Title: Activation of TRPV3 by Wood Smoke Particles and Roles in Pneumotoxicity.
Journal: Chemical research in toxicology 20180521
Title: A novel TRPV4-specific agonist inhibits monocyte adhesion and atherosclerosis.
Journal: Oncotarget 20160621
Title: Identification of potent Yes1 kinase inhibitors using a library screening approach.
Journal: Bioorganic & medicinal chemistry letters 20130801
Title: Optical recording reveals novel properties of GSK1016790A-induced vanilloid transient receptor potential channel TRPV4 activity in primary human endothelial cells.
Journal: Molecular pharmacology 20120901
Title: TRPV4 in porcine lens epithelium regulates hemichannel-mediated ATP release and Na-K-ATPase activity.
Journal: American journal of physiology. Cell physiology 20120615
Title: Elementary Ca2+ signals through endothelial TRPV4 channels regulate vascular function.
Journal: Science (New York, N.Y.) 20120504
Title: Hypotonicity-induced TRPV4 function in renal collecting duct cells: modulation by progressive cross-talk with Ca2+-activated K+ channels.
Journal: Cell calcium 20120201
Title: Effects of TRPV4 cation channel activation on the primary bladder afferent activities of the rat.
Journal: Neurourology and urodynamics 20120101
Title: Characterization of transient receptor potential vanilloid channel 4 (TRPV4) in human corneal endothelial cells.
Journal: Experimental eye research 20111101
Title: Mutations in TRPV4 cause an inherited arthropathy of hands and feet.
Journal: Nature genetics 20111002
Title: Transient receptor potential vanilloid 4 (TRPV4)-dependent calcium influx and ATP release in mouse oesophageal keratinocytes.
Journal: The Journal of physiology 20110715
Title: The polymodal ion channel transient receptor potential vanilloid 4 modulates calcium flux, spiking rate, and apoptosis of mouse retinal ganglion cells.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20110511
Title: Determinants of TRPV4 activity following selective activation by small molecule agonist GSK1016790A.
Journal: PloS one 20110101
Title: Inhibition of the cation channel TRPV4 improves bladder function in mice and rats with cyclophosphamide-induced cystitis.
Journal: Proceedings of the National Academy of Sciences of the United States of America 20101102
Title: Activation of Trpv4 reduces the hyperproliferative phenotype of cystic cholangiocytes from an animal model of ARPKD.
Journal: Gastroenterology 20100701
Title: TRPV4-mediated endothelial Ca2+ influx and vasodilation in response to shear stress.
Journal: American journal of physiology. Heart and circulatory physiology 20100201
Title: Functional TRPV4 channels and an absence of capsaicin-evoked currents in freshly-isolated, guinea-pig urothelial cells.
Journal: Channels (Austin, Tex.) 20090101
Title: N-((1S)-1-{[4-((2S)-2-{[(2,4-dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I.
Journal: The Journal of pharmacology and experimental therapeutics 20080801
Title: Systemic activation of the transient receptor potential vanilloid subtype 4 channel causes endothelial failure and circulatory collapse: Part 2.
Journal: The Journal of pharmacology and experimental therapeutics 20080801
Title: Kevin S Thorneloe, et al. N-((1S)-1-{-((2S)-2-{[(2,4-dichlorophenyl)sulfonylamino}-3-hydroxypropanoyl)-1-piperazinylcarbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I. J Pharmacol Exp Ther. 2008 Aug;326(2):432-42.
Title: J Fichna, et al. Transient receptor potential vanilloid 4 inhibits mouse colonic motility by activating NO-dependent enteric neurotransmission. J Mol Med (Berl). 2015 Dec;93(12):1297-309.
