Title: Activation of transmembrane bile acid receptor TGR5 stimulates insulin secretion in pancreatic β cells.
Journal: Biochemical and biophysical research communications 20121026
Title: Effect of development on [Ca2+]i transients to ATP in petrosal ganglion neurons: a pharmacological approach using optical recording.
Journal: Journal of applied physiology (Bethesda, Md. : 1985) 20120415
Title: Molecular basis of selective antagonism of the P2X1 receptor for ATP by NF449 and suramin: contribution of basic amino acids in the cysteine-rich loop.
Journal: British journal of pharmacology 20120101
Title: Prostaglandin E2 induces spontaneous rhythmic activity in mouse urinary bladder independently of efferent nerves.
Journal: British journal of pharmacology 20120101
Title: Study of the reversal effect of NF449 on neuromuscular blockade induced by d-tubocurarine.
Journal: Life sciences 20110606
Title: Ionotropic NMDA and P2X1/5 receptors mediate synaptically induced Ca2+ signalling in cortical astrocytes.
Journal: Cell calcium 20101001
Title: NF449 is a novel inhibitor of fibroblast growth factor receptor 3 (FGFR3) signaling active in chondrocytes and multiple myeloma cells.
Journal: The Journal of biological chemistry 20100702
Title: Low doses of bisphenol A promote human seminoma cell proliferation by activating PKA and PKG via a membrane G-protein-coupled estrogen receptor.
Journal: Environmental health perspectives 20090701
Title: Bradykinin inhibits the transient outward K+ current in mouse Schwann cells via the cAMP/PKA pathway.
Journal: American journal of physiology. Cell physiology 20090601
Title: Spontaneous purinergic neurotransmission in the mouse urinary bladder.
Journal: The Journal of physiology 20081201
Title: Ectodomain lysines and suramin block of P2X1 receptors.
Journal: The Journal of biological chemistry 20081031
Title: Characterization of pharmacologically active compounds that inhibit poliovirus and enterovirus 71 infectivity.
Journal: The Journal of general virology 20081001
Title: Genistein potentiates protein kinase A activity in porcine coronary artery.
Journal: Molecular and cellular biochemistry 20080401
Title: Inhibition of human and mouse plasma membrane bound NTPDases by P2 receptor antagonists.
Journal: Biochemical pharmacology 20071115
Title: Primary and secondary agonists can use P2X(1) receptors as a major pathway to increase intracellular Ca(2+) in the human platelet.
Journal: Journal of thrombosis and haemostasis : JTH 20070501
Title: P2X purinergic receptor-mediated ionic current in cardiac myocytes of calsequestrin model of cardiomyopathy: implications for the treatment of heart failure.
Journal: American journal of physiology. Heart and circulatory physiology 20070201
Title: Histamine decreases myogenic tone in rat cerebral arteries by H2-receptor-mediated KV channel activation, independent of endothelium and cyclic AMP.
Journal: European journal of pharmacology 20061010
Title: Mechanisms of disease: role of purinergic signaling in the pathophysiology of bladder dysfunction.
Journal: Nature clinical practice. Urology 20060401
Title: Inhibition of platelet functions and thrombosis through selective or nonselective inhibition of the platelet P2 receptors with increasing doses of NF449 [4,4',4'',4'''-(carbonylbis(imino-5,1,3-benzenetriylbis-(carbonylimino)))tetrakis-benzene-1,3-disulfonic acid octasodium salt].
Journal: The Journal of pharmacology and experimental therapeutics 20050701
Title: Profiling at recombinant homomeric and heteromeric rat P2X receptors identifies the suramin analogue NF449 as a highly potent P2X1 receptor antagonist.
Journal: Neuropharmacology 20050301
Title: Progesterone upregulates calcitonin gene-related peptide and adrenomedullin receptor components and cyclic adenosine 3'5'-monophosphate generation in Eker rat uterine smooth muscle cell line.
Journal: Biology of reproduction 20050201
Title: Structure-activity relationships of analogues of NF449 confirm NF449 as the most potent and selective known P2X1 receptor antagonist.
Journal: European journal of medicinal chemistry 20040401
Title: ATP-induced ATP release from astrocytes.
Journal: Journal of neurochemistry 20040101
Title: NF449, a novel picomolar potency antagonist at human P2X1 receptors.
Journal: European journal of pharmacology 20030530
Title: Development of Gs-selective inhibitory compounds.
Journal: Methods in enzymology 20020101
Title: NF449: a subnanomolar potency antagonist at recombinant rat P2X1 receptors.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20010901
Title: Induction of Galphas contributes to the paradoxical stimulation of cytosolic phospholipase A2alpha expression by cortisol in human amnion fibroblasts.
Journal: Molecular endocrinology (Baltimore, Md.)
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Title: Hechler B, et al. Inhibition of platelet functions and thrombosis through selective or nonselective inhibition of the platelet P2 receptors with increasing doses of NF449 ,4',4'',4'''-(carbonylbis(imino-5,1,3-benzenetriylbis-(carbonylimino)))tetrakis-benzene-1,3-disulfonic acid octasodium salt J Pharmacol Exp Ther. 2005;314(1):232-243.
