Title: Zhou B, et al. Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression. J Med Chem. 2018 Jan 25;61(2):462-481.
2093388-33-9
2093388-62-4
2140289-17-2
943764-99-6 | Acebilustat | AA01EO1J | MFCD30496703
1799506-30-1 | PROTAC Linker 4 | AA01EO52 | MFCD31692394
2134602-45-0 | SR17018 | AA01EO9M | MFCD31657392
1699720-85-8 | BCRP-IN-1 | AA01EOFW | MFCD30533375
290814-68-5 | PBOX 6 | AA01EOLM | MFCD31382391
254435-95-5 | Alisporivir | AA01EOQ2 | MFCD28411375
1843184-38-2 | 2-(2-chlorophenyl)-1-[1-(4-hydroxypentyl)-1H-indol-3-yl]-ethanone | AA01EOZA
1219798-88-5 | 2,3-dihydro-5,6-dimethoxy-2[[1-(phenylmethyl-d2)-4-piperidinyl]methyl-d2]-1H-inden-1-one,monohydrochloride | AA01EPAK | MFCD08704900
663625-18-1 | 2,2'-((2-(2-(2-(bis(carboxylatomethyl)amino)-5-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)phenoxy)ethoxy)-4-methylphenyl)azanediyl)diacetate,tripotassiumsalt | AA01EPI0
862073-79-8 | (2S,4aR,6aR,7R,9S,10aS,10bR)-2-(3-furanyl)dodecahydro-6a,10b-dimethyl-9-[(methylsulfonyl)oxy]-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylicacid,methylester | AA01EPN2