Title: The translocator protein (peripheral benzodiazepine receptor) mediates rat-selective activation of the mitochondrial permeability transition by norbormide.
Journal: Biochimica et biophysica acta 20111201
Title: On the path from chemistry to neuroscience: early explorations in chemical medicine under the mentorship of Dr. Erminio Costa, a neuroscientist with a big brain and a bigger heart.
Journal: Pharmacological research 20111001
Title: Modulation of constitutive androstane receptor (CAR) and pregnane X receptor (PXR) by 6-arylpyrrolo[2,1-d][1,5]benzothiazepine derivatives, ligands of peripheral benzodiazepine receptor (PBR).
Journal: Toxicology letters 20110425
Title: Regulation of the inner membrane mitochondrial permeability transition by the outer membrane translocator protein (peripheral benzodiazepine receptor).
Journal: The Journal of biological chemistry 20110114
Title: Effects of neurosteroid actions at N-methyl-D-aspartate and GABA A receptors in the midbrain ventral tegmental area for anxiety-like and mating behavior of female rats.
Journal: Psychopharmacology 20110101
Title: Midazolam inhibits hippocampal long-term potentiation and learning through dual central and peripheral benzodiazepine receptor activation and neurosteroidogenesis.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20101215
Title: Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Journal: Nature chemical biology 20091001
Title: The translocator protein (18 kDa): central nervous system disease and drug design.
Journal: Journal of medicinal chemistry 20090212
Title: Increasing 3alpha,5alpha-THP following inhibition of neurosteroid biosynthesis in the ventral tegmental area reinstates anti-anxiety, social, and sexual behavior of naturally receptive rats.
Journal: Reproduction (Cambridge, England) 20090101
Title: The 18-kDa translocator protein, formerly known as the peripheral-type benzodiazepine receptor, confers proapoptotic and antineoplastic effects in a human colorectal cancer cell line.
Journal: Pharmacogenetics and genomics 20081101
Title: Synthesis, fluorine-18 radiolabeling, and in vitro characterization of 1-iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivatives as potential PET radioligands for imaging peripheral benzodiazepine receptor.
Journal: Bioorganic & medicinal chemistry 20080601
Title: The potential anticancer agent PK11195 induces apoptosis irrespective of p53 and ATM status in chronic lymphocytic leukemia cells.
Journal: Haematologica 20071201
Title: Preparation of indoles from alpha-aminonitriles: A short synthesis of FGIN-1-27.
Journal: Organic letters 20060928
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Mechanisms of mitochondrial apoptosis induced by peripheral benzodiazepine receptor ligands in human colorectal cancer cells.
Journal: Biochemical and biophysical research communications 20050708
Title: A cDNA encoding diazepam-binding inhibitor/acyl-CoA-binding protein in Helicoverpa armigera: molecular characterization and expression analysis associated with pupal diapause.
Journal: Comparative biochemistry and physiology. Toxicology & pharmacology : CBP 20050601
Title: In the ventral tegmental area picrotoxin blocks FGIN 1-27-induced increases in sexual behavior of rats and hamsters.
Journal: Psychopharmacology 20050301
Title: Peripheral benzodiazepine receptor (PBR) ligand cytotoxicity unrelated to PBR expression.
Journal: Biochemical pharmacology 20050301
Title: Peripheral benzodiazepine receptor ligands induce apoptosis and cell cycle arrest in human hepatocellular carcinoma cells and enhance chemosensitivity to paclitaxel, docetaxel, doxorubicin and the Bcl-2 inhibitor HA14-1.
Journal: Journal of hepatology 20041101
Title: GABA(A)/central benzodiazepine receptor and peripheral benzodiazepine receptor ligands as inducers of phenobarbital-inducible CYP2B and CYP3A.
Journal: Biochemical pharmacology 20041001
Title: Enhancement of peripheral benzodiazepine receptor ligand-induced apoptosis and cell cycle arrest of esophageal cancer cells by simultaneous inhibition of MAPK/ERK kinase.
Journal: Biochemical pharmacology 20040501
Title: Design, synthesis and structure-affinity relationships of aryloxyanilide derivatives as novel peripheral benzodiazepine receptor ligands.
Journal: Bioorganic & medicinal chemistry 20040115
Title: Ligands of the peripheral benzodiazepine receptor induce apoptosis and cell cycle arrest in oesophageal cancer cells: involvement of the p38MAPK signalling pathway.
Journal: British journal of cancer 20030804
Title: Mitochondrial benzodiazepine receptors in the ventral tegmental area modulate sexual behaviour of cycling or hormone-primed hamsters.
Journal: Journal of neuroendocrinology 20030701
Title: Lordosis of rats is modified by neurosteroidogenic effects of membrane benzodiazepine receptors in the ventral tegmental area.
Journal: Neuroendocrinology 20030101
Title: Mitochondrial benzodiazepine receptors regulate oxygen homeostasis in the early mouse embryo.
Journal: Reproductive toxicology (Elmsford, N.Y.) 20030101
Title: Specific ligands of the peripheral benzodiazepine receptor induce apoptosis and cell cycle arrest in human esophageal cancer cells.
Journal: International journal of cancer 20021201
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: Binding of [3H]CB 34, a selective ligand for peripheral benzodiazepine receptors, to rat brain membranes.
Journal: European journal of pharmacology 20011207
Title: Synthesis and preliminary behavioural evaluation in mice of new 3-aryl-3-pyrrol-1-ylpropanamides, analogues of FGIN-1-27 and FGIN-1-43.
Journal: The Journal of pharmacy and pharmacology 20011101
Title: Specific ligands of the peripheral benzodiazepine receptor induce apoptosis and cell cycle arrest in human colorectal cancer cells.
Journal: British journal of cancer 20011101
Title: Cataleptic effect of neurosteroid 3alpha-hydroxy-5alpha-pregnan-20-one in mice: modulation by serotonergic agents.
Journal: Brain research 20010413
Title: Mitochondrial diazepam-binding inhibitor receptor complex agonists antagonize dizocilpine amnesia: putative role for allopregnanolone.
Journal: The Journal of pharmacology and experimental therapeutics 19940701
Title: 2-Aryl-3-indoleacetamides (FGIN-1): a new class of potent and specific ligands for the mitochondrial DBI receptor (MDR).
Journal: The Journal of pharmacology and experimental therapeutics 19920901