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58822-25-6,MFCD00076406
Catalog No.:AA01DNMM

58822-25-6 | 1-5-b-Neoendorphin (human)

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Purity
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10mg
98%
in stock  
$150.00   $105.00
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25mg
98
in stock  
$254.00   $178.00
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100mg
98%
in stock  
$816.00   $572.00
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  • Technical Information
  • Properties
  • Literature
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  • Technical Information
  • Properties
  • Literature
Technical Information
Catalog Number:
AA01DNMM
Chemical Name:
1-5-b-Neoendorphin (human)
CAS Number:
58822-25-6
Molecular Formula:
C28H37N5O7
Molecular Weight:
555.6227
MDL Number:
MFCD00076406
SMILES:
O=C(CNC(=O)C(Cc1ccc(cc1)O)N)NCC(=O)NC(C(=O)NC(C(=O)O)CC(C)C)Cc1ccccc1
Properties
Computed Properties
 
Complexity:
854  
Covalently-Bonded Unit Count:
1  
Defined Atom Stereocenter Count:
3  
Heavy Atom Count:
40  
Hydrogen Bond Acceptor Count:
8  
Hydrogen Bond Donor Count:
7  
Rotatable Bond Count:
15  
XLogP3:
-2.3  

Literature

Title: In vivo and in vitro evaluation of novel μ-opioid receptor agonist compounds.

Journal: European journal of pharmacology 20151115

Title: Superoxide reaction with tyrosyl radicals generates para-hydroperoxy and para-hydroxy derivatives of tyrosine.

Journal: Journal of the American Chemical Society 20121010

Title: Oxidative and nitrative modifications of enkephalins by human neutrophils: effect of nitroenkephalin on leukocyte functional responses.

Journal: Amino acids 20120801

Title: Neuroendocrine system of the digestive tract in Rhamdia quelen juvenile: an immunohistochemical study.

Journal: Tissue & cell 20120801

Title: Quantitative multiple reaction monitoring of peptide abundance introduced via a capillary zone electrophoresis-electrospray interface.

Journal: Analytical chemistry 20120717

Title: New insights into the neuroanatomical distribution and phylogeny of opioids and POMC-derived peptides in fish.

Journal: General and comparative endocrinology 20120701

Title: Conformation-specific spectroscopy of peptide fragment ions in a low-temperature ion trap.

Journal: Journal of the American Society for Mass Spectrometry 20120601

Title: Covalent and non-covalent binding in the ion/ion charge inversion of peptide cations with benzene-disulfonic acid anions.

Journal: Journal of mass spectrometry : JMS 20120601

Title: Direct peptide bioconjugation/PEGylation at tyrosine with linear and branched polymeric diazonium salts.

Journal: Journal of the American Chemical Society 20120502

Title: Design and self-assembly of a leucine-enkephalin analogue in different nanostructures: application of nanovesicles.

Journal: Small (Weinheim an der Bergstrasse, Germany) 20120410

Title: Conformational space exploration of Met- and Leu-enkephalin using the MOLS method, molecular dynamics, and Monte Carlo simulation--a comparative study.

Journal: Biopolymers 20120301

Title: How hot are your ions in TWAVE ion mobility spectrometry?

Journal: Journal of the American Society for Mass Spectrometry 20120301

Title: Fast, selective, and sensitive analysis of low-abundance peptides in human plasma by electromembrane extraction.

Journal: Analytica chimica acta 20120224

Title: Microfluidic dual emitter electrospray ionization source for accurate mass measurements.

Journal: Analytical chemistry 20120207

Title: Hypoxic preconditioning attenuates global cerebral ischemic injury following asphyxial cardiac arrest through regulation of delta opioid receptor system.

Journal: Neuroscience 20120127

Title: N-Protonated isomers as gateways to peptide ion fragmentation.

Journal: Journal of the American Society for Mass Spectrometry 20111201

Title: Adaptation of a 3-D quadrupole ion trap for dipolar DC collisional activation.

Journal: Journal of the American Society for Mass Spectrometry 20110901

Title: [Affection of acupotomy lysis on leu-enkephalin (L-ENK) content in different parts of centrum of rats with knee osteoarthritis].

Journal: Zhongguo gu shang = China journal of orthopaedics and traumatology 20110801

Title: Peptide synthesis 'in water' by a solution-phase method using water-dispersible nanoparticle Boc-amino acid.

Journal: Journal of peptide science : an official publication of the European Peptide Society 20110701

Title: Microdialysis and mass spectrometric monitoring of dopamine and enkephalins in the globus pallidus reveal reciprocal interactions that regulate movement.

Journal: Journal of neurochemistry 20110701

Title: The effect of hydrothermal treatment on column performance for monolithic silica capillary columns.

Journal: Journal of chromatography. A 20110610

Title: Oxytocin in the periaqueductal gray participates in pain modulation in the rat by influencing endogenous opiate peptides.

Journal: Peptides 20110601

Title: HPLC/MS/MS for quantification of two types of neurotransmitters in rat brain and application: myocardial ischemia and protection of Sheng-Mai-San.

Journal: Journal of pharmaceutical and biomedical analysis 20110428

Title: Differentiation between Aδ and C fibre evoked nociceptive reflexes by TTX resistance and opioid sensitivity in the cat.

Journal: Neuroscience research 20110301

Title: Regulated proenkephalin expression in human skin and cultured skin cells.

Journal: The Journal of investigative dermatology 20110301

Title: Lipophilic derivatives of leu-enkephalinamide: in vitro permeability, stability and in vivo nasal delivery.

Journal: Bioorganic & medicinal chemistry 20110215

Title: Micro-opioid receptor activation in the basolateral amygdala mediates the learning of increases but not decreases in the incentive value of a food reward.

Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20110202

Title: [The extended amygdala system and self-stimulation of the lateral hypothalamus in rats: modulation with opiates and opioids].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20110201

Title: Cavitation of liquid flow in electrospray mass spectrometry especially for addition of internal calibrant in 'accurate mass' measurements.

Journal: Rapid communications in mass spectrometry : RCM 20110115

Title: Leucine enkephalin--a mass spectrometry standard.

Journal: Mass spectrometry reviews 20110101

Title: Intrathecal herpes simplex virus type 1 amplicon vector-mediated human proenkephalin reduces chronic constriction injury-induced neuropathic pain in rats.

Journal: Molecular medicine reports 20110101

Title: [Role of serotonin receptors in the delta-opioid immunosuppression].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20101201

Title: Axonal branching patterns of nucleus accumbens neurons in the rat.

Journal: The Journal of comparative neurology 20101115

Title: A bioinspired synthetic approach for building metal-organic frameworks with accessible metal centers.

Journal: Inorganic chemistry 20101115

Title: Multi-component signaling complexes of the delta-opioid receptor with STAT5B and G proteins.

Journal: Neuropharmacology 20100901

Title: Oxazolone versus macrocycle structures for Leu-enkephalin b2-b4: insights from infrared multiple-photon dissociation spectroscopy and gas-phase hydrogen/deuterium exchange.

Journal: Journal of the American Society for Mass Spectrometry 20100801

Title: Electroosmotic sampling. Application to determination of ectopeptidase activity in organotypic hippocampal slice cultures.

Journal: Analytical chemistry 20100801

Title: Measuring internal energy deposition in collisional activation using hydrated ion nanocalorimetry to obtain peptide dissociation energies and entropies.

Journal: Journal of the American Society for Mass Spectrometry 20100701

Title: Dissociation kinetics of singly protonated leucine enkephalin investigated by time-resolved photodissociation tandem mass spectrometry.

Journal: Journal of the American Society for Mass Spectrometry 20100701

Title: [Methionine-enkephalin (Met5-Enk) and leucine-enkephalin (Leu5-Enk)].

Journal: Nihon rinsho. Japanese journal of clinical medicine 20100701

Title: Stable isotope labeling method targeting terminal tyrosine for relative peptide quantitation using mass spectrometry.

Journal: Analytical biochemistry 20100601

Title: Delivery of neuropeptides from the periphery to the brain: studies with enkephalin.

Journal: ACS chemical neuroscience 20100519

Title: A high recovery microsampling device based on a microdialysis probe for peptide sampling.

Journal: Analytical biochemistry 20100415

Title: 'Carba'-analogues of fentanyl are opioid receptor agonists.

Journal: Journal of medicinal chemistry 20100408

Title: Analogues of both Leu- and Met-enkephalin containing a constrained dipeptide isostere prepared from a Baylis-Hillman adduct.

Journal: Amino acids 20100401

Title: Immunohistochemical characterization of neurones in the hypoglossal nucleus of the pig.

Journal: Anatomia, histologia, embryologia 20100401

Title: Coordination of trivalent metal cations to peptides: results from IRMPD spectroscopy and theory.

Journal: The journal of physical chemistry. A 20100121

Title: Interactions of tyrosine in Leu-enkephalin at a membrane-water interface: an ultrafast two-dimensional infrared study combined with density functional calculations and molecular dynamics simulations.

Journal: The journal of physical chemistry. B 20100121

Title: Laser-induced acoustic desorption coupled with a linear quadrupole ion trap mass spectrometer.

Journal: Analytical chemistry 20100115

Title: Opioid and non-opioid receptor-mediated immunoregulatory role of leucine-enkephalin in teleost Channa punctatus.

Journal: Fish & shellfish immunology 20100101

Title: Mean daily plasma concentrations of beta-endorphin, leu-enkephalin, ACTH, cortisol, and DHEAS in epileptic patients with complex partial seizures evolving to generalized tonic-clonic seizures.

Journal: Endokrynologia Polska 20100101

Title: Plasma endogenous enkephalin levels in early systemic sclerosis: clinical and laboratory associations.

Journal: Clinical and experimental rheumatology 20100101

Title: Immune response of submissive and aggressive mice under conditions of opioid receptor activation.

Journal: Bulletin of experimental biology and medicine 20091201

Title: Synthesis and receptor binding of opioid peptide analogues containing beta3-homo-amino acids.

Journal: Journal of peptide science : an official publication of the European Peptide Society 20091101

Title: Rapid magnetic catch-and-release purification by hydrophobic interactions.

Journal: Langmuir : the ACS journal of surfaces and colloids 20090915

Title: Modification with organometallic compounds improves crossing of the blood-brain barrier of [Leu5]-enkephalin derivatives in an in vitro model system.

Journal: Chembiochem : a European journal of chemical biology 20090720

Title: Arginine vasopressin antinociception in the rat nucleus raphe magnus is involved in the endogenous opiate peptide and serotonin system.

Journal: Peptides 20090701

Title: Opioid and progesterone signaling is obligatory for early human embryogenesis.

Journal: Stem cells and development 20090601

Title: Direct quantitation of peptide mixtures without standards using clusters formed by electrospray ionization mass spectrometry.

Journal: Analytical chemistry 20090515

Title: Central administration of somatostatin stimulates feeding behavior in chicks.

Journal: General and comparative endocrinology 20090501

Title: Does the endogenous opiate system play a role in the Restless Legs Syndrome? A pilot post-mortem study.

Journal: Journal of the neurological sciences 20090415

Title: Hypertensive state, independent of hypertrophy, exhibits an attenuated decrease in systolic function on cardiac kappa-opioid receptor stimulation.

Journal: American journal of physiology. Heart and circulatory physiology 20090401

Title: Practical aspects of in vivo detection of neuropeptides by microdialysis coupled off-line to capillary LC with multistage MS.

Journal: Analytical chemistry 20090315

Title: Benzotriazole-assisted solid-phase assembly of Leu-enkephalin, amyloid beta segment 34-42, and other 'difficult' peptide sequences.

Journal: The Journal of organic chemistry 20090306

Title: Novel role for the delta-opioid receptor in hypoxic preconditioning in rat retinas.

Journal: Journal of neurochemistry 20090201

Title: A neuropathological study of autosomal-dominant chorea-acanthocytosis with a mutation of VPS13A.

Journal: Acta neuropathologica 20090101

Title: Spiny versus stubby: 3D reconstruction of human myenteric (type I) neurons.

Journal: Histochemistry and cell biology 20090101

Title: [The influence of leu-enkephalin on the bile secretion function in the rat liver during pharmacological modulation of the autonomous nervous system].

Journal: Fiziolohichnyi zhurnal (Kiev, Ukraine : 1994) 20090101

Title: Dilution-free analysis from picoliter droplets by nano-electrospray ionization mass spectrometry.

Journal: Angewandte Chemie (International ed. in English) 20090101

Title: The relationship and co-localization of vasoactive intestinal peptide (VIP)- and Leu5-enkephalin (LENK)-immunoreactivity in the female genital tract of the pig.

Journal: Polish journal of veterinary sciences 20090101

Title: Peptide-phospholipid complex formation at liquid-liquid interfaces.

Journal: Analytical chemistry 20081215

Title: Ovarian steroids modulate leu-enkephalin levels and target leu-enkephalinergic profiles in the female hippocampal mossy fiber pathway.

Journal: Brain research 20080926

Title: Identification of leucine-enkephalin radical oxidation products by liquid chromatography tandem mass spectrometry.

Journal: Biomedical chromatography : BMC 20080901

Title: Distinct morphological and immunohistochemical features and different growth rates among four human neuroblastomas heterotransplanted into nude mice.

Journal: Medical molecular morphology 20080901

Title: Arylation of Phe and Tyr side chains of unprotected peptides by a Suzuki-Miyaura reaction in water.

Journal: Organic letters 20080807

Title: An in vitro comparison of microdialysis relative recovery of Met- and Leu-enkephalin using cyclodextrins and antibodies as affinity agents.

Journal: Analytica chimica acta 20080714

Title: Conformational dynamics of free and catalytically active thermolysin are indistinguishable by hydrogen/deuterium exchange mass spectrometry.

Journal: Biochemistry 20080617

Title: Identification of modulating residues defining the catalytic cleft of insulin-regulated aminopeptidase.

Journal: Biochemistry and cell biology = Biochimie et biologie cellulaire 20080601

Title: Evidence for effect of GM1 on opioid peptide conformation: NMR study on leucine enkephalin in ganglioside-containing isotropic phospholipid bicelles.

Journal: Langmuir : the ACS journal of surfaces and colloids 20080520

Title: Internalisation of the mu-opioid receptor by endomorphin-1 and leu-enkephalin is dependant on aromatic amino acid residues.

Journal: Bioorganic & medicinal chemistry 20080415

Title: Effects of leucine-enkephalin on catalase activity and hydrogen peroxide levels in the haemolymph of the Pacific Oyster (Crassostrea gigas).

Journal: Molecules (Basel, Switzerland) 20080415

Title: Hydrolysis of various bioactive peptides by goat brain dipeptidylpeptidase-III homologue.

Journal: Cell biochemistry and function 20080401

Title: On-line electrogeneration of copper-peptide complexes in microspray mass spectrometry.

Journal: Journal of the American Society for Mass Spectrometry 20080401

Title: A selective fluorescence reaction for peptides and chromatographic analysis.

Journal: Peptides 20080301

Title: Surface-induced dissociation of peptides and protein complexes in a quadrupole/time-of-flight mass spectrometer.

Journal: Analytical chemistry 20080301

Title: On the dynamics of fragment isomerization in collision-induced dissociation of peptides.

Journal: The journal of physical chemistry. A 20080214

Title: Reactivity and oxidative potential of fructose and glucose in enkephalin-sugar model systems.

Journal: Amino acids 20080201

Title: Use of preproenkephalin knockout mice and selective inhibitors of enkephalinases to investigate the role of enkephalins in various behaviours.

Journal: Psychopharmacology 20080201

Title: Great increase in antinociceptive potency of [Leu5]enkephalin after peptidase inhibition.

Journal: Journal of pharmacological sciences 20080201

Title: CE hydrogen deuterium exchange-MS in peptide analysis.

Journal: Electrophoresis 20080101

Title: Central inhibition of opioid receptor subtypes and its effect on haemorrhagic hypotension in conscious sheep.

Journal: Acta physiologica (Oxford, England) 20070901

Title: Two-photon excitation fluorescence cross-correlation assay for ligand-receptor binding: cell membrane nanopatches containing the human micro-opioid receptor.

Journal: Analytical chemistry 20070901

Title: Experimental design optimization of the capillary electrophoresis separation of leucine enkephalin and its immune complex.

Journal: Journal of separation science 20070901

Title: Effects of leucine-enkephalin on potassium currents in neurons in the rat respiratory center in vitro.

Journal: Neuroscience and behavioral physiology 20070901

Title: Reaction products in mass spectrometry elucidated with infrared spectroscopy.

Journal: Physical chemistry chemical physics : PCCP 20070807

Title: Detection and characterization of N-alpha-chloramines by electrospray tandem mass spectrometry.

Journal: Analytical biochemistry 20070715

Title: Dynamic collision-induced dissociation of peptides in a quadrupole ion trap mass spectrometer.

Journal: Analytical chemistry 20070715

Title: Arginine vasopressin induces periaqueductal gray release of enkephalin and endorphin relating to pain modulation in the rat.

Journal: Regulatory peptides 20070705

Title: Solid-phase peptide synthesis using nanoparticulate amino acids in water.

Journal: Journal of peptide science : an official publication of the European Peptide Society 20070701

Title: Structure-activity relationships of Leu-Enkephalin analog with (4-Carboxamido)phenylalanine substituted for tyrosine: a molecular dynamics study.

Journal: Biopolymers 20070615

Title: Infrared spectroscopy and theoretical studies on gas-phase protonated leu-enkephalin and its fragments: direct experimental evidence for the mobile proton.

Journal: Journal of the American Chemical Society 20070509

Title: Microsphere entrapped emitters for sample preconcentration and electrospray ionization mass spectrometry.

Journal: Analytical chemistry 20070501

Title: Quantitative conformationally sampled pharmacophore for delta opioid ligands: reevaluation of hydrophobic moieties essential for biological activity.

Journal: Journal of medicinal chemistry 20070419

Title: Fragmentation of leucine enkephalin as a function of laser fluence in a MALDI TOF-TOF.

Journal: Journal of the American Society for Mass Spectrometry 20070401

Title: Opioid peptides as possible neuromodulators in the frog peripheral nerve system.

Journal: Neuropeptides 20070401

Title: Insulin-regulated aminopeptidase: analysis of peptide substrate and inhibitor binding to the catalytic domain.

Journal: Biological chemistry 20070401

Title: Molecular basis of branched peptides resistance to enzyme proteolysis.

Journal: Chemical biology & drug design 20070301

Title: Opioid limbic circuit for reward: interaction between hedonic hotspots of nucleus accumbens and ventral pallidum.

Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20070214

Title: Influence of acute and chronic treadmill exercise on rat plasma lactate and brain NPY, L-ENK, DYN A1-13.

Journal: Cellular and molecular neurobiology 20070201

Title: Presynaptic delta opioid receptors regulate ethanol actions in central amygdala.

Journal: The Journal of pharmacology and experimental therapeutics 20070201

Title: Dual-source mass spectrometer with MALDI-LIT-ESI configuration.

Journal: Journal of proteome research 20070201

Title: Lowering the concentration limits of detection by on-line solid-phase extraction-capillary electrophoresis-electrospray mass spectrometry.

Journal: Journal of chromatography. A 20070126

Title: Reactions of hydrogen atoms with met-enkephalin and related peptides.

Journal: Chemistry (Weinheim an der Bergstrasse, Germany) 20070101

Title: Immunohistochemical organization of the forebrain in the white sturgeon, Acipenser transmontanus.

Journal: Brain, behavior and evolution 20070101

Title: RB101-mediated protection of endogenous opioids: potential therapeutic utility?

Journal: CNS drug reviews 20070101

Title: Plasma met-enkephalin, beta-endorphin and leu-enkephalin levels in human hepatic encephalopathy.

Journal: Eastern Mediterranean health journal = La revue de sante de la Mediterranee orientale = al-Majallah al-sihhiyah li-sharq al-mutawassit 20070101

Title: Novel non-PEG derived polyethers as solid supports. 2. Solid-phase synthesis studies.

Journal: Journal of combinatorial chemistry 20070101

Title: Arginine vasopressin enhances periaqueductal gray synthesis and secretion of enkephalin and endorphin in the rat.

Journal: Brain research bulletin 20061211

Title: Chemical coding of myenteric neurons with different axonal projection patterns in the porcine ileum.

Journal: Journal of anatomy 20061201

Title: Use of an aromatase inhibitor in patients with polycystic ovary syndrome: a prospective randomized trial.

Journal: Fertility and sterility 20061101

Title: Thiophene backbone amide linkers, a new class of easily prepared and highly acid-labile linkers for solid-phase synthesis.

Journal: The Journal of organic chemistry 20060901

Title: Modeling the amide I bands of small peptides.

Journal: The Journal of chemical physics 20060728

Title: Transformations of bioactive peptides in the presence of sugars--characterization and stability studies of the adducts generated via the Maillard reaction.

Journal: Bioorganic & medicinal chemistry 20060715

Title: Energetics and dynamics of fragmentation of protonated leucine enkephalin from time- and energy-resolved surface-induced dissociation studies.

Journal: The journal of physical chemistry. A 20060713

Title: Determination of cooling rates in a quadrupole ion trap.

Journal: Journal of the American Society for Mass Spectrometry 20060701

Title: The effects of leucine-enkephalin on the membrane potential and activity of rat respiratory center neurons in vitro.

Journal: Neuroscience and behavioral physiology 20060701

Title: Oxidative and nitrative modifications of enkephalins by reactive nitrogen species.

Journal: Free radical research 20060701

Title: Enkephalinergic afferents of the centromedial amygdala in the rat.

Journal: The Journal of comparative neurology 20060620

Title: A pulsed field gradient NMR diffusion investigation of enkephalin peptide-sodium dodecyl sulfate micelle association.

Journal: Magnetic resonance in chemistry : MRC 20060601

Title: In vitro evaluation of the potential of thiomers for the nasal administration of Leu-enkephalin.

Journal: Amino acids 20060601

Title: Vibrational dynamics of morphine in relation to Leu5--and Met5-enkephalins.

Journal: Indian journal of biochemistry & biophysics 20060601

Title: Delta and mu opioid receptors from the brain of a urodele amphibian, the rough-skinned newt Taricha granulosa: cloning, heterologous expression, and pharmacological characterization.

Journal: General and comparative endocrinology 20060501

Title: Peptide-phospholipid cross-linking reactions: identification of leucine enkephalin-alka(e)nal-glycerophosphatidylcholine adducts by tandem mass spectrometry.

Journal: Journal of the American Society for Mass Spectrometry 20060501

Title: The existence of opioid receptors in the cochlea of guinea pigs.

Journal: The European journal of neuroscience 20060501

Title: [Effect of leu-enkephalin on potassium currents in neurons of the respiratory center of rats in vitro].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20060501

Title: Reversible lipidization for the oral delivery of leu-enkephalin.

Journal: Journal of drug targeting 20060401

Title: Investigation of interaction of Leu-enkephalin with lipid membranes.

Journal: Colloids and surfaces. B, Biointerfaces 20060315

Title: Modulation of cardiovascular excitatory responses in rats by transcutaneous magnetic stimulation: role of the spinal cord.

Journal: Journal of applied physiology (Bethesda, Md. : 1985) 20060301

Title: Determination of enkephalin peptides by nonaqueous capillary electrophoresis with electrochemical detection.

Journal: Electrophoresis 20060301

Title: Investigation of the route of absorption of lipid and sugar modified leu-enkephalin analogues and their enzymatic stability using the caco-2 cell monolayer system.

Journal: Medicinal chemistry (Shariqah (United Arab Emirates)) 20060301

Title: Only arginine vasopressin, not oxytocin and endogenous opiate peptides, in hypothalamic paraventricular nucleus play a role in acupuncture analgesia in the rat.

Journal: Brain research bulletin 20060215

Title: Synthesis and biological evaluation of leucine enkephalin turn mimetics.

Journal: Organic & biomolecular chemistry 20060207

Title: Three-dimensional representation of the neurotransmitter systems of the human hypothalamus: inputs of the gonadotrophin hormone-releasing hormone neuronal system.

Journal: Journal of neuroendocrinology 20060201

Title: The superior colliculus of the camel: a neuronal-specific nuclear protein (NeuN) and neuropeptide study.

Journal: Journal of anatomy 20060201

Title: A new electrochemical HPLC method for analysis of enkephalins and endomorphins.

Journal: Journal of neuroscience methods 20060115

Title: Orientation and conformational preference of leucine-enkephalin at the surface of a hydrated dimyristoylphosphatidylcholine bilayer: NMR and MD simulation.

Journal: Journal of the American Chemical Society 20060111

Title: Through central arginine vasopressin, not oxytocin and endogenous opiate peptides, glutamate sodium induces hypothalamic paraventricular nucleus enhancing acupuncture analgesia in the rat.

Journal: Neuroscience research 20060101

Title: Ultra-performance liquid chromatography coupled to time-of-flight mass spectrometry for robust, high-throughput quantitative analysis of an automated metabolic stability assay, with simultaneous determination of metabolic data.

Journal: Rapid communications in mass spectrometry : RCM 20060101

Title: Extrahypothalamic corticoliberin receptors regulate the reinforcing effects of self-stimulation.

Journal: Doklady biological sciences : proceedings of the Academy of Sciences of the USSR, Biological sciences sections 20060101

Title: [Evenly tritium-labeled peptides and their in vivo and in vitro biodegradation].

Journal: Bioorganicheskaia khimiia 20060101

Title: Top-down analysis of basic proteins by microchip capillary electrophoresis mass spectrometry.

Journal: Rapid communications in mass spectrometry : RCM 20060101

Title: Endogenous signaling complexity in neuropeptides- leucine- and methionine-enkephalin.

Journal: Cellular and molecular neurobiology 20060101

Title: [Astressin blockade of amygdaloid corticoliberin receptors eliminates the stimulating effects of amphetamine, morphine and leu-enkephalin on brain self-stimulation].

Journal: Eksperimental'naia i klinicheskaia farmakologiia 20060101

Title: [Leu-enkephalin modulates gastric secretion activated by various stimulants].

Journal: Eksperimental'naia i klinicheskaia farmakologiia 20060101

Title: Effect of co-solvents on the characteristics of enkephalin microcapsules.

Journal: Journal of biomaterials science. Polymer edition 20060101

Title: Combination of sustained off-resonance irradiation and on-resonance excitation in FT-ICR.

Journal: Analytical chemistry 20051201

Title: Multiplex multidimensional nanoLC-MS system for targeted proteomic analyses.

Journal: Electrophoresis 20051201

Title: Subclass opioid receptors associated with the cardiovascular depression after traumatic shock and the antishock effects of its specific receptor antagonists.

Journal: Shock (Augusta, Ga.) 20051101

Title: Ischemic preconditioning increases the bioavailability of cardiac enkephalins.

Journal: American journal of physiology. Heart and circulatory physiology 20051001

Title: Capillary liquid chromatography and tandem mass spectrometry for the quantification of enkephalins in cerebrospinal fluid.

Journal: Journal of separation science 20050901

Title: Reduced kappa-opioid activity in a rat model of cholestasis.

Journal: European journal of pharmacology 20050822

Title: [Methionine-enkephalin (Met-Enk) and leucine-enkephalin (Leu-Enk)].

Journal: Nihon rinsho. Japanese journal of clinical medicine 20050801

Title: Microglial NADPH oxidase mediates leucine enkephalin dopaminergic neuroprotection.

Journal: Annals of the New York Academy of Sciences 20050801

Title: Double labelling immunohistochemistry on the nerve fibres of retractor clitoridis muscle of the sow.

Journal: Veterinary research communications 20050801

Title: Analysis and separation of enkephalin and dalargin analogues and fragments by capillary zone electrophoresis.

Journal: Journal of chromatography. A 20050715

Title: MALDI of individual biomolecule-containing airborne particles in an ion trap mass spectrometer.

Journal: Analytical chemistry 20050701

Title: [The effect of leu-enkephalin on membrane potential and activity of the rat respiratory center neurons in vitro].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20050601

Title: Oxygen-sensitive {delta}-opioid receptor-regulated survival and death signals: novel insights into neuronal preconditioning and protection.

Journal: The Journal of biological chemistry 20050422

Title: Ionic-liquid-supported peptide synthesis demonstrated by the synthesis of Leu(5)-enkephalin.

Journal: The Journal of organic chemistry 20050415

Title: Inverse agonism and neutral antagonism at wild-type and constitutively active mutant delta opioid receptors.

Journal: The Journal of pharmacology and experimental therapeutics 20050401

Title: Induction of delta-opioid receptor function in the midbrain after chronic morphine treatment.

Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20050323

Title: Internalization and Src activity regulate the time course of ERK activation by delta opioid receptor ligands.

Journal: The Journal of biological chemistry 20050304

Title: Differential mechanisms of antianalgesia induced by endomorphin-1 and endomorphin-2 in the ventral periaqueductal gray of the rat.

Journal: The Journal of pharmacology and experimental therapeutics 20050301

Title: Substance P and opioid peptidergic innervation of the anterior eye segment of the rat: an immunohistochemical study.

Journal: Journal of anatomy 20050301

Title: Sugar amino acids in designing new molecules.

Journal: Glycoconjugate journal 20050301

Title: Striatal opioid peptide content in an animal model of spontaneous stereotypic behavior.

Journal: Behavioural brain research 20050227

Title: Capillary liquid chromatography with MS3 for the determination of enkephalins in microdialysis samples from the striatum of anesthetized and freely-moving rats.

Journal: Journal of mass spectrometry : JMS 20050201

Title: Morphology of enkephalin-immunoreactive myenteric neurons in the human gut.

Journal: Histochemistry and cell biology 20050201

Title: Structural characterization of methionine and leucine enkephalins by hydrogen/deuterium exchange and electrospray ionization tandem mass spectrometry.

Journal: Rapid communications in mass spectrometry : RCM 20050101

Title: Internal energy distribution in electrospray ionization.

Journal: Journal of mass spectrometry : JMS 20050101

Title: Tissue levels of leu-enkephalin in rats with adjuvant arthritis.

Journal: Journal of neuroimmunology 20050101

Title: [Changes in systemic and local vascular reactivity in hemorrhagic shock and the therapeutic effect of delta opioid receptor antagonist ICI174,864].

Journal: Zhongguo wei zhong bing ji jiu yi xue = Chinese critical care medicine = Zhongguo weizhongbing jijiuyixue 20050101

Title: Parallel synthesis and biological evaluation of different sizes of bicyclo[2,3]-Leu-enkephalin analogues.

Journal: Biopolymers 20050101

Title: [Effect of opiod peptides on free radical oxidation in a bone regenerate after fracture].

Journal: Patologicheskaia fiziologiia i eksperimental'naia terapiia 20050101

Title: delta-opioid receptor-mediated actions on rostral ventromedial medulla neurons.

Journal: Neuroscience 20050101

Title: Interactions among mu- and delta-opioid receptors, especially putative delta1- and delta2-opioid receptors, promote dopamine release in the nucleus accumbens.

Journal: Neuroscience 20050101

Title: Specific photodissociation of peptides with multi-stage mass spectrometry.

Journal: Rapid communications in mass spectrometry : RCM 20050101

Title: Fasting-induced changes of neuropeptide immunoreactivity in the lateral septum of male rats.

Journal: Acta biologica Hungarica 20050101

Title: Distribution of methionine and leucine enkephalin neurons within the social behavior circuitry of the male Syrian hamster brain.

Journal: Brain research 20041224

Title: The effect of glycation on the chemical and enzymatic stability of the endogenous opioid peptide, leucine-enkephalin, and related fragments.

Journal: Bioorganic chemistry 20041201

Title: Investigation into factors affecting precision in ion trap mass spectrometry using different scan directions and axial modulation potential amplitudes.

Journal: Journal of mass spectrometry : JMS 20041101

Title: Facile incorporation of urea pseudopeptides into protease substrate analogue inhibitors.

Journal: Bioorganic & medicinal chemistry letters 20041018

Title: Infrared atmospheric pressure MALDI ion trap mass spectrometry of frozen samples using a Peltier-cooled sample stage.

Journal: Analytical chemistry 20041001

Title: Delta-opioid receptor antagonists exhibit properties of partial delta-receptor agonists in isolated perfused heart.

Journal: Bulletin of experimental biology and medicine 20041001

Title: Conjugation of a novel histidine derivative to biomolecules and labelling with [99mTc(OH2)3(CO)3]+.

Journal: Organic & biomolecular chemistry 20040921

Title: Novel design of bicyclic beta-turn dipeptides on solid-phase supports and synthesis of [3.3.0]-Bicyclo([2,3])-leu-enkephalin analogues.

Journal: Organic letters 20040916

Title: Water network dynamics at the critical moment of a peptide's beta-turn formation: a molecular dynamics study.

Journal: The Journal of chemical physics 20040908

Title: The antinociceptive effect of Delta9-tetrahydrocannabinol in the arthritic rat.

Journal: European journal of pharmacology 20040616

Title: Synthesis and conformational studies of a beta-turn mimetic incorporated in Leu-enkephalin.

Journal: The Journal of organic chemistry 20040514

Title: Ultrastructural localization of Leu5-enkephalin immunoreactivity in mesocortical neurons and their input terminals in rat ventral tegmental area.

Journal: Synapse (New York, N.Y.) 20040401

Title: Peptide synthesis in water IV. Preparation of N-ethanesulfonylethoxycarbonyl (Esc) amino acids and their application to solid phase peptide synthesis.

Journal: Chemical & pharmaceutical bulletin 20040401

Title: Half-life of leu-enkephalin in the serum of infants of the first year of life on different types of feeding: relationship with temperament.

Journal: Bulletin of experimental biology and medicine 20040401

Title: Immunohistochemistry, histopathology and ultrastructure of Gasterosteus aculeatus tissues infected with Glugea anomala.

Journal: Diseases of aquatic organisms 20040310

Title: Conformational search of peptides and proteins: Monte Carlo minimization with an adaptive bias method applied to the heptapeptide deltorphin.

Journal: Journal of computational chemistry 20040301

Title: Changes of central norepinephrine, beta-endorphin, LEU-enkephalin, peripheral arginine-vasopressin, and angiotensin II levels in acute and chronic phases of sino-aortic denervation in rats.

Journal: Journal of cardiovascular pharmacology 20040201

Title: 2',6'-dimethylphenylalanine (Dmp) can mimic the N-terminal Tyr in opioid peptides.

Journal: Biological & pharmaceutical bulletin 20040201

Title: Use of NMR and fluorescence spectroscopy as well as theoretical conformational analysis in conformation-activity studies of cyclic enkephalin analogues.

Journal: Current topics in medicinal chemistry 20040101

Title: Conformational analysis of opioid peptides in the solid states and the membrane environments by NMR spectroscopy.

Journal: Current topics in medicinal chemistry 20040101

Title: Antagonism in opioid peptides: the role of conformation.

Journal: Current topics in medicinal chemistry 20040101

Title: Cloning of prodynorphin cDNAs from the brain of Australian and African lungfish: implications for the evolution of the prodynorphin gene.

Journal: Neuroendocrinology 20040101

Title: [Leu-enkephalin homogeneously labeled with tritium in studying the Selank inhibiting effect on the enkephalin-degrading enzymes of human plasma].

Journal: Bioorganicheskaia khimiia 20040101

Title: High sensitivity and broad dynamic range infrared multiphoton dissociation for a quadrupole ion trap.

Journal: Rapid communications in mass spectrometry : RCM 20040101

Title: [Antiarrhythmic and cardioprotective effect of stimulation of delta1-opiate receptors in myocardial ischemia and reperfusion].

Journal: Patologicheskaia fiziologiia i eksperimental'naia terapiia 20040101

Title: [Correction of temperature homeostasis and microcirculation under the stress-protection anesthesia in hip replacement].

Journal: Anesteziologiia i reanimatologiia 20040101

Title: Inhibition of human plasma leucine5-enkephalin aminopeptidase hydrolysis by various endogenous peptides and a select number of clinically used drugs.

Journal: American journal of therapeutics 20040101

Title: Gas-phase dissociation pathways of multiply charged peptide clusters.

Journal: Journal of the American Society for Mass Spectrometry 20031201

Title: The role of acidic residues and of sodium ion adduction on the gas-phase H/D exchange of peptides and peptide dimers.

Journal: Journal of the American Society for Mass Spectrometry 20031201

Title: Stress applied during primary immunization affects the secondary humoral immune response in the rat: involvement of opioid peptides.

Journal: Stress (Amsterdam, Netherlands) 20031201

Title: A possible role for an enkephalinergic system in the internal defense mechanism of Biomphalaria alexandrina exposed to Schistosoma mansoni.

Journal: Journal of the Egyptian Society of Parasitology 20031201

Title: Relations between Leu(5)-enkephalin- (LENK) and VIP-immunoreactive nerve fibres during human drug-resistant colitis. A case study.

Journal: Folia morphologica 20031101

Title: [Absence of the effect of opioid peptides on muscarine receptors in the frog vestibular apparatus].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20031101

Title: The use of static pressures of heavy gases within a quadrupole ion trap.

Journal: Journal of the American Society for Mass Spectrometry 20031001

Title: The regulation of steroidogenesis by opioid peptides in porcine theca cells.

Journal: Animal reproduction science 20030915

Title: Leucine-enkephalin interrupts sympathetically mediated tachycardia prejunctionally in the canine sinoatrial node.

Journal: Experimental biology and medicine (Maywood, N.J.) 20030901

Title: Analgesic effects of intra-nasal enkephalins.

Journal: The Journal of pharmacy and pharmacology 20030901

Title: A genetic algorithm with conformational memories for structure prediction of polypeptides.

Journal: Journal of biomolecular structure & dynamics 20030801

Title: Effect of synthetic oligopeptides on osteoporosis.

Journal: Preparative biochemistry & biotechnology 20030801

Title: Stereoselective synthesis of individual isomers of Leu-enkephalin analogues containing substituted beta-turn bicyclic dipeptide mimetics.

Journal: Chemical communications (Cambridge, England) 20030707

Title: Gradient liquid chromatography of leucine-enkephalin peptide and its metabolites with electrochemical detection using highly boron-doped diamond electrode.

Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20030705

Title: Activation of peripheral delta opioid receptors eliminates cardiac electrical instability in a rat model of post-infarction cardiosclerosis via mitochondrial ATP-dependent K+ channels.

Journal: Life sciences 20030704

Title: 'Fast excitation' CID in a quadrupole ion trap mass spectrometer.

Journal: Journal of the American Society for Mass Spectrometry 20030701

Title: Contribution of organic anion transporting polypeptide OATP-C to hepatic elimination of the opioid pentapeptide analogue [D-Ala2, D-Leu5]-enkephalin.

Journal: The Journal of pharmacy and pharmacology 20030701

Title: The neuropeptide-degrading enzyme NL1 is expressed in specific neurons of mouse brain.

Journal: Peptides 20030701

Title: Manipulating internal energy of protonated biomolecules in electrospray ionization Fourier transform ion cyclotron resonance mass spectrometry.

Journal: Journal of mass spectrometry : JMS 20030601

Title: The selective action of opioid peptides on excitability and the various sensory inputs of defensive behavior command neurons LPl1 and RPl1 of the common snail.

Journal: Neuroscience and behavioral physiology 20030601

Title: Structure-activity relationships of dynorphin a analogues modified in the address sequence.

Journal: Journal of medicinal chemistry 20030522

Title: Soluble proteolytic enzyme release by naive and HIV-infected cultured T-cells.

Journal: International immunopharmacology 20030501

Title: DSLET and ACTH(4-10) increase mitotic activity of hepatocytes and suppress antibody production.

Journal: Bulletin of experimental biology and medicine 20030501

Title: Topography and associations of leu-enkephalin and luteinizing hormone-releasing hormone neuronal systems in the human diencephalon.

Journal: The Journal of clinical endocrinology and metabolism 20030401

Title: New development in the tritium labelling of peptides and proteins using solid catalytic isotopic exchange with spillover-tritium.

Journal: Amino acids 20030401

Title: Synthesis and binding affinity of neuropeptide Y at opiate receptors.

Journal: Bioorganic & medicinal chemistry letters 20030324

Title: Peptide separations and dissociation constants in nonaqueous capillary electrophoresis: comparison of methanol and aqueous buffers.

Journal: Electrophoresis 20030301

Title: A comparison between electrokinetic capillary chromatography and absorption spectroscopy for the analysis of peptide-micelle association by weak hydrophobic interactions.

Journal: Electrophoresis 20030301

Title: Switched-angle spinning applied to bicelles containing phospholipid-associated peptides.

Journal: Journal of biomolecular NMR 20030201

Title: Studies on the synthesis and anti-Osteoporosis of estrogen-GHRPs linkers.

Journal: Bioorganic & medicinal chemistry letters 20030106

Title: In vitro human plasma leucine(5)-enkephalin degradation is inhibited by a select number of drugs with the phenothiazine molecule in their chemical structure.

Journal: Pharmacology 20030101

Title: Product ion spectral simplification using time-delayed fragment ion capture with tandem linear ion traps.

Journal: Rapid communications in mass spectrometry : RCM 20030101

Title: Parallel high-throughput accurate mass measurement using a nine-channel multiplexed electrospray liquid chromatography ultraviolet time-of-flight mass spectrometry system.

Journal: Rapid communications in mass spectrometry : RCM 20030101

Title: [Effect of new peptide bioregulators livagen and epitalon on enkephalin-degrading enzymes in human serum].

Journal: Izvestiia Akademii nauk. Seriia biologicheskaia 20030101

Title: Synthesis and evaluation of derivatives of leucine enkephalin as potential affinity labels for delta opioid receptors.

Journal: Biopolymers 20030101

Title: The probability distribution of side-chain conformations in [Leu] and [Met]enkephalin determines the potency and selectivity to mu and delta opiate receptors.

Journal: Biopolymers 20030101

Title: Differences in the chemical coding of nerve fibres supplying major populations of neurons between the caudal mesenteric ganglion and anterior pelvic ganglion in the male pig.

Journal: Folia histochemica et cytobiologica 20030101

Title: Lack of evidence of an interaction between leu-enkephalin and muscarinic-like responses in the frog semicircular canal.

Journal: Neuro-Signals 20030101

Title: [The role of opiate receptors and ATP-dependent potassium channels of mitochondria in the formation of myocardial adaptive resistance to the arrhythmogenic effect of ischemia and reperfusion].

Journal: Izvestiia Akademii nauk. Seriia biologicheskaia 20030101

Title: Methionine-enkephalin and leucine-enkephalin increase interleukin-1 beta release in mixed glia cultures.

Journal: Neuropeptides 20021201

Title: [Study on the relationship between endogenous opioid peptides and fetal distress].

Journal: Zhonghua fu chan ke za zhi 20021201

Title: Correlated morphological and chemical phenotyping in myenteric type V neurons of porcine ileum.

Journal: The Journal of comparative neurology 20021104

Title: Opioid activity of 4-imidazolidinone positional analogues of Leu-Enkephalin.

Journal: Bioorganic & medicinal chemistry letters 20021104

Title: The effect of opioid agonists of delta-class DSLET, mu-class DAMGO, kappa-class U-69593 and an opioid antagonist, naloxone, on MTT activity of NALM-1 leukemic cells.

Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie 20021101

Title: Solid-phase synthesis of fullerene-peptides.

Journal: Journal of the American Chemical Society 20021023

Title: Integration of solid-phase extraction membranes for sample multiplexing: application to rapid protein identification from gel-isolated protein extracts.

Journal: Electrophoresis 20021001

Title: Effect of in vivo and in vitro stimulation of delta1-opioid receptors on myocardial resistance to arrhythmogenic action of ischemia and reperfusion.

Journal: Bulletin of experimental biology and medicine 20021001

Title: The structure of an endomorphin analogue incorporating 1-aminocyclohexane-1-carboxlylic acid for proline is similar to the beta-turn of Leu-enkephalin.

Journal: Biochemical and biophysical research communications 20020913

Title: Efficiency of the multicanonical simulation method as applied to peptides of increasing size: the heptapeptide deltorphin.

Journal: Journal of computational chemistry 20020901

Title: Fabrication of microchannel structures in fluorinated ethylene propylene.

Journal: Analytical chemistry 20020901

Title: A conformational analysis of leucine enkephalin as a function of pH.

Journal: Biopolymers 20020805

Title: Determination of transport in the Caco-2 cell assay of compounds varying in lipophilicity using LC-MS: enhanced transport of Leu-enkephalin analogues.

Journal: European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20020801

Title: Distribution of leucine-enkephalin in bone and joint tissues.

Journal: Neuropeptides 20020801

Title: Effect of synthetic oligopeptides on osteoporosis.

Journal: Preparative biochemistry & biotechnology 20020801

Title: Surface-induced dissociation in a Fourier transform ion cyclotron resonance mass spectrometer: instrument design and evaluation.

Journal: Analytical chemistry 20020715

Title: Labelling of [Leu5]-enkephalin with organometallic Mo complexes by solid-phase synthesis.

Journal: Chemical communications (Cambridge, England) 20020707

Title: Neurons with mu opioid receptors interact indirectly with enkephalin-containing neurons in the rat dentate gyrus.

Journal: Experimental neurology 20020701

Title: The longitudinal smooth muscle layer of the pig small intestine is innervated by both myenteric and submucous neurons.

Journal: Histochemistry and cell biology 20020601

Title: Characterization of human nasal primary culture systems to investigate peptide metabolism.

Journal: International journal of pharmaceutics 20020515

Title: Nasal absorption enhancement strategies for therapeutic peptides: an in vitro study using cultured human nasal epithelium.

Journal: International journal of pharmaceutics 20020426

Title: Ligands act as pharmacological chaperones and increase the efficiency of delta opioid receptor maturation.

Journal: The EMBO journal 20020402

Title: Evidence for changes in brain enkephalin contents associated to male rat sexual activity.

Journal: Behavioural brain research 20020401

Title: Enkephalinergic control of the secretory activity of neurons producing stereoisomers of crustacean hyperglycemic hormone in the eyestalk of the crayfish Orconectes limosus.

Journal: The Journal of comparative neurology 20020225

Title: Peptidase activity on the surface of the porcine buccal mucosa.

Journal: International journal of pharmaceutics 20020221

Title: MALDI-TOF-MS analysis of droplets prepared in an electrodynamic balance: 'wall-less' sample preparation.

Journal: Analytical chemistry 20020201

Title: Effects of Selank on behavioral reactions and activities of plasma enkephalin-degrading enzymes in mice with different phenotypes of emotional and stress reactions.

Journal: Bulletin of experimental biology and medicine 20020201

Title: [The postburn change in hypothalamic paraventricular beta-endorphin and the roles of delta-receptor in scalded rats].

Journal: Zhonghua shao shang za zhi = Zhonghua shaoshang zazhi = Chinese journal of burns 20020201

Title: [Selectivity of opioid peptide effects on excitability and various sensory inputs in LPl1 and PPl1 command neurons participating in defensive behavior of the snail Helix lucorum].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20020101

Title: Multi-stage tandem mass spectrometry of metal cationized leucine enkephalin and leucine enkephalin amide.

Journal: Rapid communications in mass spectrometry : RCM 20020101

Title: [Effect of opioid peptides on the repair regeneration of the bone tissue].

Journal: Arkhiv patologii 20020101

Title: Delta opioid activation of the mitogen-activated protein kinase cascade does not require transphosphorylation of receptor tyrosine kinases.

Journal: BMC pharmacology 20020101

Title: [Opiatergic modulation of cardiac resistance to arrhythmogenic exposures].

Journal: Patologicheskaia fiziologiia i eksperimental'naia terapiia 20020101

Title: The ortho backbone amide linker (o-BAL) is an easily prepared and highly acid-labile handle for solid-phase synthesis.

Journal: Journal of combinatorial chemistry 20020101

Title: [Stimulation of delta1-opioid receptors increases the ventricular fibrillation threshold in post-infarct cardiosclerosis: the role of K(ATP)-channels].

Journal: Eksperimental'naia i klinicheskaia farmakologiia 20020101

Title: Leu-enkephalin immunoreactivity in the pig pineal gland.

Journal: Folia histochemica et cytobiologica 20020101

Title: Neither axotomy nor target-tissue inflammation changes the NOS- or VIP-synthesis rate in distal bowel-projecting neurons of the porcine inferior mesenteric ganglion (IMG).

Journal: Folia histochemica et cytobiologica 20020101

Title: Identification and characterization of an oligopeptide transport system in Leuconostoc mesenteroides subsp. mesenteroides CNRZ 1463.

Journal: Letters in applied microbiology 20020101

Title: Water structure around enkephalin near a GeO2 surface: a molecular dynamics study.

Journal: Journal of biomaterials science. Polymer edition 20020101

Title: [Effect of opioid peptides on proliferation and differentiation of skeletogenic cells of rabbit bone marrow in vitro].

Journal: Tsitologiia 20020101

Title: Solid-phase synthesis of oligourea peptidomimetics employing the Fmoc protection strategy.

Journal: The Journal of organic chemistry 20011214

Title: Improved blood-brain barrier penetration and enhanced analgesia of an opioid peptide by glycosylation.

Journal: The Journal of pharmacology and experimental therapeutics 20011201

Title: A novel tandem quadrupole mass spectrometer allowing gaseous collisional activation and surface induced dissociation.

Journal: Journal of mass spectrometry : JMS 20011201

Title: Spinorphin, an endogenous inhibitor of enkephalin-degrading enzymes, potentiates leu-enkephalin-induced anti-allodynic and antinociceptive effects in mice.

Journal: Japanese journal of pharmacology 20011201

Title: [Role of delta opioid receptors and their ligands in the development of adaptive heart protection against arrhythmogenesis].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20011201

Title: Parallel nociceptive reflex pathways with negative and positive feedback functions to foot extensors in the cat.

Journal: The Journal of physiology 20011015

Title: Short-term inverse-agonist treatment induces reciprocal changes in delta-opioid agonist and inverse-agonist binding capacity.

Journal: Molecular pharmacology 20011001

Title: Endorphin and enkephalin ameliorate excessive synovial cell functions in patients with rheumatoid arthritis.

Journal: The Journal of rheumatology 20011001

Title: Differential antinociceptive effects induced by intrathecally administered endomorphin-1 and endomorphin-2 in the mouse.

Journal: European journal of pharmacology 20010921

Title: Agonist-, antagonist-, and inverse agonist-regulated trafficking of the delta-opioid receptor correlates with, but does not require, G protein activation.

Journal: The Journal of pharmacology and experimental therapeutics 20010901

Title: Naloxone blocks transferred preconditioning in isolated rabbit hearts.

Journal: Journal of molecular and cellular cardiology 20010901

Title: Neuropeptide degradation in naive and steroid-treated allergic saliva.

Journal: International immunopharmacology 20010901

Title: Cross-checking of nanoelectrospray ionization mass spectrometry and computer simulation for the evaluation of the interaction strength of non-covalently bound enkephalins in solution.

Journal: Journal of mass spectrometry : JMS 20010801

Title: The role of leucine-enkephalin on insulin and glucagon secretion from pancreatic tissue fragments of normal and diabetic rats.

Journal: Archives of physiology and biochemistry 20010701

Title: [Clinical study on analgesic mechanism of bitongxiao in treating neck pain due to cervical spondylitis].

Journal: Zhongguo Zhong xi yi jie he za zhi Zhongguo Zhongxiyi jiehe zazhi = Chinese journal of integrated traditional and Western medicine 20010701

Title: Rostral ventrolateral medullary opioid receptor subtypes in the inhibitory effect of electroacupuncture on reflex autonomic response in cats.

Journal: Autonomic neuroscience : basic & clinical 20010620

Title: Antisera against endogenous opioids increase the nocifensive response to formalin: demonstration of inhibitory beta-endorphinergic control.

Journal: European journal of pharmacology 20010601

Title: Inverse agonist action of Leu-enkephalin at delta(2)-opioid receptors mediates spinal antianalgesia.

Journal: The Journal of pharmacology and experimental therapeutics 20010501

Title: Derivatization and fluorescence detection of amino acids and peptides with 9-fluorenylmethyl chloroformate on the surface of a solid adsorbent.

Journal: Analytical chemistry 20010501

Title: [The role of mu- and delta-opiate receptors in resistance of the myocardium to free radical damage].

Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova 20010501

Title: Monitoring receptor oligomerization using time-resolved fluorescence resonance energy transfer and bioluminescence resonance energy transfer. The human delta -opioid receptor displays constitutive oligomerization at the cell surface, which is not regulated by receptor occupancy.

Journal: The Journal of biological chemistry 20010427

Title: An immunoassay for Leu-enkephalin based on a C-terminal aequorin-peptide fusion.

Journal: Analytical chemistry 20010415

Title: Characterization of opioid receptors modulating neurogenic contractions of circular muscle from porcine ileum and evidence that delta- and kappa-opioid receptors are coexpressed in myenteric neurons.

Journal: The Journal of pharmacology and experimental therapeutics 20010401

Title: Probing opioid receptor-ligand interactions by employment of indolizidin-9-one amino acid as a constrained Gly(2)-Gly(3) surrogate in a leucine-enkephalin mimic.

Journal: The journal of peptide research : official journal of the American Peptide Society 20010401

Title: Stimulation of mu and delta-Opiate Receptors and Tolerance of Isolated Heart to Oxidative Stress: the Role of NO-Synthase.

Journal: Biochemistry. Biokhimiia 20010401

Title: Stereospecific synthesis of (2S)-2-methyl-3-(2',6'-dimethyl-4'-hydroxyphenyl)-propionic acid (Mdp) and its incorporation into an opioid peptide.

Journal: Bioorganic & medicinal chemistry letters 20010212

Title: Enkephalin analogues with 2',6'-dimethylphenylalanine replacing phenylalanine in position 4.

Journal: Bioorganic & medicinal chemistry letters 20010212

Title: The metabolic evidence of synergistic effect between ohmefentanyl and [D-Pen2, D-Pen5] enkephalin on differentiated SH-SY5Y cells in humans.

Journal: Neuroscience letters 20010209

Title: Role of endogenous opioid peptides in protection of ischemic preconditioning in rat small intestine.

Journal: Life sciences 20010119

Title: Antianalgesic action of nociceptin originating in the brain is mediated by spinal prostaglandin E(2) in mice.

Journal: The Journal of pharmacology and experimental therapeutics 20010101

Title: Chloramine-T in radiolabeling techniques. IV. Penta-O-acetyl-N-chloro-N-methylglucamine as an oxidizing agent in radiolabelling techniques.

Journal: Analytical biochemistry 20010101

Title: C-terminal and n-terminal fusions of aequorin with small peptides in immunoassay development.

Journal: Bioconjugate chemistry 20010101

Title: Electrospray ionization detection of inherently nonresponsive epoxides by peptide binding.

Journal: Rapid communications in mass spectrometry : RCM 20010101

Title: An apparatus to assay opioid activity in the infused lumen of the intact isolated guinea pig ileum.

Journal: Journal of pharmacological and toxicological methods 20010101

Title: Identification of dipeptidyl peptidase III in human neutrophils.

Journal: Biochemical and biophysical research communications 20000705

Title: Chromatographic detection using tris(2,2'-bipyridyl)ruthenium(III) as a fluorogenic electron-transfer reagent.

Journal: Analytical chemistry 19990415

Title: Delta-opioid receptor antagonist inhibits immunomodulation by Met-enkephalin analogs.

Journal: Neuroimmunomodulation 19990101

Title: Regulation of delta opioid receptors by delta9-tetrahydrocannabinol in NG108-15 hybrid cells.

Journal: Life sciences 19980101

Title: [The participation of the mu-, delta- and kappa-opioid receptors in the realization of the anti-arrhythmia effect of Rhodiola rosea].

Journal: Eksperimental'naia i klinicheskaia farmakologiia 19970101

Title: Lipid-induced secondary structures and orientations of (Leu5)-enkephalin: helical and crystallographic double-bend conformers revealed by IRATR and molecular modelling.

Journal: Journal of peptide science : an official publication of the European Peptide Society 19970101

Title: Fate of peptides in peptidase mutants of Lactococcus lactis.

Journal: Molecular microbiology 19960701

Title: New theoretical methodology for elucidating the solution structure of peptides from NMR data. II. Free energy of dominant microstates of Leu-enkephalin and population-weighted average nuclear Overhauser effects intensities.

Journal: Biopolymers 19960101

Title: Isolation and characterization of opioid peptides in the avian brain.

Journal: The Journal of experimental zoology 19951001

Title: Acute tolerance to the excitatory effects of opioids in the rat hippocampus.

Journal: Journal of neuroscience research 19950101

Title: Conserved delta-activity in reverse enantiomeric opioid peptide.

Journal: Life sciences 19950101

Title: Differential regulation of mu and delta opiate receptors by morphine, selective agonists and antagonists and differentiating agents in SH-SY5Y human neuroblastoma cells.

Journal: The Journal of pharmacology and experimental therapeutics 19940901

Title: TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity.

Journal: Journal of medicinal chemistry 19931015

Title: Differential regulation of adenylyl cyclase activity by mu and delta opioids in rat caudate putamen and nucleus accumbens.

Journal: The Journal of pharmacology and experimental therapeutics 19931001

Title: Involvement of mu-opioid receptors in alcohol drinking by alcohol-preferring AA rats.

Journal: Pharmacology, biochemistry, and behavior 19930701

Title: Agonist and antagonist profiles of [D-Ala2,Glu4]deltorphin and its [Cys4]- and [Ser4]-substituted derivatives: further evidence of opioid delta receptor multiplicity.

Journal: The Journal of pharmacology and experimental therapeutics 19930501

Title: Dipeptidyl peptidase I from goat brain: purification, characterization and its action on Leu-enkephalin.

Journal: Neurochemistry international 19930101

Title: Conformationally restricted deltorphin analogues.

Journal: Journal of medicinal chemistry 19921016

Title: Neuroanatomical sites mediating the central actions of beta-endorphin as mapped by changes in glucose utilization: involvement of mu opioid receptors.

Journal: The Journal of pharmacology and experimental therapeutics 19920701

Title: Binding to opioid receptors of enkephalin derivatives taking alpha-helical conformation and its dimer.

Journal: International journal of peptide and protein research 19911001

Title: Human brain leucyl aminopeptidase: isolation, characterization and specificity against some neuropeptides.

Journal: Neuropeptides 19910701

Title: The opioid activity and receptor selectivity of fluorinated Leu5 enkephalin analogues in vitro and in vivo.

Journal: Journal of pharmacobio-dynamics 19910201

Title: Influence of peptidase inhibitors on the apparent agonist potency of delta selective opioid peptides in vitro.

Journal: Life sciences 19910101

Title: Transdermal delivery of bioactive peptides: the effect of n-decylmethyl sulfoxide, pH, and inhibitors on enkephalin metabolism and transport.

Journal: Pharmaceutical research 19901101

Title: Involvement of multiple opiate receptors in opioid kindling.

Journal: Brain research 19900528

Title: Modulation of mu, delta and kappa opioid receptors in rat brain by metal ions and histidine.

Journal: Neuropharmacology 19900501

Title: Effects of thioamide substitution for the enkephalin conformation. Crystal structure of Boc-Tyr-Gly-Gly-Phe psi [CSNH]Leu-OBzl.

Journal: International journal of peptide and protein research 19891101

Title: Inhibition of vagal transmission by cardiac sympathetic nerve stimulation in the dog: possible involvement of opioid receptor.

Journal: The Journal of pharmacology and experimental therapeutics 19890901

Title: Synthesis of peptide amides by Fmoc-solid-phase peptide synthesis and acid labile anchor groups.

Journal: International journal of peptide and protein research 19890901

Title: Guanine nucleotide regulation of [125I]beta-endorphin binding to NG108-15 and SK-N-SH cell membranes: specific cation requirements.

Journal: Brain research 19890724

Title: Paradoxical analgesia produced by low doses of the opiate-antagonist naloxone is mediated by interaction at a site with characteristics of the delta opioid receptor.

Journal: The Journal of pharmacology and experimental therapeutics 19890401

Title: [Highly active analogs of opiate-like peptides historphin and kapporphin].

Journal: Voprosy meditsinskoi khimii 19890101

Title: Mu and delta opioid receptors inhibit serotonin release in rat hippocampus.

Journal: The Journal of pharmacology and experimental therapeutics 19890101

Title: Purification and assay of opioid activity of low molecular weight enkephalin-immunoreactive peptides generated by peptic digestion of rat plasma proteins.

Journal: Neuropeptides 19890101

Title: Selectivity of various opioid peptides towards delta-, kappa; and mu-opioid receptors mediating presynaptic inhibition of neurotransmitter release in the brain.

Journal: Neuropeptides 19890101

Title: Opioid receptor selectivity of beta-endorphin in vitro and in vivo: mu, delta and epsilon receptors.

Journal: The Journal of pharmacology and experimental therapeutics 19880901

Title: Inhibition of exocrine pancreatic secretion by opiates is mediated by suppression of cholinergic transmission: characterization of receptor subtypes.

Journal: The Journal of pharmacology and experimental therapeutics 19880701

Title: [Bioavailability of dalargin and its metabolism during intranasal administration to rats].

Journal: Biulleten' eksperimental'noi biologii i meditsiny 19880701

Title: Endogenous opioids and immune responses: an experimental study.

Journal: NIDA research monograph 19880101

Title: [Biosynthesis of opioid peptides].

Journal: Annales d'endocrinologie 19880101

Title: Hybrid bivalent ligands with opiate and enkephalin pharmacophores.

Journal: Journal of medicinal chemistry 19871101

Title: Morphine and enkephalins potently inhibit [3H]noradrenaline release from rat brain cortex synaptosomes: further evidence for a presynaptic localization of mu-opioid receptors.

Journal: Journal of neurochemistry 19870401

Title: Opposite effects of delta and mu opioid receptor agonists on the in vitro release of substance P-like material from the rat spinal cord.

Journal: Journal of neurochemistry 19870201

Title: Opioid peptides. Biological study of [D-MetO2] dermorphin analogues in relation to the plurality of opioid receptors. XI.

Journal: Il Farmaco; edizione scientifica 19870201

Title: Normalization of blood pressure and plasma concentrations of beta-endorphin and leucine-enkephalin in patients with primary hypertension after treatment with clonidine.

Journal: Journal of cardiovascular pharmacology 19870101

Title: Effects of bestatin and phosphoramidon on the hypertensive response to physostigmine in the rat.

Journal: Fundamental & clinical pharmacology 19870101

Title: Purification and characterization of an enkephalin-degrading dipeptidyl-aminopeptidase from porcine brain.

Journal: Biochemistry 19861216

Title: Evidence that endogenous enkephalins produce delta-opiate receptor mediated neuronal inhibitions in rat dorsal horn.

Journal: Neuroscience letters 19861212

Title: Audiogenic seizures during ethanol withdrawal can be blocked by a delta opioid agonist.

Journal: Drug and alcohol dependence 19861201

Title: Opiate-induced seizures: a study of mu and delta specific mechanisms.

Journal: Experimental neurology 19860801

Title: Opioid-mediated cardiovascular effects of clonidine in spontaneously hypertensive rats: elimination by neonatal treatment with monosodium glutamate.

Journal: Endocrinology 19860501

Title: Metorphamide levels in chromaffin cells increase after treatment with reserpine.

Journal: Journal of neurochemistry 19860501

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Journal: Bioorganicheskaia khimiia 19860101

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Tags:58822-25-6 Molecular Formula|58822-25-6 MDL|58822-25-6 SMILES|58822-25-6 1-5-b-Neoendorphin (human)