[1]Shinkai;Maeda;Yamasaki;Okamoto;Uchida[JournalofMedicinalChemistry,2000,vol.43,#19,p.3566-3572]
[2]CurrentPatentAssignee:JAPANTOBACCOINC-US6426365,2002,B1
[1]Shinkai;Maeda;Yamasaki;Okamoto;Uchida[JournalofMedicinalChemistry,2000,vol.43,#19,p.3566-3572]
[1]Shinkai;Maeda;Yamasaki;Okamoto;Uchida[JournalofMedicinalChemistry,2000,vol.43,#19,p.3566-3572]
[1]Shinkai;Maeda;Yamasaki;Okamoto;Uchida[JournalofMedicinalChemistry,2000,vol.43,#19,p.3566-3572]
[1]Shinkai;Maeda;Yamasaki;Okamoto;Uchida[JournalofMedicinalChemistry,2000,vol.43,#19,p.3566-3572]
Title: Cholesteryl ester-transfer protein inhibitors stimulate aldosterone biosynthesis in adipocytes through Nox-dependent processes.
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Title: Future of cholesteryl ester transfer protein inhibitors.
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Title: Cholesteryl ester transfer protein inhibition as a strategy to reduce cardiovascular risk.
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Title: Dalcetrapib , a cholesteryl ester transfer protein modulator.
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Title: HDL and CETP Inhibition: Will This DEFINE the Future?
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Title: Lipid and apoprotein composition of HDL in partial or complete CETP deficiency.
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Title: Determination of dalcetrapib by liquid chromatography-tandem mass spectrometry.
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Title: Increasing high-density lipoprotein cholesterol by cholesteryl ester transfer protein-inhibition: a rocky road and lessons learned? The early demise of the dal-HEART programme.
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Title: An update on the clinical development of dalcetrapib (RO4607381), a cholesteryl ester transfer protein modulator that increases HDL cholesterol levels.
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Title: Current status of CETP inhibitors in the treatment of hyperlipidemia: an update.
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Title: Design, synthesis and structure-activity-relationship of 1,5-tetrahydronaphthyridines as CETP inhibitors.
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Title: Dalcetrapib--restoring belief in modulating CETP as a beneficial mechanism in cardiovascular disease.
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Title: Vascular effects and safety of dalcetrapib in patients with or at risk of coronary heart disease: the dal-VESSEL randomized clinical trial.
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Title: Cholesteryl ester transfer protein inhibition and endothelial function: enough with the surrogates.
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Title: No clinically relevant drug-drug interactions when dalcetrapib is co-administered with a monophasic oral contraceptive (Microgynon® 30).
Journal: International journal of clinical pharmacology and therapeutics 20120401
Title: Monitoring Cyp2b10 mRNA expression at cessation of 2-year carcinogenesis bioassay in mouse liver provides evidence for a carcinogenic mechanism devoid of human relevance: the dalcetrapib experience.
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Title: Pharmacotherapy. Elevating HDL-cholesterol levels with dalcetrapib is safe.
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Title: Effect of dalcetrapib plus pravastatin on lipoprotein metabolism and high-density lipoprotein composition and function in dyslipidemic patients: results of a phase IIb dose-ranging study.
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Title: Multidimensional profiling of plasma lipoproteins by size exclusion chromatography followed by reverse-phase protein arrays.
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Title: Effect of dalcetrapib, a CETP modulator, on non-cholesterol sterol markers of cholesterol homeostasis in healthy subjects.
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Title: Safety and efficacy of dalcetrapib on atherosclerotic disease using novel non-invasive multimodality imaging (dal-PLAQUE): a randomised clinical trial.
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Title: Dalcetrapib: turning the tide for CETP inhibition?
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Title: Lack of effect of dalcetrapib on QT interval in healthy subjects following multiple dosing.
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Title: Dalcetrapib: JTT 705; JTT-705; R 1658; R1658; RG1658; RO 4607381; RO4607381.
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Title: MARCO, a macrophage scavenger receptor highly expressed in rodents, mediates dalcetrapib-induced uptake of lipids by rat and mouse macrophages.
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