Title: Structure-activity relationship of boronic acid derivatives of tyropeptin: proteasome inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20101001
Title: Proline isosteres in a series of 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitors of IGF-1R kinase and IR kinase.
Journal: Bioorganic & medicinal chemistry letters 20100901