechanism of action.
Journal: Pharmacology, biochemistry, and behavior 20050701
Title: Serotonin (1A) receptor involvement in acute 3,4-methylenedioxymethamphetamine (MDMA) facilitation of social interaction in the rat.
Journal: Progress in neuro-psychopharmacology & biological psychiatry 20050601
Title: Modulation of dopamine release by striatal 5-HT2C receptors.
Journal: Synapse (New York, N.Y.) 20050315
Title: Partial 5-HT(1A) receptor agonist activity by the 5-HT(2C) receptor antagonist SB 206,553 is revealed in rats spinalized as neonates.
Journal: Experimental neurology 20050201
Title: The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo.
Journal: British journal of pharmacology 20041101
Title: Serotonin-GABA interactions modulate MDMA-induced mesolimbic dopamine release.
Journal: Journal of neurochemistry 20041101
Title: Mechanisms intrinsic to 5-HT2B receptor-induced potentiation of NMDA receptor responses in frog motoneurones.
Journal: British journal of pharmacology 20041001
Title: Involvement of the serotonin 5-HT2B receptor in cardiac hypertrophy linked to sympathetic stimulation: control of interleukin-6, interleukin-1beta, and tumor necrosis factor-alpha cytokine production by ventricular fibroblasts.
Journal: Circulation 20040824
Title: Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20040801
Title: Effect of estrogen on the lordosis-inhibiting action of ketanserin and SB 206553.
Journal: Behavioural brain research 20040604
Title: Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
Journal: Pharmacology 20040601
Title: Constitutive activity of the serotonin2C receptor inhibits in vivo dopamine release in the rat striatum and nucleus accumbens.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20040331
Title: In vivo evidence that 5-HT2C receptor antagonist but not agonist modulates cocaine-induced dopamine outflow in the rat nucleus accumbens and striatum.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040201
Title: Agomelatine(S 20098) antagonizes the penile erections induced by the stimulation of 5-HT2C receptors in Wistar rats.
Journal: Psychopharmacology 20031001
Title: Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
Journal: Behavioral neuroscience 20030401
Title: Anxiolytic-like effects of 5-HT2 ligands on three mouse models of anxiety.
Journal: Behavioural brain research 20030318
Title: Wistar-Kyoto rats are sensitive to the hypolocomotor and anxiogenic effects of mCPP.
Journal: Behavioural pharmacology 20030301
Title: Discriminative stimulus properties of 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane [(+/-)DOI] in C57BL/6J mice.
Journal: Psychopharmacology 20030201
Title: Conserved helix 7 tyrosine acts as a multistate conformational switch in the 5HT2C receptor. Identification of a novel 'locked-on' phenotype and double revertant mutations.
Journal: The Journal of biological chemistry 20020927
Title: Vasodilator and vasoconstrictor responses induced by 5-hydroxytryptamine in the in situ blood autoperfused hindquarters of the anaesthetized rat.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20020801
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: Attenuation of ischemic efflux of endogenous amino acids by the novel 5-HT(1A)/5-HT(2) receptor ligand adatanserin.
Journal: Neurochemistry international 20020301
Title: Pharmacological studies of the acute effects of (+)-3,4-methylenedioxymethamphetamine on locomotor activity: role of 5-HT(1B/1D) and 5-HT(2) receptors.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020101
Title: Effects of 5-HT(2) receptor antagonists on the anti-immobility effects of imipramine in the forced swimming test with mice.
Journal: European journal of pharmacology 20010921
Title: Role of 5-HT(2) receptor subtypes in depletion of 5-HT induced by p-chloroamphetamine in the mouse frontal cortex.
Journal: Brain research 20010824
Title: Strain-dependent effects of diazepam and the 5-HT2B/2C receptor antagonist SB 206553 in spontaneously hypertensive and Lewis rats tested in the elevated plus-maze.
Journal: Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20010501
Title: Role of 5-HT(2a) and 5-HT(2B/2C) receptors in the behavioral interactions between serotonin and catecholamine reuptake inhibitors.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20010301
Title: Effects of the 5-HT2C/2B antagonist SB 206553 on hyperactivity induced by cocaine.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 19990601
Title: Potentiation of fluoxetine-induced penile erections by combined blockade of 5-HT1A and 5-HT1B receptors.
Journal: European journal of pharmacology 19970305
Title: In vitro and in vivo profile of SB 206553, a potent 5-HT2C/5-HT2B receptor antagonist with anxiolytic-like properties.
Journal: British journal of pharmacology 19960201