Title: Identification of potent Yes1 kinase inhibitors using a library screening approach.
Journal: Bioorganic & medicinal chemistry letters 20130801
Title: Synthesis and pharmacological properties of novel hydrophilic 5-HT4 receptor antagonists.
Journal: Bioorganic & medicinal chemistry 20101215
Title: Effect of piboserod, a 5-HT4 serotonin receptor antagonist, on left ventricular function in patients with symptomatic heart failure.
Journal: European journal of heart failure 20090801
Title: Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
Journal: Bioorganic & medicinal chemistry 20090315
Title: Measurement of 5-HT4 receptor-mediated esophageal responses by digital sonomicrometry in the anesthetized rat.
Journal: Journal of pharmacological and toxicological methods 20060101
Title: Piboserod (SB 207266), a selective 5-HT4 receptor antagonist, reduces serotonin potentiation of neurally-mediated contractile responses of human detrusor muscle.
Journal: World journal of urology 20050601
Title: Identification of a 5-HT4 receptor antagonist clinical candidate through side-chain modification.
Journal: Bioorganic & medicinal chemistry letters 20050315
Title: The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo.
Journal: British journal of pharmacology 20041101
Title: Trials of new antiarrhythmic drugs for maintenance of sinus rhythm in patients with atrial fibrillation.
Journal: Journal of interventional cardiac electrophysiology : an international journal of arrhythmias and pacing 20040101
Title: Regulatory role of 5-HT and muscarinic receptor antagonists on the migrating myoelectric complex in rats.
Journal: European journal of pharmacology 20030425
Title: 5-HT4 receptor ligands: applications and new prospects.
Journal: Journal of medicinal chemistry 20030130
Title: Synthesis and pharmacological activity of metabolites of the 5-HT(4) receptor antagonist SB-207266.
Journal: Bioorganic & medicinal chemistry 20010801
Title: Serotonin-4 receptor antagonists reverse cocaine-induced cardiac arrhythmia.
Journal: Life sciences 19980101
Title: Cloning and expression of human 5-HT4S receptors. Effect of receptor density on their coupling to adenylyl cyclase.
Journal: Neuroreport 19971020
Title: Darblade B, et al. Piboserod (SB 207266), a selective 5-HT4 receptor antagonist, reduces serotonin potentiation of neurally-mediated contractile responses of human detrusor muscle. World J Urol. 2005 Jun;23(2):147-51.
Title: Kjekshus JK, et al. Effect of piboserod, a 5-HT4 serotonin receptor antagonist, on left ventricular function in patients with symptomatic heart failure. Eur J Heart Fail. 2009 Aug;11(8):771-8.
Title: Nirogi R, et al. In-vivo rat striatal 5-HT4 receptor occupancy using non-radiolabelled SB207145. J Pharm Pharmacol. 2013 May;65(5):704-12.
