19875-60-6,MFCD28166478
Catalog No.:AA002BNG

19875-60-6 | Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)

Pack Size
Purity
Availability
Price(USD)
Quantity
  
1mg
99%
1 week  
$447.00   $313.00
- +
5mg
99%
1 week  
$1,241.00   $869.00
- +
10mg
99%
1 week  
$2,082.00   $1,458.00
- +
  • Technical Information
  • Properties
  • Literature
  • Request for Quotation
  • Download SDS
Technical Information
Catalog Number:
AA002BNG
Chemical Name:
Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)
CAS Number:
19875-60-6
Molecular Formula:
C24H30N4O5
Molecular Weight:
454.5188
MDL Number:
MFCD28166478
SMILES:
OC(=O)/C=C\C(=O)O.CCN(C(=O)N[C@@H]1CN(C)[C@H]2C(=C1)c1cccc3c1c(C2)c[nH]3)CC
Properties
Computed Properties
 
Complexity:
663  
Covalently-Bonded Unit Count:
2  
Defined Atom Stereocenter Count:
2  
Defined Bond Stereocenter Count:
1  
Formal Charge:
0  
Heavy Atom Count:
33  
Hydrogen Bond Acceptor Count:
6  
Hydrogen Bond Donor Count:
4  
Isotope Atom Count:
0  
Rotatable Bond Count:
5  
Undefined Atom Stereocenter Count:
0  
Undefined Bond Stereocenter Count:
0  

Literature

Title: Pathways in pulmonary arterial hypertension: the future is here.

Journal: European respiratory review : an official journal of the European Respiratory Society 20121201

Title: [Prescription of ergot derivatives for lactation inhibition in France: Current practices].

Journal: Journal de gynecologie, obstetrique et biologie de la reproduction 20120401

Title: Antiserotonergic properties of terguride in blood vessels, platelets, and valvular interstitial cells.

Journal: The Journal of pharmacology and experimental therapeutics 20120201

Title: Terguride for pulmonary arterial hypertension.

Journal: Expert opinion on therapeutic targets 20111101

Title: Effects of lisuride hydrogen maleate on pericontusional tissue metabolism, brain edema formation, and contusion volume development after experimental traumatic brain injury in rats.

Journal: Neuroscience letters 20110725

Title: Terguride ameliorates monocrotaline-induced pulmonary hypertension in rats.

Journal: The European respiratory journal 20110501

Title: The dopamine D(2) partial agonist and antagonist terguride decreases heroin self-administration on fixed- and progressive-ratio schedules.

Journal: Pharmacology, biochemistry, and behavior 20101201

Title: Increased expression of 5-hydroxytryptamine2A/B receptors in idiopathic pulmonary fibrosis: a rationale for therapeutic intervention.

Journal: Thorax 20101101

Title: Anticonvulsive effects of the dopamine agonist lisuride maleate after experimental traumatic brain injury.

Journal: Neuroscience letters 20100212

Title: LSD but not lisuride disrupts prepulse inhibition in rats by activating the 5-HT(2A) receptor.

Journal: Psychopharmacology 20100201

Title: Evaluation of the efficacy and safety of terguride in patients with fibromyalgia syndrome: results of a twelve-week, multicenter, randomized, double-blind, placebo-controlled, parallel-group study.

Journal: Arthritis and rheumatism 20100101

Title: Co-administration of the partial dopamine D2 agonist terguride with L-dopa attenuates L-dopa-induced locomotor sensitization in hemiparkinsonian mice.

Journal: Behavioural brain research 20090914

Title: Use of apomorphine in Parkinson's disease.

Journal: Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology 20081201

Title: The effect of terguride in carbon tetrachloride-induced liver fibrosis in rat.

Journal: Experimental biology and medicine (Maywood, N.J.) 20081101

Title: Both mild hypothermia and dopamine D(2) agonist are neuroprotective against hyperthermia-induced injury in PC12 cells.

Journal: Neuroscience letters 20081010

Title: Effect of dopaminergic substances on sleep/wakefulness in saline- and MPTP-treated mice.

Journal: Journal of sleep research 20080301

Title: Effects of aripiprazole and terguride on dopamine synthesis in the dorsal striatum and medial prefrontal cortex of preweanling rats.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20080101

Title: [A case of ruptured internal carotid artery aneurysm mimicking pituitary apoplexy].

Journal: No shinkei geka. Neurological surgery 20071201

Title: Long-term serotonin effects in the rat are prevented by terguride.

Journal: Regulatory peptides 20071004

Title: In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling.

Journal: Journal of psychopharmacology (Oxford, England) 20070801

Title: Hallucinogens recruit specific cortical 5-HT(2A) receptor-mediated signaling pathways to affect behavior.

Journal: Neuron 20070201

Title: In vitro characterization of SLV308 (7-[4-methyl-1-piperazinyl]-2(3H)-benzoxazolone, monohydrochloride): a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist.

Journal: Synapse (New York, N.Y.) 20061215

Title: Striking differences of action of lisuride stereoisomers at histamine H1 receptors.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 20061201

Title: Observed smoking in cars: a method and differences by socioeconomic area.

Journal: Tobacco control 20061001

Title: Glutamate-induced cell death and formation of radicals can be reduced by lisuride in mesencephalic primary cell culture.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20060901

Title: Dopamine stimulation via infusion in the lateral ventricle.

Journal: Annals of the New York Academy of Sciences 20060801

Title: Homology modelling of the serotoninergic 5-HT2c receptor.

Journal: Journal of enzyme inhibition and medicinal chemistry 20060601

Title: Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.

Journal: European journal of pharmacology 20060327

Title: The partial dopamine D2-like receptor agonist terguride functions as an agonist in preweanling rats after a 5-day reserpine regimen.

Journal: Psychopharmacology 20060301

Title: Effects of terguride, ropinirole, and acetyl-L-carnitine on methamphetamine withdrawal in the rat.

Journal: Pharmacology, biochemistry, and behavior 20060301

Title: Effects of a partial D2-like receptor agonist on striatal dopamine autoreceptor functioning in preweanling rats.

Journal: Brain research 20060216

Title: Transdermal lisuride: short-term efficacy and tolerability study in patients with severe restless legs syndrome.

Journal: Sleep medicine 20060101

Title: Lisuride treatment of restless legs syndrome: first studies with monotherapy in de novo patients and in combination with levodopa in advanced disease.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20060101

Title: Lisuride, a dopamine receptor agonist with 5-HT2B receptor antagonist properties: absence of cardiac valvulopathy adverse drug reaction reports supports the concept of a crucial role for 5-HT2B receptor agonism in cardiac valvular fibrosis.

Journal: Clinical neuropharmacology 20060101

Title: Dopamine and serotonin modulate the onset of metamorphosis in the ascidian Phallusia mammillata.

Journal: Developmental biology 20050601

Title: Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.

Journal: European journal of pharmacology 20050516

Title: Levodopa in the treatment of Parkinson's disease: current controversies.

Journal: Movement disorders : official journal of the Movement Disorder Society 20050501

Title: Evidence-based medical review update: pharmacological and surgical treatments of Parkinson's disease: 2001 to 2004.

Journal: Movement disorders : official journal of the Movement Disorder Society 20050501

Title: Influence of steric hindrance on enantioseparation of Dns-amino acids and pesticides on terguride based chiral selectors in capillary electrophoresis.

Journal: Journal of separation science 20050501

Title: The partial D2-like dopamine receptor agonist terguride acts as a functional antagonist in states of high and low dopaminergic tone: evidence from preweanling rats.

Journal: Psychopharmacology 20050401

Title: Capillary zone electrophoresis separation of enantiomers of lisuride.

Journal: Journal of chromatography. A 20050225

Title: Buprenorphine and a CRF1 antagonist block the acquisition of opiate withdrawal-induced conditioned place aversion in rats.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20050101

Title: Regulation of serotonin 5-HT2C receptors by chronic ligand exposure.

Journal: European journal of pharmacology 20040913

Title: The effects of dopamine receptor agonists and antagonists on the secretory rate of cockroach (Periplaneta americana) salivary glands.

Journal: Journal of insect physiology 20040901

Title: 8R-lisuride is a potent stereospecific histamine H1-receptor partial agonist.

Journal: Molecular pharmacology 20040301

Title: No evidence of the usefulness of eye blinking as a marker for central dopaminergic activity.

Journal: Journal of psychopharmacology (Oxford, England) 20040301

Title: Pergolide, terguride and N,N'-spacer-linked oligomers of both interact with 5-HT2A receptors of rat tail artery.

Journal: Physiological research 20040101

Title: LSD, 5-HT (serotonin), and the evolution of a behavioral assay.

Journal: Neuroscience and biobehavioral reviews 20040101

Title: Transdermal lisuride delivery in the treatment of Parkinson's disease.

Journal: Journal of neural transmission. Supplementum 20040101

Title: Effects of terguride treatment on glucose abnormalities induced by ischemic brain damage in SHR/N-cp lean Koletsky strain and in rats of Wistar strain.

Journal: Bratislavske lekarske listy 20040101

Title: The dopamine receptor agonist lisuride attenuates iron-mediated dopaminergic neurodegeneration.

Journal: Experimental neurology 20031101

Title: Management of restless legs syndrome by the partial D2-agonist terguride.

Journal: Sleep medicine 20030901

Title: Cortisol as an indicator of dopaminergic effects on nicotine craving.

Journal: Human psychopharmacology 20030801

Title: Effects of a partial dopamine D2-like agonist on the cocaine-induced behavioral sensitization of preweanling rats.

Journal: Pharmacology, biochemistry, and behavior 20030801

Title: [Pharmacokinetic/pharmacodynamic analysis of anti-hyperprolactinemic effect of terguride based on dopamine D2 receptor occupancy].

Journal: Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20030401

Title: Suppression of cocaine- and food-maintained behavior by the D2-like receptor partial agonist terguride in squirrel monkeys.

Journal: Psychopharmacology 20030301

Title: Inhibition of growth hormone excess reduces insulin resistance and ovarian dysfunction in a lean case of polycystic ovary syndrome with a growth-hormone-producing pituitary adenoma.

Journal: Hormone research 20030101

Title: [Arrest of lactation after 2nd trimester abortion with a single dose of cabergoline in comparison with 10-day administration of teguride].

Journal: Ceska gynekologie 20030101

Title: [Results of treatment for male prolactinomas].

Journal: No shinkei geka. Neurological surgery 20021201

Title: Re-evaluation of lisuride pharmacology: 5-hydroxytryptamine1A receptor-mediated behavioral effects overlap its other properties in rats.

Journal: Psychopharmacology 20021001

Title: Prospective randomized trial of lisuride infusion versus oral levodopa in patients with Parkinson's disease.

Journal: Brain : a journal of neurology 20020901

Title: The trigonometric responder approach: a new method for detecting responders to pharmacological or experimental challenges.

Journal: Pharmacopsychiatry 20020901

Title: Terguride treatment attenuated prolactin release and enhanced insulin receptor affinity and GLUT 4 content in obese spontaneously hypertensive female, but not male rats.

Journal: Annals of the New York Academy of Sciences 20020601

Title: Is the 5-HT(7) receptor involved in the pathogenesis and prophylactic treatment of migraine?

Journal: European journal of pharmacology 20020329

Title: Clustered ergot alkaloids modulate cell-mediated cytotoxicity.

Journal: Bioorganic & medicinal chemistry 20020201

Title: Lisuride, a dopamine D2 receptor agonist, and anticraving drug expectancy as modifiers of relapse in alcohol dependence.

Journal: Progress in neuro-psychopharmacology & biological psychiatry 20020201

Title: Protection of dopaminergic neurons in primary culture by lisuride.

Journal: Journal of neural transmission (Vienna, Austria : 1996) 20020201

Title: DA agonists -- ergot derivatives: bromocriptine: management of Parkinson's disease.

Journal: Movement disorders : official journal of the Movement Disorder Society 20020101

Title: DA agonists -- ergot derivatives: lisuride: management of Parkinson's disease.

Journal: Movement disorders : official journal of the Movement Disorder Society 20020101

Title: [Use of dopamine agonists in the treatment of Parkinson's disease].

Journal: Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova 20020101

Title: Quantitative analysis of striatal dopamine D2 receptors with 123 I-iodolisuride SPECT in degenerative extrapyramidal diseases.

Journal: Nuclear medicine communications 20011101

Title: Dopaminergic modulation of grooming behavior in virgin and pregnant rats.

Journal: Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas 20011101

Title: Dopamine partial agonist reverses amphetamine withdrawal in rats.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20011101

Title: Poetic talent unmasked by treatment of Parkinson's disease.

Journal: Movement disorders : official journal of the Movement Disorder Society 20011101

Title: Real-time analysis of dopamine: antagonist interactions at recombinant human D2long receptor upon modulation of its activation state.

Journal: British journal of pharmacology 20010901

Title: Symptomatic treatment of premenstrual mastalgia in premenopausal women with lisuride maleate: a double-blind placebo-controlled randomized study.

Journal: Fertility and sterility 20010401

Title: A dopamine partial agonist and antagonist block amphetamine self-administration in a progressive ratio schedule.

Journal: Pharmacology, biochemistry, and behavior 20010401

Title: [Parkinson disease: diagnostic and therapeutic criteria].

Journal: Presse medicale (Paris, France : 1983) 20010303

Title: Long-duration effect and the postsynaptic compartment: study using a dopamine agonist with a short half-life.

Journal: Movement disorders : official journal of the Movement Disorder Society 20010301

Title: Efficacy and tolerability of dopamine agonists in a parkinsonian population.

Journal: Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology 20010201

Title: The influence of personality on nicotine craving: a hierarchical multivariate statistical prediction model.

Journal: Neuropsychobiology 20010101

Title: Clinical features and medical treatment of male prolactinomas.

Journal: Acta neurochirurgica 20010101

Title: Nonlinear analysis of partial dopamine agonist effects on cAMP in C6 glioma cells.

Journal: Journal of pharmacological and toxicological methods 20010101

Title: Atypical polypoid adenomyoma in a patient with hyperprolactinemia.

Journal: International journal of gynecological cancer : official journal of the International Gynecological Cancer Society 20010101

Title: Terguride attenuates prolactin levels and ameliorates insulin sensitivity and insulin binding in obese spontaneously hypertensive rats.

Journal: Physiological research 20010101

Title: Sleep attacks and Parkinson's disease treatment.

Journal: Lancet (London, England) 20000415

Title: Pharmacological effects of BAM-1120, a novel ergoline derivative, on central dopaminergic functions in rats.

Journal: Methods and findings in experimental and clinical pharmacology 19980901

Title: Characterization of enhanced behavioral responses to L-DOPA following repeated administration in the 6-hydroxydopamine-lesioned rat model of Parkinson's disease.

Journal: Experimental neurology 19980601

Title: Postpartum cerebral angiopathy with intracerebral hemorrhage in a patient receiving lisuride.

Journal: Neurology 19980401

Title: Agonist activity of antimigraine drugs at recombinant human 5-HT1A receptors: potential implications for prophylactic and acute therapy.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19970601

Title: Involvement of dopamine D2 receptors in the effect of cocaine on sexual behaviour and stretching-yawning of male rats.

Journal: Neuropharmacology 19970601

Title: Effects of terguride on anterior pituitary function in parkinsonian patients treated with L-dopa: a double-blind study versus placebo.

Journal: Clinical neuropharmacology 19960201

Title: Is alpha-methyldopa-type autoimmune hemolytic anemia mediated by interferon-gamma?

Journal: Annals of hematology 19941101

Title: [Therapeutic effect of lisuride maleate on post-stroke depression].

Journal: Nihon Ronen Igakkai zasshi. Japanese journal of geriatrics 19940101

Title: Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.

Journal: European journal of pharmacology 19930624

Title: Effects of terguride, a partial D2 agonist, on MPTP-lesioned parkinsonian cynomolgus monkeys.

Journal: Annals of neurology 19930501

Title: Extrapyramidal syndrome responsive to dopaminergic treatment following recovery from central pontine myelinolysis.

Journal: European neurology 19930101

Title: Transient left bundle branch block following intravenous lisuride bolus.

Journal: Fundamental & clinical pharmacology 19930101

Title: Partial dopamine agonist therapy of levodopa-induced dyskinesias.

Journal: Neurology 19920601

Title: Levodopa-induced dyskinesias in Parkinson's disease: clinical and pharmacological classification.

Journal: Movement disorders : official journal of the Movement Disorder Society 19920101

Title: Antagonist effect of terguride in Parkinson's disease.

Journal: Clinical neuropharmacology 19911001

Title: Behavioural profile of partial D2 dopamine receptor agonists. 1. Atypical inhibition of d-amphetamine-induced locomotor hyperactivity and stereotypy.

Journal: Psychopharmacology 19910101

Title: Subcutaneous administration of lisuride in the treatment of complex motor fluctuations in Parkinson's disease.

Journal: Journal of neural transmission. Supplementum 19880101

Title: Continuous subcutaneous lisuride infusions in Parkinson's disease.

Journal: Journal of neural transmission. Supplementum 19880101

Title: Treatment of Parkinson's disease with subcutaneous lisuride infusions.

Journal: Journal of neural transmission. Supplementum 19880101

Title: Lisuride infusion pump in Parkinson's disease. A report of two cases.

Journal: Journal of neural transmission. Supplementum 19880101

Title: Transdihydrolisuride in parkinsonism.

Journal: Clinical neuropharmacology 19870101

Title: Studies on the involvement of dopamine D-1 and D-2 receptors in the anticonvulsant effect of dopamine agonists in various rodent models of epilepsy.

Journal: European journal of pharmacology 19860822

Title: The use of pergolide and lisuride, two experimental dopamine agonists, in patients with advanced Parkinson disease.

Journal: The American journal of the medical sciences 19850901

Title: Novel 8 alpha-ergolines with inhibitory and stimulatory effects on prolactin secretion in rats.

Journal: Life sciences 19841029

Title: Drug-induced modulation of locomotor hyperactivity induced by picrotoxin in nucleus accumbens.

Journal: Pharmacology, biochemistry, and behavior 19841001

Title: Use of ergot derivative lisuride in Parkinson's disease.

Journal: Advances in neurology 19840101

Title: [Acid lysuride maleate in the prevention of migraine headache. Clinical experience].

Journal: Minerva medica 19830714

Title: Anwesenheit: psychopathology and clinical associations.

Journal: The British journal of psychiatry : the journal of mental science 19821201

Title: Influence of lisuride on morphine withdrawal signs in the rat: a dopamine-mimetic effect.

Journal: Psychopharmacology 19820101

Title: Action of lisuride on reserpine-induced muscular rigidity in rats after local application into the striatum, ventricular space or the spinal subarachnoid space.

Journal: Arzneimittel-Forschung 19820101

Title: Depression of reserpine-induced muscular rigidity in rats after administration of lisuride into the spinal subarachnoid space.

Journal: Naunyn-Schmiedeberg's archives of pharmacology 19800101

Title: Suppression of prolactin secretion by lisuride throughout the menstrual cycle and in hyperprolactinaemic menstrual disorders.

Journal: Acta endocrinologica 19790901

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Related Products of 19875-60-6
Tags:19875-60-6 Molecular Formula|19875-60-6 MDL|19875-60-6 SMILES|19875-60-6 Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)
Catalog No.: AA002BNG
19875-60-6,MFCD28166478
19875-60-6 | Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)
Pack Size: 1mg
Purity: 99%
1 week
$447.00 $313.00
Pack Size: 5mg
Purity: 99%
1 week
$1,241.00 $869.00
Pack Size: 10mg
Purity: 99%
1 week
$2,082.00 $1,458.00
Quantity
- +
Add to Card
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Technical Information
Catalog Number: AA002BNG
Chemical Name: Urea, N'-[(8α)-9,10-didehydro-6-methylergolin-8-yl]-N,N-diethyl-, (2Z)-2-butenedioate (1:1)
CAS Number: 19875-60-6
Molecular Formula: C24H30N4O5
Molecular Weight: 454.5188
MDL Number: MFCD28166478
SMILES: OC(=O)/C=C\C(=O)O.CCN(C(=O)N[C@@H]1CN(C)[C@H]2C(=C1)c1cccc3c1c(C2)c[nH]3)CC
Properties
Complexity: 663  
Covalently-Bonded Unit Count: 2  
Defined Atom Stereocenter Count: 2  
Defined Bond Stereocenter Count: 1  
Formal Charge: 0  
Heavy Atom Count: 33  
Hydrogen Bond Acceptor Count: 6  
Hydrogen Bond Donor Count: 4  
Isotope Atom Count: 0  
Rotatable Bond Count: 5  
Undefined Atom Stereocenter Count: 0  
Undefined Bond Stereocenter Count: 0  
Literature fold

Title: Pathways in pulmonary arterial hypertension: the future is here.

Journal: European respiratory review : an official journal of the European Respiratory Society20121201

Title: [Prescription of ergot derivatives for lactation inhibition in France: Current practices].

Journal: Journal de gynecologie, obstetrique et biologie de la reproduction20120401

Title: Antiserotonergic properties of terguride in blood vessels, platelets, and valvular interstitial cells.

Journal: The Journal of pharmacology and experimental therapeutics20120201

Title: Terguride for pulmonary arterial hypertension.

Journal: Expert opinion on therapeutic targets20111101

Title: Effects of lisuride hydrogen maleate on pericontusional tissue metabolism, brain edema formation, and contusion volume development after experimental traumatic brain injury in rats.

Journal: Neuroscience letters20110725

Title: Terguride ameliorates monocrotaline-induced pulmonary hypertension in rats.

Journal: The European respiratory journal20110501

Title: The dopamine D(2) partial agonist and antagonist terguride decreases heroin self-administration on fixed- and progressive-ratio schedules.

Journal: Pharmacology, biochemistry, and behavior20101201

Title: Increased expression of 5-hydroxytryptamine2A/B receptors in idiopathic pulmonary fibrosis: a rationale for therapeutic intervention.

Journal: Thorax20101101

Title: Anticonvulsive effects of the dopamine agonist lisuride maleate after experimental traumatic brain injury.

Journal: Neuroscience letters20100212

Title: LSD but not lisuride disrupts prepulse inhibition in rats by activating the 5-HT(2A) receptor.

Journal: Psychopharmacology20100201

Title: Evaluation of the efficacy and safety of terguride in patients with fibromyalgia syndrome: results of a twelve-week, multicenter, randomized, double-blind, placebo-controlled, parallel-group study.

Journal: Arthritis and rheumatism20100101

Title: Co-administration of the partial dopamine D2 agonist terguride with L-dopa attenuates L-dopa-induced locomotor sensitization in hemiparkinsonian mice.

Journal: Behavioural brain research20090914

Title: Use of apomorphine in Parkinson's disease.

Journal: Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology20081201

Title: The effect of terguride in carbon tetrachloride-induced liver fibrosis in rat.

Journal: Experimental biology and medicine (Maywood, N.J.)20081101

Title: Both mild hypothermia and dopamine D(2) agonist are neuroprotective against hyperthermia-induced injury in PC12 cells.

Journal: Neuroscience letters20081010

Title: Effect of dopaminergic substances on sleep/wakefulness in saline- and MPTP-treated mice.

Journal: Journal of sleep research20080301

Title: Effects of aripiprazole and terguride on dopamine synthesis in the dorsal striatum and medial prefrontal cortex of preweanling rats.

Journal: Journal of neural transmission (Vienna, Austria : 1996)20080101

Title: [A case of ruptured internal carotid artery aneurysm mimicking pituitary apoplexy].

Journal: No shinkei geka. Neurological surgery20071201

Title: Long-term serotonin effects in the rat are prevented by terguride.

Journal: Regulatory peptides20071004

Title: In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling.

Journal: Journal of psychopharmacology (Oxford, England)20070801

Title: Hallucinogens recruit specific cortical 5-HT(2A) receptor-mediated signaling pathways to affect behavior.

Journal: Neuron20070201

Title: In vitro characterization of SLV308 (7-[4-methyl-1-piperazinyl]-2(3H)-benzoxazolone, monohydrochloride): a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist.

Journal: Synapse (New York, N.Y.)20061215

Title: Striking differences of action of lisuride stereoisomers at histamine H1 receptors.

Journal: Naunyn-Schmiedeberg's archives of pharmacology20061201

Title: Observed smoking in cars: a method and differences by socioeconomic area.

Journal: Tobacco control20061001

Title: Glutamate-induced cell death and formation of radicals can be reduced by lisuride in mesencephalic primary cell culture.

Journal: Journal of neural transmission (Vienna, Austria : 1996)20060901

Title: Dopamine stimulation via infusion in the lateral ventricle.

Journal: Annals of the New York Academy of Sciences20060801

Title: Homology modelling of the serotoninergic 5-HT2c receptor.

Journal: Journal of enzyme inhibition and medicinal chemistry20060601

Title: Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.

Journal: European journal of pharmacology20060327

Title: The partial dopamine D2-like receptor agonist terguride functions as an agonist in preweanling rats after a 5-day reserpine regimen.

Journal: Psychopharmacology20060301

Title: Effects of terguride, ropinirole, and acetyl-L-carnitine on methamphetamine withdrawal in the rat.

Journal: Pharmacology, biochemistry, and behavior20060301

Title: Effects of a partial D2-like receptor agonist on striatal dopamine autoreceptor functioning in preweanling rats.

Journal: Brain research20060216

Title: Transdermal lisuride: short-term efficacy and tolerability study in patients with severe restless legs syndrome.

Journal: Sleep medicine20060101

Title: Lisuride treatment of restless legs syndrome: first studies with monotherapy in de novo patients and in combination with levodopa in advanced disease.

Journal: Journal of neural transmission (Vienna, Austria : 1996)20060101

Title: Lisuride, a dopamine receptor agonist with 5-HT2B receptor antagonist properties: absence of cardiac valvulopathy adverse drug reaction reports supports the concept of a crucial role for 5-HT2B receptor agonism in cardiac valvular fibrosis.

Journal: Clinical neuropharmacology20060101

Title: Dopamine and serotonin modulate the onset of metamorphosis in the ascidian Phallusia mammillata.

Journal: Developmental biology20050601

Title: Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.

Journal: European journal of pharmacology20050516

Title: Levodopa in the treatment of Parkinson's disease: current controversies.

Journal: Movement disorders : official journal of the Movement Disorder Society20050501

Title: Evidence-based medical review update: pharmacological and surgical treatments of Parkinson's disease: 2001 to 2004.

Journal: Movement disorders : official journal of the Movement Disorder Society20050501

Title: Influence of steric hindrance on enantioseparation of Dns-amino acids and pesticides on terguride based chiral selectors in capillary electrophoresis.

Journal: Journal of separation science20050501

Title: The partial D2-like dopamine receptor agonist terguride acts as a functional antagonist in states of high and low dopaminergic tone: evidence from preweanling rats.

Journal: Psychopharmacology20050401

Title: Capillary zone electrophoresis separation of enantiomers of lisuride.

Journal: Journal of chromatography. A20050225

Title: Buprenorphine and a CRF1 antagonist block the acquisition of opiate withdrawal-induced conditioned place aversion in rats.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20050101

Title: Regulation of serotonin 5-HT2C receptors by chronic ligand exposure.

Journal: European journal of pharmacology20040913

Title: The effects of dopamine receptor agonists and antagonists on the secretory rate of cockroach (Periplaneta americana) salivary glands.

Journal: Journal of insect physiology20040901

Title: 8R-lisuride is a potent stereospecific histamine H1-receptor partial agonist.

Journal: Molecular pharmacology20040301

Title: No evidence of the usefulness of eye blinking as a marker for central dopaminergic activity.

Journal: Journal of psychopharmacology (Oxford, England)20040301

Title: Pergolide, terguride and N,N'-spacer-linked oligomers of both interact with 5-HT2A receptors of rat tail artery.

Journal: Physiological research20040101

Title: LSD, 5-HT (serotonin), and the evolution of a behavioral assay.

Journal: Neuroscience and biobehavioral reviews20040101

Title: Transdermal lisuride delivery in the treatment of Parkinson's disease.

Journal: Journal of neural transmission. Supplementum20040101

Title: Effects of terguride treatment on glucose abnormalities induced by ischemic brain damage in SHR/N-cp lean Koletsky strain and in rats of Wistar strain.

Journal: Bratislavske lekarske listy20040101

Title: The dopamine receptor agonist lisuride attenuates iron-mediated dopaminergic neurodegeneration.

Journal: Experimental neurology20031101

Title: Management of restless legs syndrome by the partial D2-agonist terguride.

Journal: Sleep medicine20030901

Title: Cortisol as an indicator of dopaminergic effects on nicotine craving.

Journal: Human psychopharmacology20030801

Title: Effects of a partial dopamine D2-like agonist on the cocaine-induced behavioral sensitization of preweanling rats.

Journal: Pharmacology, biochemistry, and behavior20030801

Title: [Pharmacokinetic/pharmacodynamic analysis of anti-hyperprolactinemic effect of terguride based on dopamine D2 receptor occupancy].

Journal: Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan20030401

Title: Suppression of cocaine- and food-maintained behavior by the D2-like receptor partial agonist terguride in squirrel monkeys.

Journal: Psychopharmacology20030301

Title: Inhibition of growth hormone excess reduces insulin resistance and ovarian dysfunction in a lean case of polycystic ovary syndrome with a growth-hormone-producing pituitary adenoma.

Journal: Hormone research20030101

Title: [Arrest of lactation after 2nd trimester abortion with a single dose of cabergoline in comparison with 10-day administration of teguride].

Journal: Ceska gynekologie20030101

Title: [Results of treatment for male prolactinomas].

Journal: No shinkei geka. Neurological surgery20021201

Title: Re-evaluation of lisuride pharmacology: 5-hydroxytryptamine1A receptor-mediated behavioral effects overlap its other properties in rats.

Journal: Psychopharmacology20021001

Title: Prospective randomized trial of lisuride infusion versus oral levodopa in patients with Parkinson's disease.

Journal: Brain : a journal of neurology20020901

Title: The trigonometric responder approach: a new method for detecting responders to pharmacological or experimental challenges.

Journal: Pharmacopsychiatry20020901

Title: Terguride treatment attenuated prolactin release and enhanced insulin receptor affinity and GLUT 4 content in obese spontaneously hypertensive female, but not male rats.

Journal: Annals of the New York Academy of Sciences20020601

Title: Is the 5-HT(7) receptor involved in the pathogenesis and prophylactic treatment of migraine?

Journal: European journal of pharmacology20020329

Title: Clustered ergot alkaloids modulate cell-mediated cytotoxicity.

Journal: Bioorganic & medicinal chemistry20020201

Title: Lisuride, a dopamine D2 receptor agonist, and anticraving drug expectancy as modifiers of relapse in alcohol dependence.

Journal: Progress in neuro-psychopharmacology & biological psychiatry20020201

Title: Protection of dopaminergic neurons in primary culture by lisuride.

Journal: Journal of neural transmission (Vienna, Austria : 1996)20020201

Title: DA agonists -- ergot derivatives: bromocriptine: management of Parkinson's disease.

Journal: Movement disorders : official journal of the Movement Disorder Society20020101

Title: DA agonists -- ergot derivatives: lisuride: management of Parkinson's disease.

Journal: Movement disorders : official journal of the Movement Disorder Society20020101

Title: [Use of dopamine agonists in the treatment of Parkinson's disease].

Journal: Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova20020101

Title: Quantitative analysis of striatal dopamine D2 receptors with 123 I-iodolisuride SPECT in degenerative extrapyramidal diseases.

Journal: Nuclear medicine communications20011101

Title: Dopaminergic modulation of grooming behavior in virgin and pregnant rats.

Journal: Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas20011101

Title: Dopamine partial agonist reverses amphetamine withdrawal in rats.

Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20011101

Title: Poetic talent unmasked by treatment of Parkinson's disease.

Journal: Movement disorders : official journal of the Movement Disorder Society20011101

Title: Real-time analysis of dopamine: antagonist interactions at recombinant human D2long receptor upon modulation of its activation state.

Journal: British journal of pharmacology20010901

Title: Symptomatic treatment of premenstrual mastalgia in premenopausal women with lisuride maleate: a double-blind placebo-controlled randomized study.

Journal: Fertility and sterility20010401

Title: A dopamine partial agonist and antagonist block amphetamine self-administration in a progressive ratio schedule.

Journal: Pharmacology, biochemistry, and behavior20010401

Title: [Parkinson disease: diagnostic and therapeutic criteria].

Journal: Presse medicale (Paris, France : 1983)20010303

Title: Long-duration effect and the postsynaptic compartment: study using a dopamine agonist with a short half-life.

Journal: Movement disorders : official journal of the Movement Disorder Society20010301

Title: Efficacy and tolerability of dopamine agonists in a parkinsonian population.

Journal: Neurological sciences : official journal of the Italian Neurological Society and of the Italian Society of Clinical Neurophysiology20010201

Title: The influence of personality on nicotine craving: a hierarchical multivariate statistical prediction model.

Journal: Neuropsychobiology20010101

Title: Clinical features and medical treatment of male prolactinomas.

Journal: Acta neurochirurgica20010101

Title: Nonlinear analysis of partial dopamine agonist effects on cAMP in C6 glioma cells.

Journal: Journal of pharmacological and toxicological methods20010101

Title: Atypical polypoid adenomyoma in a patient with hyperprolactinemia.

Journal: International journal of gynecological cancer : official journal of the International Gynecological Cancer Society20010101

Title: Terguride attenuates prolactin levels and ameliorates insulin sensitivity and insulin binding in obese spontaneously hypertensive rats.

Journal: Physiological research20010101

Title: Sleep attacks and Parkinson's disease treatment.

Journal: Lancet (London, England)20000415

Title: Pharmacological effects of BAM-1120, a novel ergoline derivative, on central dopaminergic functions in rats.

Journal: Methods and findings in experimental and clinical pharmacology19980901

Title: Characterization of enhanced behavioral responses to L-DOPA following repeated administration in the 6-hydroxydopamine-lesioned rat model of Parkinson's disease.

Journal: Experimental neurology19980601

Title: Postpartum cerebral angiopathy with intracerebral hemorrhage in a patient receiving lisuride.

Journal: Neurology19980401

Title: Agonist activity of antimigraine drugs at recombinant human 5-HT1A receptors: potential implications for prophylactic and acute therapy.

Journal: Naunyn-Schmiedeberg's archives of pharmacology19970601

Title: Involvement of dopamine D2 receptors in the effect of cocaine on sexual behaviour and stretching-yawning of male rats.

Journal: Neuropharmacology19970601

Title: Effects of terguride on anterior pituitary function in parkinsonian patients treated with L-dopa: a double-blind study versus placebo.

Journal: Clinical neuropharmacology19960201

Title: Is alpha-methyldopa-type autoimmune hemolytic anemia mediated by interferon-gamma?

Journal: Annals of hematology19941101

Title: [Therapeutic effect of lisuride maleate on post-stroke depression].

Journal: Nihon Ronen Igakkai zasshi. Japanese journal of geriatrics19940101

Title: Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.

Journal: European journal of pharmacology19930624

Title: Effects of terguride, a partial D2 agonist, on MPTP-lesioned parkinsonian cynomolgus monkeys.

Journal: Annals of neurology19930501

Title: Extrapyramidal syndrome responsive to dopaminergic treatment following recovery from central pontine myelinolysis.

Journal: European neurology19930101

Title: Transient left bundle branch block following intravenous lisuride bolus.

Journal: Fundamental & clinical pharmacology19930101

Title: Partial dopamine agonist therapy of levodopa-induced dyskinesias.

Journal: Neurology19920601

Title: Levodopa-induced dyskinesias in Parkinson's disease: clinical and pharmacological classification.

Journal: Movement disorders : official journal of the Movement Disorder Society19920101

Title: Antagonist effect of terguride in Parkinson's disease.

Journal: Clinical neuropharmacology19911001

Title: Behavioural profile of partial D2 dopamine receptor agonists. 1. Atypical inhibition of d-amphetamine-induced locomotor hyperactivity and stereotypy.

Journal: Psychopharmacology19910101

Title: Subcutaneous administration of lisuride in the treatment of complex motor fluctuations in Parkinson's disease.

Journal: Journal of neural transmission. Supplementum19880101

Title: Continuous subcutaneous lisuride infusions in Parkinson's disease.

Journal: Journal of neural transmission. Supplementum19880101

Title: Treatment of Parkinson's disease with subcutaneous lisuride infusions.

Journal: Journal of neural transmission. Supplementum19880101

Title: Lisuride infusion pump in Parkinson's disease. A report of two cases.

Journal: Journal of neural transmission. Supplementum19880101

Title: Transdihydrolisuride in parkinsonism.

Journal: Clinical neuropharmacology19870101

Title: Studies on the involvement of dopamine D-1 and D-2 receptors in the anticonvulsant effect of dopamine agonists in various rodent models of epilepsy.

Journal: European journal of pharmacology19860822

Title: The use of pergolide and lisuride, two experimental dopamine agonists, in patients with advanced Parkinson disease.

Journal: The American journal of the medical sciences19850901

Title: Novel 8 alpha-ergolines with inhibitory and stimulatory effects on prolactin secretion in rats.

Journal: Life sciences19841029

Title: Drug-induced modulation of locomotor hyperactivity induced by picrotoxin in nucleus accumbens.

Journal: Pharmacology, biochemistry, and behavior19841001

Title: Use of ergot derivative lisuride in Parkinson's disease.

Journal: Advances in neurology19840101

Title: [Acid lysuride maleate in the prevention of migraine headache. Clinical experience].

Journal: Minerva medica19830714

Title: Anwesenheit: psychopathology and clinical associations.

Journal: The British journal of psychiatry : the journal of mental science19821201

Title: Influence of lisuride on morphine withdrawal signs in the rat: a dopamine-mimetic effect.

Journal: Psychopharmacology19820101

Title: Action of lisuride on reserpine-induced muscular rigidity in rats after local application into the striatum, ventricular space or the spinal subarachnoid space.

Journal: Arzneimittel-Forschung19820101

Title: Depression of reserpine-induced muscular rigidity in rats after administration of lisuride into the spinal subarachnoid space.

Journal: Naunyn-Schmiedeberg's archives of pharmacology19800101

Title: Suppression of prolactin secretion by lisuride throughout the menstrual cycle and in hyperprolactinaemic menstrual disorders.

Journal: Acta endocrinologica19790901

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