Title: Increased binding of peripheral benzodiazepine receptor in mild cognitive impairment-dementia converters measured by positron emission tomography with [¹¹C]DAA1106.
Journal: Psychiatry research 20120730
Title: Fully automated synthesis of PET TSPO radioligands [11C]DAA1106 and [18F]FEDAA1106.
Journal: Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine 20120601
Title: Peripheral benzodiazepine receptors in patients with chronic schizophrenia: a PET study with [11C]DAA1106.
Journal: The international journal of neuropsychopharmacology 20100801
Title: Evaluation of [11C]-DAA1106 for imaging and quantification of neuroinflammation in a rat model of herpes encephalitis.
Journal: Nuclear medicine and biology 20100101
Title: Visualization of brain amyloid and microglial activation in mouse models of Alzheimer's disease.
Journal: Current Alzheimer research 20090401
Title: Single-step high-yield radiosynthesis and evaluation of a sensitive 18F-labeled ligand for imaging brain peripheral benzodiazepine receptors with PET.
Journal: Journal of medicinal chemistry 20090212
Title: A comparative autoradiography study in post mortem whole hemisphere human brain slices taken from Alzheimer patients and age-matched controls using two radiolabelled DAA1106 analogues with high affinity to the peripheral benzodiazepine receptor (PBR) system.
Journal: Neurochemistry international 20090101
Title: Imaging of peripheral benzodiazepine receptor expression as biomarkers of detrimental versus beneficial glial responses in mouse models of Alzheimer's and other CNS pathologies.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20081119
Title: Increased binding of peripheral benzodiazepine receptor in Alzheimer's disease measured by positron emission tomography with [11C]DAA1106.
Journal: Biological psychiatry 20081115
Title: The positron emission tomography ligand DAA1106 binds with high affinity to activated microglia in human neurological disorders.
Journal: Journal of neuropathology and experimental neurology 20081001
Title: The high affinity peripheral benzodiazepine receptor ligand DAA1106 binds to activated and infected brain macrophages in areas of synaptic degeneration: implications for PET imaging of neuroinflammation in lentiviral encephalitis.
Journal: Neurobiology of disease 20080201
Title: A comparison of the high-affinity peripheral benzodiazepine receptor ligands DAA1106 and (R)-PK11195 in rat models of neuroinflammation: implications for PET imaging of microglial activation.
Journal: Journal of neurochemistry 20070901
Title: The high affinity peripheral benzodiazepine receptor ligand DAA1106 binds specifically to microglia in a rat model of traumatic brain injury: implications for PET imaging.
Journal: Experimental neurology 20070901
Title: Phase-dependent roles of reactive microglia and astrocytes in nervous system injury as delineated by imaging of peripheral benzodiazepine receptor.
Journal: Brain research 20070709
Title: Strategy for improved [(11)C]DAA1106 radiosynthesis and in vivo peripheral benzodiazepine receptor imaging using microPET, evaluation of [(11)C]DAA1106.
Journal: Nuclear medicine and biology 20070501
Title: N-(5-Fluoro-2-phenoxyphenyl)-N-(2-[(131)I]iodo-5-me thoxybenzyl)acetamide: a potent iodinated radioligand for the peripheral-type benzodiazepine receptor in brain.
Journal: Journal of medicinal chemistry 20070222
Title: PET imaging with [11C]PBR28 can localize and quantify upregulated peripheral benzodiazepine receptors associated with cerebral ischemia in rat.
Journal: Neuroscience letters 20070116
Title: Quantitative analysis for estimating binding potential of the peripheral benzodiazepine receptor with [(11)C]DAA1106.
Journal: Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20070101
Title: [2-11C]isopropyl-, [1-11C]ethyl-, and [11C]methyl-labeled phenoxyphenyl acetamide derivatives as positron emission tomography ligands for the peripheral benzodiazepine receptor: radiosynthesis, uptake, and in vivo binding in brain.
Journal: Journal of medicinal chemistry 20060504
Title: [Imaging of glial cells by positron-emitted peripheral benzodiazepine receptor ligands].
Journal: Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology 20060201
Title: Novel peripheral benzodiazepine receptor ligand [11C]DAA1106 for PET: an imaging tool for glial cells in the brain.
Journal: Synapse (New York, N.Y.) 20040615
Title: Development of a new radioligand, N-(5-fluoro-2-phenoxyphenyl)-N-(2-[18F]fluoroethyl-5-methoxybenzyl)acetamide, for pet imaging of peripheral benzodiazepine receptor in primate brain.
Journal: Journal of medicinal chemistry 20040422
Title: Design, synthesis and structure-affinity relationships of aryloxyanilide derivatives as novel peripheral benzodiazepine receptor ligands.
Journal: Bioorganic & medicinal chemistry 20040115
Title: [(11)C]DAA1106: radiosynthesis and in vivo binding to peripheral benzodiazepine receptors in mouse brain.
Journal: Nuclear medicine and biology 20030701
Title: [18F]FMDAA1106 and [18F]FEDAA1106: two positron-emitter labeled ligands for peripheral benzodiazepine receptor (PBR).
Journal: Bioorganic & medicinal chemistry letters 20030120
Title: Yasuno F, et al. Increased binding of peripheral benzodiazepine receptor in mild cognitive impairment-dementia converters measured by positron emission tomography with 1CDAA1106. Psychiatry Res. 2012 Jul 30;203(1):67-74.
Title: DAA1106
