Title: Behavioral and neurochemical profile of some novel phenacyl based isonipecotamide derivatives.
Journal: Pakistan journal of pharmaceutical sciences20121001
Title: Anti-AIDS agents 90. novel C-28 modified bevirimat analogues as potent HIV maturation inhibitors.
Journal: Journal of medicinal chemistry20120927
Title: A β-tryptase inhibitor with a tropanylamide scaffold to improve in vitro stability and to lower hERG channel binding affinity.
Journal: Bioorganic & medicinal chemistry letters20120215
Title: Development of Metarhizium anisopliae and Beauveria bassiana formulations for control of malaria mosquito larvae.
Journal: Parasites & vectors20110101
Title: New classes of alanine racemase inhibitors identified by high-throughput screening show antimicrobial activity against Mycobacterium tuberculosis.
Journal: PloS one20110101
Title: A conformationally constrained inhibitor with an enhanced potency for β-tryptase and stability against semicarbazide-sensitive amine oxidase (SSAO).
Journal: Bioorganic & medicinal chemistry letters20101115
Title: Non-peptidic antagonists of the CGRP receptor, BIBN4096BS and MK-0974, interact with the calcitonin receptor-like receptor via methionine-42 and RAMP1 via tryptophan-74.
Journal: Biochemical and biophysical research communications20100101
Title: Discovery of 4-morpholino-6-aryl-1H-pyrazolo[3,4-d]pyrimidines as highly potent and selective ATP-competitive inhibitors of the mammalian target of rapamycin (mTOR): optimization of the 6-aryl substituent.
Journal: Journal of medicinal chemistry20091224
Title: Optimization of 2-piperidin-4-yl-acetamides as melanin-concentrating hormone receptor 1 (MCH-R1) antagonists: Designing out hERG inhibition.
Journal: Bioorganic & medicinal chemistry letters20090801
Title: Optimization of piperidin-4-yl-urea-containing melanin-concentrating hormone receptor 1 (MCH-R1) antagonists: Reducing hERG-associated liabilities.
Journal: Bioorganic & medicinal chemistry letters20090801
Title: Synthesis and structure-activity relationship of novel diarylpyrazole imide analogues as CB1 cannabinoid receptor ligands.
Journal: Bioorganic & medicinal chemistry20090415
Title: The design and discovery of novel amide CCR5 antagonists.
Journal: Bioorganic & medicinal chemistry letters20090215
Title: Casopitant: a novel NK(1)-receptor antagonist in the prevention of chemotherapy-induced nausea and vomiting.
Journal: Therapeutics and clinical risk management20090101
Title: 1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor.
Journal: Bioorganic & medicinal chemistry20080315
Title: Functional antagonism between endogenous neuropeptide Y and calcitonin gene-related peptide in mesenteric resistance arteries.
Journal: The Journal of pharmacology and experimental therapeutics20080301
Title: Methoxy- and fluorine-substituted analogs of O-1302: synthesis and in vitro binding affinity for the CB1 cannabinoid receptor.
Journal: Chemical & pharmaceutical bulletin20070801
Title: Piperidine amides as 11beta-hydroxysteroid dehydrogenase type 1 inhibitors.
Journal: Bioorganic & medicinal chemistry letters20070615
Title: Pharmacological characterisation of capsaicin-induced relaxations in human and porcine isolated arteries.
Journal: Naunyn-Schmiedeberg's archives of pharmacology20070301
Title: Enantioselective strecker reaction of phosphinoyl ketoimines catalyzed by in situ prepared chiral N,N'-dioxides.
Journal: The Journal of organic chemistry20070105
Title: Determinants of 1-piperidinecarboxamide, N-[2-[[5-amino-l-[[4-(4-pyridinyl)-l-piperazinyl]carbonyl]pentyl]amino]-1-[(3,5-dibromo-4-hydroxyphenyl)methyl]-2-oxoethyl]-4-(1,4-dihydro-2-oxo-3(2H)-quinazolinyl) (BIBN4096BS) affinity for calcitonin gene-related peptide and amylin receptors--the role of receptor activity modifying protein 1.
Journal: Molecular pharmacology20061201
Title: A key role for transmembrane prolines in calcitonin receptor-like receptor agonist binding and signalling: implications for family B G-protein-coupled receptors.
Journal: Molecular pharmacology20050101
Title: Noncompetitive antagonism of BIBN4096BS on CGRP-induced responses in human subcutaneous arteries.
Journal: British journal of pharmacology20041201
Title: Structure activity relationship by NMR and by computer: a comparative study.
Journal: Journal of the American Chemical Society20020918
Title: GC/MS investigations of the minor constituents of Piper guineense stem.
Journal: Die Pharmazie20020901
Title: A piperidine amide extracted from Piper longum L. fruit shows activity against Aedes aegypti mosquito larvae.
Journal: Journal of agricultural and food chemistry20020619
Title: Tandem mass spectrum of a growth hormone secretagogue: amide bond cleavage and resultant gas-phase rearrangement.
Journal: Journal of the American Society for Mass Spectrometry20020401
