Title: Carbonic anhydrase inhibitors: synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety.
Journal: Bioorganic & medicinal chemistry 20131001
Title: Single and mixed poloxamine micelles as nanocarriers for solubilization and sustained release of ethoxzolamide for topical glaucoma therapy.
Journal: Journal of the Royal Society, Interface 20120907
Title: Methazolamide is a new hepatic insulin sensitizer that lowers blood glucose in vivo.
Journal: Diabetes 20120801
Title: Molecular cloning, characterization, and inhibition studies of a β-carbonic anhydrase from Malassezia globosa, a potential antidandruff target.
Journal: Journal of medicinal chemistry 20120412
Title: Mutation of active site residues Asn67 to Ile, Gln92 to Val and Leu204 to Ser in human carbonic anhydrase II: influences on the catalytic activity and affinity for inhibitors.
Journal: Bioorganic & medicinal chemistry 20120401
Title: Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI.
Journal: European journal of medicinal chemistry 20120301
Title: Cloning, characterization and sulfonamide inhibition studies of an α-carbonic anhydrase from the living fossil sponge Astrosclera willeyana.
Journal: Bioorganic & medicinal chemistry 20120215
Title: Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives.
Journal: Bioorganic & medicinal chemistry letters 20120201
Title: Dependence of avidity on linker length for a bivalent ligand-bivalent receptor model system.
Journal: Journal of the American Chemical Society 20120111
Title: Topiramate and the vision: a systematic review.
Journal: Clinical ophthalmology (Auckland, N.Z.) 20120101
Title: Differential scanning fluorometry signatures as indicators of enzyme inhibitor mode of action: case study of glutathione S-transferase.
Journal: PloS one 20120101
Title: Thermodynamics of aryl-dihydroxyphenyl-thiadiazole binding to human Hsp90.
Journal: PloS one 20120101
Title: Regulation of the cyanobacterial CO2-concentrating mechanism involves internal sensing of NADP+ and α-ketogutarate levels by transcription factor CcmR.
Journal: PloS one 20120101
Title: Carbonic anhydrase activity in Arabidopsis thaliana thylakoid membrane and fragments enriched with PSI or PSII.
Journal: Photosynthesis research 20111201
Title: Testing the limits of sensitivity in a solid-state structural investigation by combined X-ray powder diffraction, solid-state NMR, and molecular modelling.
Journal: Physical chemistry chemical physics : PCCP 20111028
Title: Photosynthetic characteristics of a multicellular green alga Volvox carteri in response to external CO2 levels possibly regulated by CCM1/CIA5 ortholog.
Journal: Photosynthesis research 20110901
Title: Evidence for the occurrence of photorespiration in synurophyte algae.
Journal: Photosynthesis research 20110901
Title: Carbonic anhydrase inhibitors. Synthesis, molecular structures, and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with novel 3-pyridinesulfonamide derivatives.
Journal: European journal of medicinal chemistry 20110901
Title: Inhibition studies of the β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium with sulfonamides and sulfamates.
Journal: Bioorganic & medicinal chemistry 20110815
Title: Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.
Journal: Bioorganic & medicinal chemistry 20110515
Title: Carbonate precipitates and bicarbonate secretion in the intestine of sea bass, Dicentrarchus labrax.
Journal: Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20110501
Title: Extracellular β-class carbonic anhydrase of the alkaliphilic cyanobacterium Microcoleus chthonoplastes.
Journal: Journal of photochemistry and photobiology. B, Biology 20110404
Title: Evaluation of the reproductive and developmental risks of caffeine.
Journal: Birth defects research. Part B, Developmental and reproductive toxicology 20110401
Title: Purification and inhibition studies with anions and sulfonamides of an α-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii.
Journal: Bioorganic & medicinal chemistry 20110315
Title: Bioinspired imprinted PHEMA-hydrogels for ocular delivery of carbonic anhydrase inhibitor drugs.
Journal: Biomacromolecules 20110314
Title: (R)-/(S)-10-camphorsulfonyl-substituted aromatic/heterocyclic sulfonamides selectively inhibit mitochondrial over cytosolic carbonic anhydrases.
Journal: Bioorganic & medicinal chemistry letters 20110301
Title: A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth.
Journal: Bioorganic & medicinal chemistry 20110201
Title: Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata.
Journal: Bioorganic & medicinal chemistry letters 20110115
Title: A high throughput screen identifies chemical modulators of the laminin-induced clustering of dystroglycan and aquaporin-4 in primary astrocytes.
Journal: PloS one 20110101
Title: Treat ankylosing spondylitis with methazolamide.
Journal: International journal of medical sciences 20110101
Title: Bacterial carbonic anhydrases as drug targets: toward novel antibiotics?
Journal: Frontiers in pharmacology 20110101
Title: Transport activity of the sodium bicarbonate cotransporter NBCe1 is enhanced by different isoforms of carbonic anhydrase.
Journal: PloS one 20110101
Title: Sharpey-Schafer lecture: gas channels.
Journal: Experimental physiology 20101201
Title: Carbonic anhydrase II regulates differentiation of ameloblasts via intracellular pH-dependent JNK signaling pathway.
Journal: Journal of cellular physiology 20101101
Title: Carbonic anhydrase inhibitors. Regioselective synthesis of novel 1-substituted 1,4-dihydro-4-oxo-3-pyridinesulfonamides and their inhibition of the human cytosolic isozymes I and II and transmembrane cancer-associated isozymes IX and XII.
Journal: European journal of medicinal chemistry 20100901
Title: Mutation of Phe91 to Asn in human carbonic anhydrase I unexpectedly enhanced both catalytic activity and affinity for sulfonamide inhibitors.
Journal: Bioorganic & medicinal chemistry 20100801
Title: Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV.
Journal: Bioorganic & medicinal chemistry letters 20100615
Title: New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20100615
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with 4-substituted 3-pyridinesulfonamides.
Journal: European journal of medicinal chemistry 20100601
Title: Carbonic anhydrase inhibitors. The beta-carbonic anhydrases from the fungal pathogens Cryptococcus neoformans and Candida albicans are strongly inhibited by substituted-phenyl-1H-indole-5-sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20100415
Title: Nonenzymatic augmentation of lactate transport via monocarboxylate transporter isoform 4 by carbonic anhydrase II.
Journal: The Journal of membrane biology 20100401
Title: Cloning, characterization, and inhibition studies of a beta-carbonic anhydrase from Brucella suis.
Journal: Journal of medicinal chemistry 20100311
Title: Differences in transcription between free-living and CO2-activated third-stage larvae of Haemonchus contortus.
Journal: BMC genomics 20100101
Title: Alterations in osteoclast function and phenotype induced by different inhibitors of bone resorption--implications for osteoclast quality.
Journal: BMC musculoskeletal disorders 20100101
Title: Saccharomyces cerevisiae β-carbonic anhydrase: inhibition and activation studies.
Journal: Current pharmaceutical design 20100101
Title: Role of carbonic anhydrase IV in the bicarbonate-mediated activation of murine and human sperm.
Journal: PloS one 20100101
Title: Increased expression of carbonic anhydrase I in the synovium of patients with ankylosing spondylitis.
Journal: BMC musculoskeletal disorders 20100101
Title: T tubules and surface membranes provide equally effective pathways of carbonic anhydrase-facilitated lactic acid transport in skeletal muscle.
Journal: PloS one 20100101
Title: Cyclodextrins in delivery systems: Applications.
Journal: Journal of pharmacy & bioallied sciences 20100101
Title: Ocular inserts - Advancement in therapy of eye diseases.
Journal: Journal of advanced pharmaceutical technology & research 20100101
Title: Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.
Journal: Bioorganic & medicinal chemistry letters 20091201
Title: A pea mutant (costata) expressing higher activity in thylakoid membrane-bound carbonic anhydrase alters PSII downregulation mechanisms.
Journal: Cell biology international 20090801
Title: Carbonic anhydrase inhibitors. Inhibition studies of a coral secretory isoform by sulfonamides.
Journal: Bioorganic & medicinal chemistry 20090715
Title: Carbonic anhydrase inhibitors. Inhibition and homology modeling studies of the fungal beta-carbonic anhydrase from Candida albicans with sulfonamides.
Journal: Bioorganic & medicinal chemistry 20090701
Title: Carbonic anhydrase inhibitors. Phenacetyl-, pyridylacetyl- and thienylacetyl-substituted aromatic sulfonamides act as potent and selective isoform VII inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20090615
Title: Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII.
Journal: Bioorganic & medicinal chemistry letters 20090601
Title: Measurement of nanomolar dissociation constants by titration calorimetry and thermal shift assay - radicicol binding to Hsp90 and ethoxzolamide binding to CAII.
Journal: International journal of molecular sciences 20090601
Title: Titration calorimetry standards and the precision of isothermal titration calorimetry data.
Journal: International journal of molecular sciences 20090601
Title: Carbonic anhydrase inhibitors. Cloning, characterization, and inhibition studies of a new beta-carbonic anhydrase from Mycobacterium tuberculosis.
Journal: Journal of medicinal chemistry 20090514
Title: Ligand-directed tosyl chemistry for protein labeling in vivo.
Journal: Nature chemical biology 20090501
Title: Manganese-dependent carboanhydrase activity of photosystem II proteins.
Journal: Biochemistry. Biokhimiia 20090501
Title: Molecular cloning, characterization, and inhibition studies of the Rv1284 beta-carbonic anhydrase from Mycobacterium tuberculosis with sulfonamides and a sulfamate.
Journal: Journal of medicinal chemistry 20090423
Title: Carbonic anhydrase inhibitors. The nematode alpha-carbonic anhydrase of Caenorhabditis elegans CAH-4b is highly inhibited by 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides.
Journal: Bioorganic & medicinal chemistry 20090415
Title: QSAR studies for the inhibition of the transmembrane carbonic anhydrase isozyme XIV with sulfonamides using PRECLAV software.
Journal: Journal of enzyme inhibition and medicinal chemistry 20090401
Title: A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases.
Journal: Bioorganic & medicinal chemistry letters 20090301
Title: Design of a carbonic anhydrase IX active-site mimic to screen inhibitors for possible anticancer properties.
Journal: Biochemistry 20090217
Title: Carbonic anhydrase inhibitors. Comparison of chlorthalidone, indapamide, trichloromethiazide, and furosemide X-ray crystal structures in adducts with isozyme II, when several water molecules make the difference.
Journal: Bioorganic & medicinal chemistry 20090201
Title: Carbonic anhydrase inhibitors: inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with sulfonamides and sulfamates.
Journal: Bioorganic & medicinal chemistry 20090201
Title: Carbonic anhydrase inhibitors. Comparison of chlorthalidone and indapamide X-ray crystal structures in adducts with isozyme II: when three water molecules and the keto-enol tautomerism make the difference.
Journal: Journal of medicinal chemistry 20090122
Title: Inhibition of aquaporin 4 by antiepileptic drugs.
Journal: Bioorganic & medicinal chemistry 20090101
Title: Label-free determination of protein-ligand binding constants using mass spectrometry and validation using surface plasmon resonance and isothermal titration calorimetry.
Journal: Journal of molecular recognition : JMR 20090101
Title: Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions.
Journal: Bioorganic & medicinal chemistry letters 20081215
Title: The bicarbonate transporter is essential for Bacillus anthracis lethality.
Journal: PLoS pathogens 20081101
Title: Lack of aquaporin-4 water transport inhibition by antiepileptics and arylsulfonamides.
Journal: Bioorganic & medicinal chemistry 20080801
Title: Carbonic anhydrase inhibitors: design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes.
Journal: Bioorganic & medicinal chemistry letters 20080615
Title: Isolation and characterization of a gene encoding carbonic anhydrase from Ostertagia ostertagi and quantitative measurement of expression during in vivo exsheathment.
Journal: Veterinary parasitology 20080614
Title: Carbonic anhydrase inhibitors: bioreductive nitro-containing sulfonamides with selectivity for targeting the tumor associated isoforms IX and XII.
Journal: Journal of medicinal chemistry 20080612
Title: Antagonistic effect of juvenile hormone on hemocyte-spreading behavior of Spodoptera exigua in response to an insect cytokine and its putative membrane action.
Journal: Journal of insect physiology 20080601
Title: Diversity of inorganic carbon acquisition mechanisms by intact microbial mats of Microcoleus chthonoplastes (Cyanobacteriae, Oscillatoriaceae).
Journal: Physiologia plantarum 20080501
Title: Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20080415
Title: Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct.
Journal: Bioorganic & medicinal chemistry letters 20080415
Title: Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry 20080401
Title: Inhibition of carbonic anhydrases with glycosyltriazole benzene sulfonamides.
Journal: Journal of medicinal chemistry 20080327
Title: Carbonic anhydrase inhibitors: interactions of phenols with the 12 catalytically active mammalian isoforms (CA I-XIV).
Journal: Bioorganic & medicinal chemistry letters 20080301
Title: Fluid and osmolyte recovery in the common pond snail Lymnaea stagnalis following full-body withdrawal.
Journal: The Journal of experimental biology 20080201
Title: Carbonic anhydrase inhibitors: copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII.
Journal: Bioorganic & medicinal chemistry letters 20080115
Title: The alpha and beta classes carbonic anhydrases from Helicobacter pylori as novel drug targets.
Journal: Current pharmaceutical design 20080101
Title: The development of topically acting carbonic anhydrase inhibitors as antiglaucoma agents.
Journal: Current pharmaceutical design 20080101
Title: Direct non-cyclooxygenase-2 targets of celecoxib and their potential relevance for cancer therapy.
Journal: British journal of cancer 20071203
Title: Carbonic anhydrase inhibitors: cloning, characterization, and inhibition studies of the cytosolic isozyme III with sulfonamides.
Journal: Bioorganic & medicinal chemistry 20071201
Title: Carbonic anhydrase inhibitors: Selective inhibition of the extracellular, tumor-associated isoforms IX and XII over isozymes I and II with glycosyl-thioureido-sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20070915
Title: Carbonic anhydrase inhibitors. Interaction of the antiepileptic drug sulthiame with twelve mammalian isoforms: kinetic and X-ray crystallographic studies.
Journal: Bioorganic & medicinal chemistry letters 20070901
Title: Carbonic anhydrase inhibitors: inhibition of human, bacterial, and archaeal isozymes with benzene-1,3-disulfonamides--solution and crystallographic studies.
Journal: Bioorganic & medicinal chemistry letters 20070801
Title: Acclimation of wild-type cells and CO2-insensitive mutants of the green alga Chlorella ellipsoidea to elevated [CO2].
Journal: Plant, cell & environment 20070801
Title: Electrical parameters and ion species for active transport in human esophageal stratified squamous epithelium and Barrett's specialized columnar epithelium.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20070701
Title: Carbonic anhydrases as targets for medicinal chemistry.
Journal: Bioorganic & medicinal chemistry 20070701
Title: Carbonic anhydrase inhibitors: the beta-carbonic anhydrase from Helicobacter pylori is a new target for sulfonamide and sulfamate inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20070701
Title: Carbonic anhydrase II increases the activity of the human electrogenic Na+/HCO3- cotransporter.
Journal: The Journal of biological chemistry 20070504
Title: Carbonic anhydrase inhibitors: inhibition of isozymes I, II, and IX with triazole-linked O-glycosides of benzene sulfonamides.
Journal: Journal of medicinal chemistry 20070405
Title: Inhibition of hypoxia-induced calcium responses in pulmonary arterial smooth muscle by acetazolamide is independent of carbonic anhydrase inhibition.
Journal: American journal of physiology. Lung cellular and molecular physiology 20070401
Title: Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated isoforms I, II, and IX with iminodiacetic carboxylates/hydroxamates also incorporating benzenesulfonamide moieties.
Journal: Bioorganic & medicinal chemistry letters 20070315
Title: Identification of arylsulfonamides as Aquaporin 4 inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20070301
Title: Carbonic anhydrase inhibition prevents and reverts cardiomyocyte hypertrophy.
Journal: The Journal of physiology 20070215
Title: Inhibition of membrane-associated carbonic anhydrase isozymes IX, XII and XIV with a library of glycoconjugate benzenesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20070215
Title: Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors.
Journal: Journal of medicinal chemistry 20070125
Title: Pulmonary vasodilation by acetazolamide during hypoxia is unrelated to carbonic anhydrase inhibition.
Journal: American journal of physiology. Lung cellular and molecular physiology 20070101
Title: Multiple sources of carbonic anhydrase activity in pea thylakoids: soluble and membrane-bound forms.
Journal: Photosynthesis research 20070101
Title: The development of topically acting carbonic anhydrase inhibitors as anti-glaucoma agents.
Journal: Current topics in medicinal chemistry 20070101
Title: Carbonic anhydrase inhibitors: clash with Ala65 as a means for designing inhibitors with low affinity for the ubiquitous isozyme II, exemplified by the crystal structure of the topiramate sulfamide analogue.
Journal: Journal of medicinal chemistry 20061130
Title: A novel class of carbonic anhydrase inhibitors: glycoconjugate benzene sulfonamides prepared by 'click-tailing'.
Journal: Journal of medicinal chemistry 20061102
Title: Carbonic anhydrase inhibitors: Hypoxia-activatable sulfonamides incorporating disulfide bonds that target the tumor-associated isoform IX.
Journal: Journal of medicinal chemistry 20060907
Title: Expression, purification, kinetic, and structural characterization of an alpha-class carbonic anhydrase from Aedes aegypti (AaCA1).
Journal: Biochimica et biophysica acta 20060801
Title: Effect of human carbonic anhydrase II on the activity of the human electrogenic Na/HCO3 cotransporter NBCe1-A in Xenopus oocytes.
Journal: The Journal of biological chemistry 20060714
Title: Evidence for a plasmalemma-based CO2 concentrating mechanism in Laminaria saccharina.
Journal: Photosynthesis research 20060601
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Heterogeneous origin of carbonic anhydrase activity of thylakoid membranes.
Journal: Biochemistry. Biokhimiia 20060501
Title: Carbonic anhydrase inhibitors: cloning and sulfonamide inhibition studies of a carboxyterminal truncated alpha-carbonic anhydrase from Helicobacter pylori.
Journal: Bioorganic & medicinal chemistry letters 20060415
Title: Carbonic anhydrase inhibitors: DNA cloning and inhibition studies of the alpha-carbonic anhydrase from Helicobacter pylori, a new target for developing sulfonamide and sulfamate gastric drugs.
Journal: Journal of medicinal chemistry 20060323
Title: Characterization of H+ and HCO3- transporters in CFPAC-1 human pancreatic duct cells.
Journal: World journal of gastroenterology 20060214
Title: Carbonic anhydrase inhibitors ameliorate the symptoms of hypokalaemic periodic paralysis in rats by opening the muscular Ca2+-activated-K+ channels.
Journal: Neuromuscular disorders : NMD 20060101
Title: Cryptococcus neoformans senses CO2 through the carbonic anhydrase Can2 and the adenylyl cyclase Cac1.
Journal: Eukaryotic cell 20060101
Title: Pea leaf thylakoids contain several carbonic anhydrases.
Journal: Doklady. Biochemistry and biophysics 20060101
Title: Transport activity of MCT1 expressed in Xenopus oocytes is increased by interaction with carbonic anhydrase.
Journal: The Journal of biological chemistry 20051202
Title: Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors.
Journal: Journal of medicinal chemistry 20051201
Title: Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20051101
Title: Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozymes IX and XII with a library of aromatic and heteroaromatic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20051101
Title: Modulation of carbonic anhydrase activity in two nitrogen fixing cyanobacteria, Nostoc calcicola and Anabaena sp.
Journal: Journal of plant physiology 20051001
Title: Carbonic anhydrase inhibitors: inhibition of the transmembrane isozyme XIV with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050901
Title: Carbonic anhydrase inhibitors: design of thioureido sulfonamides with potent isozyme II and XII inhibitory properties and intraocular pressure lowering activity in a rabbit model of glaucoma.
Journal: Bioorganic & medicinal chemistry letters 20050901
Title: Carbonic anhydrase inhibitors. Inhibition of red blood cell ostrich (Struthio camelus) carbonic anhydrase with a series of aromatic and heterocyclic sulfonamides.
Journal: Journal of enzyme inhibition and medicinal chemistry 20050801
Title: Carbonic anhydrase inhibitors. Design of fluorescent sulfonamides as probes of tumor-associated carbonic anhydrase IX that inhibit isozyme IX-mediated acidification of hypoxic tumors.
Journal: Journal of medicinal chemistry 20050728
Title: Carbonic anhydrase inhibitors. Synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with boron-containing sulfonamides, sulfamides, and sulfamates: toward agents for boron neutron capture therapy of hypoxic tumors.
Journal: Bioorganic & medicinal chemistry letters 20050701
Title: Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.
Journal: Bioorganic & medicinal chemistry letters 20050615
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes.
Journal: Bioorganic & medicinal chemistry letters 20050615
Title: Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.
Journal: Bioorganic & medicinal chemistry letters 20050502
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating thioureido-sulfanilyl scaffolds.
Journal: Bioorganic & medicinal chemistry letters 20050502
Title: HCO3- secretion in the esophageal submucosal glands.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20050401
Title: Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs?
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with bis-sulfamates.
Journal: Bioorganic & medicinal chemistry letters 20050201
Title: Carbonic anhydrase inhibitors. Novel sulfanilamide/acetazolamide derivatives obtained by the tail approach and their interaction with the cytosolic isozymes I and II, and the tumor-associated isozyme IX.
Journal: Bioorganic & medicinal chemistry letters 20050117
Title: Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20041220
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide.
Journal: Bioorganic & medicinal chemistry letters 20041206
Title: Photosystem II associated carbonic anhydrase activity in higher plants is situated in core complex.
Journal: FEBS letters 20041105
Title: Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.
Journal: Bioorganic & medicinal chemistry letters 20041101
Title: Theoretical study of gas-phase acidity, pKa, lipophilicity, and solubility of some biologically active sulfonamides.
Journal: Bioorganic & medicinal chemistry 20041015
Title: Carbonic anhydrase inhibitors: the first on-resin screening of a 4-sulfamoylphenylthiourea library.
Journal: Journal of medicinal chemistry 20041007
Title: Roles of carbonic anhydrase in photosynthesis of Skeletonema costatum.
Journal: Zhi wu sheng li yu fen zi sheng wu xue xue bao = Journal of plant physiology and molecular biology 20041001
Title: pH microdomains in oligodendrocytes.
Journal: The Journal of biological chemistry 20040827
Title: Carbonic anhydrase isoform expression and functional role in rodent extraocular muscle.
Journal: Pflugers Archiv : European journal of physiology 20040801
Title: Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20040621
Title: Inhibition of alpha(1E) Ca(2+) channels by carbonic anhydrase inhibitors.
Journal: Journal of pharmacological sciences 20040601
Title: Benzolamide is not a membrane-impermeant carbonic anhydrase inhibitor.
Journal: Journal of enzyme inhibition and medicinal chemistry 20040601
Title: Carbonic anhydrase inhibitors: synthesis and topical intraocular pressure lowering effects of fluorine-containing inhibitors devoid of enhanced reactivity.
Journal: Journal of medicinal chemistry 20040520
Title: Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with fluorine-containing sulfonamides. The first subnanomolar CA IX inhibitor discovered.
Journal: Bioorganic & medicinal chemistry letters 20040503
Title: Inhibition of 3T3-L1 adipocyte differentiation by 6-ethoxyzolamide: repressed peroxisome proliferator-activated receptor gamma mRNA and enhanced CCAAT/enhancer binding protein beta mRNA levels.
Journal: Biochemical pharmacology 20040501
Title: Carbonic anhydrase inhibitors are specific openers of skeletal muscle BK channel of K+-deficient rats.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20040401
Title: Carbonic anhydrase inhibitors. Inhibition of mitochondrial isozyme V with aromatic and heterocyclic sulfonamides.
Journal: Journal of medicinal chemistry 20040226
Title: Pdcd4 inhibits growth of tumor cells by suppression of carbonic anhydrase type II.
Journal: Molecular and cellular endocrinology 20040212
Title: Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20040105
Title: Sodium and chloride transport in soft water and hard water acclimated zebrafish (Danio rerio).
Journal: Biochimica et biophysica acta 20031230
Title: Carbonic anhydrase inhibitors: inhibition of transmembrane, tumor-associated isozyme IX, and cytosolic isozymes I and II with aliphatic sulfamates.
Journal: Journal of medicinal chemistry 20031204
Title: Inorganic carbon limitation induces transcripts encoding components of the CO(2)-concentrating mechanism in Synechococcus sp. PCC7942 through a redox-independent pathway.
Journal: Plant physiology 20031201
Title: Bicarbonate-dependent depolarizing potentials in pyramidal cells and interneurons during epileptiform activity.
Journal: The European journal of neuroscience 20030901
Title: Carbonic anhydrase inhibitors: topically acting antiglaucoma sulfonamides incorporating esters and amides of 3- and 4-carboxybenzolamide.
Journal: Bioorganic & medicinal chemistry letters 20030901
Title: Carbonic anhydrase inhibitors. Inhibition of tumor-associated isozyme IX by halogenosulfanilamide and halogenophenylaminobenzolamide derivatives.
Journal: Journal of medicinal chemistry 20030522
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Journal: Journal of medicinal chemistry 20030522
Title: Spinal carbonic anhydrase contributes to nociceptive reflex enhancement by midazolam, pentobarbital, and propofol.
Journal: Anesthesiology 20030401
Title: Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20030324
Title: Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives.
Journal: Bioorganic & medicinal chemistry letters 20030310
Title: Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV.
Journal: Bioorganic & medicinal chemistry letters 20030310
Title: Transepithelial sulfate transport by avian renal proximal tubule epithelium in primary culture.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20021201
Title: Inhibition of muscle carbonic anhydrase slows the Ca(2+) transient in rat skeletal muscle fibers.
Journal: American journal of physiology. Cell physiology 20021001
Title: Proton pump activity is required for active uptake of chloride in isolated amphibian skin exposed to freshwater.
Journal: Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology 20020801
Title: Carbonic anhydrase inhibitors. Preparation of potent sulfonamides inhibitors incorporating bile acid tails.
Journal: Bioorganic & medicinal chemistry letters 20020617
Title: Biochemical and molecular inhibition of plastidial carbonic anhydrase reduces the incorporation of acetate into lipids in cotton embryos and tobacco cell suspensions and leaves.
Journal: Plant physiology 20020401
Title: Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties.
Journal: Journal of medicinal chemistry 20020328
Title: Potassium drives daily reversible thallus enlargement in the marine red alga Porphyra leucosticta (Rhodophyta).
Journal: Planta 20020301
Title: Inhibition of muscle carbonic anhydrase increases rise and relaxation times of twitches in rat skeletal muscle fibres.
Journal: Pflugers Archiv : European journal of physiology 20020301
Title: Role of carbon dioxide and ion transport in the formation of sub-embryonic fluid by the blastoderm of the Japanese quail.
Journal: British poultry science 20020301
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