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Journal: Toxicology and applied pharmacology 20180801
Title: Galunisertib modifies the liver fibrotic composition in the Abcb4Ko mouse model.
Journal: Archives of toxicology 20180701
Title: Preclinical assessment of galunisertib (LY2157299 monohydrate), a first-in-class transforming growth factor-β receptor type I inhibitor.
Journal: Oncotarget 20180123
Title: Discovery of N-((4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-5-(6-methylpyridin-2-yl)-1H-imidazol-2-yl)methyl)-2-fluoroaniline (EW-7197): a highly potent, selective, and orally bioavailable inhibitor of TGF-β type I receptor kinase as cancer immunotherapeutic/antifibrotic agent.
Journal: Journal of medicinal chemistry 20140522
Title: Optimization of a dihydropyrrolopyrazole series of transforming growth factor-beta type I receptor kinase domain inhibitors: discovery of an orally bioavailable transforming growth factor-beta receptor type I inhibitor as antitumor agent.
Journal: Journal of medicinal chemistry 20080410
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