Title: Bactericidal activity and mechanism of action of AZD5847, a novel oxazolidinone for treatment of tuberculosis.
Journal: Antimicrobial agents and chemotherapy20140101
Title: Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
Journal: Bioorganic & medicinal chemistry20121115
Title: FLO11 expression and lipid biosynthesis are required for air-liquid biofilm formation in a Saccharomyces cerevisiae flor strain.
Journal: FEMS yeast research20121101
Title: Inhibition of fatty-acid synthase suppresses P-AKT and induces apoptosis in bladder cancer.
Journal: Urology20120801
Title: Involvement of the AtoSCDAEB regulon in the high molecular weight poly-(R)-3-hydroxybutyrate biosynthesis in phaCAB(+)Escherichia coli.
Journal: Metabolic engineering20120701
Title: Therapeutic and toxicologic evaluation of anti-lipogenic agents in cancer cells compared with non-neoplastic cells.
Journal: Basic & clinical pharmacology & toxicology20120601
Title: Cerulenin-induced apoptosis is mediated by disrupting the interaction between AIF and hexokinase II.
Journal: International journal of oncology20120601
Title: Crystal structures of Xanthomonas campestris OleA reveal features that promote head-to-head condensation of two long-chain fatty acids.
Journal: Biochemistry20120522
Title: Enhanced antitumor activity of epirubicin combined with cerulenin in osteosarcoma.
Journal: Molecular medicine reports20120201
Title: Search method for inhibitors of Staphyloxanthin production by methicillin-resistant Staphylococcus aureus.
Journal: Biological & pharmaceutical bulletin20120101
Title: Inhibition of fatty acid synthase supresses osteosarcoma cell invasion and migration.
Journal: Indian journal of pathology & microbiology20120101
Title: A combination of flow cytometry and traditional screening using chemicals to isolate high glutathione-producing yeast mutants.
Journal: Bioscience, biotechnology, and biochemistry20120101
Title: Inhibition of fatty acid metabolism reduces human myeloma cells proliferation.
Journal: PloS one20120101
Title: Similarities between exogenously- and endogenously-induced envelope stress: the effects of a new antibacterial molecule, TPI1609-10.
Journal: PloS one20120101
Title: Discovery of BI 99179, a potent and selective inhibitor of type I fatty acid synthase with central exposure.
Journal: Bioorganic & medicinal chemistry letters20111001
Title: Lipid droplet formation protects against gluco/lipotoxicity in Candida parapsilosis: an essential role of fatty acid desaturase Ole1.
Journal: Cell cycle (Georgetown, Tex.)20110915
Title: The lipogenesis pathway as a cancer target.
Journal: Journal of medicinal chemistry20110825
Title: Pyrazinamide, but not pyrazinoic acid, is a competitive inhibitor of NADPH binding to Mycobacterium tuberculosis fatty acid synthase I.
Journal: Bioorganic & medicinal chemistry letters20110815
Title: Malonyl-CoA mediates leptin hypothalamic control of feeding independent of inhibition of CPT-1a.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20110701
Title: A novel positive feedback loop involving FASN/p-ERK1/2/5-LOX/LTB4/FASN sustains high growth of breast cancer cells.
Journal: Acta pharmacologica Sinica20110701
Title: AtoSC two-component system is involved in cPHB biosynthesis through fatty acid metabolism in E. coli.
Journal: Biochimica et biophysica acta20110501
Title: Inhibition of fatty acid synthase in melanoma cells activates the intrinsic pathway of apoptosis.
Journal: Laboratory investigation; a journal of technical methods and pathology20110201
Title: Suppression of phospholipid biosynthesis by cerulenin in the condensed Single-Protein-Production (cSPP) system.
Journal: Journal of biomolecular NMR20110201
Title: DGK1-encoded diacylglycerol kinase activity is required for phospholipid synthesis during growth resumption from stationary phase in Saccharomyces cerevisiae.
Journal: The Journal of biological chemistry20110114
Title: Glucose stimulation of protein acylation in the pancreatic β-cell.
Journal: Life sciences20101218
Title: The construction and application of diploid sake yeast with a homozygous mutation in the FAS2 gene.
Journal: Journal of bioscience and bioengineering20101201
Title: Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Journal: Bioorganic & medicinal chemistry letters20101101
Title: Endogenous H2O2 produced by Streptococcus pneumoniae controls FabF activity.
Journal: Biochimica et biophysica acta20100901
Title: Canola oil inhibits breast cancer cell growth in cultures and in vivo and acts synergistically with chemotherapeutic drugs.
Journal: Lipids20100901
Title: Hypothalamic AMPK and fatty acid metabolism mediate thyroid regulation of energy balance.
Journal: Nature medicine20100901
Title: Fatty acid synthase inhibitor cerulenin suppresses liver metastasis of colon cancer in mice.
Journal: Cancer science20100801
Title: Fatty acid synthase as a novel target for meningioma therapy.
Journal: Neuro-oncology20100801
Title: Fatty acid synthesis is a therapeutic target in human liposarcoma.
Journal: International journal of oncology20100501
Title: Inhibition of fatty acid biosynthesis prevents adipocyte lipotoxicity on human osteoblasts in vitro.
Journal: Journal of cellular and molecular medicine20100401
Title: Fatty acid synthase as a potential therapeutic target in cancer.
Journal: Future oncology (London, England)20100401
Title: Visfatin gene expression in chickens is sex and tissue dependent.
Journal: Domestic animal endocrinology20100201
Title: The TGL2 gene of Saccharomyces cerevisiae encodes an active acylglycerol lipase located in the mitochondria.
Journal: The Journal of biological chemistry20100129
Title: Striatal dopamine in the response of brain and liver unsaturated and saturated free fatty acids following administration of C75 in CD-1 mice.
Journal: Neuroscience letters20100129
Title: Differentiation inducing factors in Dictyostelium discoideum: a novel low molecular factor functions at an early stage(s) of differentiation.
Journal: Development, growth & differentiation20091201
Title: Analysis of potato virus X replicase and TGBp3 subcellular locations.
Journal: Virology20091025
Title: Fatty acid oxidation and meiotic resumption in mouse oocytes.
Journal: Molecular reproduction and development20090901
Title: Design, synthesis, and structure-activity relationships of benzophenone-based tetraamides as novel antibacterial agents.
Journal: Journal of medicinal chemistry20090827
Title: Chemical genetic profiling and characterization of small-molecule compounds that affect the biosynthesis of unsaturated fatty acids in Candida albicans.
Journal: The Journal of biological chemistry20090717
Title: Cerulenin analogues as inhibitors of efflux pumps in drug-resistant Candida albicans.
Journal: Archiv der Pharmazie20090301
Title: Transepithelial transport of Cerulenin across Caco-2 cell monolayers.
Journal: European journal of drug metabolism and pharmacokinetics20090101
Title: Fatty acid synthase inhibitors modulate energy balance via mammalian target of rapamycin complex 1 signaling in the central nervous system.
Journal: Diabetes20081201
Title: Cerulenin inhibits de novo sophorolipid synthesis of Candida bombicola.
Journal: Biotechnology letters20081001
Title: Fatty acid synthase inhibition results in a magnetic resonance-detectable drop in phosphocholine.
Journal: Molecular cancer therapeutics20080801
Title: Fatty acid synthase is a novel therapeutic target in multiple myeloma.
Journal: British journal of haematology20080601
Title: Increased fatty acid synthase as a potential therapeutic target in multiple myeloma.
Journal: Journal of Zhejiang University. Science. B20080601
Title: A malonyl-CoA-dependent switch in the bacterial response to a dysfunction of lipid metabolism.
Journal: Molecular microbiology20080501
Title: Dietary soy protein inhibits DNA damage and cell survival of colon epithelial cells through attenuated expression of fatty acid synthase.
Journal: American journal of physiology. Gastrointestinal and liver physiology20080401
Title: The synthetic triterpenoid CDDO-Im inhibits fatty acid synthase expression and has antiproliferative and proapoptotic effects in human liposarcoma cells.
Journal: Cancer investigation20080301
Title: Monosaccharide-induced lipogenesis regulates the human hepatic sex hormone-binding globulin gene.
Journal: The Journal of clinical investigation20071203
Title: The human fatty acid synthase: a new therapeutic target for coxsackievirus B3-induced diseases?
Journal: Antiviral research20071101
Title: Cryptosporidium parvum long-chain fatty acid elongase.
Journal: Eukaryotic cell20071101
Title: Expression of prenylated Rab acceptor 1 domain family, member 2 (PRAF2) in neuroblastoma: correlation with clinical features, cellular localization, and cerulenin-mediated apoptosis regulation.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research20071101
Title: Inhibition of Fatty Acid Synthase (FASN) synergistically enhances the efficacy of 5-fluorouracil in breast carcinoma cells.
Journal: Oncology reports20071001
Title: Fatty acid synthase inhibitors cerulenin and C75 retard growth and induce caspase-dependent apoptosis in human melanoma A-375 cells.
Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie20071001
Title: Structural and mechanistic analysis of protein interactions in module 3 of the 6-deoxyerythronolide B synthase.
Journal: Chemistry & biology20070801
Title: The inhibitors of protein acylation, cerulenin and tunicamycin, increase voltage-dependent Ca(2+) currents in the insulin-secreting INS 832/13 cell.
Journal: Biochemical pharmacology20070715
Title: S-acylation regulates Kv1.5 channel surface expression.
Journal: American journal of physiology. Cell physiology20070701
Title: Inhibition of isolated Mycobacterium tuberculosis fatty acid synthase I by pyrazinamide analogs.
Journal: Antimicrobial agents and chemotherapy20070701
Title: An antifungal agent inhibits an aminoacyl-tRNA synthetase by trapping tRNA in the editing site.
Journal: Science (New York, N.Y.)20070622
Title: [Cerulenin changes apoptosis related genes expression in multiple myeloma cell line U266].
Journal: Zhonghua xue ye xue za zhi = Zhonghua xueyexue zazhi20070401
Title: Anti-Candida metabolites from endophytic fungi.
Journal: Phytochemistry20070301
Title: Links between de novo fatty acid synthesis and leptin secretion in bovine adipocytes.
Journal: The Journal of veterinary medical science20070301
Title: Inhibition of insulin secretion by cerulenin might be due to impaired glucose metabolism.
Journal: Diabetes/metabolism research and reviews20070201
Title: Structure of the human beta-ketoacyl [ACP] synthase from the mitochondrial type II fatty acid synthase.
Journal: Protein science : a publication of the Protein Society20070201
Title: Inhibition of fatty acid synthase induces endoplasmic reticulum stress in tumor cells.
Journal: Cancer research20070201
Title: Identification of a cerulenin resistance gene from Monascus pilosus.
Journal: DNA sequence : the journal of DNA sequencing and mapping20070201
Title: The regulation of stearoyl-CoA desaturase gene expression is tissue specific in chickens.
Journal: The Journal of endocrinology20070101
Title: Cerulenin-mediated apoptosis is involved in adenine metabolic pathway.
Journal: Biochemical and biophysical research communications20061027
Title: Fatty acid synthase: a novel target for antiglioma therapy.
Journal: British journal of cancer20061009
Title: [Study on proliferation inhibiting and apoptosis inducing effects of cerulenin on multiple myeloma cells].
Journal: Zhonghua xue ye xue za zhi = Zhonghua xueyexue zazhi20061001
Title: Fatty acid synthase inhibitory activity of acylphloroglucinols isolated from Dryopteris crassirhizoma.
Journal: Bioorganic & medicinal chemistry letters20060915
Title: Inhibitors of fatty acid biosynthesis in sunflower seeds.
Journal: Journal of plant physiology20060901
Title: Inositol induces a profound alteration in the pattern and rate of synthesis and turnover of membrane lipids in Saccharomyces cerevisiae.
Journal: The Journal of biological chemistry20060811
Title: FAS inhibitor cerulenin reduces food intake and melanocortin receptor gene expression without modulating the other (an)orexigenic neuropeptides in chickens.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20060701
Title: Biosynthetic requirements for the repair of sublethal membrane damage in Escherichia coli cells after pulsed electric fields.
Journal: Journal of applied microbiology20060301
Title: Inhibition of the phosphatidylinositol 3-kinase/Akt pathway sensitizes MDA-MB468 human breast cancer cells to cerulenin-induced apoptosis.
Journal: Molecular cancer therapeutics20060301
Title: Discovery of bacterial fatty acid synthase inhibitors from a Phoma species as antimicrobial agents using a new antisense-based strategy.
Journal: Journal of natural products20060301
Title: Changes in composition and content of mycolic acids in glutamate-overproducing Corynebacterium glutamicum.
Journal: Bioscience, biotechnology, and biochemistry20060101
Title: Lipid biosynthesis and its coordination with cell cycle progression.
Journal: Plant & cell physiology20051201
Title: Identification of a plastid acyl-acyl carrier protein synthetase in Arabidopsis and its role in the activation and elongation of exogenous fatty acids.
Journal: The Plant journal : for cell and molecular biology20051101
Title: YaeT (Omp85) affects the assembly of lipid-dependent and lipid-independent outer membrane proteins of Escherichia coli.
Journal: Molecular microbiology20050901
Title: Subinhibitory cerulenin inhibits staphylococcal exoprotein production by blocking transcription rather than by blocking secretion.
Journal: Microbiology (Reading, England)20050901
Title: Biological and molecular variability of Sarocladium oryzae, the sheath rot pathogen of rice (Oryza sativa L.).
Journal: Current microbiology20050601
Title: Fatty acid metabolism as a target for obesity treatment.
Journal: Physiology & behavior20050519
Title: Cloning, expression, and characterization of the human mitochondrial beta-ketoacyl synthase. Complementation of the yeast CEM1 knock-out strain.
Journal: The Journal of biological chemistry20050401
Title: Inhibition of fatty acid synthase prevents preadipocyte differentiation.
Journal: Biochemical and biophysical research communications20050325
Title: Enhancement of polyunsaturated fatty acid production by cerulenin treatment in polyunsaturated fatty acid-producing bacteria.
Journal: Biotechnology letters20050301
Title: Proliferation of fibroblasts cultured from normal gingiva and hereditary gingival fibromatosis is dependent on fatty acid synthase activity.
Journal: Journal of periodontology20050201
Title: A pilot study of fatty acid metabolism in oral squamous cell carcinoma.
Journal: International journal of oral and maxillofacial surgery20050101
Title: Transcutaneous delivery of levodopa: enhancement by fatty acid synthesis inhibition.
Journal: Molecular pharmaceutics20050101
Title: Targeting fatty acid synthase: potential for therapeutic intervention in her-2/neu-overexpressing breast cancer.
Journal: Drug news & perspectives20050101
Title: Vitamin D3 inhibits fatty acid synthase expression by stimulating the expression of long-chain fatty-acid-CoA ligase 3 in prostate cancer cells.
Journal: FEBS letters20041119
Title: Pharmacological inhibition of fatty acid synthase (FAS): a novel therapeutic approach for breast cancer chemoprevention through its ability to suppress Her-2/neu (erbB-2) oncogene-induced malignant transformation.
Journal: Molecular carcinogenesis20041101
Title: Conspecificity of the cerulenin and helvolic acid producing 'Cephalosporium caerulens', and the hypocrealean fungus Sarocladium oryzae.
Journal: Mycological research20041101
Title: Metabolic regulation of leptin production in adipocytes: a role of fatty acid synthesis intermediates.
Journal: The Journal of nutritional biochemistry20041101
Title: Androgens, lipogenesis and prostate cancer.
Journal: The Journal of steroid biochemistry and molecular biology20041101
Title: Influence of molecule CD 11b blockade on the course of acute ceruleine pancreatitis in rats.
Journal: Experimental and molecular pathology20040801
Title: Inhibition of tumor-associated fatty acid synthase activity enhances vinorelbine (Navelbine)-induced cytotoxicity and apoptotic cell death in human breast cancer cells.
Journal: Oncology reports20040801
Title: Carnitine palmitoyltransferase-1 (CPT-1) activity stimulation by cerulenin via sympathetic nervous system activation overrides cerulenin's peripheral effect.
Journal: Endocrinology20040701
Title: Overexpression and hyperactivity of breast cancer-associated fatty acid synthase (oncogenic antigen-519) is insensitive to normal arachidonic fatty acid-induced suppression in lipogenic tissues but it is selectively inhibited by tumoricidal alpha-linolenic and gamma-linolenic fatty acids: a novel mechanism by which dietary fat can alter mammary tumorigenesis.
Journal: International journal of oncology20040601
Title: Biosynthesis and dietary uptake of polyunsaturated fatty acids by piezophilic bacteria.
Journal: Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology20040401
Title: Expression and functional characterization of a giant Type I fatty acid synthase (CpFAS1) gene from Cryptosporidium parvum.
Journal: Molecular and biochemical parasitology20040301
Title: Novel signaling molecules implicated in tumor-associated fatty acid synthase-dependent breast cancer cell proliferation and survival: Role of exogenous dietary fatty acids, p53-p21WAF1/CIP1, ERK1/2 MAPK, p27KIP1, BRCA1, and NF-kappaB.
Journal: International journal of oncology20040301
Title: Inhibition of tumor-associated fatty acid synthase hyperactivity induces synergistic chemosensitization of HER -2/ neu -overexpressing human breast cancer cells to docetaxel (taxotere).
Journal: Breast cancer research and treatment20040301
Title: Identification and molecular characterization of the beta-ketoacyl-[acyl carrier protein] synthase component of the Arabidopsis mitochondrial fatty acid synthase.
Journal: The Journal of biological chemistry20040227
Title: Self-cloning yeast strains containing novel FAS2 mutations produce a higher amount of ethyl caproate in Japanese sake.
Journal: Bioscience, biotechnology, and biochemistry20040101
Title: Nutrient modulation of palmitoylated 24-kilodalton protein in rat pancreatic islets.
Journal: Endocrinology20031201
Title: Increased fatty acid synthase expression and activity during progression of prostate cancer in the TRAMP model.
Journal: The Prostate20031101
Title: Novel roles for palmitoylation of Ras in IL-1 beta-induced nitric oxide release and caspase 3 activation in insulin-secreting beta cells.
Journal: Biochemical pharmacology20031101
Title: The fatty acid synthase inhibitor cerulenin and feeding, like leptin, activate hypothalamic pro-opiomelanocortin (POMC) neurons.
Journal: Brain research20030919
Title: Requirement for kasB in Mycobacterium mycolic acid biosynthesis, cell wall impermeability and intracellular survival: implications for therapy.
Journal: Molecular microbiology20030901
Title: Futile cycling of intermediates of fatty acid biosynthesis toward peroxisomal beta-oxidation in Saccharomyces cerevisiae.
Journal: The Journal of biological chemistry20030829
Title: Protein acylation in the inhibition of insulin secretion by norepinephrine, somatostatin, galanin, and PGE2.
Journal: American journal of physiology. Endocrinology and metabolism20030801
Title: Effects of cerulenin on the endogenous fatty acid synthetic activity in squamous cell carcinoma of the oral cavity.
Journal: Journal of oral and maxillofacial surgery : official journal of the American Association of Oral and Maxillofacial Surgeons20030801
Title: CT2108A and B: New fatty acid synthase inhibitors as antifungal agents.
Journal: Journal of natural products20030801
Title: Regulation of the CDP-choline pathway by sterol regulatory element binding proteins involves transcriptional and post-transcriptional mechanisms.
Journal: The Biochemical journal20030615
Title: Inhibition of fatty acid synthase expression by 1alpha,25-dihydroxyvitamin D3 in prostate cancer cells.
Journal: The Journal of steroid biochemistry and molecular biology20030501
Title: Phenolic compounds from Nymphaea odorata.
Journal: Journal of natural products20030401
Title: Bacterial beta-ketoacyl-acyl carrier protein synthases as targets for antibacterial agents.
Journal: Current protein & peptide science20030201
Title: [Fatty acid synthase: specific target for cancer therapy].
Journal: Sheng wu hua xue yu sheng wu wu li xue bao Acta biochimica et biophysica Sinica20030101
Title: Flavanone glycosides from Miconia trailii.
Journal: Journal of natural products20030101
Title: Characterization and inhibition of fatty acid synthase in pediatric tumor cell lines.
Journal: Anticancer research20030101
Title: Fatty acid synthase inhibitors from plants: isolation, structure elucidation, and SAR studies.
Journal: Journal of natural products20021201
Title: Effect of 2-fluoropalmitate, cerulenin and tunicamycin on the palmitoylation and intracellular translocation of myelin proteolipid protein.
Journal: Neurochemical research20021201
Title: Time-dependent stimulation of insulin exocytosis by 3',5'-cyclic adenosine monophosphate in the rat islet beta-cell.
Journal: Endocrinology20021101
Title: Protein acylation in the cardiac muscle like cell line, H9c2.
Journal: Molecular and cellular biochemistry20021001
Title: Key role of mitochondria in cerulenin-mediated apoptosis.
Journal: Cell death and differentiation20020901
Title: [Biosynthesis and accumulation of poly(3-hydroxybutyrate) in Vibrio natriegens].
Journal: Sheng wu gong cheng xue bao = Chinese journal of biotechnology20020901
Title: Biosynthesis of triacylglycerol molecular species in an oleaginous fungus, Mortierella ramanniana var. angulispora.
Journal: Journal of biochemistry20020701
Title: Block the FAS, lose the fat.
Journal: Nature medicine20020401
Title: The effects of cerulenin, an inhibitor of protein acylation, on the two phases of glucose-stimulated insulin secretion.
Journal: Diabetes20020201
Title: Time-dependent potentiation of the beta-cell is a Ca2+-independent phenomenon.
Journal: The Journal of endocrinology20020201
Title: Use of a YAP1 overexpression cassette conferring specific resistance to cerulenin and cycloheximide as an efficient selectable marker in the yeast Saccharomyces cerevisiae.
Journal: Yeast (Chichester, England)20020115
Title: Detection and quantification of phytotoxic metabolites of Sarocladium oryzae in sheath rot-infected grains of rice.
Journal: Letters in applied microbiology20020101
Title: Purification and biochemical characterization of the Mycobacterium tuberculosis beta-ketoacyl-acyl carrier protein synthases KasA and KasB.
Journal: The Journal of biological chemistry20011214
Title: An unusual seed-specific 3-ketoacyl-ACP synthase associated with the biosynthesis of petroselinic acid in coriander.
Journal: Plant molecular biology20011101
Title: Cellular pharmacology of cerulenin analogs that inhibit protein palmitoylation.
Journal: Biochemical pharmacology20011015
Title: Purification and some properties of an inhibitor for a yeast pleiotropic drug resistant pump from Kitasatospora sp. E-420.
Journal: Bioscience, biotechnology, and biochemistry20011001
Title: Regulation of catalytic activity of a multifunctional polyketide biosynthetic enzyme, 6-hydroxymellein synthase, by interaction between NADPH and phenylglyoxal-sensitive amino acid residue at the reaction center.
Journal: Biochimica et biophysica acta20010910
Title: Fatty acid synthase inhibition in human breast cancer cells leads to malonyl-CoA-induced inhibition of fatty acid oxidation and cytotoxicity.
Journal: Biochemical and biophysical research communications20010713
Title: Astaxanthin accumulation in Haematococcus requires a cytochrome P450 hydroxylase and an active synthesis of fatty acids.
Journal: FEBS letters20010706
Title: Mechanisms of fluconazole resistance in Candida albicans isolates from Japanese AIDS patients.
Journal: The Journal of antimicrobial chemotherapy20010501
Title: Cerulenin mimics effects of leptin on metabolic rate, food intake, and body weight independent of the melanocortin system, but unlike leptin, cerulenin fails to block neuroendocrine effects of fasting.
Journal: Diabetes20010401
Title: Biosynthesis of fattiviracin FV-8, an antiviral agent.
Journal: Bioscience, biotechnology, and biochemistry20010401
Title: Inhibition of beta-ketoacyl-acyl carrier protein synthases by thiolactomycin and cerulenin. Structure and mechanism.
Journal: The Journal of biological chemistry20010302
Title: ND9P, a novel protein with armadillo-like repeats involved in exocytosis: physiological studies using allelic mutants in paramecium.
Journal: Genetics20010201
Title: Increased fatty acid synthase is a therapeutic target in mesothelioma.
Journal: Clinical cancer research : an official journal of the American Association for Cancer Research20010101
Title: A new class of antituberculosis agents.
Journal: Journal of medicinal chemistry20000824
Title: Thiolactomycin and related analogues as novel anti-mycobacterial agents targeting KasA and KasB condensing enzymes in Mycobacterium tuberculosis.
Journal: The Journal of biological chemistry20000602
Title: [An experimental study on cerulenin induced apoptosis of human colonic cancer cells].
Journal: Zhonghua bing li xue za zhi = Chinese journal of pathology20000401
Title: Novel approaches to the treatment of hepatitis C virus infection.
Journal: Antiviral chemistry & chemotherapy20000301
Title: Antimycobacterial activity of cerulenin and its effects on lipid biosynthesis.
Journal: The Journal of antimicrobial chemotherapy19990201
Title: Synergistic activities of antituberculous drugs with cerulenin and trans-cinnamic acid against Mycobacterium tuberculosis.
Journal: FEMS immunology and medical microbiology19980601
Title: In vitro activities of free and liposomal drugs against Mycobacterium avium-M. intracellulare complex and M. tuberculosis.
Journal: Antimicrobial agents and chemotherapy19931201
Title: Thiolactomycin resistance in Escherichia coli is associated with the multidrug resistance efflux pump encoded by emrAB.
Journal: Journal of bacteriology19930601
Title: Activities of fluoroquinolone, macrolide, and aminoglycoside drugs combined with inhibitors of glycosylation and fatty acid and peptide biosynthesis against Mycobacterium avium.
Journal: Antimicrobial agents and chemotherapy19930401
Title: Inhibitors of HIV-1 protease.
Journal: Journal of enzyme inhibition19920101
Title: Characterization of N-myristoyl transferase inhibitors and their effect on HIV release.
Journal: AIDS (London, England)19910801
Title: In vitro inhibition of HIV-1 proteinase by cerulenin.
Journal: FEBS letters19900226
Title: Synthetic non-peptide inhibitors of HIV protease.
Journal: Biochemical and biophysical research communications19890915
Title: Processing of the structural proteins of human immunodeficiency virus type 1 in the presence of monensin and cerulenin.
Journal: Proceedings of the National Academy of Sciences of the United States of America19881201
Title: Cerulenin resistance in a cerulenin-producing fungus. III. Studies on active-site peptides of fatty acid synthetase from Cephalosporium caerulens.
Journal: Journal of biochemistry19840601
Title: Inhibitory effect of cerulenin and sodium butyrate on germination of Candida albicans.
Journal: Antimicrobial agents and chemotherapy19830901
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