176-73-8 
 
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cisracemate-1-3-(3-{7-azaspiro4.5decane-7-carbonyl}cyclohexyl)phenyl-5-cyclopropyl-1H-pyrazole-4-carboxylicacidmethylester 
[1]CurrentPatentAssignee:OTSUKAHOLDINGSCOLTD-WO2017/60855,2017,A1Locationinpatent:Page/Pagecolumn80
176-73-8 
 
1-3-((1R,3S)-3-carboxycyclohexyl)phenyl-5-cyclopropyl-1H-pyrazole-4-carboxylicacidmethylester 
 
cisracemate-1-3-(3-{7-azaspiro4.5decane-7-carbonyl}cyclohexyl)phenyl-5-cyclopropyl-1H-pyrazole-4-carboxylicacid 
[1]CurrentPatentAssignee:OTSUKAHOLDINGSCOLTD-WO2017/60855,2017,A1
176-73-8 
 
1-(3'-carboxy-2'-fluoro-biphenyl-3-yl)-5-cyclopropyl-1H-pyrazole-4-carboxylicacidmethylester 
 
1-3-(3-{7-azaspiro4.5decane-7-carbonyl}-2-fluorophenyl)phenyl-5-cyclopropyl-1H-pyrazole-4-carboxylicacidmethylester 
[1]CurrentPatentAssignee:OTSUKAHOLDINGSCOLTD-WO2017/60854,2017,A1Locationinpatent:Page/Pagecolumn219
[2]Norton,David;Bonnette,WilliamG.;Callahan,JamesF.;Carr,MariaG.;Griffiths-Jones,CharlotteM.;Heightman,TomD.;Kerns,JeffreyK.;Nie,Hong;Rich,SharnaJ.;Richardson,Caroline;Rumsey,William;Sanchez,Yolanda;Verdonk,MarcelL.;Willems,HenriëtteM.G.;Wixted,WilliamE.;Wolfe,Lawrence;Woolford,AlisonJ.-A.;Wu,Zining;Davies,ThomasG.[JournalofMedicinalChemistry,2021,vol.64,#21,p.15949-15972]
176-73-8 
 
1-(3'-carboxy-2'-fluoro-biphenyl-3-yl)-5-cyclopropyl-1H-pyrazole-4-carboxylicacidmethylester 
 
1-3-(3-{7-azaspiro4.5decane-7-carbonyl}-2-fluorophenyl)phenyl-5-cyclopropyl-1H-pyrazole-4-carboxylicacid 
[1]CurrentPatentAssignee:OTSUKAHOLDINGSCOLTD-WO2017/60854,2017,A1