[1]Prasad,RajNandan;Bariana,DilbaghS.;Fung,Anthony;Savic,Milica;Tietje,Karin;etal.[JournalofMedicinalChemistry,1980,vol.23,#3,p.313-319]
[1]Gallo-Rodriguez,Carola;Ji,Xiao-duo;Melman,Neli;Siegman,BarryD.;Sanders,LawrenceH.;etal.[JournalofMedicinalChemistry,1994,vol.37,#5,p.636-646]
[1]Gallo-Rodriguez,Carola;Ji,Xiao-duo;Melman,Neli;Siegman,BarryD.;Sanders,LawrenceH.;etal.[JournalofMedicinalChemistry,1994,vol.37,#5,p.636-646]
[1]Prasad,RajNandan;Bariana,DilbaghS.;Fung,Anthony;Savic,Milica;Tietje,Karin;etal.[JournalofMedicinalChemistry,1980,vol.23,#3,p.313-319]
[1]Olsson;Kusachi;Thompson;Ukena;Padgett;Daly[Journalofmedicinalchemistry,1986,vol.29,#9,p.1683-1689]
Title: The wakefulness promoting drug Modafinil causes adenosine receptor-mediated upregulation of receptor activator of nuclear factor κB ligand in osteoblasts: Negative impact of the drug on peak bone accrual in rats.
Journal: Toxicology and applied pharmacology 20180601
Title: Enhanced A2A adenosine receptor-mediated increase in coronary flow in type I diabetic mice.
Journal: Journal of molecular and cellular cardiology 20160101
Title: Structure-activity relationship in a purine-scaffold compound series with selectivity for the endoplasmic reticulum Hsp90 paralog Grp94.
Journal: Journal of medicinal chemistry 20150514
Title: The effects of A2B receptor modulators on vascular endothelial growth factor and nitric oxide axis in chronic cyclosporine nephropathy.
Journal: Journal of pharmacology & pharmacotherapeutics 20150101
Title: Adenosine A2A receptor as a drug discovery target.
Journal: Journal of medicinal chemistry 20140508
Title: Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Journal: European journal of medicinal chemistry 20130501
Title: Inhibitory effects of benzodiazepines on the adenosine A(2B) receptor mediated secretion of interleukin-8 in human mast cells.
Journal: European journal of pharmacology 20130130
Title: Adenosine A2A receptor modulates vascular response in soluble epoxide hydrolase-null mice through CYP-epoxygenases and PPARγ.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20130101
Title: Downregulation of A(1) and A(2B) adenosine receptors in human trisomy 21 mesenchymal cells from first-trimester chorionic villi.
Journal: Biochimica et biophysica acta 20121101
Title: Structural sweet spot for A1 adenosine receptor activation by truncated (N)-methanocarba nucleosides: receptor docking and potent anticonvulsant activity.
Journal: Journal of medicinal chemistry 20120927
Title: Adenosine signaling promotes regeneration of pancreatic β cells in vivo.
Journal: Cell metabolism 20120606
Title: The A2B adenosine receptor modulates pulmonary hypertension associated with interstitial lung disease.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20120601
Title: Optimization of adenosine 5'-carboxamide derivatives as adenosine receptor agonists using structure-based ligand design and fragment screening.
Journal: Journal of medicinal chemistry 20120510
Title: Loss of adenosine A2B receptor mediated relaxant responses in the aged female rat bladder; effects of dietary phytoestrogens.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20120501
Title: Opposing effects of ATP and adenosine on barrier function of rat coronary microvasculature.
Journal: Journal of molecular and cellular cardiology 20120501
Title: 3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A₂B adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20120223
Title: The role of mechanical forces and adenosine in the regulation of intestinal enterochromaffin cell serotonin secretion.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20120201
Title: The effect of adenosine on pro-inflammatory cytokine production by porcine T cells.
Journal: Veterinary immunology and immunopathology 20120115
Title: Evaluation of molecular modeling of agonist binding in light of the crystallographic structure of an agonist-bound A₂A adenosine receptor.
Journal: Journal of medicinal chemistry 20120112
Title: Enhanced IL-6 transcriptional response to adenosine receptor ligands in horses with lower airway inflammation.
Journal: Equine veterinary journal 20120101
Title: Adenosine promotes alternative macrophage activation via A2A and A2B receptors.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20120101
Title: Adora2b adenosine receptor engagement enhances regulatory T cell abundance during endotoxin-induced pulmonary inflammation.
Journal: PloS one 20120101
Title: Adenosine reduces cell surface expression of toll-like receptor 4 and inflammation in response to lipopolysaccharide and matrix products.
Journal: Journal of cardiovascular translational research 20111201
Title: Pharmacological characterization of adenosine receptors on isolated human bronchi.
Journal: American journal of respiratory cell and molecular biology 20111201
Title: Purinergic regulation of high-glucose-induced caspase-1 activation in the rat retinal Müller cell line rMC-1.
Journal: American journal of physiology. Cell physiology 20111101
Title: Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20111001
Title: Regulation of innate immunity by the nucleotide pathway in children with idiopathic nephrotic syndrome.
Journal: Clinical and experimental immunology 20111001
Title: Reciprocal modulation of anti-IgE induced histamine release from human mast cells by A₁ and A(2B) adenosine receptors.
Journal: British journal of pharmacology 20110901
Title: Adenosine receptor subtype expression and activation influence the differentiation of mesenchymal stem cells to osteoblasts and adipocytes.
Journal: Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research 20110901
Title: Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.
Journal: European journal of medicinal chemistry 20110901
Title: Adenosine activation of A(2B) receptor(s) is essential for stimulated epithelial ciliary motility and clearance.
Journal: American journal of physiology. Lung cellular and molecular physiology 20110801
Title: 5'-(N-ethylcarboxamido) adenosine improves angiogenesis in transplanted human ovarian tissue.
Journal: Fertility and sterility 20110630
Title: Thermostabilisation of an agonist-bound conformation of the human adenosine A(2A) receptor.
Journal: Journal of molecular biology 20110610
Title: Agonist-bound adenosine A2A receptor structures reveal common features of GPCR activation.
Journal: Nature 20110518
Title: GPCR structure and activation: an essential role for the first extracellular loop in activating the adenosine A2B receptor.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20110201
Title: Links between insulin resistance, adenosine A2B receptors, and inflammatory markers in mice and humans.
Journal: Diabetes 20110201
Title: Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20110127
Title: Effect of fluoxetine or adenosine receptor NECA agonist on G-proteins of C6 glioma cells or NK immunocytes.
Journal: Neuro endocrinology letters 20110101
Title: Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: design, synthesis, and structure-activity relationships.
Journal: Bioorganic & medicinal chemistry 20101101
Title: Both A2a and A2b adenosine receptors at reperfusion are necessary to reduce infarct size in mouse hearts.
Journal: American journal of physiology. Heart and circulatory physiology 20101001
Title: Contraction-induced secretion of VEGF from skeletal muscle cells is mediated by adenosine.
Journal: American journal of physiology. Heart and circulatory physiology 20100901
Title: Inhibition of neutrophil-mediated production of reactive oxygen species (ROS) by endothelial cells is not impaired in anti-neutrophil cytoplasmic autoantibodies (ANCA)-associated vasculitis patients.
Journal: Clinical and experimental immunology 20100801
Title: Multivalent dendrimeric and monomeric adenosine agonists attenuate cell death in HL-1 mouse cardiomyocytes expressing the A(3) receptor.
Journal: Biochemical pharmacology 20100715
Title: The critical role of intracellular zinc in adenosine A(2) receptor activation induced cardioprotection against reperfusion injury.
Journal: Journal of molecular and cellular cardiology 20100701
Title: Involvement of Cx43 phosphorylation in 5'-N-ethylcarboxamide-induced migration and proliferation of mouse embryonic stem cells.
Journal: Journal of cellular physiology 20100701
Title: Involvement of A1 adenosine receptors in altered vascular responses and inflammation in an allergic mouse model of asthma.
Journal: American journal of physiology. Heart and circulatory physiology 20100701
Title: Modulation by salt intake of the vascular response mediated through adenosine A(2A) receptor: role of CYP epoxygenase and soluble epoxide hydrolase.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20100701
Title: Adenosine A(3) receptor stimulation induces protection of skeletal muscle from eccentric exercise-mediated injury.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20100701
Title: Fibroblast-specific expression of AC6 enhances beta-adrenergic and prostacyclin signaling and blunts bleomycin-induced pulmonary fibrosis.
Journal: American journal of physiology. Lung cellular and molecular physiology 20100601
Title: Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation.
Journal: Journal of medicinal chemistry 20100527
Title: Oxidative/nitrosative stress selectively altered A(2B) adenosine receptors in chronic obstructive pulmonary disease.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20100401
Title: Stimulation of adenosine A(2B) receptors induces interleukin-6 secretion in cardiac fibroblasts via the PKC-delta-P38 signalling pathway.
Journal: British journal of pharmacology 20100401
Title: Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions.
Journal: Molecular pharmacology 20100401
Title: A new role for the A2b adenosine receptor in regulating platelet function.
Journal: Journal of thrombosis and haemostasis : JTH 20100401
Title: Novel 8-(furan-2-yl)-3-substituted thiazolo [5,4-e][1,2,4] triazolo[1,5-c] pyrimidine-2(3H)-thione derivatives as potential adenosine A(2A) receptor antagonists.
Journal: Bioorganic & medicinal chemistry 20100401
Title: A volume regulatory response can be triggered by nucleosides in human erythrocytes, a perfect osmometer no longer.
Journal: The Journal of biological chemistry 20100226
Title: Adenosine mediated desensitization of cAMP signaling enhances T-cell responses.
Journal: European journal of immunology 20100201
Title: Synthesis and evaluation of two series of 4'-aza-carbocyclic nucleosides as adenosine A2A receptor agonists.
Journal: Bioorganic & medicinal chemistry letters 20100201
Title: Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands.
Journal: British journal of pharmacology 20100201
Title: 2-Dialkynyl derivatives of (N)-methanocarba nucleosides: 'Clickable' A(3) adenosine receptor-selective agonists.
Journal: Bioorganic & medicinal chemistry 20100115
Title: Pharmacological validation of a telemetric model for the measurement of bronchoconstriction in conscious rats.
Journal: Journal of pharmacological and toxicological methods 20100101
Title: Elevated cAMP opposes (TNF-alpha)-induced loss in the barrier integrity of corneal endothelium.
Journal: Molecular vision 20100101
Title: Theophylline inhibits the differentiation of human monocyte into dendritic cell potentially via adenosine receptor antagonism.
Journal: Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20091201
Title: Purinergic modulation in the development of the rat uncrossed retinotectal pathway.
Journal: Neuroscience 20091110
Title: Adenosine A2A and A2B receptors work in concert to induce a strong protection against reperfusion injury in rat hearts.
Journal: Journal of molecular and cellular cardiology 20091101
Title: Absence of adenosine-mediated aortic relaxation in A(2A) adenosine receptor knockout mice.
Journal: American journal of physiology. Heart and circulatory physiology 20091101
Title: Cholesterol-dependent regulation of adenosine A(2A) receptor-mediated anion secretion in colon epithelial cells.
Journal: Experimental cell research 20091015
Title: Adenosine-evoked hyperpolarization of retinal ganglion cells is mediated by G-protein-coupled inwardly rectifying K+ and small conductance Ca2+-activated K+ channel activation.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20090909
Title: Differential regulation of HIF-1alpha isoforms in murine macrophages by TLR4 and adenosine A(2A) receptor agonists.
Journal: Journal of leukocyte biology 20090901
Title: 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity.
Journal: Journal of medicinal chemistry 20090709
Title: Synthesis of hybrid analogues of caffeine and eudistomin D and its affinity for adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20090701
Title: Intranasal administration of NECA can induce both anti-inflammatory and pro-inflammatory effects in BALB/c mice: evidence for A 2A receptor sub-type mediation of NECA-induced anti-inflammatory effects.
Journal: Pulmonary pharmacology & therapeutics 20090601
Title: 5'-N-ethylcarboxamide induces IL-6 expression via MAPKs and NF-kappaB activation through Akt, Ca(2+)/PKC, cAMP signaling pathways in mouse embryonic stem cells.
Journal: Journal of cellular physiology 20090601
Title: Adenosine signaling mediates SUMO-1 modification of IkappaBalpha during hypoxia and reoxygenation.
Journal: The Journal of biological chemistry 20090515
Title: Vascular endothelial growth factors synthesized by human lung mast cells exert angiogenic effects.
Journal: The Journal of allergy and clinical immunology 20090501
Title: Regulation of cardiac fibroblast collagen synthesis by adenosine: roles for Epac and PI3K.
Journal: American journal of physiology. Cell physiology 20090501
Title: Novel 2- and 4-substituted 1H-imidazo[4,5-c]quinolin-4-amine derivatives as allosteric modulators of the A3 adenosine receptor.
Journal: Journal of medicinal chemistry 20090409
Title: High-salt diet enhances mouse aortic relaxation through adenosine A2A receptor via CYP epoxygenases.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20090301
Title: Involvement of NO and KATP channel in adenosine A2B receptors induced cardiovascular regulation in the posterior hypothalamus of rats.
Journal: Journal of cardiovascular pharmacology 20090201
Title: Adenosine induces loss of actin stress fibers and inhibits contraction in hepatic stellate cells via Rho inhibition.
Journal: Hepatology (Baltimore, Md.) 20090101
Title: In vitro induction of T cells that are resistant to A2 adenosine receptor-mediated immunosuppression.
Journal: British journal of pharmacology 20090101
Title: Contribution of NO, ATP-sensitive K+ channels and prostaglandins to adenosine receptor agonists-induced relaxation of the rat tail artery.
Journal: Pharmacological reports : PR 20090101
Title: The A(2B)-D(2) receptor interaction that controls carotid body catecholamines release locates between the last two steps of hypoxic transduction cascade.
Journal: Advances in experimental medicine and biology 20090101
Title: An antagonistic interaction between A2B adenosine and D2 dopamine receptors modulates the function of rat carotid body chemoreceptor cells.
Journal: Journal of neurochemistry 20081201
Title: Modulation of insulin release by adenosine A1 receptor agonists and antagonists in INS-1 cells: the possible contribution of 86Rb+ efflux and 45Ca2+ uptake.
Journal: Cell biochemistry and function 20081201
Title: cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Journal: Journal of medicinal chemistry 20081127
Title: Role of CYP epoxygenases in A2A AR-mediated relaxation using A2A AR-null and wild-type mice.
Journal: American journal of physiology. Heart and circulatory physiology 20081101
Title: A new chemical tool (C0036E08) supports the role of adenosine A(2B) receptors in mediating human mast cell activation.
Journal: Biochemical pharmacology 20081001
Title: Selective inhibitory effect of adenosine A1 receptor agonists on the proliferation of human tumor cell lines.
Journal: Iranian biomedical journal 20081001
Title: Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC.
Journal: European journal of pharmacology 20080820
Title: 2-Amino-6-furan-2-yl-4-substituted nicotinonitriles as A2A adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20080814
Title: N6-1,3-diphenylurea derivatives of 2-phenyl-9-benzyladenines and 8-azaadenines: synthesis and biological evaluation as allosteric modulators of A2A adenosine receptors.
Journal: European journal of medicinal chemistry 20080801
Title: A2B adenosine receptors regulate the mucus clearance component of the lung's innate defense system.
Journal: American journal of respiratory cell and molecular biology 20080801
Title: Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
Journal: Journal of medicinal chemistry 20080724
Title: Adenosine induces airway hyperresponsiveness through activation of A3 receptors on mast cells.
Journal: The Journal of allergy and clinical immunology 20080701
Title: Adenosine receptor agonists attenuate the development of diazepam withdrawal-induced sensitization in mice.
Journal: European journal of pharmacology 20080624
Title: Effects of IL-4 and IL-13 on adenosine receptor expression and responsiveness of the human mast cell line 1.
Journal: International immunopharmacology 20080601
Title: Modulation of murine dendritic cell function by adenine nucleotides and adenosine: involvement of the A(2B) receptor.
Journal: European journal of immunology 20080601
Title: Local stimulation of the adenosine A2B receptors induces an increased release of IL-6 in mouse striatum: an in vivo microdialysis study.
Journal: Journal of neurochemistry 20080501
Title: Up-regulation of A 2B adenosine receptor in A 2A adenosine receptor knockout mouse coronary artery.
Journal: Journal of molecular and cellular cardiology 20080501
Title: Design of (N)-methanocarba adenosine 5'-uronamides as species-independent A3 receptor-selective agonists.
Journal: Bioorganic & medicinal chemistry letters 20080501
Title: Probing distal regions of the A2B adenosine receptor by quantitative structure-activity relationship modeling of known and novel agonists.
Journal: Journal of medicinal chemistry 20080410
Title: Synthesis of eudistomin D analogues and its effects on adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20080401
Title: Derivatives of 4-amino-6-hydroxy-2-mercaptopyrimidine as novel, potent, and selective A3 adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20080327
Title: [Advances in the study of A2B adenosine receptor antagonists].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20080301
Title: Adenosine A2A receptor agonists inhibit lipopolysaccharide-induced production of tumor necrosis factor-alpha by equine monocytes.
Journal: Veterinary immunology and immunopathology 20080115
Title: Involvement of adenosine receptor agonists on the development of hypersensitivity to acute dose of morphine during morphine withdrawal period.
Journal: Pharmacological reports : PR 20080101
Title: Flexible modulation of agonist efficacy at the human A3 adenosine receptor by the imidazoquinoline allosteric enhancer LUF6000.
Journal: BMC pharmacology 20080101
Title: Structure-activity relationships of adenosines with heterocyclic N6-substituents.
Journal: Bioorganic & medicinal chemistry letters 20071215
Title: In vivo adenosine A(2B) receptor desensitization in guinea-pig airway smooth muscle: implications for asthma.
Journal: European journal of pharmacology 20071201
Title: 5-amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a versatile scaffold to obtain potent and selective A3 adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20071115
Title: Adenosine A1 but not A2a receptor agonist reduces hyperalgesia caused by a surgical incision in rats: a pertussis toxin-sensitive G protein-dependent process.
Journal: Anesthesiology 20071101
Title: Adenosine deaminase 1 and concentrative nucleoside transporters 2 and 3 regulate adenosine on the apical surface of human airway epithelia: implications for inflammatory lung diseases.
Journal: Biochemistry 20070911
Title: Protein kinase C protects preconditioned rabbit hearts by increasing sensitivity of adenosine A2b-dependent signaling during early reperfusion.
Journal: Journal of molecular and cellular cardiology 20070901
Title: Pharmacologic characterization of novel adenosine A2A receptor agonists in equine neutrophils.
Journal: American journal of veterinary research 20070901
Title: A(2b) receptor mediates adenosine inhibition of taurine efflux from pituicytes.
Journal: Biology of the cell 20070801
Title: Adenosine receptor activation ameliorates type 1 diabetes.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20070801
Title: Involvement of guanylate cyclase in the cardiovascular response induced by adenosine A2B receptor stimulation in the posterior hypothalamus of the anesthetized rats.
Journal: Autonomic neuroscience : basic & clinical 20070731
Title: Rapid stimulation of presynaptic serotonin transport by A(3) adenosine receptors.
Journal: The Journal of pharmacology and experimental therapeutics 20070701
Title: Involvement of A1 adenosine receptors and neural pathways in adenosine-induced bronchoconstriction in mice.
Journal: American journal of physiology. Lung cellular and molecular physiology 20070701
Title: ATP modulates the release of noradrenaline through two different prejunctional receptors on the adrenergic nerves of rat prostate.
Journal: Clinical and experimental pharmacology & physiology 20070701
Title: Effects of stimulation of adenosine A2A receptors on lipopolysaccharide-induced production of reactive oxygen species by equine neutrophils.
Journal: American journal of veterinary research 20070601
Title: Synthesis of hybrid molecules of caffeine and eudistomin D and its effects on adenosine receptors.
Journal: Bioorganic & medicinal chemistry 20070501
Title: Adenosine is not a direct GHSR agonist--artificial cross-talk between GHSR and adenosine receptor pathways.
Journal: Acta physiologica (Oxford, England) 20070501
Title: Cross-regulation of carbon monoxide and the adenosine A2a receptor in macrophages.
Journal: Journal of immunology (Baltimore, Md. : 1950) 20070501
Title: Structure-activity relationships of 2,N(6),5'-substituted adenosine derivatives with potent activity at the A2B adenosine receptor.
Journal: Journal of medicinal chemistry 20070419
Title: N(6)-[(hetero)aryl/(cyclo)alkyl-carbamoyl-methoxy-phenyl]-(2-chloro)-5'-N-ethylcarboxamido-adenosines: the first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor.
Journal: Bioorganic & medicinal chemistry 20070401
Title: Adenosine opposes thrombin-induced inhibition of intercellular calcium wave in corneal endothelial cells.
Journal: Investigative ophthalmology & visual science 20070401
Title: Effect of a specific and selective A(2B) adenosine receptor antagonist on adenosine agonist AMP and allergen-induced airway responsiveness and cellular influx in a mouse model of asthma.
Journal: The Journal of pharmacology and experimental therapeutics 20070301
Title: New fluorescent adenosine A1-receptor agonists that allow quantification of ligand-receptor interactions in microdomains of single living cells.
Journal: Journal of medicinal chemistry 20070222
Title: Role of adenosine receptors in the regulation of angiogenic factors and neovascularization in hypoxia.
Journal: The Journal of pharmacology and experimental therapeutics 20070201
Title: Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]- 9H-purin-9-yl]-N-ethyl-beta-D-ribofuranuronamide derivatives as useful templates for the development of A2B adenosine receptor agonists.
Journal: Journal of medicinal chemistry 20070125
Title: Structure-activity relationship study of prion inhibition by 2-aminopyridine-3,5-dicarbonitrile-based compounds: parallel synthesis, bioactivity, and in vitro pharmacokinetics.
Journal: Journal of medicinal chemistry 20070111
Title: Evidence for the involvement of nitric oxide in A2B receptor-mediated vasorelaxation of mouse aorta.
Journal: American journal of physiology. Heart and circulatory physiology 20070101
Title: The thyroid disruptor 1,1,1-trichloro-2,2-bis(p-chlorophenyl)-ethane appears to be an uncompetitive inverse agonist for the thyrotropin receptor.
Journal: The Journal of pharmacology and experimental therapeutics 20070101
Title: Intratumoral lymphatic vessels and VEGF-C expression are predictive factors of lymph node relapse in T1-T4 N0 laryngopharyngeal squamous cell carcinoma.
Journal: Annals of surgical oncology 20070101
Title: Human micro- and macrovessel-derived endothelial cells: a comparative study on the effects of adrenaline and a selective adenosine A2-type receptor agonist under normoxic and hypoxic conditions.
Journal: Pharmacological reports : PR 20070101
Title: Regulation of pharmacology by hetero-oligomerization between A1 adenosine receptor and P2Y2 receptor.
Journal: Biochemical and biophysical research communications 20061215
Title: Loss of vascular adenosine A1 receptors with age in the rat heart.
Journal: Vascular pharmacology 20061201
Title: The impact of adenosine and A(2B) receptors on glucose homoeostasis.
Journal: The Journal of pharmacy and pharmacology 20061201
Title: Expression of adenosine receptors in cardiac fibroblasts as a function of insulin and glucose level.
Journal: Archives of biochemistry and biophysics 20061101
Title: Adenosine A1 receptors mediate mobilization of calcium in human bronchial smooth muscle cells.
Journal: American journal of respiratory cell and molecular biology 20061001
Title: Corpus cavernosum from men with vasculogenic impotence is partially resistant to adenosine relaxation due to endothelial A(2B) receptor dysfunction.
Journal: The Journal of pharmacology and experimental therapeutics 20061001
Title: Cross-talk between G(s)- and G(q)-coupled pathways in regulation of interleukin-4 by A(2B) adenosine receptors in human mast cells.
Journal: Molecular pharmacology 20060801
Title: Real-time and high throughput monitoring of cAMP in live cells using a fluorescent membrane potential-sensitive dye.
Journal: Assay and drug development technologies 20060801
Title: NECA at reperfusion limits infarction and inhibits formation of the mitochondrial permeability transition pore by activating p70S6 kinase.
Journal: Basic research in cardiology 20060701
Title: Orthogonal activation of the reengineered A3 adenosine receptor (neoceptor) using tailored nucleoside agonists.
Journal: Journal of medicinal chemistry 20060504
Title: N6-ethyl-2-alkynyl NECAs, selective human A3 adenosine receptor agonists.
Journal: Bioorganic & medicinal chemistry letters 20060501
Title: Postconditioning protects rabbit hearts through a protein kinase C-adenosine A2b receptor cascade.
Journal: Cardiovascular research 20060501
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Characterization of adenosine receptors in the human bladder carcinoma T24 cell line.
Journal: European journal of pharmacology 20060424
Title: Astrocytes promote myelination in response to electrical impulses.
Journal: Neuron 20060316
Title: Moderate hypoxia induces xanthine oxidoreductase activity in arterial endothelial cells.
Journal: Free radical biology & medicine 20060315
Title: Role of the second transmembrane domain of rat adenosine A1 receptor in ligand-receptor interaction.
Journal: Biochemical pharmacology 20060314
Title: Solid phase synthesis and antiprotozoal evaluation of di- and trisubstituted 5'-carboxamidoadenosine analogues.
Journal: Bioorganic & medicinal chemistry 20060301
Title: A membrane-permeable peptide containing the last 21 residues of the G alpha(s) carboxyl terminus inhibits G(s)-coupled receptor signaling in intact cells: correlations between peptide structure and biological activity.
Journal: Molecular pharmacology 20060301
Title: Binding of the viral immunogenic octapeptide VSV8 to native glucose-regulated protein Grp94 (gp96) and its inhibition by the physiological ligands ATP and Ca2+.
Journal: The FEBS journal 20060201
Title: Purinergic substances promote murine keratinocyte proliferation and enhance impaired wound healing in mice.
Journal: Wound repair and regeneration : official publication of the Wound Healing Society [and] the European Tissue Repair Society 20060101
Title: 2-(Benzimidazol-2-yl)quinoxalines: a novel class of selective antagonists at human A(1) and A(3) adenosine receptors designed by 3D database searching.
Journal: Journal of medicinal chemistry 20051229
Title: Pharmacological characterization of novel adenosine ligands in recombinant and native human A2B receptors.
Journal: Biochemical pharmacology 20051125
Title: Influence of adenosine receptor agonists on benzodiazepine withdrawal signs in mice.
Journal: European journal of pharmacology 20051031
Title: Neuroprotective effect of paeoniflorin on cerebral ischemic rat by activating adenosine A1 receptor in a manner different from its classical agonists.
Journal: British journal of pharmacology 20051001
Title: Caffeine intake induces an alteration in human neutrophil A2A adenosine receptors.
Journal: Cellular and molecular life sciences : CMLS 20051001
Title: Gs protein-coupled adenosine receptor signaling and lytic function of activated NK cells.
Journal: Journal of immunology (Baltimore, Md. : 1950) 20051001
Title: Mast cell involvement in the adenosine mediated airway hyper-reactivity in a murine model of ovalbumin-induced lung inflammation.
Journal: British journal of pharmacology 20050801
Title: Adenosine signaling promotes neuronal, catecholaminergic differentiation of primary neural crest cells and CNS-derived CAD cells.
Journal: Molecular and cellular neurosciences 20050701
Title: Involvement of p38-mitogen-activated protein kinase in adenosine receptor-mediated relaxation of coronary artery.
Journal: American journal of physiology. Heart and circulatory physiology 20050601
Title: Expression, pharmacological profile, and functional coupling of A2B receptors in a recombinant system and in peripheral blood cells using a novel selective antagonist radioligand, [3H]MRE 2029-F20.
Journal: Molecular pharmacology 20050601
Title: A2B adenosine receptor mediates human chorionic vasoconstriction and signals through arachidonic acid cascade.
Journal: American journal of physiology. Heart and circulatory physiology 20050501
Title: Human breast cancer cell line MDA-MB-231 expresses endogenous A2B adenosine receptors mediating a Ca2+ signal.
Journal: British journal of pharmacology 20050501
Title: Involvement of mast cells in adenosine-mediated bronchoconstriction and inflammation in an allergic mouse model.
Journal: The Journal of pharmacology and experimental therapeutics 20050401
Title: Adenosine agonist regulation of outward active transport of fluorescein across retinal pigment epithelium in rabbits.
Journal: Experimental eye research 20050401
Title: Binding thermodynamics as a tool to investigate the mechanisms of drug-receptor interactions: thermodynamics of cytoplasmic steroid/nuclear receptors in comparison with membrane receptors.
Journal: Journal of medicinal chemistry 20050324
Title: The role of adenosine A2A and A2B receptors in the regulation of TNF-alpha production by human monocytes.
Journal: Biochemical pharmacology 20050315
Title: Synthesis, biological evaluation, and molecular modeling of ribose-modified adenosine analogues as adenosine receptor agonists.
Journal: Journal of medicinal chemistry 20050310
Title: Role of A1 adenosine receptors in regulation of vascular tone.
Journal: American journal of physiology. Heart and circulatory physiology 20050301
Title: Adenosine receptor mediates nicotine-induced antinociception in formalin test.
Journal: Pharmacological research 20050301
Title: Different modulation of inhibitory and stimulatory pathways mediated by adenosine after chronic in vivo agonist exposure.
Journal: Brain research 20050121
Title: A2B adenosine receptor activity is reduced in neutrophils from patients with systemic sclerosis.
Journal: Arthritis research & therapy 20050101
Title: Modulation of cytokine release by purine receptors in patients with rheumatoid arthritis.
Journal: Clinical and experimental rheumatology 20050101
Title: Participation of adenosine system in the ketamine-induced motor activity in mice.
Journal: Pharmacological reports : PR 20050101
Title: New 8-substituted xanthiene derivatives as potent bronchodilators.
Journal: Farmaco (Societa chimica italiana : 1989) 20050101
Title: Ring opening reactions: synthesis of AICAR analogs as potential antimetabolite agents.
Journal: Nucleosides, nucleotides & nucleic acids 20050101
Title: Functional effects of enhancing or silencing adenosine A2b receptors in cardiac fibroblasts.
Journal: American journal of physiology. Heart and circulatory physiology 20041201
Title: Regulation of A2B adenosine receptor functioning by tumour necrosis factor a in human astroglial cells.
Journal: Journal of neurochemistry 20041201
Title: 2-Substituted adenosine derivatives: affinity and efficacy at four subtypes of human adenosine receptors.
Journal: Biochemical pharmacology 20041115
Title: Adenosine receptors involved in modulation of noradrenaline release in isolated rat tail artery.
Journal: European journal of pharmacology 20041103
Title: Coupling of the human A1 adenosine receptor to different heterotrimeric G proteins: evidence for agonist-specific G protein activation.
Journal: British journal of pharmacology 20041101
Title: Synthesis and biological evaluation of novel N6-[4-(substituted)sulfonamidophenylcarbamoyl]adenosine-5'-uronamides as A3 adenosine receptor agonists.
Journal: Journal of medicinal chemistry 20041021
Title: Influence of the combined treatment of LY 300164 (an AMPA/kainate receptor antagonist) with adenosine receptor agonists on the electroconvulsive threshold in mice.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20041001
Title: Negative chronotropic response to adenosine receptor stimulation in rat right atria after run training.
Journal: Clinical and experimental pharmacology & physiology 20041001
Title: Purine modulation of cytokine release during diuretic therapy of rheumatoid arthritis.
Journal: Nucleosides, nucleotides & nucleic acids 20041001
Title: ATP-sensitive potassium channels and endogenous adenosine are involved in spinal antinociception produced by locus coeruleus stimulation.
Journal: The International journal of neuroscience 20040801
Title: Synthesis and biological activity of new potential agonists for the human adenosine A2A receptor.
Journal: Journal of medicinal chemistry 20040729
Title: [3H]OSIP339391, a selective, novel, and high affinity antagonist radioligand for adenosine A2B receptors.
Journal: Biochemical pharmacology 20040715
Title: New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with an improved selectivity profile compared to the reference agonist N-ethylcarboxamidoadenosine.
Journal: Journal of medicinal chemistry 20040715
Title: 1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.
Journal: Journal of medicinal chemistry 20040701
Title: Adenosine-activated mast cells induce IgE synthesis by B lymphocytes: an A2B-mediated process involving Th2 cytokines IL-4 and IL-13 with implications for asthma.
Journal: Journal of immunology (Baltimore, Md. : 1950) 20040615
Title: Comparative analysis of putative agonist-binding modes in the human A1 adenosine receptor.
Journal: Chembiochem : a European journal of chemical biology 20040607
Title: Adenosine receptor, protein kinase G, and p38 mitogen-activated protein kinase-dependent up-regulation of serotonin transporters involves both transporter trafficking and activation.
Journal: Molecular pharmacology 20040601
Title: An IgM class anti-neutrophil cytoplasm antibody inhibits neutrophil adhesion and apoptosis via a Syk dependent signaling cascade.
Journal: Molecular immunology 20040601
Title: Characterization of glycine N-methyltransferase from rabbit liver.
Journal: Biochemistry and cell biology = Biochimie et biologie cellulaire 20040601
Title: Development of a sensitive and HTS-compatible reporter gene assay for functional analysis of human adenosine A2a receptors in CHO-K1 cells.
Journal: Assay and drug development technologies 20040601
Title: [(3)H]Adenosine uptake in brainstem membranes of CD-1 mice lacking the adenosine A(2a) receptor.
Journal: Life sciences 20040528
Title: The role of intraspinal adenosine A1 receptors in sympathetic regulation.
Journal: European journal of pharmacology 20040510
Title: Novel amino acid derived natural products from the ascidian Atriolum robustum: identification and pharmacological characterization of a unique adenosine derivative.
Journal: Journal of medicinal chemistry 20040422
Title: Regional and endothelial differences in cyclosporine attenuation of adenosine receptor-mediated vasorelaxations.
Journal: Journal of cardiovascular pharmacology 20040401
Title: NECA and bradykinin at reperfusion reduce infarction in rabbit hearts by signaling through PI3K, ERK, and NO.
Journal: Journal of molecular and cellular cardiology 20040301
Title: Pulmonary surfactant secretion in briefly cultured mouse type II cells.
Journal: American journal of physiology. Lung cellular and molecular physiology 20040201
Title: A1 and A2A adenosine receptor modulation of alpha 1-adrenoceptor-mediated contractility in human cultured prostatic stromal cells.
Journal: British journal of pharmacology 20040101
Title: A2B adenosine receptor agonists: synthesis and biological evaluation of 2-phenylhydroxypropynyl adenosine and NECA derivatives.
Journal: Nucleosides, nucleotides & nucleic acids 20040101
Title: Effects of stable adenosine receptor agonists on bone marrow hematopoietic cells as inferred from the cytotoxic action of 5-fluorouracil.
Journal: Physiological research 20040101
Title: The role of the basolateral outwardly rectifying chloride channel in human airway epithelial anion secretion.
Journal: American journal of respiratory cell and molecular biology 20031201
Title: Structure of the N-terminal domain of GRP94. Basis for ligand specificity and regulation.
Journal: The Journal of biological chemistry 20031128
Title: A(2A) adenosine receptor ligands and proinflammatory cytokines induce PC 12 cell death through apoptosis.
Journal: Biochemical pharmacology 20031115
Title: Modeling the adenosine receptors: comparison of the binding domains of A2A agonists and antagonists.
Journal: Journal of medicinal chemistry 20031106
Title: Oligodendrocytes express functional A1 adenosine receptors that stimulate cellular migration.
Journal: Glia 20031101
Title: Comparative pharmacological studies on the A2 adenosine receptor agonist 5'-n-ethyl-carboxamidoadenosine and its F19 isotope labelled derivative.
Journal: Journal of pharmacological sciences 20031101
Title: Adenosine receptor agonists: from basic medicinal chemistry to clinical development.
Journal: Expert opinion on emerging drugs 20031101
Title: Effect of taurine deficiency on adenosine receptor-mediated relaxation of the rat aorta.
Journal: Vascular pharmacology 20031101
Title: The G(s)-coupled adenosine A(2B) receptor recruits divergent pathways to regulate ERK1/2 and p38.
Journal: Experimental cell research 20031015
Title: Adenosine-induced IL-6 expression in pituitary folliculostellate cells is mediated via A2b adenosine receptors coupled to PKC and p38 MAPK.
Journal: British journal of pharmacology 20031001
Title: Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor antagonists. Influence of the N5 substituent on the affinity at the human A 3 and A 2B adenosine receptor subtypes: a molecular modeling investigation.
Journal: Journal of medicinal chemistry 20030925
Title: Antagonist pharmacology of adenosine A2B receptors from rat, guinea pig and dog.
Journal: European journal of pharmacology 20030815
Title: Blockade of A2A adenosine receptors prevents basic fibroblast growth factor-induced reactive astrogliosis in rat striatal primary astrocytes.
Journal: Glia 20030801
Title: An angiogenic switch in macrophages involving synergy between Toll-like receptors 2, 4, 7, and 9 and adenosine A(2A) receptors.
Journal: The American journal of pathology 20030801
Title: Adenosine slows migration of dendritic cells but does not affect other aspects of dendritic cell maturation.
Journal: The Journal of investigative dermatology 20030801
Title: Activation of mast cells by immunoglobulin E-receptor cross-linkage, but not through adenosine receptors, induces A1 expression and promotes survival.
Journal: Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20030801
Title: Adenosine A 2B receptors modulate cAMP levels and induce CREB but not ERK1/2 and p38 phosphorylation in rat skeletal muscle cells.
Journal: Biochemical and biophysical research communications 20030718
Title: Characterization of adenosine receptor(s) involved in adenosine-induced bronchoconstriction in an allergic mouse model.
Journal: American journal of physiology. Lung cellular and molecular physiology 20030601
Title: Purinergic receptors on microglial cells: functional expression in acute brain slices and modulation of microglial activation in vitro.
Journal: The European journal of neuroscience 20030601
Title: Adenosine affects the calcium dynamics of rat portal vein.
Journal: Autonomic & autacoid pharmacology 20030601
Title: Binding of HTLV-1 virions to T cells occurs by a temperature and calcium-dependent process and is blocked by certain type 2 adenosine receptor antagonists.
Journal: Virus research 20030501
Title: N6-cyclopentyl-2-(3-phenylaminocarbonyltriazene-1-yl)adenosine (TCPA), a very selective agonist with high affinity for the human adenosine A1 receptor.
Journal: Journal of medicinal chemistry 20030410
Title: Adenosine stimulates anion secretion across cultured and native adult human vas deferens epithelia.
Journal: Biology of reproduction 20030301
Title: Central nervous system effects of caffeine and adenosine on fatigue.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology 20030201
Title: Regional differences in the adenosine A(2) receptor-mediated modulation of contractions in rat vas deferens.
Journal: European journal of pharmacology 20030124
Title: Adenosine receptor subtypes mediating coronary vasodilation in rat hearts.
Journal: Journal of cardiovascular pharmacology 20030101
Title: Synthesis of carbocyclic analogues of MECA and NECA 1,2-disubstituted as potential adenosine receptor agonists.
Journal: Nucleosides, nucleotides & nucleic acids 20030101
Title: Effects of doxazosin and propranolol on A2A adenosine receptors in essential hypertension.
Journal: Hypertension (Dallas, Tex. : 1979) 20021201
Title: Possible role of mast cells in cineole-induced scratching behavior in mice.
Journal: Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association 20021001
Title: Structural determinants of A(3) adenosine receptor activation: nucleoside ligands at the agonist/antagonist boundary.
Journal: Journal of medicinal chemistry 20020926
Title: The effects of adenosine receptor agonists and antagonists on morphine state-dependent memory of passive avoidance.
Journal: Neurobiology of learning and memory 20020901
Title: Involvement of mitogen protein kinase cascade in agonist-mediated human A(3) adenosine receptor regulation.
Journal: Biochimica et biophysica acta 20020819
Title: Relaxation of the mouse isolated aorta and carotid artery in response to adenosine analogues in genetically-modified mice lacking the adenosine A(2A) receptor.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20020801
Title: Induction of interleukin 8 release from the HMC-1 mast cell line: synergy between stem cell factor and activators of the adenosine A(2b) receptor.
Journal: Biochemical pharmacology 20020715
Title: Synergistic up-regulation of vascular endothelial growth factor expression in murine macrophages by adenosine A(2A) receptor agonists and endotoxin.
Journal: The American journal of pathology 20020601
Title: [The [18F]-FNECA serves as a suitable radioligand for PET investigation of purinergic receptor expression].
Journal: Orvosi hetilap 20020526
Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
Journal: The Journal of biological chemistry 20020419
Title: Adenosine receptor-mediated control of in vitro release of pain-related neuropeptides from the rat spinal cord.
Journal: European journal of pharmacology 20020419
Title: Role of vasodilator-stimulated phosphoprotein in PKA-induced changes in endothelial junctional permeability.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20020401
Title: Dopaminergic mechanism for caffeine-produced cocaine seeking in rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20020401
Title: Rhythmic gene expression in pituitary depends on heterologous sensitization by the neurohormone melatonin.
Journal: Nature neuroscience 20020301
Title: Basolateral potassium channels of rabbit colon epithelium: role in sodium absorption and chloride secretion.
Journal: Biochimica et biophysica acta 20020218
Title: Cardiac effects of adenosine in A(2A) receptor knockout hearts: uncovering A(2B) receptors.
Journal: American journal of physiology. Heart and circulatory physiology 20020201
Title: Evidence for an atypical receptor mediating the augmented bronchoconstrictor response to adenosine induced by allergen challenge in actively sensitized Brown Norway rats.
Journal: British journal of pharmacology 20020201
Title: Effects of adenosine on bacterial lipopolysaccharide- and interleukin 1-induced nitric oxide release from equine articular chondrocytes.
Journal: American journal of veterinary research 20020201
Title: Effects of adenosine agonists on consumptive behaviour and body temperature.
Journal: The Journal of pharmacy and pharmacology 20020201
Title: 2,5'-Disubstituted adenosine derivatives: evaluation of selectivity and efficacy for the adenosine A(1), A(2A), and A(3) receptor.
Journal: Journal of medicinal chemistry 20020117
Title: Comparison of the vascular effects of adenosine in isolated mouse heart and aorta.
Journal: American journal of physiology. Heart and circulatory physiology 20020101
Title: Cocaine-induced hyperactivity is more influenced by adenosine receptor agonists than amphetamine-induced hyperactivity.
Journal: Polish journal of pharmacology 20020101
Title: 7-Nitrobenzofurazan (NBD) derivatives of 5'-N-ethylcarboxamidoadenosine (NECA) as new fluorescent probes for human A(3) adenosine receptors.
Journal: Bioorganic & medicinal chemistry letters 20011203
Title: Regulation of SP-B and SP-C secretion in rat type II cells in primary culture.
Journal: American journal of physiology. Lung cellular and molecular physiology 20011201
Title: Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides.
Journal: Journal of medicinal chemistry 20011122
Title: Effects of adenosine receptor agonists and antagonists on pentylenetetrazole-induced amnesia.
Journal: European journal of pharmacology 20011102
Title: Inhibition of human mast cell activation with the novel selective adenosine A(2B) receptor antagonist 3-isobutyl-8-pyrrolidinoxanthine (IPDX)(2).
Journal: Biochemical pharmacology 20011101
Title: Adenosine-mediated hypotension in in vivo guinea-pig: receptors involved and role of NO.
Journal: British journal of pharmacology 20011001
Title: The plasma protein extravasation induced by adenosine and its analogues in the rat dorsal skin: evidence for the involvement of capsaicin sensitive primary afferent neurones and mast cells.
Journal: British journal of pharmacology 20010901
Title: Pharmacological characterization of adenosine receptors in PGT-beta mouse pineal gland tumour cells.
Journal: British journal of pharmacology 20010901
Title: Arrestin specificity for G protein-coupled receptors in human airway smooth muscle.
Journal: The Journal of biological chemistry 20010831
Title: P2Y(11) receptor expression by human lymphocytes: evidence for two cAMP-linked purinoceptors.
Journal: European journal of pharmacology 20010831
Title: 5'-O-alkyl ethers of N,2-substituted adenosine derivatives: partial agonists for the adenosine A1 and A3 receptors.
Journal: Journal of medicinal chemistry 20010830
Title: Why do asthmatic subjects respond so strongly to inhaled adenosine?
Journal: Life sciences 20010803
Title: Proliferation, migration, and ERK activation in human retinal endothelial cells through A(2B) adenosine receptor stimulation.
Journal: Investigative ophthalmology & visual science 20010801
Title: Functional characterization of coronary vascular adenosine receptors in the mouse.
Journal: British journal of pharmacology 20010801
Title: Introduction of alkynyl chains on C-8 of adenosine led to very selective antagonists of the A(3) adenosine receptor.
Journal: Bioorganic & medicinal chemistry letters 20010723
Title: Withdrawal and bidirectional cross-withdrawal responses in rats treated with adenosine agonists and morphine.
Journal: Life sciences 20010706
Title: Role of cyclic nucleotides in vasodilations of the rat thoracic aorta induced by adenosine analogues.
Journal: British journal of pharmacology 20010701
Title: Modulation of ethanol-induced motor incoordination by mouse striatal A(1) adenosinergic receptor.
Journal: Brain research bulletin 20010701
Title: Protective effect of adenosine receptor agonists in a new model of epilepsy--seizures evoked by mitochondrial toxin, 3-nitropropionic acid, in mice.
Journal: Neuroscience letters 20010608
Title: Differential effects of UTP, ATP, and adenosine on ciliary activity of human nasal epithelial cells.
Journal: American journal of physiology. Cell physiology 20010601
Title: Ring-Constrained (N)-methanocarba nucleosides as adenosine receptor agonists: independent 5'-uronamide and 2'-deoxy modifications.
Journal: Bioorganic & medicinal chemistry letters 20010521
Title: Age-related changes in adenosine-mediated relaxation of coronary and aortic smooth muscle.
Journal: American journal of physiology. Heart and circulatory physiology 20010501
Title: Aberrant amplification of A(2A) receptor signaling in striatal cells expressing mutant huntingtin.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20010501
Title: Glucocorticoid enhances the response of type II cells from newborn rats to surfactant secretagogues.
Journal: Biochimica et biophysica acta 20010430
Title: Pharmacology of a unique adenosine binding site in rat brain using a selective ligand.
Journal: Clinical and experimental pharmacology & physiology 20010401
Title: Effect of 9-(6,7-dideoxy-beta-D-allo-hept-5-ynofuranosyl)adenine on noradrenaline release from vascular sympathetic nerves.
Journal: Clinical and experimental pharmacology & physiology 20010401
Title: Adenosine inhibits neutrophil vascular endothelial growth factor release and transendothelial migration via A2B receptor activation.
Journal: Shock (Augusta, Ga.) 20010401
Title: Adenosine agonists CGS 21680 and NECA inhibit the initiation of cocaine self-administration.
Journal: Pharmacology, biochemistry, and behavior 20010401
Title: [3H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors.
Journal: Biochemical pharmacology 20010315
Title: Adenosine enhances neuroexcitability by inhibiting a slow postspike afterhyperpolarization in rabbit vagal afferent neurons.
Journal: Circulation 20010306
Title: Design, synthesis, and evaluation of novel A2A adenosine receptor agonists.
Journal: Journal of medicinal chemistry 20010215
Title: Extracellular adenosine-induced apoptosis in mouse neuroblastoma cells: studies on involvement of adenosine receptors and adenosine uptake.
Journal: Biochemical pharmacology 20010215
Title: Regulation of G protein-coupled receptor-adenylyl cyclase responsiveness in human airway smooth muscle by exogenous and autocrine adenosine.
Journal: American journal of respiratory cell and molecular biology 20010201
Title: 3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: a new class of selective A1 adenosine receptor antagonists.
Journal: Journal of medicinal chemistry 20010201
Title: Nucleosides and nucleotides. 200. Reinvestigation of 5'-N-ethylcarboxamidoadenosine derivatives: structure-activity relationships for P(3) purinoceptor-like proteins.
Journal: Journal of medicinal chemistry 20010118
Title: Adenosine A2B receptors behave as an alternative anchoring protein for cell surface adenosine deaminase in lymphocytes and cultured cells.
Journal: Molecular pharmacology 20010101
Title: Cloning of a chick A3 adenosine receptor: characterization of ligand binding and receptor-effector coupling of chick A1 and A3 adenosine receptors.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20010101
Title: Characterization of prejunctional purinoceptors inhibiting noradrenaline release in rat mesenteric arteries.
Journal: Japanese journal of pharmacology 20010101
Title: Synthesis and adenosine receptor affinity and potency of 8-alkynyl derivatives of adenosine.
Journal: Nucleosides, nucleotides & nucleic acids 20010101
Title: Role of endothelium in ischaemia-induced myocardial dysfunction of isolated working hearts: cardioprotection by activation of adenosine A(2A) receptors.
Journal: Journal of autonomic pharmacology 20010101
Title: Why are A(2B) receptors low-affinity adenosine receptors? Mutation of Asn273 to Tyr increases affinity of human A(2B) receptor for 2-(1-Hexynyl)adenosine.
Journal: Molecular pharmacology 20001201
Title: [(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.
Journal: Molecular pharmacology 20000501
Title: Activation of the A3 adenosine receptor affects cell cycle progression and cell growth.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 20000301
Title: Characterization of human A(2B) adenosine receptors: radioligand binding, western blotting, and coupling to G(q) in human embryonic kidney 293 cells and HMC-1 mast cells.
Journal: Molecular pharmacology 19991001
Title: 2-Substituted N-ethylcarboxamidoadenosine derivatives as high-affinity agonists at human A3 adenosine receptors.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 19990801
Title: Identification of the adenine binding site of the human A1 adenosine receptor.
Journal: The Journal of biological chemistry 19990205
Title: Differences in the order of potency for agonists but not antagonists at human and rat adenosine A2A receptors.
Journal: Biochemical pharmacology 19990101
Title: 2'-C-Methyl analogues of selective adenosine receptor agonists: synthesis and binding studies.
Journal: Journal of medicinal chemistry 19980507
Title: Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 19980101
Title: Effect of adenosine receptor agonists and antagonists on morphine-induced catalepsy in mice.
Journal: European journal of pharmacology 19971029
Title: Mechanism and pressor relevance of the short-term cardiovascular and renin excitatory actions of the selective A2A-adenosine receptor agonists.
Journal: Journal of cardiovascular pharmacology 19970901
Title: Pharmacological characterization of novel A3 adenosine receptor-selective antagonists.
Journal: Neuropharmacology 19970901
Title: Adenosine A2 receptors modulate haloperidol-induced catalepsy in rats.
Journal: European journal of pharmacology 19970611
Title: Characterization of human A2A adenosine receptors with the antagonist radioligand [3H]-SCH 58261.
Journal: British journal of pharmacology 19970501
Title: Characterization of the human brain putative A2B adenosine receptor expressed in Chinese hamster ovary (CHO.A2B4) cells.
Journal: British journal of pharmacology 19961101
Title: Effects of adenosine analogues on apomorphine-induced penile erection in rats.
Journal: General pharmacology 19951201
Title: Site-directed mutagenesis identifies residues involved in ligand recognition in the human A2a adenosine receptor.
Journal: The Journal of biological chemistry 19950609
Title: Species difference in the G protein selectivity of the human and bovine A1-adenosine receptor.
Journal: The Journal of biological chemistry 19941223
Title: Role of the second extracellular loop of adenosine receptors in agonist and antagonist binding. Analysis of chimeric A1/A3 adenosine receptors.
Journal: The Journal of biological chemistry 19941007
Title: Structure-activity relationships of N6-benzyladenosine-5'-uronamides as A3-selective adenosine agonists.
Journal: Journal of medicinal chemistry 19940304
Title: Functional characterization of the A2b adenosine receptor in NIH 3T3 fibroblasts.
Journal: Biochemical pharmacology 19940302
Title: A threonine residue in the seventh transmembrane domain of the human A1 adenosine receptor mediates specific agonist binding.
Journal: The Journal of biological chemistry 19940128
Title: Noradrenaline but not dopamine involved in NMDA receptor-mediated hyperalgesia induced by theophylline in awake rats.
Journal: European journal of pharmacology 19940124
Title: Molecular cloning and characterization of the human A3 adenosine receptor.
Journal: Proceedings of the National Academy of Sciences of the United States of America 19931101
Title: N-ethyl-carboxamide adenosine inhibits perioral dyskinesias induced by sulpiride + SKF 38393 in rabbits.
Journal: European journal of pharmacology 19921113
Title: [Effects of agonists and antagonists of benzodiazepine, GABA and NMDA receptors, on caffeine-induced seizures in mice].
Journal: Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology 19920801
Title: Enhanced fatty acid biosynthesis and normal surfactant secretion in hypertrophic rat type II cells.
Journal: The American journal of physiology 19910601
Title: Allosteric enhancement of adenosine A1 receptor binding and function by 2-amino-3-benzoylthiophenes.
Journal: Molecular pharmacology 19901201
Title: Binding of the adenosine A2 receptor ligand [3H]CGS 21680 to human and rat brain: evidence for multiple affinity sites.
Journal: Journal of neurochemistry 19901101
Title: Hemodynamic effects of adenosine agonists in the conscious spontaneously hypertensive rat.
Journal: The Journal of pharmacology and experimental therapeutics 19900901
Title: Caffeine-induced seizures: apparent proconvulsant action of N-ethyl carboxamidoadenosine (NECA).
Journal: Life sciences 19900101
Title: [3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain.
Journal: The Journal of pharmacology and experimental therapeutics 19891201
Title: Comparison of the behavioral effects of adenosine agonists and dopamine antagonists in mice.
Journal: Psychopharmacology 19890101
Title: Potent convulsant actions of the adenosine receptor antagonist, xanthine amine congener (XAC).
Journal: Life sciences 19890101
Title: Doxofylline, an antiasthmatic drug lacking affinity for adenosine receptors.
Journal: Archives internationales de pharmacodynamie et de therapie 19880101
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Title: Elsherbiny NM, et al. Reno-protective effect of NECA in diabetic nephropathy: implication of IL-18 and ICAM-1. Eur Cytokine Netw. 2012 Jul-Sep;23(3):78-86.
