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Title: The novel mu-opioid antagonist, GSK1521498, reduces ethanol consumption in C57BL/6J mice.
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Title: Orally active opioid μ/δ dual agonist MGM-16, a derivative of the indole alkaloid mitragynine, exhibits potent antiallodynic effect on neuropathic pain in mice.
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Title: Powerful inhibitory action of mu opioid receptors (MOR) on cholinergic interneuron excitability in the dorsal striatum.
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Title: Accumbal core: essential link in feed-forward spiraling striato-nigro-striatal in series connected loop.
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Title: Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
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Title: A G protein-biased ligand at the μ-opioid receptor is potently analgesic with reduced gastrointestinal and respiratory dysfunction compared with morphine.
Journal: The Journal of pharmacology and experimental therapeutics20130301
Title: Deciphering µ-opioid receptor phosphorylation and dephosphorylation in HEK293 cells.
Journal: British journal of pharmacology20121101
Title: Pontine μ-opioid receptors mediate bradypnea caused by intravenous remifentanil infusions at clinically relevant concentrations in dogs.
Journal: Journal of neurophysiology20121101
Title: Direct regulation of GnRH neuron excitability by arcuate nucleus POMC and NPY neuron neuropeptides in female mice.
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Title: Pain-facilitating medullary neurons contribute to opioid-induced respiratory depression.
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Title: Enkephalin surges in dorsal neostriatum as a signal to eat.
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Title: The effect of Pro(2) modifications on the structural and pharmacological properties of endomorphin-2.
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Title: The mu opioid receptor modulates neurotransmission in the rat spinal ventral horn.
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Title: Disturbances in behavior and cortical enkephalin gene expression during the anticipation of ethanol in rats characterized as high drinkers.
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Title: Effects of peripheral μ, δ, and Κ-opioid receptor agonists on the levels of anxiety and motor activity of rats.
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Title: A118G Mu Opioid Receptor polymorphism increases inhibitory effects on CaV2.2 channels.
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Title: Endomorphin-2: a biased agonist at the μ-opioid receptor.
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Title: Inhibition of forebrain μ-opioid receptor signaling by low concentrations of rimonabant does not require cannabinoid receptors and directly involves μ-opioid receptors.
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Title: Selective impairment of spinal mu-opioid receptor mechanism by plasticity of serotonergic facilitation mediated by 5-HT2A and 5-HT2B receptors.
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Title: Quantitative analysis of the opioid peptide DAMGO in rat plasma and microdialysis samples using liquid chromatography-tandem mass spectrometry.
Journal: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences20120701
Title: Differences in the characteristics of tolerance to μ-opioid receptor agonists in the colon from wild type and β-arrestin2 knockout mice.
Journal: European journal of pharmacology20120615
Title: What and when to 'want'? Amygdala-based focusing of incentive salience upon sugar and sex.
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Title: Modulation of tight junction proteins in the perineurium to facilitate peripheral opioid analgesia.
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Title: Genetic differences in response properties of rostral ventromedial medulla neurons to the μ-opioid receptor agonist DAMGO in mouse inbred strains.
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Title: Effects of muscimol, amphetamine, and DAMGO injected into the nucleus accumbens shell on food-reinforced lever pressing by undeprived rats.
Journal: Pharmacology, biochemistry, and behavior20120501
Title: An examination of the effects of subthalamic nucleus inhibition or μ-opioid receptor stimulation on food-directed motivation in the non-deprived rat.
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Title: Which cue to 'want'? Opioid stimulation of central amygdala makes goal-trackers show stronger goal-tracking, just as sign-trackers show stronger sign-tracking.
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Title: Fast modulation of μ-opioid receptor (MOR) recycling is mediated by receptor agonists.
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Title: Synthesis, binding affinity, and functional in vitro activity of 3-benzylaminomorphinan and 3-benzylaminomorphine ligands at opioid receptors.
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Title: GRK2 protein-mediated transphosphorylation contributes to loss of function of μ-opioid receptors induced by neuropeptide FF (NPFF2) receptors.
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Title: Regulatory mechanism of body temperature in the central nervous system during the maintenance phase of hibernation in Syrian hamsters: involvement of β-endorphin.
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Title: A critical period in the supraspinal control of pain: opioid-dependent changes in brainstem rostroventral medulla function in preadolescence.
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Title: Probes for narcotic receptor mediated phenomena. 44. Synthesis of an N-substituted 4-hydroxy-5-(3-hydroxyphenyl)morphan with high affinity and selective μ-antagonist activity.
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Title: Opioid-related (ORL1) receptors are enriched in a subpopulation of sensory neurons and prolonged activation produces no functional loss of surface N-type calcium channels.
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Title: Ethanol alters opioid regulation of Ca(2+) influx through L-type Ca(2+) channels in PC12 cells.
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Title: [(35)S]GTPγS binding and opioid tolerance and efficacy in mouse spinal cord.
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Title: Activation of mu opioid receptors in the striatum differentially augments methamphetamine-induced gene expression and enhances stereotypic behavior.
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Title: Protein kinase C activity alters the effect of μ-opioid receptors on inhibitory postsynaptic current in the striosomes.
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Title: The central versus peripheral antinociceptive effects of μ-opioid receptor agonists in the new model of rat visceral pain.
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Title: Opioidergic modulation of ethanol self-administration in the ventral pallidum.
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Title: Tonic GABAA receptor conductance in medial subnucleus of the tractus solitarius neurons is inhibited by activation of μ-opioid receptors.
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Title: Opiate agonist-induced re-distribution of Wntless, a mu-opioid receptor interacting protein, in rat striatal neurons.
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Title: Regional and cell-type-specific effects of DAMGO on striatal D1 and D2 dopamine receptor-expressing medium-sized spiny neurons.
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Title: Importance of GluA1 subunit-containing AMPA glutamate receptors for morphine state-dependency.
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Title: [Effect of opioid peptides on oxygen-dependent microbicidity of peripheral blood neutrophils].
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Title: A novel µ-opioid receptor ligand with high in vitro and in vivo agonist efficacy.
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Title: Discovery of aminobenzyloxyarylamides as κ opioid receptor selective antagonists: application to preclinical development of a κ opioid receptor antagonist receptor occupancy tracer.
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Title: Involvement of NOX1/NADPH oxidase in morphine-induced analgesia and tolerance.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20111207
Title: Role of gonadal hormones on mu-opioid-stimulated [³⁵S]GTPγS binding and morphine-mediated antinociception in male and female Sprague-Dawley rats.
Journal: Psychopharmacology20111201
Title: Effect of ΔFosB overexpression on opioid and cannabinoid receptor-mediated signaling in the nucleus accumbens.
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Title: Opioid-sensitive GABA inputs from rostromedial tegmental nucleus synapse onto midbrain dopamine neurons.
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Title: Superpotent [Dmt¹] dermorphin tetrapeptides containing the 4-aminotetrahydro-2-benzazepin-3-one scaffold with mixed μ/δ opioid receptor agonistic properties.
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Title: Ivy and neurogliaform interneurons are a major target of μ-opioid receptor modulation.
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Title: Structural determinants of opioid and NOP receptor activity in derivatives of buprenorphine.
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Title: Neuroadaptation of GABAergic transmission in the central amygdala during chronic morphine treatment.
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Title: Activation of spinal mu- and delta-opioid receptors potently inhibits substance P release induced by peripheral noxious stimuli.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20110914
Title: Agonist-directed interactions with specific beta-arrestins determine mu-opioid receptor trafficking, ubiquitination, and dephosphorylation.
Journal: The Journal of biological chemistry20110909
Title: Agonist-selective patterns of µ-opioid receptor phosphorylation revealed by phosphosite-specific antibodies.
Journal: British journal of pharmacology20110901
Title: μ-Opioid modulation in the rostral solitary nucleus and reticular formation alters taste reactivity: evidence for a suppressive effect on consummatory behavior.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20110901
Title: RGS9-2 modulates nociceptive behaviour and opioid-mediated synaptic transmission in the spinal dorsal horn.
Journal: Neuroscience letters20110821
Title: Chronic neuropathic pain in mice reduces μ-opioid receptor-mediated G-protein activity in the thalamus.
Journal: Brain research20110811
Title: Dynamic mass redistribution as a means to measure and differentiate signaling via opioid and cannabinoid receptors.
Journal: Assay and drug development technologies20110801
Title: Opioid receptor modulation of GABAergic and serotonergic spinally projecting neurons of the rostral ventromedial medulla in mice.
Journal: Journal of neurophysiology20110801
Title: Distinct cellular properties of identified dopaminergic and GABAergic neurons in the mouse ventral tegmental area.
Journal: The Journal of physiology20110801
Title: Activation of opioid μ-receptors in the commissural subdivision of the nucleus tractus solitarius abolishes the ventilatory response to hypoxia in anesthetized rats.
Journal: Anesthesiology20110801
Title: A μ-opioid receptor agonist DAMGO induces rapid breathing in the arterially perfused in situ preparation of rat.
Journal: Respiratory physiology & neurobiology20110731
Title: mu-Opioid receptor stimulation in the nucleus accumbens elevates fatty tastant intake by increasing palatability and suppressing satiety signals.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20110701
Title: Generation of novel radiolabeled opiates through site-selective iodination.
Journal: Bioorganic & medicinal chemistry letters20110701
Title: Protein kinase Czeta mediates micro-opioid receptor-induced cross-desensitization of chemokine receptor CCR5.
Journal: The Journal of biological chemistry20110610
Title: Nucleus accumbens dopamine and mu-opioid receptors modulate the reinstatement of food-seeking behavior by food-associated cues.
Journal: Behavioural brain research20110601
Title: Nucleus accumbens facilitates nociception.
Journal: Experimental neurology20110601
Title: Spinal motor actions of the μ-opioid receptor agonist DAMGO in the cat.
Journal: Neuroscience research20110501
Title: Discovery of a potent and efficacious peptide derivative for δ/μ opioid agonist/neurokinin 1 antagonist activity with a 2',6'-dimethyl-L-tyrosine: in vitro, in vivo, and NMR-based structural studies.
Journal: Journal of medicinal chemistry20110414
Title: Modulating micro-opioid receptor phosphorylation switches agonist-dependent signaling as reflected in PKCepsilon activation and dendritic spine stability.
Journal: The Journal of biological chemistry20110408
Title: Aminothiazolomorphinans with mixed κ and μ opioid activity.
Journal: Journal of medicinal chemistry20110324
Title: Opioid-induced down-regulation of RGS4: role of ubiquitination and implications for receptor cross-talk.
Journal: The Journal of biological chemistry20110311
Title: Design, synthesis, pharmacological evaluation, and structure-activity study of novel endomorphin analogues with multiple structural modifications.
Journal: Journal of medicinal chemistry20110310
Title: Induction of hyperphagia and carbohydrate intake by μ-opioid receptor stimulation in circumscribed regions of frontal cortex.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20110302
Title: Gi/o-coupled receptors compete for signaling to adenylyl cyclase in SH-SY5Y cells and reduce opioid-mediated cAMP overshoot.
Journal: Molecular pharmacology20110301
Title: Differentiation between Aδ and C fibre evoked nociceptive reflexes by TTX resistance and opioid sensitivity in the cat.
Journal: Neuroscience research20110301
Title: Involvement of the lateral amygdala in the antiallodynic and reinforcing effects of heroin in rats after peripheral nerve injury.
Journal: Anesthesiology20110301
Title: Micro-opioid receptor activation in the basolateral amygdala mediates the learning of increases but not decreases in the incentive value of a food reward.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20110202
Title: Opioid-induced chemokine expression requires NF-κB activity: the role of PKCζ.
Journal: Journal of leukocyte biology20110201
Title: Morphine induces μ opioid receptor endocytosis in guinea pig enteric neurons following prolonged receptor activation.
Journal: Gastroenterology20110201
Title: Multiple targets of μ-opioid receptor-mediated presynaptic inhibition at primary afferent Aδ- and C-fibers.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20110126
Title: Involvement of mouse μ-opioid receptor splice variants in the spinal antinociception induced by the dermorphin tetrapeptide analog amidino-TAPA.
Journal: European journal of pharmacology20110125
Title: Development of potent μ and δ opioid agonists with high lipophilicity.
Journal: Journal of medicinal chemistry20110113
Title: μ-Opioid receptors in the nucleus accumbens shell region mediate the effects of amphetamine on inhibitory control but not impulsive choice.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20110105
Title: Differential expression and sensitivity of presynaptic and postsynaptic opioid receptors regulating hypothalamic proopiomelanocortin neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20110105
Title: Identification and modulation of voltage-gated Ca2+ currents in zebrafish Rohon-Beard neurons.
Journal: Journal of neurophysiology20110101
Title: Sevoflurane inhibits the µ-opioid receptor function expressed in Xenopus oocytes.
Journal: Pharmacology20110101
Title: Involvement of peripheral mu opioid receptors in scratching behavior in mice.
Journal: European journal of pharmacology20101215
Title: Tolerance to the antinociceptive effect of morphine in the absence of short-term presynaptic desensitization in rat periaqueductal gray neurons.
Journal: The Journal of pharmacology and experimental therapeutics20101201
Title: Mu and delta opioid receptors on nociceptors attenuate mechanical hyperalgesia in rat.
Journal: Neuroscience20101124
Title: The effects of daikenchuto (DKT) on propulsive motility in the colon.
Journal: The Journal of surgical research20101101
Title: CB1 receptors modulate the intake of a sweetened-fat diet in response to μ-opioid receptor stimulation of the nucleus accumbens.
Journal: Pharmacology, biochemistry, and behavior20101101
Title: The μ-opioid receptor variant N190K is unresponsive to peptide agonists yet can be rescued by small-molecule drugs.
Journal: Molecular pharmacology20101101
Title: Opioid-Induced GABA potentiation after chronic morphine attenuates the rewarding effects of opioids in the ventral tegmental area.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20101020
Title: Voltage-dependent kappa-opioid modulation of action potential waveform-elicited calcium currents in neurohypophysial terminals.
Journal: Journal of cellular physiology20101001
Title: Differential modulation of N-type calcium channels by micro-opioid receptors in oxytocinergic versus vasopressinergic neurohypophysial terminals.
Journal: Journal of cellular physiology20101001
Title: Morphine induces the release of CCL5 from astrocytes: potential neuroprotective mechanism against the HIV protein gp120.
Journal: Glia20101001
Title: Depression of cough reflex by microinjections of antitussive agents into caudal ventral respiratory group of the rabbit.
Journal: Journal of applied physiology (Bethesda, Md. : 1985)20101001
Title: Implication of dopaminergic projection from the ventral tegmental area to the anterior cingulate cortex in μ-opioid-induced place preference.
Journal: Addiction biology20101001
Title: Opioid inhibition of N-type Ca2+ channels and spinal analgesia couple to alternative splicing.
Journal: Nature neuroscience20101001
Title: High-fat intake induced by mu-opioid activation of the nucleus accumbens is inhibited by Y1R-blockade and MC3/4R- stimulation.
Journal: Brain research20100902
Title: Src family kinases mediate the inhibition of substance P release in the rat spinal cord by μ-opioid receptors and GABA(B) receptors, but not α2 adrenergic receptors.
Journal: The European journal of neuroscience20100901
Title: beta-Arrestin 2-mediated heterologous desensitization of IGF-IR by prolonged exposure of SH-SY5Y neuroblastoma cells to a mu opioid agonist.
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Title: G-protein-independent modulation of P-type calcium channels by mu-opioids in Purkinje neurons of rat.
Journal: Neuroscience letters20100816
Title: Characteristics of tolerance in the guinea pig ileum produced by chronic in vivo exposure to opioid versus cannabinoid agonists.
Journal: Biochemical pharmacology20100815
Title: Biological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillamines.
Journal: Journal of medicinal chemistry20100812
Title: Ethanol blocks long-term potentiation of GABAergic synapses in the ventral tegmental area involving mu-opioid receptors.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20100801
Title: Ex vivo delta opioid receptor autoradiography: CNS receptor occupancy of two novel compounds over their antihyperalgesic dose range.
Journal: Pharmacology, biochemistry, and behavior20100801
Title: micro-Opioid receptor stimulation in the medial subnucleus of the tractus solitarius inhibits gastric tone and motility by reducing local GABA activity.
Journal: American journal of physiology. Gastrointestinal and liver physiology20100801
Title: Peripheral mu-opioid receptors attenuate the augmented exercise pressor reflex in rats with chronic femoral artery occlusion.
Journal: American journal of physiology. Heart and circulatory physiology20100801
Title: Involvement of kappa opioid receptors in the formalin-induced inhibition of analgesic tolerance to morphine via suppression of conventional protein kinase C activation.
Journal: The Journal of pharmacy and pharmacology20100801
Title: Long-term adaptation to high doses of morphine causes desensitization of mu-OR- and delta-OR-stimulated G-protein response in forebrain cortex but does not decrease the amount of G-protein alpha subunits.
Journal: Medical science monitor : international medical journal of experimental and clinical research20100801
Title: Methylxanthine reversal of opioid-evoked inspiratory depression via phosphodiesterase-4 blockade.
Journal: Respiratory physiology & neurobiology20100731
Title: Evaluation of N-substitution in 6,7-benzomorphan compounds.
Journal: Bioorganic & medicinal chemistry20100715
Title: Modulation of feeding and locomotion through mu and delta opioid receptor signaling in the nucleus accumbens.
Journal: Neuropeptides20100601
Title: Hasubanan alkaloids with delta-opioid binding affinity from the aerial parts of Stephania japonica.
Journal: Journal of natural products20100528
Title: Agonist-selective dynamic compartmentalization of human Mu opioid receptor as revealed by resolutive FRAP analysis.
Journal: The Journal of biological chemistry20100507
Title: Opioids affect focal contact-mediated cell-substrate adhesion.
Journal: European journal of cancer prevention : the official journal of the European Cancer Prevention Organisation (ECP)20100501
Title: Correlation of the time course of development and decay of tolerance to morphine with alterations in sodium pump protein isoform abundance.
Journal: Biochemical pharmacology20100401
Title: Agonist-dependent mu-opioid receptor signaling can lead to heterologous desensitization.
Journal: Cellular signalling20100401
Title: Sigma 1 receptor modulation of G-protein-coupled receptor signaling: potentiation of opioid transduction independent from receptor binding.
Journal: Molecular pharmacology20100401
Title: Shared mechanisms for opioid tolerance and a transition to chronic pain.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20100331
Title: Opioid-induced long-term potentiation in the spinal cord is a presynaptic event.
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Title: Preference for a high fat diet, but not hyperphagia following activation of mu opioid receptors is blocked in AgRP knockout mice.
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Title: Phosphorylation of the mu-opioid receptor at tyrosine 166 (Tyr3.51) in the DRY motif reduces agonist efficacy.
Journal: Molecular pharmacology20100301
Title: The effect of protein kinase C and G protein-coupled receptor kinase inhibition on tolerance induced by mu-opioid agonists of different efficacy.
Journal: The Journal of pharmacology and experimental therapeutics20100301
Title: Nociceptive behaviour upon modulation of mu-opioid receptors in the ventrobasal complex of the thalamus of rats.
Journal: Pain20100301
Title: Standard opioid agonists activate heteromeric opioid receptors: evidence for morphine and [d-Ala(2)-MePhe(4)-Glyol(5)]enkephalin as selective μ-δ agonists.
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Title: Synthesis and opioid activity of enantiomeric N-substituted 2,3,4,4a,5,6,7,7a-octahydro-1H-benzofuro[3,2-e]isoquinolines.
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Title: Opioids in the hypothalamus control dopamine and acetylcholine levels in the nucleus accumbens.
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Title: Opioids in the hypothalamic paraventricular nucleus stimulate ethanol intake.
Journal: Alcoholism, clinical and experimental research20100201
Title: Differential modulation of mu-opioid receptor signaling to adenylyl cyclase by regulators of G protein signaling proteins 4 or 8 and 7 in permeabilised C6 cells is Galpha subtype dependent.
Journal: Journal of neurochemistry20100201
Title: Activation of spinal alpha-2 adrenoceptors, but not mu-opioid receptors, reduces the intrathecal N-methyl-D-aspartate-induced increase in spinal NR1 subunit phosphorylation and nociceptive behaviors in the rat.
Journal: Anesthesia and analgesia20100201
Title: Ethanol exposure selectively alters beta-endorphin content but not [3H]-DAMGO binding in discrete regions of the rat brain.
Journal: Neuropeptides20100201
Title: Novel approach to demonstrate high efficacy of mu opioids in the rat vas deferens: a simple model of predictive value.
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Title: The role of nucleus accumbens adenosine-opioid interaction in mediating palatable food intake.
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Title: CB1 receptor blockade decreases ethanol intake and associated neurochemical changes in fawn-hooded rats.
Journal: Alcoholism, clinical and experimental research20100101
Title: Muscarinic acetylcholine receptor modulation of mu (mu) opioid receptors in adult rat sphenopalatine ganglion neurons.
Journal: Journal of neurophysiology20100101
Title: Clinically relevant infusion rates of mu-opioid agonist remifentanil cause bradypnea in decerebrate dogs but not via direct effects in the pre-Bötzinger complex region.
Journal: Journal of neurophysiology20100101
Title: Cholecystokinin receptors mediate tolerance to the analgesic effect of TENS in arthritic rats.
Journal: Pain20100101
Title: Opiate-induced suppression of rat hypoglossal motoneuron activity and its reversal by ampakine therapy.
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Title: Modulation by neuropeptide FF of the interaction of mu-opioid (MOP) receptor with G-proteins.
Journal: Neurochemistry international20100101
Title: Analysis of the effects of anesthetics and ethanol on mu-opioid receptor.
Journal: Journal of pharmacological sciences20100101
Title: The functional antiopioid action of the ventrolateral periaqueductal gray nociceptin/orphanin FQ and nociceptin receptor system underlies DAMGO analgesic tolerance.
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Title: Regulation of mu opioid receptor internalization by the scaffold protein RanBPM.
Journal: Neuroscience letters20091211
Title: Probes for narcotic receptor mediated phenomena. 39. Enantiomeric N-substituted benzofuro[2,3-c]pyridin-6-ols: synthesis and topological relationship to oxide-bridged phenylmorphans.
Journal: Journal of medicinal chemistry20091210
Title: The unconditioned fear produced by morphine withdrawal is regulated by mu- and kappa-opioid receptors in the midbrain tectum.
Journal: Behavioural brain research20091201
Title: Electroacupuncture attenuates visceral hyperalgesia and inhibits the enhanced excitability of colon specific sensory neurons in a rat model of irritable bowel syndrome.
Journal: Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society20091201
Title: Feeding association between the nucleus of the solitary tract and the ventral tegmental area.
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Title: Design, synthesis and biological evaluation of a bivalent micro opiate and adenosine A1 receptor antagonist.
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Title: Cocaine-induced mu opioid receptor occupancy within the striatum is mediated by dopamine D2 receptors.
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Title: Involvement of Ca2+-dependent PKCs in the adaptive changes of mu-opioid pathways to sympathetic denervation in the guinea pig colon.
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Title: Immunoneutralization of agmatine sensitizes mice to micro-opioid receptor tolerance.
Journal: The Journal of pharmacology and experimental therapeutics20091101
Title: Opioid microinjection into raphe magnus modulates cardiorespiratory function in mice and rats.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20091101
Title: Micro-opioid receptor agonist injections into the presumed pre-Botzinger complex and the surrounding region of awake goats do not alter eupneic breathing.
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Title: Opioids in the nucleus accumbens stimulate ethanol intake.
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Title: The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety.
Journal: Bioorganic & medicinal chemistry20091015
Title: Opioid mu-receptors in medullary raphe region affect the hypoxic ventilation in anesthetized rats.
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Title: Purification and functional reconstitution of monomeric mu-opioid receptors: allosteric modulation of agonist binding by Gi2.
Journal: The Journal of biological chemistry20090925
Title: Synthesis and pharmacological evaluation of 6-naltrexamine analogs for alcohol cessation.
Journal: Bioorganic & medicinal chemistry20090915
Title: Cell aggregation on agar as an indicator for cell-matrix adhesion: effects of opioids.
Journal: In vitro cellular & developmental biology. Animal20090901
Title: Involvement of PKC alpha and G-protein-coupled receptor kinase 2 in agonist-selective desensitization of mu-opioid receptors in mature brain neurons.
Journal: British journal of pharmacology20090901
Title: Temporal lobe epilepsy causes selective changes in mu opioid and nociceptin receptor binding and functional coupling to G-proteins in human temporal neocortex.
Journal: Neurobiology of disease20090901
Title: Effects of opioid receptor activation on thermal antinociception in red-eared slider turtles (Trachemys scripta).
Journal: American journal of veterinary research20090901
Title: Activating mu-opioid receptors in the lateral parabrachial nucleus increases c-Fos expression in forebrain areas associated with caloric regulation, reward and cognition.
Journal: Neuroscience20090818
Title: Synthesis and characterizations of novel quinoline derivatives having mixed ligand activities at the kappa and mu receptors: Potential therapeutic efficacy against morphine dependence.
Journal: Bioorganic & medicinal chemistry20090815
Title: Capsaicin-evoked iCGRP release from human dental pulp: a model system for the study of peripheral neuropeptide secretion in normal healthy tissue.
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Title: CB1 receptor-independent actions of SR141716 on G-protein signaling: coapplication with the mu-opioid agonist Tyr-D-Ala-Gly-(NMe)Phe-Gly-ol unmasks novel, pertussis toxin-insensitive opioid signaling in mu-opioid receptor-Chinese hamster ovary cells.
Journal: The Journal of pharmacology and experimental therapeutics20090801
Title: Behavioral characterization of amygdala involvement in mediating intra-accumbens opioid-driven feeding behavior.
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Title: Induction of synaptic long-term potentiation after opioid withdrawal.
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Title: Convergent, not serial, striatal and pallidal circuits regulate opioid-induced food intake.
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Title: Differential modulation of mu- and delta-opioid receptor agonists by endogenous RGS4 protein in SH-SY5Y cells.
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Title: Lung respiratory rhythm and pattern generation in the bullfrog: role of neurokinin-1 and mu-opioid receptors.
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Title: Role of mu- and delta-opioid receptors in the nucleus accumbens in cocaine-seeking behavior.
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Title: Delta receptors are required for full inhibitory coupling of mu-receptors to voltage-dependent Ca(2+) channels in dorsal root ganglion neurons.
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Title: Inhibition of EGF-induced ERK/MAP kinase-mediated astrocyte proliferation by mu opioids: integration of G protein and beta-arrestin 2-dependent pathways.
Journal: Journal of neurochemistry20090701
Title: Regulation of interleukin-1beta and interleukin-8 production by agonists of mu and delta opiate receptors in vitro.
Journal: Neuroscience and behavioral physiology20090701
Title: Mu opioid receptor modulation of somatodendritic dopamine overflow: GABAergic and glutamatergic mechanisms.
Journal: The European journal of neuroscience20090701
Title: Activation of mu-opioid receptors in thalamic nucleus submedius depresses bee venom-evoked spinal c-Fos expression and flinching behavior.
Journal: Neuroscience20090630
Title: Mouse model of OPRM1 (A118G) polymorphism has sex-specific effects on drug-mediated behavior.
Journal: Proceedings of the National Academy of Sciences of the United States of America20090630
Title: Seizure activity involved in the up-regulation of BDNF mRNA expression by activation of central mu opioid receptors.
Journal: Neuroscience20090616
Title: Sex differences in the activation of the spinoparabrachial circuit by visceral pain.
Journal: Physiology & behavior20090525
Title: Which cue to 'want?' Central amygdala opioid activation enhances and focuses incentive salience on a prepotent reward cue.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20090520
Title: Antinociceptive effects of nociceptin/orphanin FQ administered intrathecally in monkeys.
Journal: The journal of pain : official journal of the American Pain Society20090501
Title: Activation of opioid micro-receptors in medullary raphe depresses sighs.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20090501
Title: A functional link between T-type calcium channels and mu-opioid receptor expression in adult primary sensory neurons.
Journal: Journal of neurochemistry20090501
Title: Functional interaction between TRPV1 and mu-opioid receptors in the descending antinociceptive pathway activates glutamate transmission and induces analgesia.
Journal: Journal of neurophysiology20090501
Title: Comparison of five benzodiazepine-receptor agonists on buprenorphine-induced mu-opioid receptor regulation.
Journal: Journal of pharmacological sciences20090501
Title: Syntheses of novel high affinity ligands for opioid receptors.
Journal: Bioorganic & medicinal chemistry letters20090415
Title: Neuropeptide modulation of a lumbar spinal reflex: potential implications for female sexual function.
Journal: The journal of sexual medicine20090401
Title: Neutral antagonist activity of naltrexone and 6beta-naltrexol in naïve and opioid-dependent C6 cells expressing a mu-opioid receptor.
Journal: British journal of pharmacology20090401
Title: Shadows across mu-Star? Constitutively active mu-opioid receptors revisited.
Journal: British journal of pharmacology20090401
Title: GABA and opioid mechanisms of the central amygdala underlie the withdrawal-potentiated startle from acute morphine.
Journal: Progress in neuro-psychopharmacology & biological psychiatry20090317
Title: Design, synthesis, and biological evaluation of 6alpha- and 6beta-N-heterocyclic substituted naltrexamine derivatives as mu opioid receptor selective antagonists.
Journal: Journal of medicinal chemistry20090312
Title: A common human micro-opioid receptor genetic variant diminishes the receptor signaling efficacy in brain regions processing the sensory information of pain.
Journal: The Journal of biological chemistry20090306
Title: p38 MAPK and beta-arrestin 2 mediate functional interactions between endogenous micro-opioid and alpha2A-adrenergic receptors in neurons.
Journal: The Journal of biological chemistry20090306
Title: G proteins in rat prefrontal cortex (PFC) are differentially activated as a function of oxygen status and PFC region.
Journal: Journal of chemical neuroanatomy20090301
Title: Allosteric modulation of metabotropic glutamate receptor 5 affects phosphorylation, internalization, and desensitization of the micro-opioid receptor.
Journal: Neuropharmacology20090301
Title: Epileptiform synchronization in the cingulate cortex.
Journal: Epilepsia20090301
Title: Beta-endorphin fragments DTgammaE and DEgammaE reduced morphine inhibition of electrically-induced contractions and opiate withdrawal.
Journal: Medicinal chemistry (Shariqah (United Arab Emirates))20090301
Title: Morphine increases brain levels of ferritin heavy chain leading to inhibition of CXCR4-mediated survival signaling in neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20090225
Title: Activation of micro, delta or kappa opioid receptors by DAMGO, DPDPE, U-50488 or U-69593 respectively causes antinociception in the formalin test in the naked mole-rat (Heterocephalus glaber).
Journal: Pharmacology, biochemistry, and behavior20090201
Title: Muscarinic receptor antagonism causes a functional alteration in nucleus accumbens mu-opiate-mediated feeding behavior.
Journal: Behavioural brain research20090130
Title: Morphine enhances microglial migration through modulation of P2X4 receptor signaling.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20090128
Title: Binding studies of novel, non-mammalian enkephalins, structures predicted from frog and lungfish brain cDNA sequences.
Journal: Neuroscience20090123
Title: Induced association of mu opioid (MOP) and type 2 cholecystokinin (CCK2) receptors by novel bivalent ligands.
Journal: Journal of medicinal chemistry20090122
Title: Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 7: syntheses and opioid receptor properties of cyclic variants of cyclazocine.
Journal: Bioorganic & medicinal chemistry letters20090115
Title: Neurokinin 1 receptors regulate morphine-induced endocytosis and desensitization of mu-opioid receptors in CNS neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20090107
Title: Syntheses and opioid receptor binding properties of carboxamido-substituted opioids.
Journal: Bioorganic & medicinal chemistry letters20090101
Title: Persistent inflammatory pain decreases the antinociceptive effects of the mu opioid receptor agonist DAMGO in the locus coeruleus of male rats.
Journal: Neuropharmacology20090101
Title: [Mu-opioidergic immunomodulation: the neurochemical basis].
Journal: Uspekhi fiziologicheskikh nauk20090101
Title: Respiratory pattern in midline-lesioned brainstems and hemibrainstems from adult turtles.
Journal: Respiratory physiology & neurobiology20081231
Title: Effect of agmatine on DAMGO-induced mu-opioid receptor down-regulation and internalization via activation of IRAS, a candidate for imidazoline I(1) receptor.
Journal: European journal of pharmacology20081203
Title: A pharmacological comparison of the cloned frog and human mu opioid receptors reveals differences in opioid affinity and function.
Journal: European journal of pharmacology20081203
Title: Depression of C fibre-evoked spinal field potentials by the spinal delta opioid receptor is enhanced in the spinal nerve ligation model of neuropathic pain: involvement of the mu-subtype.
Journal: Neuropharmacology20081201
Title: CB(2) cannabinoid receptor antagonist SR144528 decreases mu-opioid receptor expression and activation in mouse brainstem: role of CB(2) receptor in pain.
Journal: Neurochemistry international20081201
Title: cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Journal: Journal of medicinal chemistry20081127
Title: A naloxonazine sensitive (mu1 receptor) mechanism in the parabrachial nucleus modulates eating.
Journal: Brain research20081113
Title: The role of amygdalar mu-opioid receptors in anxiety-related responses in two rat models.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20081101
Title: The S218L familial hemiplegic migraine mutation promotes deinhibition of Ca(v)2.1 calcium channels during direct G-protein regulation.
Journal: Pflugers Archiv : European journal of physiology20081101
Title: Sustained inhibition of neurotransmitter release from nontransient receptor potential vanilloid type 1-expressing primary afferents by mu-opioid receptor activation-enkephalin in the spinal cord.
Journal: The Journal of pharmacology and experimental therapeutics20081101
Title: Inhibitory and excitatory effects of micro-, delta-, and kappa-opioid receptor activation on breathing in awake turtles, Trachemys scripta.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20081101
Title: G protein betagamma subunits modulate the number and nature of exocytotic fusion events in adrenal chromaffin cells independent of calcium entry.
Journal: Journal of neurophysiology20081101
Title: mu-Opioid receptor forms a functional heterodimer with cannabinoid CB1 receptor: electrophysiological and FRET assay analysis.
Journal: Journal of pharmacological sciences20081101
Title: Morphine attenuates the expression of sensitization to ethanol, but opioid antagonists do not.
Journal: Neuroscience20081028
Title: The importance of micelle-bound states for the bioactivities of bifunctional peptide derivatives for delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists.
Journal: Journal of medicinal chemistry20081023
Title: Activation of the mu opioid receptor involves conformational rearrangements of multiple transmembrane domains.
Journal: Biochemistry20081007
Title: Filamin A mutant lacking actin-binding domain restores mu opioid receptor regulation in melanoma cells.
Journal: Neurochemical research20081001
Title: Mu-opioid receptor activation in live cells.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology20081001
Title: Differential activation and trafficking of micro-opioid receptors in brain slices.
Journal: Molecular pharmacology20081001
Title: Capsaicin inhibits the in vitro binding of peptides selective for mu- and kappa-opioid, and nociceptin-receptors.
Journal: Brain research bulletin20080930
Title: Activating parabrachial cannabinoid CB1 receptors selectively stimulates feeding of palatable foods in rats.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20080924
Title: Differential effects of opioid agonists on G protein expression in CHO cells expressing cloned human opioid receptors.
Journal: Brain research bulletin20080905
Title: Morphine-induced mu-opioid receptor rapid desensitization is independent of receptor phosphorylation and beta-arrestins.
Journal: Cellular signalling20080901
Title: Possible involvement of dynorphin A release via mu1-opioid receptor on supraspinal antinociception of endomorphin-2.
Journal: Peptides20080901
Title: Spatial information processing consequences of DAMGO injections into the dorsal striatum.
Journal: Neurobiology of learning and memory20080901
Title: Involvement of kappa opioid receptors in the inhibition of receptor desensitization and PKC activation induced by repeated morphine treatment.
Journal: The Journal of pharmacy and pharmacology20080901
Title: Acute delta- and kappa-opioid agonist pretreatment potentiates opioid antagonist-induced suppression of water consumption.
Journal: Brain research bulletin20080815
Title: Structure-antitussive activity relationships of naltrindole derivatives. Identification of novel and potent antitussive agents.
Journal: Journal of medicinal chemistry20080814
Title: Opioid activation in the lateral parabrachial nucleus induces hypertonic sodium intake.
Journal: Neuroscience20080813
Title: Insulin acts at different CNS sites to decrease acute sucrose intake and sucrose self-administration in rats.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20080801
Title: Shell/core differences in mu- and delta-opioid receptor modulation of dopamine efflux in nucleus accumbens.
Journal: Neuropharmacology20080801
Title: Intrathecal clonidine suppresses phosphorylation of the N-methyl-D-aspartate receptor NR1 subunit in spinal dorsal horn neurons of rats with neuropathic pain.
Journal: Anesthesia and analgesia20080801
Title: Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
Journal: Journal of medicinal chemistry20080724
Title: Micro-opioid receptor agonist diminishes POMC gene expression and anorexia by central insulin in neonatal chicks.
Journal: Neuroscience letters20080718
Title: Modulation of the cough reflex by antitussive agents within the caudal aspect of the nucleus tractus solitarii in the rabbit.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20080701
Title: [Regulation of IL-1beta and IL-8 production by mu-, delta-opiate receptors agonists in vitro].
Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova20080701
Title: Morphine-nicotine interaction in conditioned place preference in mice after chronic nicotine exposure.
Journal: European journal of pharmacology20080610
Title: Distinct roles of adenylyl cyclases 1 and 8 in opiate dependence: behavioral, electrophysiological, and molecular studies.
Journal: Biological psychiatry20080601
Title: The spinal antinociceptive effects of endomorphins in rats: behavioral and G protein functional studies.
Journal: Anesthesia and analgesia20080601
Title: [Analysis of central mechanisms involved in gastric mucosal integrity].
Journal: Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology20080601
Title: Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 6: Opioid receptor binding properties of cyclic variants of 8-carboxamidocyclazocine.
Journal: Bioorganic & medicinal chemistry20080515
Title: Effects of chronic treatment with citalopram on cannabinoid and opioid receptor-mediated G-protein coupling in discrete rat brain regions.
Journal: Psychopharmacology20080501
Title: Endogenous regulators of G protein signaling differentially modulate full and partial mu-opioid agonists at adenylyl cyclase as predicted by a collision coupling model.
Journal: Molecular pharmacology20080501
Title: Constitutive activity of the cannabinoid CB1 receptor regulates the function of co-expressed Mu opioid receptors.
Journal: The Journal of biological chemistry20080425
Title: Direct evidence for the involvement of endogenous beta-endorphin in the suppression of the morphine-induced rewarding effect under a neuropathic pain-like state.
Journal: Neuroscience letters20080425
Title: Herkinorin analogues with differential beta-arrestin-2 interactions.
Journal: Journal of medicinal chemistry20080424
Title: Multiple actions of spinophilin regulate mu opioid receptor function.
Journal: Neuron20080424
Title: Ethanol dually modulates GABAergic synaptic transmission onto dopaminergic neurons in ventral tegmental area: role of mu-opioid receptors.
Journal: Neuroscience20080422
Title: Presynaptic actions of opioid receptor agonists in ventromedial hypothalamic neurons in estrogen- and oil-treated female mice.
Journal: Neuroscience20080409
Title: Agonist-specific down regulation of mu-opioid receptors: Different cellular pathways are activated by different opioid agonists.
Journal: Life sciences20080409
Title: DAMGO-induced expression of chemokines and chemokine receptors: the role of TGF-beta1.
Journal: Journal of leukocyte biology20080401
Title: Opioid modulation of ferret vagal afferent mechanosensitivity.
Journal: American journal of physiology. Gastrointestinal and liver physiology20080401
Title: Sex-dependent effects of periadolescent exposure to the cannabinoid agonist CP-55,940 on morphine self-administration behaviour and the endogenous opioid system.
Journal: Neuropharmacology20080401
Title: A structure-activity relationship study and combinatorial synthetic approach of C-terminal modified bifunctional peptides that are delta/mu opioid receptor agonists and neurokinin 1 receptor antagonists.
Journal: Journal of medicinal chemistry20080313
Title: Acute amphetamine exposure selectively desensitizes kappa-opioid receptors in the nucleus accumbens.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20080301
Title: ATP sensitivity of preBötzinger complex neurones in neonatal rat in vitro: mechanism underlying a P2 receptor-mediated increase in inspiratory frequency.
Journal: The Journal of physiology20080301
Title: GTPgammaS incorporation in the rat brain: a study on mu-opioid receptors and CXCR4.
Journal: Journal of neuroimmune pharmacology : the official journal of the Society on NeuroImmune Pharmacology20080301
Title: Peripherally-acting opioids.
Journal: Pain physician20080301
Title: The effects of local perfusion of DAMGO on extracellular GABA and glutamate concentrations in the rostral ventromedial medulla.
Journal: Journal of neurochemistry20080201
Title: Modulation of extracellular signal-regulated kinase (ERK) by opioid and cannabinoid receptors that are expressed in the same cell.
Journal: Brain research20080116
Title: Layer selective presynaptic modulation of excitatory inputs to hippocampal cornu Ammon 1 by mu-opioid receptor activation.
Journal: Neuroscience20080102
Title: Noladin ether, a putative endocannabinoid, inhibits mu-opioid receptor activation via CB2 cannabinoid receptors.
Journal: Neurochemistry international20080101
Title: Manipulation of fatty acid amide hydrolase functional activity alters sensitivity and dependence to ethanol.
Journal: Journal of neurochemistry20080101
Title: Activation of mu-opioid receptor selectively potentiates NMDA-induced outward currents in rat locus coeruleus neurons.
Journal: Neuroscience research20080101
Title: Opioid regulation of spinal cord plasticity: evidence the kappa-2 opioid receptor agonist GR89696 inhibits learning within the rat spinal cord.
Journal: Neurobiology of learning and memory20080101
Title: Modulation of Ca2+ channel current by mu opioid receptors in prefrontal cortex pyramidal neurons in rats.
Journal: Acta neurobiologiae experimentalis20080101
Title: Comparison of liquid chromatography-mass spectrometry and radioimmunoassay for measurement of fentanyl and determination of pharmacokinetics in equine plasma.
Journal: Journal of analytical toxicology20080101
Title: Opioid-induced depression in the lamprey respiratory network.
Journal: Neuroscience20071212
Title: Differential effects of mu-opioid receptor agonists in a hippocampal hypoxia/hypoglycemia model.
Journal: Brain research20071205
Title: Mu opioid receptor mutant, T394A, abolishes opioid-mediated adenylyl cyclase superactivation.
Journal: Neuroreport20071203
Title: Maternal separation leads to persistent reductions in pain sensitivity in female rats.
Journal: The journal of pain : official journal of the American Pain Society20071201
Title: RGS14 prevents morphine from internalizing Mu-opioid receptors in periaqueductal gray neurons.
Journal: Cellular signalling20071201
Title: Activity of murine raphe magnus cells predicts tachypnea and on-going nociceptive responsiveness.
Journal: Journal of neurophysiology20071201
Title: Trafficking of preassembled opioid mu-delta heterooligomer-Gz signaling complexes to the plasma membrane: coregulation by agonists.
Journal: Biochemistry20071113
Title: [Opioids and spinal analgesia].
Journal: Masui. The Japanese journal of anesthesiology20071101
Title: Differential presynaptic effects of opioid agonists on Adelta- and C-afferent glutamatergic transmission to the spinal dorsal horn.
Journal: Anesthesiology20071101
Title: Chronic morphine treatment up-regulates mu opioid receptor binding in cells lacking filamin A.
Journal: Brain research20071026
Title: DAMGO and 6beta-glycine substituted 14-O-methyloxymorphone but not morphine show peripheral, preemptive antinociception after systemic administration in a mouse visceral pain model and high intrinsic efficacy in the isolated rat vas deferens.
Journal: Brain research bulletin20071019
Title: Low dose combination of morphine and delta9-tetrahydrocannabinol circumvents antinociceptive tolerance and apparent desensitization of receptors.
Journal: European journal of pharmacology20071001
Title: The single nucleotide polymorphism A118G alters functional properties of the human mu opioid receptor.
Journal: Journal of neurochemistry20071001
Title: Live cell monitoring of mu-opioid receptor-mediated G-protein activation reveals strong biological activity of close morphine biosynthetic precursors.
Journal: The Journal of biological chemistry20070914
Title: Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles.
Journal: Brain research bulletin20070914
Title: Neurobiology of 50-kHz ultrasonic vocalizations in rats: electrode mapping, lesion, and pharmacology studies.
Journal: Behavioural brain research20070904
Title: The differential contribution of dopamine D(1) and D (2) receptors to mu-opioidergic immunomodulation.
Journal: Neuroscience and behavioral physiology20070901
Title: Probes for narcotic receptor mediated phenomena. 34. Synthesis and structure-activity relationships of a potent mu-agonist delta-antagonist and an exceedingly potent antinociceptive in the enantiomeric C9-substituted 5-(3-hydroxyphenyl)-N-phenylethylmorphan series.
Journal: Journal of medicinal chemistry20070809
Title: Attenuation of vascular permeability by methylnaltrexone: role of mOP-R and S1P3 transactivation.
Journal: American journal of respiratory cell and molecular biology20070801
Title: Mechanisms responsible for the enhanced antinociceptive effects of micro-opioid receptor agonists in the rostral ventromedial medulla of male rats with persistent inflammatory pain.
Journal: The Journal of pharmacology and experimental therapeutics20070801
Title: Glucocorticoids plus opioids up-regulate genes that influence neuronal function.
Journal: Cellular and molecular neurobiology20070801
Title: Activation of opioid mu receptors in caudal medullary raphe region inhibits the ventilatory response to hypercapnia in anesthetized rats.
Journal: Anesthesiology20070801
Title: Lobeline, a potential pharmacotherapy for drug addiction, binds to mu opioid receptors and diminishes the effects of opioid receptor agonists.
Journal: Drug and alcohol dependence20070710
Title: micro-Opioid receptor activation prevents acute hepatic inflammation and cell death.
Journal: Gut20070701
Title: Paraventricular opioids alter intake of high-fat but not high-sucrose diet depending on diet preference in a binge model of feeding.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20070701
Title: Synthesis and biological activity of nociceptin/orphanin FQ analogues substituted in position 7 or 11 with Calpha,alpha-dialkylated amino acids.
Journal: Bioorganic & medicinal chemistry20070701
Title: Effects of ethanol on midbrain neurons: role of opioid receptors.
Journal: Alcoholism, clinical and experimental research20070701
Title: Blockade of the nociceptin/orphanin FQ/NOP receptor system in the rat ventrolateral periaqueductal gray potentiates DAMGO analgesia.
Journal: Peptides20070701
Title: In-vitro investigation of oxazol and urea analogues of morphinan at opioid receptors.
Journal: Bioorganic & medicinal chemistry20070615
Title: The chemokine CX3CL1/fractalkine interferes with the antinociceptive effect induced by opioid agonists in the periaqueductal grey of rats.
Journal: Brain research20070611
Title: The absence of endogenous beta-endorphin selectively blocks phosphorylation and desensitization of mu opioid receptors following partial sciatic nerve ligation.
Journal: Neuroscience20070608
Title: Gene transcription alterations associated with decrease of ethanol intake induced by naltrexone in the brain of Wistar rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20070601
Title: A Tyr-W-MIF-1 analog containing D-Pro2 discriminates among antinociception in mice mediated by different classes of mu-opioid receptors.
Journal: European journal of pharmacology20070601
Title: Rapid modulation of micro-opioid receptor signaling in primary sensory neurons.
Journal: The Journal of pharmacology and experimental therapeutics20070601
Title: Differential receptor binding characteristics of consecutive phenylalanines in micro-opioid specific peptide ligand endomorphin-2.
Journal: Bioorganic & medicinal chemistry20070601
Title: Analgesic tolerance to microinjection of the micro-opioid agonist DAMGO into the ventrolateral periaqueductal gray.
Journal: Neuropharmacology20070601
Title: Role of peripheral mu-opioid receptors in inflammatory orofacial muscle pain.
Journal: Neuroscience20070525
Title: Effects of local anesthetics on opioid inhibition of calcium current in rat dorsal root ganglion neurons.
Journal: Neuroscience letters20070518
Title: Conformational analysis of endomorphin-2 analogs with phenylalanine mimics by NMR and molecular modeling.
Journal: Bioorganic & medicinal chemistry20070515
Title: Presynaptic modulation of 5-HT release in the rat septal region.
Journal: Neuroscience20070511
Title: Pharmacological properties of bivalent ligands containing butorphan linked to nalbuphine, naltrexone, and naloxone at mu, delta, and kappa opioid receptors.
Journal: Journal of medicinal chemistry20070503
Title: Different effects of opioid antagonists on mu-, delta-, and kappa-opioid receptors with and without agonist pretreatment.
Journal: The Journal of pharmacology and experimental therapeutics20070501
Title: In vitro characterization of the effects of endomorphin 1 and 2, endogenous ligands for mu-opioid receptors, on mouse colonic motility.
Journal: Biochemical pharmacology20070501
Title: Biochemical anti-opioid action of NPFF2 receptors in rat spinal cord.
Journal: Neuroscience research20070501
Title: The in vitro pharmacology of the peripherally restricted opioid receptor antagonists, alvimopan, ADL 08-0011 and methylnaltrexone.
Journal: Naunyn-Schmiedeberg's archives of pharmacology20070501
Title: Staurosporine differentiation of NPFF2 receptor-transfected SH-SY5Y neuroblastoma cells induces selectivity of NPFF activity towards opioid receptors.
Journal: Peptides20070501
Title: Nucleus accumbens opioid signaling conditions short-term flavor preferences.
Journal: Neuroscience20070425
Title: Role of kappa and delta opioid receptors in mediating morphine-induced antinociception in morphine-tolerant infant rats.
Journal: Brain research20070420
Title: Involvement of endogenous opioid peptides in the antinociception induced by the novel dermorphin tetrapeptide analog amidino-TAPA.
Journal: European journal of pharmacology20070410
Title: Differential effects of opioids on sacrocaudal afferent pathways and central pattern generators in the neonatal rat spinal cord.
Journal: Journal of neurophysiology20070401
Title: CC12, a high-affinity ligand for [3H]cimetidine binding, is an improgan antagonist.
Journal: Neuropharmacology20070401
Title: Endogenous dynorphin in epileptogenesis and epilepsy: anticonvulsant net effect via kappa opioid receptors.
Journal: Brain : a journal of neurology20070401
Title: Bidirectional regulation of mu-opioid and CB1-cannabinoid receptor in rats self-administering heroin or WIN 55,212-2.
Journal: The European journal of neuroscience20070401
Title: Pain hypersensitivity induced by paradoxical sleep deprivation is not due to altered binding to brain mu-opioid receptors.
Journal: Behavioural brain research20070328
Title: Physical association between neuropeptide FF and micro-opioid receptors as a possible molecular basis for anti-opioid activity.
Journal: The Journal of biological chemistry20070316
Title: High-affinity carbamate analogues of morphinan at opioid receptors.
Journal: Bioorganic & medicinal chemistry letters20070315
Title: Adolescent cannabis exposure alters opiate intake and opioid limbic neuronal populations in adult rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20070301
Title: A comparison of noninternalizing (herkinorin) and internalizing (DAMGO) mu-opioid agonists on cellular markers related to opioid tolerance and dependence.
Journal: Synapse (New York, N.Y.)20070301
Title: Modulation of the endogenous opioid system after morphine self-administration and during its extinction: a study in Lewis and Fischer 344 rats.
Journal: Neuropharmacology20070301
Title: Effects of mu-opioid receptor modulation on GABAB receptor synaptic function in hippocampal CA1.
Journal: Journal of neurophysiology20070301
Title: Alternative splicing controls G protein-dependent inhibition of N-type calcium channels in nociceptors.
Journal: Nature neuroscience20070301
Title: Impact of 6-hydroxydopamine lesions and cocaine exposure on mu-opioid receptor expression and regulation of cholinergic transmission in the limbic-prefrontal territory of the rat dorsal striatum.
Journal: The European journal of neuroscience20070301
Title: Effects of opioid subtypes on detrusor overactivity in rats with cerebral infarction.
Journal: International journal of urology : official journal of the Japanese Urological Association20070301
Title: Suitability of the retrograde tracer Dil for electrophysiological studies of brainstem neurons: adverse ramifications for G-protein coupled receptor agonists.
Journal: Journal of neuroscience methods20070215
Title: Opioid limbic circuit for reward: interaction between hedonic hotspots of nucleus accumbens and ventral pallidum.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20070214
Title: Functional reduction in mu-opioidergic system in the spinal cord under a neuropathic pain-like state following chronic ethanol consumption in the rat.
Journal: Neuroscience20070209
Title: Integrins regulate opioid receptor signaling in trigeminal ganglion neurons.
Journal: Neuroscience20070209
Title: Salvinorin A: allosteric interactions at the mu-opioid receptor.
Journal: The Journal of pharmacology and experimental therapeutics20070201
Title: Agonist-dependent postsynaptic effects of opioids on miniature excitatory postsynaptic currents in cultured hippocampal neurons.
Journal: Journal of neurophysiology20070201
Title: Modulation of Ca2+ channels by heterologously expressed wild-type and mutant human micro-opioid receptors (hMORs) containing the A118G single-nucleotide polymorphism.
Journal: Journal of neurophysiology20070201
Title: The inhibitory effect of opioids on HepG2 cells is mediated via interaction with somatostatin receptors.
Journal: European journal of pharmacology20070119
Title: Glycosylation improves the central effects of DAMGO.
Journal: Chemical biology & drug design20070101
Title: The biochemical analysis of methadone modulation on morphine-induced tolerance and dependence in the rat brain.
Journal: Pharmacology20070101
Title: Hypoxia modulates cholinergic but not opioid activation of G proteins in rat hippocampus.
Journal: Hippocampus20070101
Title: Morphine induces endocytosis of neuronal mu-opioid receptors through the sustained transfer of Galpha subunits to RGSZ2 proteins.
Journal: Molecular pain20070101
Title: Altered gene expression and functional activity of opioid receptors in the cerebellum of CB1 cannabinoid receptor knockout mice after acute treatments with cannabinoids.
Journal: Acta biologica Hungarica20070101
Title: Functional interaction between alpha2-adrenoceptors, mu- and kappa-opioid receptors in the guinea pig myenteric plexus: effect of chronic desipramine treatment.
Journal: European journal of pharmacology20061228
Title: Black cohosh (Actaea racemosa, Cimicifuga racemosa) behaves as a mixed competitive ligand and partial agonist at the human mu opiate receptor.
Journal: Journal of agricultural and food chemistry20061227
Title: Role of CDK5 in neuroprotection from serum deprivation by mu-opioid receptor agonist.
Journal: Experimental neurology20061201
Title: Raphe magnus neurons help protect reactions to visceral pain from interruption by cutaneous pain.
Journal: Journal of neurophysiology20061201
Title: Pain sensitivity is altered in animals after subchronic ketamine treatment.
Journal: Psychopharmacology20061201
Title: The possible involvement of endogenous ligands for mu-, delta- and kappa-opioid receptors in modulating morphine-induced CPP expression in rats.
Journal: Peptides20061201
Title: Modulation of neuronal CXCR4 by the micro-opioid agonist DAMGO.
Journal: Journal of neurovirology20061201
Title: Mediation of adenylyl cyclase sensitization by PTX-insensitive GalphaoA, Galphai1, Galphai2 or Galphai3.
Journal: Journal of neurochemistry20061201
Title: Distinct populations of spinal cord lamina II interneurons expressing G-protein-gated potassium channels.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20061122
Title: Nucleus accumbens opioids regulate flavor-based preferences in food consumption.
Journal: Neuroscience20061117
Title: Mu- and kappa-opioids induce the differentiation of embryonic stem cells to neural progenitors.
Journal: The Journal of biological chemistry20061103
Title: Contingent and non-contingent effects of heroin on mu-opioid receptor-containing ventral tegmental area GABA neurons.
Journal: Experimental neurology20061101
Title: Methamphetamine-induced behavioral sensitization in mice: alterations in mu-opioid receptor.
Journal: Journal of biomedical science20061101
Title: Physiological properties of zebra finch ventral tegmental area and substantia nigra pars compacta neurons.
Journal: Journal of neurophysiology20061101
Title: Contribution of spinal mu(1)-opioid receptors and dynorphin B to the antinociception induced by Tyr-d-Arg-Phe-Sar.
Journal: Peptides20061101
Title: Role of hepatic opioid receptors in the regulation of bile excretion.
Journal: Bulletin of experimental biology and medicine20061101
Title: Mu opioid receptor-effector coupling and trafficking in dorsal root ganglia neurons.
Journal: Neuroscience20061013
Title: An antisense oligodeoxynucleotide to the mu opioid receptor attenuates cocaine-induced behavioral sensitization and reward in mice.
Journal: Neuroscience20061013
Title: Synthesis and pharmacological studies of new hybrid derivatives of fentanyl active at the mu-opioid receptor and I2-imidazoline binding sites.
Journal: Bioorganic & medicinal chemistry20061001
Title: Separation of binding affinity and intrinsic activity of the potent mu-opioid 14-methoxymetopon.
Journal: The Journal of pharmacology and experimental therapeutics20061001
Title: Alkylation of opioid receptors by 5'-naltrindole-isothiocyanate injected into the nucleus accumbens of rats: receptor selectivity and anatomical diffusion.
Journal: Synapse (New York, N.Y.)20061001
Title: Pharmacological characterization of high-fat feeding induced by opioid stimulation of the ventral striatum.
Journal: Physiology & behavior20060930
Title: The mu-opioid receptor subtype is required for the anorectic effect of an opioid receptor antagonist.
Journal: European journal of pharmacology20060918
Title: An N-methyl-D-aspartate receptor mediated large, low-frequency, spontaneous excitatory postsynaptic current in neonatal rat spinal dorsal horn neurons.
Journal: Neuroscience20060901
Title: 11 beta-hydroxysteroid dehydrogenase type 1 induction in the arcuate nucleus by high-fat feeding: A novel constraint to hyperphagia?
Journal: Endocrinology20060901
Title: Chronic prevention of mu-opioid receptor (MOR) G-protein coupling in the pontine parabrachial nucleus persistently decreases consumption of standard but not palatable food.
Journal: Psychopharmacology20060901
Title: Enhancement of morphine analgesic effect with induction of mu-opioid receptor endocytosis in rats.
Journal: Anesthesiology20060901
Title: Opiate pharmacology of intrathecal granulomas.
Journal: Anesthesiology20060901
Title: Characterization of neurons in the rat central nucleus of the amygdala: cellular physiology, morphology, and opioid sensitivity.
Journal: The Journal of comparative neurology20060820
Title: Opiate receptor binding properties of morphine-, dihydromorphine-, and codeine 6-O-sulfate ester congeners.
Journal: Bioorganic & medicinal chemistry letters20060815
Title: Differential effects of impaired mitochondrial energy production on the function of mu and delta opioid receptors in neuronal SK-N-SH cells.
Journal: Neuroscience letters20060814
Title: Agonist-selective mechanisms of mu-opioid receptor desensitization in human embryonic kidney 293 cells.
Journal: Molecular pharmacology20060801
Title: Mu-delta opioid receptor functional interaction: Insight using receptor-G protein fusions.
Journal: The Journal of pharmacology and experimental therapeutics20060801
Title: Morphine withdrawal syndrome and its prevention with baclofen: Autoradiographic study of mu-opioid receptors in prepubertal male and female mice.
Journal: Synapse (New York, N.Y.)20060801
Title: Respiration-related rhythmic activity in the rostral medulla of newborn rats.
Journal: Journal of neurophysiology20060701
Title: Involvement of spinal mu1-opioid receptors on the Tyr-d-Arg-Phe-sarcosine-induced antinociception.
Journal: European journal of pharmacology20060701
Title: Presynaptic opioid receptors on noradrenergic and serotonergic neurons in the human as compared to the rat neocortex.
Journal: British journal of pharmacology20060701
Title: Competitive displacement binding assay on rat brain sections and using a beta-imager: application to mu-opioid ligands.
Journal: Journal of neuroscience methods20060630
Title: Activation of the mu-opiate receptor by Vitex agnus-castus methanol extracts: implication for its use in PMS.
Journal: Journal of ethnopharmacology20060630
Title: Effect of opioid receptor ligands injected into the rostral lateral hypothalamus on c-fos and feeding behavior.
Journal: Brain research20060622
Title: Opioid mu receptor activation inhibits sodium currents in prefrontal cortical neurons via a protein kinase A- and C-dependent mechanism.
Journal: Brain research20060613
Title: The cardiovascular responses to mu opioid agonist and antagonist in conscious normal and obese rats.
Journal: Peptides20060601
Title: Partial and full agonism in endomorphin derivatives: comparison by null and operational model.
Journal: Peptides20060601
Title: Adenylyl cyclase type II activity is regulated by two different mechanisms: implications for acute and chronic opioid exposure.
Journal: Neuropharmacology20060601
Title: Endomorphin-2, an endogenous tetrapeptide, protects against Abeta1-42 in vitro and in vivo.
Journal: FASEB journal : official publication of the Federation of American Societies for Experimental Biology20060601
Title: Reduction of lipopolysaccharide-induced interleukin-6 production by the kappa opioid U50,488 in a mouse monocyte-like cell line.
Journal: International immunopharmacology20060601
Title: mu opioid and CB1 cannabinoid receptor interactions: reciprocal inhibition of receptor signaling and neuritogenesis.
Journal: British journal of pharmacology20060601
Title: Role of delta-opioid receptor function in neurogenesis and neuroprotection.
Journal: Journal of neurochemistry20060601
Title: Structure-activity relationships of bifunctional peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors.
Journal: Journal of medicinal chemistry20060518
Title: Delta and mu opioid receptors from the brain of a urodele amphibian, the rough-skinned newt Taricha granulosa: cloning, heterologous expression, and pharmacological characterization.
Journal: General and comparative endocrinology20060501
Title: In heterozygous GDNF knockout mice the response of striatal dopaminergic system to acute morphine is altered.
Journal: Synapse (New York, N.Y.)20060501
Title: Loss of TRPV1-expressing sensory neurons reduces spinal mu opioid receptors but paradoxically potentiates opioid analgesia.
Journal: Journal of neurophysiology20060501
Title: Anti-opioid activities of NPFF1 receptors in a SH-SY5Y model.
Journal: Peptides20060501
Title: [Differential contribution of dopamine D1 and D2 receptors in the mu-opioidergic immunomodulation].
Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova20060501
Title: In vivo evaluation of (+)-MR200 as a new selective sigma ligand modulating MOP, DOP and KOP supraspinal analgesia.
Journal: Life sciences20060418
Title: Opioid receptors in the nucleus accumbens regulate attentional learning in the blocking paradigm.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20060412
Title: Opioid-induced regulation of gene expression in PC12 cells stably transfected with mu-opioid receptor.
Journal: Neuroscience letters20060403
Title: Chronic pain induces anxiety with concomitant changes in opioidergic function in the amygdala.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20060401
Title: Mu opioid receptor activation inhibits GABAergic inputs to basolateral amygdala neurons through Kv1.1/1.2 channels.
Journal: Journal of neurophysiology20060401
Title: Mu-opioid receptors are involved in the tolerance to nicotine antinociception.
Journal: Journal of neurochemistry20060401
Title: Role of phospholipase D2 in the agonist-induced and constitutive endocytosis of G-protein coupled receptors.
Journal: Journal of neurochemistry20060401
Title: Evidence for a role of CaMKIV in the development of opioid analgesic tolerance.
Journal: The European journal of neuroscience20060401
Title: Modulation of Na, K-ATPase activity by prostaglandin E1 and [D-Ala2,N-Me-Phe4,Gly5-ol]-enkephalin.
Journal: Life sciences20060306
Title: Differential activation of G-proteins by mu-opioid receptor agonists.
Journal: British journal of pharmacology20060301
Title: Mu-opioid receptor cellular function in the nucleus accumbens is essential for hedonically driven eating.
Journal: The European journal of neuroscience20060301
Title: Mesencephalic astrocyte-derived neurotrophic factor enhances nigral gamma-aminobutyric acid release.
Journal: Neuroreport20060227
Title: Effects of prenatal cocaine, morphine, or both on postnatal opioid (mu) receptor development.
Journal: Life sciences20060223
Title: Estrogen and CCK1 receptor modification of mu-opioid receptor binding in the cortex of female rats.
Journal: Brain research20060216
Title: Different effects of opioid and cannabinoid receptor agonists on C-fiber-induced extracellular signal-regulated kinase activation in dorsal horn neurons in normal and spinal nerve-ligated rats.
Journal: The Journal of pharmacology and experimental therapeutics20060201
Title: Pharmacological characterization of inhibitory effects of postsynaptic opioid and cannabinoid receptors on calcium currents in neonatal rat nucleus tractus solitarius.
Journal: British journal of pharmacology20060201
Title: Cannabidiol is an allosteric modulator at mu- and delta-opioid receptors.
Journal: Naunyn-Schmiedeberg's archives of pharmacology20060201
Title: Medullary raphe neurons facilitate brown adipose tissue activation.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20060125
Title: Blocking polysynaptic inhibition via opioid receptor activation isolates excitatory synaptic currents without triggering epileptiform activity in organotypic hippocampal slices.
Journal: Journal of neuroscience methods20060115
Title: Mu and delta, but not kappa, opioid agonists induce spastic paraparesis after a short period of spinal cord ischaemia in rats.
Journal: British journal of anaesthesia20060101
Title: mu-Opioid receptor internalization-dependent and -independent mechanisms of the development of tolerance to mu-opioid receptor agonists: Comparison between etorphine and morphine.
Journal: Neuroscience20060101
Title: Inhibition by endomorphin-1 and endomorphin-2 of excitatory transmission in adult rat substantia gelatinosa neurons.
Journal: Neuroscience20060101
Title: [The role of monocytes in the effects of beta-endorphin and selective agonists of mu- and delta-Opiate receptors on the proliferative activity of peripheral blood lymphocytes].
Journal: Fiziologiia cheloveka20060101
Title: Methylnaltrexone inhibits opiate and VEGF-induced angiogenesis: role of receptor transactivation.
Journal: Microvascular research20060101
Title: Inhibition of AC-II activity following chronic agonist exposure is modulated by phosphorylation.
Journal: Journal of molecular neuroscience : MN20060101
Title: N-substituted cis-4a-(3-hydroxyphenyl)-8a-methyloctahydroisoquinolines are opioid receptor pure antagonists.
Journal: Journal of medicinal chemistry20051229
Title: Hedonic hot spot in nucleus accumbens shell: where do mu-opioids cause increased hedonic impact of sweetness?
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20051214
Title: Mu opioid receptor agonist DAMGO-induced suppression of saccharin intake in Lewis and Fischer rats.
Journal: Brain research20051207
Title: Antinociception following application of DAMGO to the basolateral amygdala results from a direct interaction of DAMGO with Mu opioid receptors in the amygdala.
Journal: Brain research20051207
Title: Nalmefene induced elevation in serum prolactin in normal human volunteers: partial kappa opioid agonist activity?
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20051201
Title: Hypoxia and acidosis increase the secretion of catecholamines in the neonatal rat adrenal medulla: an in vitro study.
Journal: American journal of physiology. Cell physiology20051201
Title: A role for the distal carboxyl tails in generating the novel pharmacology and G protein activation profile of mu and delta opioid receptor hetero-oligomers.
Journal: The Journal of biological chemistry20051118
Title: Morphine activates Arc expression in the mouse striatum and in mouse neuroblastoma Neuro2A MOR1A cells expressing mu-opioid receptors.
Journal: Journal of neuroscience research20051115
Title: Molecular mechanisms involved in the asymmetric interaction between cannabinoid and opioid systems.
Journal: Psychopharmacology20051101
Title: Effects of the local administration of selective mu-, delta-and kappa-opioid receptor agonists on osteosarcoma-induced hyperalgesia.
Journal: Naunyn-Schmiedeberg's archives of pharmacology20051101
Title: Reduced suppression of CO2-induced ventilatory stimulation by endomorphins relative to morphine.
Journal: Brain research20051019
Title: COMT Val108/158Met genotype affects the mu-opioid receptor system in the human brain: evidence from ligand-binding, G-protein activation and preproenkephalin mRNA expression.
Journal: NeuroImage20051015
Title: Comparison of the antinociceptive effect of acute morphine in female and male Sprague-Dawley rats using the long-lasting mu-antagonist methocinnamox.
Journal: Brain research20051005
Title: Development and validation of a radioreceptor assay for the determination of morphine and its active metabolites in serum.
Journal: Journal of pharmaceutical and biomedical analysis20051004
Title: Regulation of the extracellular signal-regulated kinases following acute and chronic opioid treatment.
Journal: Cellular and molecular life sciences : CMLS20051001
Title: Kappa- and delta-opioid receptor functional activities are increased in the caudate putamen of cannabinoid CB1 receptor knockout mice.
Journal: The European journal of neuroscience20051001
Title: Topography of 3H-DHA, 3H-QNB, 3H-dopamine, and 3H-DAGO binding sites distribution in the central part of the sinoatrial node in rat heart.
Journal: Bulletin of experimental biology and medicine20051001
Title: The ventral pallidum and hedonic reward: neurochemical maps of sucrose 'liking' and food intake.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050921
Title: Activation of delta-, kappa-, and mu-opioid receptors induces phosphorylation of tuberin in transfected HEK 293 cells and native cells.
Journal: Biochemical and biophysical research communications20050902
Title: Persistent upregulation of mu-opioid, but not adenosine, receptors in brains of long-term withdrawn escalating dose 'binge' cocaine-treated rats.
Journal: Synapse (New York, N.Y.)20050901
Title: Opioid tolerance in periaqueductal gray neurons isolated from mice chronically treated with morphine.
Journal: British journal of pharmacology20050901
Title: Peripheral axonal injury results in reduced mu opioid receptor pre- and post-synaptic action in the spinal cord.
Journal: Pain20050901
Title: Micro-opioid receptor preferentially inhibits oxytocin release from neurohypophysial terminals by blocking R-type Ca2+ channels.
Journal: Journal of neuroendocrinology20050901
Title: Activation of GPCRs modulates quantal size in chromaffin cells through G(betagamma) and PKC.
Journal: Nature neuroscience20050901
Title: Morphine promotes rapid, arrestin-dependent endocytosis of mu-opioid receptors in striatal neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050824
Title: Acute and chronic administration of clorazepate modifies the cell surface regulation of mu opioid receptors induced by buprenorphine in specific regions of the rat brain.
Journal: Brain research20050809
Title: Mu opioid receptor coupling to Gi/o proteins increases during postnatal development in rat brain.
Journal: The Journal of pharmacology and experimental therapeutics20050801
Title: Orphanin FQ/nociceptin potentiates [D-Ala2,N-Me-Phe4,Gly5-ol]-enkephalin-Induced mu-opioid receptor phosphorylation.
Journal: Molecular pharmacology20050801
Title: Mu and kappa opioid receptors activate ERK/MAPK via different protein kinase C isoforms and secondary messengers in astrocytes.
Journal: The Journal of biological chemistry20050729
Title: Mechanisms of mu opioid receptor/G-protein desensitization in brain by chronic heroin administration.
Journal: Life sciences20050722
Title: mu-Opioids disinhibit and kappa-opioids inhibit serotonin efflux in the dorsal raphe nucleus.
Journal: Brain research20050705
Title: Tramadol produces outward currents by activating mu-opioid receptors in adult rat substantia gelatinosa neurones.
Journal: British journal of pharmacology20050701
Title: Sugar solution analgesia: the effects of glucose on expressed mu opioid receptors.
Journal: Anesthesia and analgesia20050701
Title: Both kappa and mu opioid agonists inhibit glutamatergic input to ventral tegmental area neurons.
Journal: Journal of neurophysiology20050601
Title: Prolonged effects of repeated social defeat stress on mRNA expression and function of mu-opioid receptors in the ventral tegmental area of rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20050601
Title: Functional mu opioid receptors are expressed in cholinergic interneurons of the rat dorsal striatum: territorial specificity and diurnal variation.
Journal: The European journal of neuroscience20050601
Title: Alterations of prenatal morphine exposure in mu-opioid receptor density in hypothalamic nuclei associated with sexual behavior.
Journal: Brain research bulletin20050530
Title: Morphiceptin analogues containing a dipeptide mimetic structure: an investigation on the bioactive topology at the mu-receptor.
Journal: Journal of medicinal chemistry20050505
Title: Synthesis and biological evaluation of 14-alkoxymorphinans. 22.(1) Influence of the 14-alkoxy group and the substitution in position 5 in 14-alkoxymorphinan-6-ones on in vitro and in vivo activities.
Journal: Journal of medicinal chemistry20050505
Title: Maternal deprivation increases vulnerability to morphine dependence and disturbs the enkephalinergic system in adulthood.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050504
Title: Modulation of synaptic transmission in the rat nucleus of the solitary tract by endomorphin-1.
Journal: Journal of neurophysiology20050501
Title: Morphine alters the selective association between mu-opioid receptors and specific RGS proteins in mouse periaqueductal gray matter.
Journal: Neuropharmacology20050501
Title: STAT5A interacts with and is phosphorylated upon activation of the mu-opioid receptor.
Journal: Journal of neurochemistry20050501
Title: Emergence of the pre-Bötzinger respiratory rhythm generator in the mouse embryo.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050427
Title: Spinal G-protein-gated potassium channels contribute in a dose-dependent manner to the analgesic effect of mu- and delta- but not kappa-opioids.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050406
Title: Proopiomelanocortin neurons in nucleus tractus solitarius are activated by visceral afferents: regulation by cholecystokinin and opioids.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050406
Title: Inhibition by spinal mu- and delta-opioid agonists of afferent-evoked substance P release.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050406
Title: Ripple activity in the dentate gyrus of dishinibited hippocampus-entorhinal cortex slices.
Journal: Journal of neuroscience research20050401
Title: Reciprocal opioid-opioid interactions between the ventral tegmental area and nucleus accumbens regions in mediating mu agonist-induced feeding in rats.
Journal: Peptides20050401
Title: Biological activity of selected tyrosine-containing 2,5-diketopiperazines.
Journal: Die Pharmazie20050401
Title: Heterodimerization of mu- and delta-opioid receptors occurs at the cell surface only and requires receptor-G protein interactions.
Journal: The Journal of biological chemistry20050325
Title: Induction of delta-opioid receptor function in the midbrain after chronic morphine treatment.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20050323
Title: Adenosine contributes to mu-opioid synaptic inhibition in rat substantia gelatinosa in vitro.
Journal: Neuroscience letters20050311
Title: A Tyr-W-MIF-1 analog containing D-Pro2 acts as a selective mu2-opioid receptor antagonist in the mouse.
Journal: The Journal of pharmacology and experimental therapeutics20050301
Title: Characterisation of opioid receptors involved in modulating circular and longitudinal muscle contraction in the rat ileum.
Journal: British journal of pharmacology20050301
Title: Heterodimerization of opioid receptor-like 1 and mu-opioid receptors impairs the potency of micro receptor agonist.
Journal: Journal of neurochemistry20050301
Title: Ancient gill and lung oscillators may generate the respiratory rhythm of frogs and rats.
Journal: Journal of neurobiology20050215
Title: Neuronal nitric oxide modulates morphine antinociceptive tolerance by enhancing constitutive activity of the mu-opioid receptor.
Journal: Biochemical pharmacology20050215
Title: Opiate modulation of monoamines in the chick forebrain: possible role in emotional regulation?
Journal: Journal of neurobiology20050205
Title: Endogenous regulator of g protein signaling proteins reduce {mu}-opioid receptor desensitization and down-regulation and adenylyl cyclase tolerance in C6 cells.
Journal: The Journal of pharmacology and experimental therapeutics20050201
Title: Effect of the {mu} opioid on excitatory and inhibitory synaptic inputs to periaqueductal gray-projecting neurons in the amygdala.
Journal: The Journal of pharmacology and experimental therapeutics20050201
Title: Increased nociceptive response in mice lacking the adenosine A1 receptor.
Journal: Pain20050201
Title: Melatonin exerts its analgesic actions not by binding to opioid receptor subtypes but by increasing the release of beta-endorphin an endogenous opioid.
Journal: Brain research bulletin20050130
Title: Pharmacologically selective block of mu opioid antinociception by peptide nucleic acid antisense in absence of detectable ex vivo knockdown.
Journal: European journal of pharmacology20050104
Title: Receptor endocytosis counteracts the development of opioid tolerance.
Journal: Molecular pharmacology20050101
Title: Agonists at mu-opioid receptors spin the wheels to keep the action going.
Journal: Molecular pharmacology20050101
Title: Effects of long-term biogenic amine transporter blockade on receptor/G-protein coupling in rat brain.
Journal: Neuropharmacology20050101
Title: [Effect of opiod peptides on free radical oxidation in a bone regenerate after fracture].
Journal: Patologicheskaia fiziologiia i eksperimental'naia terapiia20050101
Title: delta-opioid receptor-mediated actions on rostral ventromedial medulla neurons.
Journal: Neuroscience20050101
Title: Enhanced striatal opioid receptor-mediated G-protein activation in L-DOPA-treated dyskinetic monkeys.
Journal: Neuroscience20050101
Title: Mu-opioid-mediated inhibition of glutamate synaptic transmission in rat central amygdala neurons.
Journal: Neuroscience20050101
Title: Opioid receptor stimulation does not affect cellular hypoxia-induced gene responses mediated by hypoxia-inducible factor 1 in cultured cell lines.
Journal: Journal of anesthesia20050101
Title: Ultra-low-dose naloxone suppresses opioid tolerance, dependence and associated changes in mu opioid receptor-G protein coupling and Gbetagamma signaling.
Journal: Neuroscience20050101
Title: Interactions among mu- and delta-opioid receptors, especially putative delta1- and delta2-opioid receptors, promote dopamine release in the nucleus accumbens.
Journal: Neuroscience20050101
Title: Opioid receptor binding characteristics and structure-activity studies of novel tetrapeptides in the TIPP (Tyr-Tic-Phe-Phe) series.
Journal: Neuro-Signals20050101
Title: Displacement of opioid receptor binding ligands from the rat brain by N3-(2',5'-dimethoxyphenacyl) arabinofuranosyluracil.
Journal: Research communications in molecular pathology and pharmacology20050101
Title: A bi-directional mu-opioid-opioid connection between the nucleus of the accumbens shell and the central nucleus of the amygdala in the rat.
Journal: Brain research20041210
Title: Internalization and down-regulation of mu opioid receptors by endomorphins and morphine in SH-SY5Y human neuroblastoma cells.
Journal: Brain research20041203
Title: Differential sensitivity of N- and P/Q-type Ca2+ channel currents to a mu opioid in isolectin B4-positive and -negative dorsal root ganglion neurons.
Journal: The Journal of pharmacology and experimental therapeutics20041201
Title: Opioid-like actions of neuropeptide Y in rat substantia gelatinosa: Y1 suppression of inhibition and Y2 suppression of excitation.
Journal: Journal of neurophysiology20041201
Title: Tolerance develops in spinal cord, but not in brain with chronic [Dmt1]DALDA treatment.
Journal: British journal of pharmacology20041201
Title: Mu and delta opioid-stimulated [35S]GTP gamma S binding in brain and spinal cord of polyarthritic rats.
Journal: European journal of pharmacology20041103
Title: The stimulatory effect of mu- and delta-opioid receptors on bovine pinealocyte melatonin synthesis.
Journal: Journal of pineal research20041101
Title: Hetero-oligomers of alpha2A-adrenergic and mu-opioid receptors do not lead to transactivation of G-proteins or altered endocytosis profiles.
Journal: Biochemical Society transactions20041101
Title: Selective postsynaptic inhibition of tonic-firing neurons in substantia gelatinosa by mu-opioid agonist.
Journal: Anesthesiology20041101
Title: Baclofen reestablishes micro-opioid receptor levels modified by morphine withdrawal syndrome in either sex.
Journal: Synapse (New York, N.Y.)20041001
Title: Peripheral opiate action on afferent fibres supplying the rat intestine.
Journal: Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society20041001
Title: Opioid agonist and antagonist treatment differentially regulates immunoreactive mu-opioid receptors and dynamin-2 in vivo.
Journal: European journal of pharmacology20040913
Title: Chronic antidepressant treatment causes a selective reduction of mu-opioid receptor binding and functional coupling to G Proteins in the amygdala of fawn-hooded rats.
Journal: The Journal of pharmacology and experimental therapeutics20040901
Title: The amygdala is critical for opioid-mediated binge eating of fat.
Journal: Neuroreport20040826
Title: Alterations in food intake by opioid and dopamine signaling pathways between the ventral tegmental area and the shell of the nucleus accumbens.
Journal: Brain research20040820
Title: Opioid receptors in fast and slow skeletal muscles of normal and dystrophic mice.
Journal: Neuroscience letters20040819
Title: Morphine induces terminal micro-opioid receptor desensitization by sustained phosphorylation of serine-375.
Journal: The EMBO journal20040818
Title: Activation of protein kinase C antagonizes the opioid inhibition of calcium current in rat spinal dorsal horn neurons.
Journal: Brain research20040813
Title: Activation of AP-1 and CRE-dependent gene expression via mu-opioid receptor.
Journal: Journal of neurochemistry20040801
Title: Feeding responses to mu-, delta- and kappa-opioid receptor agonists in the meat-type chick.
Journal: Pharmacology, biochemistry, and behavior20040801
Title: Modulation of anxiety-related behaviors by mu- and kappa-opioid receptor agonists depends on the social status of mice.
Journal: Peptides20040801
Title: Intra-amygdalar injection of DAMGO: effects on c-Fos levels in brain sites associated with feeding behavior.
Journal: Brain research20040723
Title: Dual effects of DAMGO [D-Ala2,N-Me-Phe4,Gly5-ol]-enkephalin and CTAP (D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2) on adenylyl cyclase activity: implications for mu-opioid receptor Gs coupling.
Journal: The Journal of pharmacology and experimental therapeutics20040701
Title: The role of central mu opioid receptors in opioid-induced itch in primates.
Journal: The Journal of pharmacology and experimental therapeutics20040701
Title: Central effects of the cannabinoid receptor agonist WIN55212-2 on respiratory and cardiovascular regulation in anaesthetised rats.
Journal: British journal of pharmacology20040701
Title: Na+ modulation, inverse agonism, and anorectic potency of 4-phenylpiperidine opioid antagonists.
Journal: European journal of pharmacology20040628
Title: Activation of mu opioid receptors in the ventrolateral periaqueductal gray inhibits reflex micturition in anesthetized rats.
Journal: Neuroscience letters20040610
Title: Opioid peptide receptor studies. 17. Attenuation of chronic morphine effects after antisense oligodeoxynucleotide knock-down of RGS9 protein in cells expressing the cloned Mu opioid receptor.
Journal: Synapse (New York, N.Y.)20040601
Title: Role of mu- and delta-opioid receptors in the nucleus accumbens in turning behaviour of rats.
Journal: Neuropharmacology20040601
Title: Nitric oxide modulates the physiological control of ciliary activity in the marine mussel Mytilus edulis via morphine: novel mu opiate receptor splice variants.
Journal: Neuro endocrinology letters20040601
Title: Opioid receptor desensitization contributes to thermal hyperalgesia in infant rats.
Journal: European journal of pharmacology20040503
Title: Activation of mu-opioid receptors inhibits synaptic inputs to spinally projecting rostral ventromedial medulla neurons.
Journal: The Journal of pharmacology and experimental therapeutics20040501
Title: Effect of the A118G polymorphism on binding affinity, potency and agonist-mediated endocytosis, desensitization, and resensitization of the human mu-opioid receptor.
Journal: Journal of neurochemistry20040501
Title: Endomorphins exit the brain by a saturable efflux system at the basolateral surface of cerebral endothelial cells.
Journal: Experimental brain research20040501
Title: Involvement of opioid receptor subtypes in both stimulatory and inhibitory effects of the opioid peptides on prolactin secretion during pregnancy.
Journal: Cellular and molecular neurobiology20040401
Title: Identification of opioid ligands possessing mixed micro agonist/delta antagonist activity among pyridomorphinans derived from naloxone, oxymorphone, and hydromorphone [correction of hydropmorphone].
Journal: Journal of medicinal chemistry20040311
Title: Increases in food intake or food-seeking behavior induced by GABAergic, opioid, or dopaminergic stimulation of the nucleus accumbens: is it hunger?
Journal: Psychopharmacology20040301
Title: Opioid partial agonist effects of 3-O-methylnaltrexone in rhesus monkeys.
Journal: The Journal of pharmacology and experimental therapeutics20040301
Title: Opioid-mediated modulation of calcium currents in striatal and pallidal neurons following reserpine treatment: focus on kappa response.
Journal: Synapse (New York, N.Y.)20040301
Title: Orexin (hypocretin)/dynorphin neurons control GABAergic inputs to tuberomammillary neurons.
Journal: The European journal of neuroscience20040301
Title: DAMGO suppresses both excitatory and inhibitory synaptic transmission in supraoptic neurones of mouse hypothalamic slice preparations.
Journal: Journal of neuroendocrinology20040301
Title: Dopamine1 receptor agonists reverse opioid respiratory network depression, increase CO2 reactivity.
Journal: Respiratory physiology & neurobiology20040225
Title: A non-peptide substance P antagonist (CP-96,345) inhibits morphine-induced NF-kappa B promoter activation in human NT2-N neurons.
Journal: Journal of neuroscience research20040215
Title: Characterization of mu opioid receptor binding and G protein coupling in rat hypothalamus, spinal cord, and primary afferent neurons during inflammatory pain.
Journal: The Journal of pharmacology and experimental therapeutics20040201
Title: Phospholipase D2 modulates agonist-induced mu-opioid receptor desensitization and resensitization.
Journal: Journal of neurochemistry20040201
Title: [Molecular pharmacology of opioid receptors].
Journal: Nihon yakurigaku zasshi. Folia pharmacologica Japonica20040201
Title: Enhanced morphine withdrawal and micro -opioid receptor G-protein coupling in A2A adenosine receptor knockout mice.
Journal: Journal of neurochemistry20040201
Title: Morphine prevents glutamate-induced death of primary rat neonatal astrocytes through modulation of intracellular redox.
Journal: Immunopharmacology and immunotoxicology20040201
Title: The influence of opioid peptides on steroidogenesis in porcine granulosa cells.
Journal: Reproduction in domestic animals = Zuchthygiene20040201
Title: Activation of mu-opioid receptors excites a population of locus coeruleus-spinal neurons through presynaptic disinhibition.
Journal: Brain research20040130
Title: Heterodimerization and cross-desensitization between the mu-opioid receptor and the chemokine CCR5 receptor.
Journal: European journal of pharmacology20040112
Title: Functional coupling, desensitization and internalization of virally expressed mu opioid receptors in cultured dorsal root ganglion neurons from mu opioid receptor knockout mice.
Journal: Neuroscience20040101
Title: Reduction in [D-Ala2, NMePhe4, Gly-ol5]enkephalin-induced peripheral antinociception in diabetic rats: the role of the L-arginine/nitric oxide/cyclic guanosine monophosphate pathway.
Journal: Anesthesia and analgesia20040101
Title: The effect of CNS opioid on autonomic nervous and cardiovascular responses in diet-induced obese rats.
Journal: Peptides20040101
Title: [d-Ala2,N-MePhe4,Gly-ol5]enkephalin-induced internalization of the micro opioid receptor in the spinal cord of morphine tolerant rats.
Journal: Neuroscience20040101
Title: Opioidergic modulation of excitability of rat trigeminal root ganglion neuron projections to the superficial layer of cervical dorsal horn.
Journal: Neuroscience20040101
Title: Neurotransmitters involved in the opioid regulation of prolactin secretion at the end of pregnancy in rats.
Journal: Neuroendocrinology20040101
Title: Opioid modulation of GABA release in the rat inferior colliculus.
Journal: BMC neuroscience20040101
Title: Enkephalinergic inhibition of raphe pallidus inputs to rat hypoglossal motoneurones in vitro.
Journal: Neuroscience20040101
Title: Mu-opioid receptor agonist effects on medullary respiratory neurons in the cat: evidence for involvement in certain types of ventilatory disturbances.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20031201
Title: Comparison of [Dmt1]DALDA and DAMGO in binding and G protein activation at mu, delta, and kappa opioid receptors.
Journal: The Journal of pharmacology and experimental therapeutics20031201
Title: DPI-3290 [(+)-3-((alpha-R)-alpha-((2S,5R)-4-allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl)-N-(3-fluorophenyl)-N-methylbenzamide]. I. A mixed opioid agonist with potent antinociceptive activity.
Journal: The Journal of pharmacology and experimental therapeutics20031201
Title: Antinociceptive effect of morphine, but not mu opioid receptor number, is attenuated in the spinal cord of diabetic rats.
Journal: Anesthesiology20031201
Title: Afferent fiber-selective shift in opiate potency following targeted opioid receptor knockdown.
Journal: Pain20031201
Title: Lack of mu-opioid receptor-mediated G-protein activation in the spinal cord of mice lacking Exon 1 or Exons 2 and 3 of the MOR-1 gene.
Journal: Journal of pharmacological sciences20031201
Title: Evidence for a mu-opioid-opioid connection between the paraventricular nucleus and ventral tegmental area in the rat.
Journal: Brain research20031121
Title: Mu-opioid receptor desensitization in mature rat neurons: lack of interaction between DAMGO and morphine.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20031119
Title: Phosphoinositide 3-kinase cascade facilitates mu-opioid desensitization in sensory neurons by altering G-protein-effector interactions.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20031112
Title: Anti-mu opioid antiserum against the third external loop of the cloned mu-opioid receptor acts as a mu receptor neutral antagonist.
Journal: Brain research. Molecular brain research20031106
Title: Kappa-opioid agonists directly inhibit midbrain dopaminergic neurons.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20031105
Title: Co-incident signalling between mu-opioid and M3 muscarinic receptors at the level of Ca2+ release from intracellular stores: lack of evidence for Ins(1,4,5)P3 receptor sensitization.
Journal: The Biochemical journal20031101
Title: Effects of the opioid antagonist naltrexone on feeding induced by DAMGO in the ventral tegmental area and in the nucleus accumbens shell region in the rat.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20031101
Title: Vivitrex, an injectable, extended-release formulation of naltrexone, provides pharmacokinetic and pharmacodynamic evidence of efficacy for 1 month in rats.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology20031101
Title: Effects of endomorphin on substantia gelatinosa neurons in rat spinal cord slices.
Journal: British journal of pharmacology20031101
Title: Neuropeptide FF exerts pro- and anti-opioid actions in the parabrachial nucleus to modulate food intake.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20031101
Title: An orexigenic role for mu-opioid receptors in the lateral parabrachial nucleus.
Journal: American journal of physiology. Regulatory, integrative and comparative physiology20031101
Title: Direct evidence for the up-regulation of spinal micro-opioid receptor function after repeated stimulation of kappa-opioid receptors in the mouse.
Journal: The European journal of neuroscience20031101
Title: Involvement of protein kinase C in the adaptive changes of cholinergic neurons to sympathetic denervation in the guinea pig myenteric plexus.
Journal: Life sciences20031003
Title: Acute ethanol administration transiently decreases [3H]-DAMGO binding to mu opioid receptors in the rat substantia nigra pars reticulata but not in the caudate-putamen.
Journal: Neuroscience research20031001
Title: Evidence for a role of dopaminergic mechanisms in the immunostimulating effect of mu-opioid receptor agonist DAGO.
Journal: The International journal of neuroscience20031001
Title: Pharmacological characterization of a 7-benzylidenenaltrexone-preferring opioid receptor in porcine ileal submucosa.
Journal: British journal of pharmacology20031001
Title: Two distinct forms of desensitization of G-protein coupled inwardly rectifying potassium currents evoked by alkaloid and peptide mu-opioid receptor agonists.
Journal: Molecular and cellular neurosciences20031001
Title: The regulation of steroidogenesis by opioid peptides in porcine theca cells.
Journal: Animal reproduction science20030915
Title: Mu-opioid-induced desensitization of opioid receptor-like 1 and mu-opioid receptors: differential intracellular signaling determines receptor sensitivity.
Journal: The Journal of pharmacology and experimental therapeutics20030901
Title: Glycinergic inputs to cardiac vagal neurons in the nucleus ambiguus are inhibited by nociceptin and mu-selective opioids.
Journal: Journal of neurophysiology20030901
Title: mu-Opioid receptor modulates peptide release from rat neurohypophysial terminals by inhibiting Ca(2+) influx.
Journal: Journal of neuroendocrinology20030901
Title: Systemic morphine-induced release of serotonin in the rostroventral medulla is not mimicked by morphine microinjection into the periaqueductal gray.
Journal: Journal of neurochemistry20030901
Title: Expression of EGFP-amino-tagged human mu opioid receptor in Drosophila Schneider 2 cells: a potential expression system for large-scale production of G-protein coupled receptors.
Journal: Protein expression and purification20030901
Title: Roles of alpha1- and alpha2-adrenoceptors in the nucleus raphe magnus in opioid analgesia and opioid abstinence-induced hyperalgesia.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20030827
Title: Presynaptic mechanism for anti-analgesic and anti-hyperalgesic actions of kappa-opioid receptors.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20030813
Title: Differences of mu-opioid receptors between Lewis and F344 rats.
Journal: Life sciences20030808
Title: Characterization of the binding of [3H][Dmt1]H-Dmt-D-Arg-Phe-Lys-NH2, a highly potent opioid peptide.
Journal: The Journal of pharmacology and experimental therapeutics20030801
Title: Effects of orexin (hypocretin) on GIRK channels.
Journal: Journal of neurophysiology20030801
Title: Painful inflammation-induced increase in mu-opioid receptor binding and G-protein coupling in primary afferent neurons.
Journal: Molecular pharmacology20030801
Title: Expression and G-protein coupling of mu-opioid receptors in the spinal cord and dorsal root ganglia of polyarthritic rats.
Journal: Neuropeptides20030801
Title: The effect of papaverine on acute opiate withdrawal in guinea pig ileum.
Journal: Phytotherapy research : PTR20030801
Title: Effects of single and dual administration of cocaine and ethanol on opioid and ORL1 receptor expression in rat CNS: an autoradiographic study.
Journal: Brain research20030718
Title: Studies of micro-, kappa-, and delta-opioid receptor density and G protein activation in the cortex and thalamus of monkeys.
Journal: The Journal of pharmacology and experimental therapeutics20030701
Title: Buprenorphine blocks epsilon- and micro-opioid receptor-mediated antinociception in the mouse.
Journal: The Journal of pharmacology and experimental therapeutics20030701
Title: Lack of intersite GABA receptor subtype antagonist effects upon mu opioid receptor agonist-induced feeding elicited from either the ventral tegmental area or nucleus accumbens shell in rats.
Journal: Physiology & behavior20030701
Title: Ligand-selective activation of mu-oid receptor: demonstrated with deletion and single amino acid mutations of third intracellular loop domain.
Journal: The Journal of pharmacology and experimental therapeutics20030601
Title: Heterologous mu-opioid receptor adaptation by repeated stimulation of kappa-opioid receptor: up-regulation of G-protein activation and antinociception.
Journal: Journal of neurochemistry20030601
Title: Rhythmic phrenic, intercostal and sympathetic activity in relation to limb and trunk motor activity in spinal cats.
Journal: Neuroscience research20030601
Title: Opioid agonists have different efficacy profiles for G protein activation, rapid desensitization, and endocytosis of mu-opioid receptors.
Journal: The Journal of biological chemistry20030523
Title: Internalization and recycling of human mu opioid receptors expressed in Sf9 insect cells.
Journal: Life sciences20030523
Title: Effect of strain and sex on mu opioid receptor-mediated G-protein activation in rat brain.
Journal: Brain research bulletin20030515
Title: New scaffolds in the development of mu opioid-receptor ligands.
Journal: Bioorganic & medicinal chemistry letters20030505
Title: Anti-inflammatory properties of the mu opioid receptor support its use in the treatment of colon inflammation.
Journal: The Journal of clinical investigation20030501
Title: Cellular actions of opioids on periaqueductal grey neurons from C57B16/J mice and mutant mice lacking MOR-1.
Journal: British journal of pharmacology20030501
Title: Effects of in vitro and in vivo opioids on the production of IL-12 and IL-10 by murine macrophages.
Journal: Annals of the New York Academy of Sciences20030501
Title: Cardiovascular responses to central administration of mu and kappa opioid receptor agonist and antagonist in normal rats.
Journal: Peptides20030501
Title: Identity of the putative delta1-opioid receptor as a delta-kappa heteromer in the mouse spinal cord.
Journal: European journal of pharmacology20030425
Title: Mu-opioid modulation of HIV-1 coreceptor expression and HIV-1 replication.
Journal: Virology20030425
Title: 14-amino, 14-alkylamino, and 14-acylamino analogs of oxymorphindole. Differential effects on opioid receptor binding and functional profiles.
Journal: Journal of medicinal chemistry20030410
Title: Morphology and axonal arborization of rat spinal inner lamina II neurons hyperpolarized by mu-opioid-selective agonists.
Journal: The Journal of comparative neurology20030407
Title: Dermorphin tetrapeptide analogues with 2',6'-dimethylphenylalanine (Dmp) substituted for aromatic amino acids have high mu opioid receptor binding and biological activities.
Journal: Bioorganic & medicinal chemistry letters20030407
Title: Hypothalamic proopiomelanocortin neurons are glucose responsive and express K(ATP) channels.
Journal: Endocrinology20030401
Title: Roles of protein kinase A and C in the opioid potentiation of the GABAA response in rat periaqueductal gray neuron.
Journal: Neuropharmacology20030401
Title: Nucleus accumbens mu-opioids regulate intake of a high-fat diet via activation of a distributed brain network.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20030401
Title: Nucleus accumbens opioid, GABaergic, and dopaminergic modulation of palatable food motivation: contrasting effects revealed by a progressive ratio study in the rat.
Journal: Behavioral neuroscience20030401
Title: Opioids and the apoptotic pathway in human cancer cells.
Journal: Neuropeptides20030401
Title: The effect of endomorphins on the release of 3H-norepinephrine from rat nucleus tractus solitarii slices.
Journal: Regulatory peptides20030328
Title: Endogenous RGS protein action modulates mu-opioid signaling through Galphao. Effects on adenylyl cyclase, extracellular signal-regulated kinases, and intracellular calcium pathways.
Journal: The Journal of biological chemistry20030314
Title: Mu-opioid receptor activation prevents apoptosis following serum withdrawal in differentiated SH-SY5Y cells and cortical neurons via phosphatidylinositol 3-kinase.
Journal: Neuropharmacology20030301
Title: Up-regulation of mu-opioid receptor-mediated G-protein activation in protein kinase Cgamma knockout mice following repeated naloxone treatment.
Journal: Neuroscience letters20030227
Title: Naloxone and its quaternary derivative, naloxone methiodide, have differing affinities for mu, delta, and kappa opioid receptors in mouse brain homogenates.
Journal: Brain research20030227
Title: The presynaptic modulation of corticostriatal afferents by mu-opioids is mediated by K+ conductances.
Journal: European journal of pharmacology20030221
Title: The mu opioid agonist DAMGO stimulates cAMP production in SK-N-SH cells through a PLC-PKC-Ca++ pathway.
Journal: Brain research. Molecular brain research20030220
Title: Blockade of mu-opioid receptor-mediated G-protein activation and antinociception by TRK-820 in mice.
Journal: European journal of pharmacology20030207
Title: (2S,3R) beta-methyl-2',6'-dimethyltyrosine-L-tetrahydroisoquinoline-3-carboxylic acid [(2S,3R)TMT-L-Tic-OH] is a potent, selective delta-opioid receptor antagonist in mouse brain.
Journal: The Journal of pharmacology and experimental therapeutics20030201
Title: Molecular evidence for the functional role of dopamine D3 receptor in the morphine-induced rewarding effect and hyperlocomotion.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20030201
Title: Opioid receptor activation attenuates nicotinic enhancement of spontaneous GABA release in lateral spiriform nucleus of the chick.
Journal: Brain research20030124
Title: Neurokinin-1 versus mu-opioid receptor binding in rat nucleus tractus solitarius after single and recurrent intermittent hypoxia.
Journal: Brain research bulletin20030115
Title: Tolerance and dependence following chronic intracerebroventricular infusions of Tyr-D-Arg2-Phe-Sar4 (TAPS).
Journal: European journal of pharmacology20030110
Title: Opioid peptide receptor studies. 16. Chronic morphine alters G-protein function in cells expressing the cloned mu opioid receptor.
Journal: Synapse (New York, N.Y.)20030101
Title: Cocaine alters mu but not delta or kappa opioid receptor-stimulated in situ [35S]GTPgammaS binding in rat brain.
Journal: Synapse (New York, N.Y.)20030101
Title: Coexpression of delta-opioid receptors with micro receptors in GH3 cells changes the functional response to micro agonists from inhibitory to excitatory.
Journal: Molecular pharmacology20030101
Title: Opioid receptor-induced GTPgamma35S binding during mouse development.
Journal: Developmental biology20030101
Title: Potency differences for D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2 as an antagonist of peptide and alkaloid micro-agonists in an antinociception assay.
Journal: The Journal of pharmacology and experimental therapeutics20030101
Title: Activity of opioid ligands in cells expressing cloned mu opioid receptors.
Journal: BMC pharmacology20030101
Title: Characterization of opioid receptors that modulate nociceptive neurotransmission in the trigeminocervical complex.
Journal: British journal of pharmacology20030101
Title: Mild thyroid hormones deficiency modifies benzodiazepine and mu-opioid receptor binding in rats.
Journal: Neuropharmacology20030101
Title: Mu opioid receptor signaling in morphine sensitization.
Journal: Neuroscience20030101
Title: Ligand-induced mu opioid receptor endocytosis and recycling in enteric neurons.
Journal: Neuroscience20030101
Title: Upregulation of mu opioid receptors by voluntary morphine administration in drinking water.
Journal: Acta biologica Hungarica20030101
Title: Effect of beta-endorphin and DAGO, a selective agonist of mu-opioid receptors, on the proliferative activity of lymphocytes.
Journal: Doklady biological sciences : proceedings of the Academy of Sciences of the USSR, Biological sciences sections20030101
Title: Loss of mu-opioid receptor-mediated G-protein activation in the pons/medulla of mice lacking the exons 2 and 3 of mu-opioid receptor gene.
Journal: Neuroscience letters20021225
Title: Modulation of melanocortin-induced changes in spinal nociception by mu-opioid receptor agonist and antagonist in neuropathic rats.
Journal: Neuroreport20021220
Title: (-)-Cannabidiol antagonizes cannabinoid receptor agonists and noradrenaline in the mouse vas deferens.
Journal: European journal of pharmacology20021205
Title: Opioid agonists differentially regulate mu-opioid receptors and trafficking proteins in vivo.
Journal: Molecular pharmacology20021201
Title: The fibroblast growth factor receptor is at the site of convergence between mu-opioid receptor and growth factor signaling pathways in rat C6 glioma cells.
Journal: The Journal of pharmacology and experimental therapeutics20021201
Title: Functional mu opioid receptors are reduced in the spinal cord dorsal horn of diabetic rats.
Journal: Anesthesiology20021201
Title: Kainic acid modifies mu-receptor binding in young, adult, and elderly rat brain.
Journal: Cellular and molecular neurobiology20021201
Title: Opioid receptor subtypes differentially modulate serotonin efflux in the rat central nervous system.
Journal: The Journal of pharmacology and experimental therapeutics20021101
Title: Spinal pretreatment with antisense oligodeoxynucleotides against exon-1, -4, or -8 of mu-opioid receptor clone leads to differential loss of spinal endomorphin-1-and endomorphin-2-induced antinociception in the mouse.
Journal: The Journal of pharmacology and experimental therapeutics20021101
Title: Induction of G protein-coupled receptor kinases 2 and 3 contributes to the cross-talk between mu and ORL1 receptors following prolonged agonist exposure.
Journal: Neuropharmacology20021101
Title: The effect of opioid agonists of delta-class DSLET, mu-class DAMGO, kappa-class U-69593 and an opioid antagonist, naloxone, on MTT activity of NALM-1 leukemic cells.
Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie20021101
Title: Turnover of mu-opioid receptors in neuroblastoma cells.
Journal: Brain research. Molecular brain research20021015
Title: The local environment at the cytoplasmic end of TM6 of the mu opioid receptor differs from those of rhodopsin and monoamine receptors: introduction of an ionic lock between the cytoplasmic ends of helices 3 and 6 by a L6.30(275)E mutation inactivates the mu opioid receptor and reduces the constitutive activity of its T6.34(279)K mutant.
Journal: Biochemistry20021008
Title: Influence of a deletion of protein kinase C gamma isoform in the G-protein activation mediated through opioid receptor-like-1 and mu-opioid receptors in the mouse pons/medulla.
Journal: Neuroscience letters20021004
Title: Estrogen modulation of mu-opioid receptor-stimulated [35S]-GTP-gamma-S binding in female rat brain visualized by in vitro autoradiography.
Journal: Neuroendocrinology20021001
Title: Dimerization of morphine and orphanin FQ/nociceptin receptors: generation of a novel opioid receptor subtype.
Journal: Biochemical and biophysical research communications20020927
Title: Quantitative stoichiometry of G-proteins activated by mu-opioid receptors in postmortem human brain.
Journal: European journal of pharmacology20020927
Title: Regulation of dihydropyridine-sensitive Ca(2+) channels during naloxone-induced opioid supersensitivity in rats.
Journal: European journal of pharmacology20020920
Title: Sympathetic denervation-induced changes in G protein expression in enteric neurons of the guinea pig colon.
Journal: Life sciences20020913
Title: Chronic muscle pain induced by repeated acid Injection is reversed by spinally administered mu- and delta-, but not kappa-, opioid receptor agonists.
Journal: The Journal of pharmacology and experimental therapeutics20020901
Title: Lack of the nociceptin receptor does not affect acute or chronic nociception in mice.
Journal: Peptides20020901
Title: Orphanin FQ/nociceptin-mediated desensitization of opioid receptor-like 1 receptor and mu opioid receptors involves protein kinase C: a molecular mechanism for heterologous cross-talk.
Journal: The Journal of pharmacology and experimental therapeutics20020801
Title: Morphine-3beta-D-glucuronide suppresses inhibitory synaptic transmission in rat substantia gelatinosa.
Journal: The Journal of pharmacology and experimental therapeutics20020801
Title: Chronic morphine-induced changes in mu-opioid receptors and G proteins of different subcellular loci in rat brain.
Journal: The Journal of pharmacology and experimental therapeutics20020801
Title: Affinities of dihydrocodeine and its metabolites to opioid receptors.
Journal: Pharmacology & toxicology20020801
Title: Quantitative autoradiographic mapping of opioid receptors in the brain of delta-opioid receptor gene knockout mice.
Journal: Brain research20020726
Title: Brain regional mu-opioid receptor function in rat lines selected for differences in alcohol preference.
Journal: European journal of pharmacology20020719
Title: Effect of MK-801 on the antinociceptive effect of [D-Ala(2),N-MePhe(4), Gly-ol(5)]enkephalin in diabetic mice.
Journal: European journal of pharmacology20020712
Title: Inhibitory effects of opioids on voltage-dependent Ca(2+) channels and catecholamine secretion in cultured porcine adrenal chromaffin cells.
Journal: Brain research20020628
Title: Endomorphin-1 analogues containing beta-proline are mu-opioid receptor agonists and display enhanced enzymatic hydrolysis resistance.
Journal: Journal of medicinal chemistry20020606
Title: Presynaptic mu-opioid receptors regulate a late step of the secretory process in rat ventral tegmental area GABAergic neurons.
Journal: Neuropharmacology20020601
Title: Heterodimerization of somatostatin and opioid receptors cross-modulates phosphorylation, internalization, and desensitization.
Journal: The Journal of biological chemistry20020531
Title: Differential effects of chronic antidepressant treatments on micro- and delta-opioid receptors in rat brain.
Journal: European journal of pharmacology20020517
Title: Potentiation of the excitatory action of NMDA in ventrolateral periaqueductal gray by the mu-opioid receptor agonist, DAMGO.
Journal: Brain research20020510
Title: mu-Opioid receptors desensitize less rapidly than delta-opioid receptors due to less efficient activation of arrestin.
Journal: The Journal of biological chemistry20020503
Title: Alterations in food intake elicited by GABA and opioid agonists and antagonists administered into the ventral tegmental area region of rats.
Journal: Physiology & behavior20020501
Title: Biosensing of opioids using frog melanophores.
Journal: Biosensors & bioelectronics20020401
Title: Characterization of mu, kappa, and delta opioid binding in amphibian whole brain tissue homogenates.
Journal: The Journal of pharmacology and experimental therapeutics20020401
Title: Specific expression of spinal Fos after PAR-2 stimulation in mast cell-depleted rats.
Journal: Neuroreport20020325
Title: Analysis of opioid receptor subtype antagonist effects upon mu opioid agonist-induced feeding elicited from the ventral tegmental area of rats.
Journal: Brain research20020301
Title: Predominance of delta-opioid-binding sites in the porcine enteric nervous system.
Journal: The Journal of pharmacology and experimental therapeutics20020301
Title: Pharmacological manipulations of the pedunculopontine tegmental nucleus in the rat reduce self-administration of both nicotine and cocaine.
Journal: Psychopharmacology20020301
Title: Deletion of CCK2 receptor in mice results in an upregulation of the endogenous opioid system.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20020301
Title: mu/delta Cooperativity and opposing kappa-opioid effects in nucleus accumbens-mediated antinociception in the rat.
Journal: The European journal of neuroscience20020301
Title: Up-regulation of central mu-opioid receptors in a model of hepatic encephalopathy: a potential mechanism for increased sensitivity to morphine in liver failure.
Journal: Life sciences20020222
Title: Ginseng and ginsenoside Rg3, a newly identified active ingredient of ginseng, modulate Ca2+ channel currents in rat sensory neurons.
Journal: European journal of pharmacology20020202
Title: [Nphe(1)]N/OFQ-(1-13)-NH(2) is a competitive and selective antagonist at nociceptin/orphanin FQ receptors mediating K(+) channel activation in rat periaqueductal gray slices.
Journal: Neuropharmacology20020201
Title: Opioid agonists inhibit excitatory neurotransmission in ganglia and at the neuromuscular junction in Guinea pig gallbladder.
Journal: Gastroenterology20020201
Title: Change of hyperexcitability of hippocampus by cyclosporin A and its modulatory action by fentanyl.
Journal: Journal of Korean medical science20020201
Title: Activation of mu-opioid receptors inhibits lordosis behavior in estrogen and progesterone-primed female rats.
Journal: Hormones and behavior20020201
Title: Regulation of opioid receptor trafficking and morphine tolerance by receptor oligomerization.
Journal: Cell20020125
Title: Relationship between rate and extent of G protein activation: comparison between full and partial opioid agonists.
Journal: The Journal of pharmacology and experimental therapeutics20020101
Title: Morphine tolerance in spinal cord is due to interaction between mu- and delta-receptors.
Journal: The Journal of pharmacology and experimental therapeutics20020101
Title: Neuroanatomical localization of receptor-activated G proteins in brain.
Journal: Methods in enzymology20020101
Title: Activation of mu-opioid receptors in rat ventrolateral medulla selectively blocks baroreceptor reflexes while activation of delta opioid receptors blocks somato-sympathetic reflexes.
Journal: Neuroscience20020101
Title: Mu and Delta opioid receptors activate the same G proteins in human neuroblastoma SH-SY5Y cells.
Journal: British journal of pharmacology20020101
Title: Mu and kappa opioid agonists modulate ventral tegmental area input to the ventral pallidum.
Journal: The European journal of neuroscience20020101
Title: [Dmt(1)]DALDA is highly selective and potent at mu opioid receptors, but is not cross-tolerant with systemic morphine.
Journal: Current medicinal chemistry20020101
Title: [Effect of opioid peptides on the repair regeneration of the bone tissue].
Journal: Arkhiv patologii20020101
Title: Endogenous morphine modulates acute thermonociception in mice.
Journal: Journal of neurochemistry20020101
Title: [Opiatergic modulation of cardiac resistance to arrhythmogenic exposures].
Journal: Patologicheskaia fiziologiia i eksperimental'naia terapiia20020101
Title: Implications of phosphoinositide 3-kinase in the mu- and delta-opioid receptor-mediated supraspinal antinociception in the mouse.
Journal: Neuroscience20020101
Title: Endomorphin-2 inhibits GABAergic inputs to cardiac parasympathetic neurons in the nucleus ambiguus.
Journal: Neuroscience20020101
Title: Expression of calcitonin gene-related peptide, substance P and protein kinase C in cultured dorsal root ganglion neurons following chronic exposure to mu, delta and kappa opiates.
Journal: Neuroscience20020101
Title: Antagonistic property of buprenorphine for putative epsilon-opioid receptor-mediated G-protein activation by beta-endorphin in pons/medulla of the mu-opioid receptor knockout mouse.
Journal: Neuroscience20020101
Title: [Effect of opioid peptides on proliferation and differentiation of skeletogenic cells of rabbit bone marrow in vitro].
Journal: Tsitologiia20020101
Title: Up-regulation of RGS4 mRNA by opioid receptor agonists in PC12 cells expressing cloned mu- or kappa-opioid receptors.
Journal: European journal of pharmacology20011214
Title: Excitatory amino acid receptor subtype agonists induce feeding in the nucleus accumbens shell in rats: opioid antagonist actions and interactions with mu-opioid agonists.
Journal: Brain research20011207
Title: Role of extracellular signal-regulated kinases in opioid-induced adenylyl cyclase superactivation in human embryonic kidney 293 cells.
Journal: Neuroscience letters20011204
Title: Studies on the antinociceptive effect of [Nphe1]nociceptin(1-13)NH2 in mice.
Journal: Neuroscience letters20011204
Title: Colocalization of mu-opioid receptors and activated G-proteins in rat cingulate cortex.
Journal: The Journal of pharmacology and experimental therapeutics20011201
Title: Acute antinociceptive tolerance and asymmetric cross-tolerance between endomorphin-1 and endomorphin-2 given intracerebroventricularly in the mouse.
Journal: The Journal of pharmacology and experimental therapeutics20011201
Title: MDR1 P-glycoprotein transports endogenous opioid peptides.
Journal: Peptides20011201
Title: Effects of a kappa-receptor agonist U-50488 on bulbar respiratory neurons and its antagonistic action against the mu receptor-induced respiratory depression in decerebrate cats.
Journal: Japanese journal of pharmacology20011201
Title: Role of protein kinase C in opioid modulation of glycine-gated Cl(-) current in rat periaqueductal gray neuron.
Journal: European journal of pharmacology20011116
Title: Morphine acutely and persistently attenuates nonvesicular GABA release in rat nucleus accumbens.
Journal: Synapse (New York, N.Y.)20011101
Title: Discriminative disulfide-bonding affinity labeling of opioid receptor subtypes.
Journal: Journal of biochemical and biophysical methods20011030
Title: Dexamethasone modulates hypotension induced by opioids in anaesthetised rats.
Journal: European journal of pharmacology20011026
Title: Antagonizing effect of protein kinase C activation on the mu-opioid agonist-induced inhibition of high voltage-activated calcium current in rat periaqueductal gray neuron.
Journal: Brain research20011019
Title: Acute ethanol administration differentially modulates mu opioid receptors in the rat meso-accumbens and mesocortical pathways.
Journal: Brain research. Molecular brain research20011019
Title: Parallel nociceptive reflex pathways with negative and positive feedback functions to foot extensors in the cat.
Journal: The Journal of physiology20011015
Title: Constitutively active mu-opioid receptors inhibit adenylyl cyclase activity in intact cells and activate G-proteins differently than the agonist [D-Ala2,N-MePhe4,Gly-ol5]enkephalin.
Journal: The Journal of biological chemistry20011012
Title: Differential in vivo internalization of MOR-1 and MOR-1C by morphine.
Journal: Neuroreport20011008
Title: Nociceptin inhibits calcium channel currents in a subpopulation of small nociceptive trigeminal ganglion neurons in mouse.
Journal: The Journal of physiology20011001
Title: Synergistic mu-opioid and 5-HT1A presynaptic inhibition of GABA release in rat periaqueductal gray neurons.
Journal: Neuropharmacology20011001
Title: The role of the hydrophilic Asn230 residue of the mu-opioid receptor in the potency of various opioid agonists.
Journal: British journal of pharmacology20011001
Title: New mu-opioid receptor agonists with piperazine moiety.
Journal: Chemical & pharmaceutical bulletin20011001
Title: Up-regulation of spinal mu-opioid receptor function to activate G-protein by chronic naloxone treatment.
Journal: Brain research20010921
Title: Differential antinociceptive effects induced by intrathecally administered endomorphin-1 and endomorphin-2 in the mouse.
Journal: European journal of pharmacology20010921
Title: Resensitization of blood pressure response to mu-opioid peptide agonists after acute desensitization.
Journal: Anesthesia and analgesia20010901
Title: Neurotrophin-3 modulates noradrenergic neuron function and opiate withdrawal.
Journal: Molecular psychiatry20010901
Title: Opioid action on respiratory neuron activity of the isolated respiratory network in newborn rats.
Journal: Anesthesiology20010901
Title: Gi- and Gs-coupled receptors up-regulate the cAMP cascade to modulate HCN2, but not HCN1 pacemaker channels.
Journal: Pflugers Archiv : European journal of physiology20010901
Title: Opioid effects on glucose and eicosanoid metabolism in isolated uterus of ovariectomized and non-ovariectomized restricted diet rats.
Journal: Prostaglandins, leukotrienes, and essential fatty acids20010901
Title: Binding of Sp1/Sp3 to the proximal promoter of the hMOR gene is enhanced by DAMGO.
Journal: Gene20010822
Title: C-terminal splice variants of the mouse mu-opioid receptor differ in morphine-induced internalization and receptor resensitization.
Journal: The Journal of biological chemistry20010817
Title: The kappa-opioid antagonist GNTI reduces U50,488-, DAMGO-, and deprivation-induced feeding, but not butorphanol- and neuropeptide Y-induced feeding in rats.
Journal: Brain research20010803
Title: Progesterone blockade of estrogen activation of mu-opioid receptors regulates reproductive behavior.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20010801
Title: Impaired inhibitory G-protein function contributes to increased calcium currents in rats with diabetic neuropathy.
Journal: Journal of neurophysiology20010801
Title: Cyclic AMP imaging in neurones in brain slice preparations.
Journal: Journal of neuroscience methods20010730
Title: Major difference in the expression of delta- and mu-opioid receptors between turtle and rat brain.
Journal: The Journal of comparative neurology20010723
Title: Quantitative autoradiographic mapping of the ORL1, mu-, delta- and kappa-receptors in the brains of knockout mice lacking the ORL1 receptor gene.
Journal: Brain research20010706
Title: gamma-Aminobutyric acid receptor subtype antagonists differentially alter opioid-induced feeding in the shell region of the nucleus accumbens in rats.
Journal: Brain research20010706
Title: L-type and T-type calcium channel blockade potentiate the analgesic effects of morphine and selective mu opioid agonist, but not to selective delta and kappa agonist at the level of the spinal cord in mice.
Journal: Pain20010701
Title: In vivo pharmacokinetics of selective mu-opioid peptide agonists.
Journal: The Journal of pharmacology and experimental therapeutics20010701
Title: Stimulation of guanosine-5'-o-(3-[35S]thio)triphosphate binding in digitonin-permeabilized C6 rat glioma cells: evidence for an organized association of mu-opioid receptors and G protein.
Journal: The Journal of pharmacology and experimental therapeutics20010701
Title: Blockade of opioid receptors in rostral ventral medulla prevents antihyperalgesia produced by transcutaneous electrical nerve stimulation (TENS).
Journal: The Journal of pharmacology and experimental therapeutics20010701
Title: Chronic exposure to mu-opioid agonists produces constitutive activation of mu-opioid receptors in direct proportion to the efficacy of the agonist used for pretreatment.
Journal: Molecular pharmacology20010701
Title: Functional expression and characterization of a voltage-gated CaV1.3 (alpha1D) calcium channel subunit from an insulin-secreting cell line.
Journal: Molecular endocrinology (Baltimore, Md.)20010701
Title: Role of opioid receptors in neurogenic dural vasodilation and sensitization of trigeminal neurones in anaesthetized rats.
Journal: British journal of pharmacology20010701
Title: SoRI 9409, a non-peptide opioid mu receptor agonist/delta receptor antagonist, fails to stimulate [35S]-GTP-gamma-S binding at cloned opioid receptors.
Journal: Brain research bulletin20010701
Title: Substance P and neurokinin A mediate sensory synaptic transmission in young rat dorsal horn neurons.
Journal: Brain research bulletin20010701
Title: Effect of intravenous injection of DAGO on neuronal activity in bulbar cardiovascular center.
Journal: Bulletin of experimental biology and medicine20010701
Title: Endomorphin-1: induction of motor behavior and lack of receptor desensitization.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20010615
Title: In vitro inhibitory effects of J-113397 on nociceptin/orphanin FQ-stimulated.
Journal: Neuroreport20010613
Title: Novel quantitative reverse-transcribed polymerase chain reaction of mu opioid receptor mRNA level.
Journal: Brain research. Brain research protocols20010601
Title: Involvement of spinal protein kinase Cgamma in the attenuation of opioid mu-receptor-mediated G-protein activation after chronic intrathecal administration of [D-Ala2,N-MePhe4,Gly-Ol(5)]enkephalin.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20010601
Title: Supraspinal delta- and mu-opioid receptors mediate gastric mucosal protection in the rat.
Journal: The Journal of pharmacology and experimental therapeutics20010601
Title: Inhibition of calcium channels by opioid- and adenosine-receptor agonists in neurons of the nucleus accumbens.
Journal: British journal of pharmacology20010601
Title: Receptor constants for endomorphin-1 and endomorphin-1-ol indicate differences in efficacy and receptor occupancy.
Journal: European journal of pharmacology20010601
Title: Differential antagonism by naloxone benzoylhydrazone of the activation of inward rectifying K+ channels by nociceptin and a mu-opioid in rat periaqueductal grey slices.
Journal: Naunyn-Schmiedeberg's archives of pharmacology20010601
Title: Functional and anatomical localization of mu opioid receptors in the striatum, amygdala, and extended amygdala of the nonhuman primate.
Journal: The Journal of comparative neurology20010514
Title: Discrimination between peptide and non-peptide opioid agonists on the transcription of opioid receptors in two cell lines.
Journal: Life sciences20010504
Title: In vivo pharmacological characterization of SoRI 9409, a nonpeptidic opioid mu-agonist/delta-antagonist that produces limited antinociceptive tolerance and attenuates morphine physical dependence.
Journal: The Journal of pharmacology and experimental therapeutics20010501
Title: Protein kinase C-mediated inhibition of mu-opioid receptor internalization and its involvement in the development of acute tolerance to peripheral mu-agonist analgesia.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20010501
Title: Opioids suppress basal and nicotine-induced catecholamine secretion via a stabilizing effect on actin filaments.
Journal: Endocrinology20010501
Title: Respiratory function in adult mice lacking the mu-opioid receptor: role of delta-receptors.
Journal: The European journal of neuroscience20010501
Title: [The role of mu- and delta-opiate receptors in resistance of the myocardium to free radical damage].
Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova20010501
Title: [Effect of stimulation of mu-opiate receptors on contractility of the isolated heart in normal oxygenation and during ischemia-reperfusion].
Journal: Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova20010501
Title: Phosphorylation of Ser363, Thr370, and Ser375 residues within the carboxyl tail differentially regulates mu-opioid receptor internalization.
Journal: The Journal of biological chemistry20010420
Title: Agonist-induced mu opioid receptor phosphorylation and functional desensitization in rat thalamus.
Journal: Brain research20010420
Title: The activation of mu opioid receptors promotes a small modulation of calcium currents in rat pallidal neurons.
Journal: Brain research20010406
Title: Interaction of co-expressed mu- and delta-opioid receptors in transfected rat pituitary GH(3) cells.
Journal: Molecular pharmacology20010401
Title: Activity of mu- and delta-opioid agonists in vas deferens from mice deficient in MOR gene.
Journal: British journal of pharmacology20010401
Title: Contribution of endogenous enkephalins to the enhanced analgesic effects of supraspinal mu opioid receptor agonists after inflammatory injury.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience20010401
Title: Non-opioid actions of lamotrigine within the rat dorsal horn after inflammation and neuropathic nerve damage.
Journal: Neuroscience research20010401
Title: Direct autocrine inhibition and cAMP-dependent potentiation of single L-type Ca2+ channels in bovine chromaffin cells.
Journal: The Journal of physiology20010401
Title: G protein-coupled receptor kinase 2 mediates mu-opioid receptor desensitization in GABAergic neurons of the nucleus raphe magnus.
Journal: Journal of neurochemistry20010401
Title: Effect of centrally administered opioid receptor agonists on CSF and plasma oxytocin concentrations in dogs.
Journal: American journal of veterinary research20010401
Title: Quantitative autoradiography of mu-opioid receptors in the CNS of high-alcohol-drinking (HAD) and low-alcohol-drinking (LAD) rats.
Journal: Alcoholism, clinical and experimental research20010401
Title: Stimulation of mu and delta-Opiate Receptors and Tolerance of Isolated Heart to Oxidative Stress: the Role of NO-Synthase.
Journal: Biochemistry. Biokhimiia20010401
Title: The metabolic evidence of synergistic interaction between DAMGO and DPDPE on undifferentiated SH-SY5Y cells.
Journal: Neuroreport20010326
Title: Factors influencing agonist potency and selectivity for the opioid delta receptor are revealed in structure-activity relationship studies of the 4-[(N-substituted-4-piperidinyl)arylamino]-N,N-diethylbenzamides.
Journal: Journal of medicinal chemistry20010315
Title: Mu opioid receptor efficacy and potency of morphine-6-glucuronide in neonatal guinea pig brainstem membranes: comparison with transfected CHO cells.
Journal: Brain research bulletin20010315
Title: Selective inactivation of guanine-nucleotide-binding regulatory protein (G-protein) alpha and betagamma subunits by urea.
Journal: The Biochemical journal20010301
Title: Opioid-mediated facilitation of long-term depression in rat hippocampus.
Journal: The Journal of pharmacology and experimental therapeutics20010301
Title: Transport of opioids from the brain to the periphery by P-glycoprotein: peripheral actions of central drugs.
Journal: Nature neuroscience20010301
Title: Expression of functional mu-opioid receptors during T cell development.
Journal: Journal of neuroimmunology20010301
Title: Neutrophil neutral endopeptidase variation and its regulation by opioid peptides.
Journal: International immunopharmacology20010301
Title: Threonine 180 is required for G-protein-coupled receptor kinase 3- and beta-arrestin 2-mediated desensitization of the mu-opioid receptor in Xenopus oocytes.
Journal: The Journal of biological chemistry20010216
Title: A single nucleotide polymorphic mutation in the human mu-opioid receptor severely impairs receptor signaling.
Journal: The Journal of biological chemistry20010202
Title: Pharmacological effects of naltriben as a ligand for opioid mu and kappa receptors in rat cerebral cortex.
Journal: Life sciences20010202
Title: Mu opiates inhibit long-term potentiation induction in the spinal cord slice.
Journal: Journal of neurophysiology20010201
Title: G protein activation in rat ponto-mesencephalic nuclei is enhanced by combined treatment with a mu opioid and an adenosine A1 receptor agonist.
Journal: Sleep20010201
Title: Interference of biocytin with opioid-evoked hyperpolarization and membrane properties of rat spinal substantia gelatinosa neurons.
Journal: Neuroscience letters20010112
Title: Cyclic AMP regulates the calcium transients released from IP(3)-sensitive stores by activation of rat kappa-opioid receptors expressed in CHO cells.
Journal: Cell calcium20010101
Title: Direct actions of cannabinoids on synaptic transmission in the nucleus accumbens: a comparison with opioids.
Journal: Journal of neurophysiology20010101
Title: Dexamethasone blocking effects on mu- and delta-opioid-induced seizures involves kappa-opioid activity in the rabbit.
Journal: Neuropsychobiology20010101
Title: Involvement of pallidothalamic circuitry in working memory.
Journal: Neuroscience20010101
Title: Characterization of kappa and delta opioid receptors in isolated organs by using type/subtype selective agonists and antagonists.
Journal: Medical science monitor : international medical journal of experimental and clinical research20010101
Title: Nicotine withdrawal hyperalgesia and opioid-mediated analgesia depend on nicotine receptors in nucleus accumbens.
Journal: Neuroscience20010101
Title: Activation of central opioid receptors may induce gastric mucosal defence in the rat.
Journal: Journal of physiology, Paris20010101
Title: Chronic in utero morphine exposure alters mu-agonist-stimulated [35S]-GTPgammaS binding in neonatal and juvenile guinea pig brainstem regions associated with breathing control.
Journal: Neurotoxicology and teratology20010101
Title: Opiates promote T cell apoptosis through JNK and caspase pathway.
Journal: Advances in experimental medicine and biology20010101
Title: Crosstalk between chemokine and opioid receptors results in downmodulation of cell migration.
Journal: Advances in experimental medicine and biology20010101
Title: [Participation of K(ATP)-channels in cardioprotective effect of mu-opioid receptor agonists in acute ischemia and reperfusion of the isolated heart].
Journal: Eksperimental'naia i klinicheskaia farmakologiia20010101
Title: [State of the opioid system in rats with different sensitivity to ethanol].
Journal: Ukrains'kyi biokhimichnyi zhurnal (1999 )20010101
Title: Autoradiographic evidence that prolonged withdrawal from intermittent cocaine reduces mu-opioid receptor expression in limbic regions of the rat brain.
Journal: Synapse (New York, N.Y.)20000915
Title: Differential cardiorespiratory effects of endomorphin 1, endomorphin 2, DAMGO, and morphine.
Journal: American journal of respiratory and critical care medicine20000901
Title: Differential effects of antisense oligodeoxynucleotides directed against g(zalpha) and g(oalpha) on antinociception produced by spinal opioid and alpha(2) adrenergic receptor agonists.
Journal: Pain20000801
Title: Synaptic actions of neuropeptide FF in the rat parabrachial nucleus: interactions with opioid receptors.
Journal: Journal of neurophysiology20000801
Title: 5'-Guanidinonaltrindole, a highly selective and potent kappa-opioid receptor antagonist.
Journal: European journal of pharmacology20000512
Title: G protein activation by endomorphins in the mouse periaqueductal gray matter.
Journal: Journal of biomedical science20000101
Title: Morphine inhibits human microglial cell production of, and migration towards, RANTES.
Journal: Journal of psychopharmacology (Oxford, England)20000101
Title: Long-lasting antinociceptive effect of DAMGO chloromethyl ketone in rats.
Journal: Peptides19991101
Title: Morphine promotes apoptosis in Jurkat cells.
Journal: Journal of leukocyte biology19991001
Title: Opioid modulation of calcium current in cultured sensory neurons: mu-modulation of baroreceptor input.
Journal: The American journal of physiology19990801
Title: Mu- and delta-opioid receptor agonists inhibit DARPP-32 phosphorylation in distinct populations of striatal projection neurons.
Journal: The European journal of neuroscience19990601
Title: [3H]ethylketocyclazocine binding to brain opioid receptor subtypes in alcohol-preferring AA and alcohol-avoiding ANA rats.
Journal: Alcohol (Fayetteville, N.Y.)19990501
Title: Time-dependent differences of repeated administration with Delta9-tetrahydrocannabinol in proenkephalin and cannabinoid receptor gene expression and G-protein activation by mu-opioid and CB1-cannabinoid receptors in the caudate-putamen.
Journal: Brain research. Molecular brain research19990406
Title: Spinal analgesic action of endomorphins in acute, inflammatory and neuropathic pain in rats.
Journal: European journal of pharmacology19990219
Title: 5-HT2A receptor or alpha1-adrenoceptor activation induces excitatory postsynaptic currents in layer V pyramidal cells of the medial prefrontal cortex.
Journal: European journal of pharmacology19990219
Title: Endomorphins fully activate a cloned human mu opioid receptor.
Journal: FEBS letters19981113
Title: Dopamine depletion reorganizes projections from the nucleus accumbens and ventral pallidum that mediate opioid-induced motor activity.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19981001
Title: Apparent thermodynamic parameters of ligand binding to the cloned rat mu-opioid receptor.
Journal: European journal of pharmacology19980807
Title: Delta opioid receptor enhancement of mu opioid receptor-induced antinociception in spinal cord.
Journal: The Journal of pharmacology and experimental therapeutics19980601
Title: Glycine and GABAA receptor-mediated synaptic transmission in rat substantia gelatinosa: inhibition by mu-opioid and GABAB agonists.
Journal: The Journal of physiology19980301
Title: Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
Journal: NIDA research monograph19980301
Title: Endogenous opioid peptides acting at mu-opioid receptors in the dorsal horn contribute to midbrain modulation of spinal nociceptive neurons.
Journal: Journal of neurophysiology19980201
Title: Differential effects of intrathecally administered delta and mu opioid receptor agonists on formalin-evoked nociception and on the expression of Fos-like immunoreactivity in the spinal cord of the rat.
Journal: The Journal of pharmacology and experimental therapeutics19980101
Title: Kappa1- and kappa2-opioid receptors mediating presynaptic inhibition of dopamine and acetylcholine release in rat neostriatum.
Journal: British journal of pharmacology19971001
Title: Kappa-opioid receptor activation modulates Ca2+ currents and secretion in isolated neuroendocrine nerve terminals.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19970901
Title: Activation of the cloned human kappa opioid receptor by agonists enhances [35S]GTPgammaS binding to membranes: determination of potencies and efficacies of ligands.
Journal: The Journal of pharmacology and experimental therapeutics19970801
Title: Differential effects of omega-conotoxin GVIA, nimodipine, calmidazolium and KN-62 injected intrathecally on the antinociception induced by beta-endorphin, morphine and [D-Ala2,N-MePhe4,Gly-ol5]-enkephalin administered intracerebroventricularly in the mouse.
Journal: The Journal of pharmacology and experimental therapeutics19970801
Title: Dissociation of tolerance and dependence for opioid peripheral antinociception in rats.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19970515
Title: A potent and selective endogenous agonist for the mu-opiate receptor.
Journal: Nature19970403
Title: Inhibition of swine microglial cell phagocytosis of Cryptococcus neoformans by femtomolar concentrations of morphine.
Journal: Biochemical pharmacology19970321
Title: Multiple receptors involved in peripheral alpha 2, mu, and A1 antinociception, tolerance, and withdrawal.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19970115
Title: Opioid peptides: simultaneous delta agonism and mu antagonism in somatostatin analogues.
Journal: Peptides19970101
Title: Competitive and non-competitive NMDA antagonists block the development of antinociceptive tolerance to morphine, but not to selective mu or delta opioid agonists in mice.
Journal: Pain19961201
Title: A single residue, Lys108, of the delta-opioid receptor prevents the mu-opioid-selective ligand [D-Ala2,N-MePhe4,Gly-ol5]enkephalin from binding to the delta-opioid receptor.
Journal: Molecular pharmacology19961101
Title: Central effects of opioid agonists and naloxone on blood pressure and heart rate in normotensive and hypertensive rats.
Journal: General pharmacology19961001
Title: The mu-opioid receptor antagonist D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2 (CTOP) [but not D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH2 (CTAP)] produces a nonopioid receptor-mediated increase in K+ conductance of rat locus ceruleus neurons.
Journal: Molecular pharmacology19960901
Title: Vincristine hyperalgesia in the rat: a model of painful vincristine neuropathy in humans.
Journal: Neuroscience19960701
Title: Differential desensitization of mu- and delta- opioid receptors in selected neural pathways following chronic morphine treatment.
Journal: British journal of pharmacology19960101
Title: Serotonin and norepinephrine uptake inhibiting activity of centrally acting analgesics: structural determinants and role in antinociception.
Journal: The Journal of pharmacology and experimental therapeutics19950901
Title: Low-dose effect of ethanol on locomotor activity induced by activation of the mesolimbic system.
Journal: Alcoholism, clinical and experimental research19950601
Title: Electrophysiological demonstration of mu, delta and kappa opioid receptors in the ventral pallidum.
Journal: The Journal of pharmacology and experimental therapeutics19950301
Title: Opioid effects on spinal [3H]5-hydroxytryptamine release are not related to their antinociceptive action.
Journal: European journal of pharmacology19950105
Title: Acute tolerance to the excitatory effects of opioids in the rat hippocampus.
Journal: Journal of neuroscience research19950101
Title: Decreased spinal morphine/clonidine antinociceptive synergism in morphine-tolerant mice.
Journal: Life sciences19950101
Title: Comparison of prostaglandin E1- and prostaglandin E2-induced hyperalgesia in the rat.
Journal: Neuroscience19940901
Title: Differential regulation of mu and delta opiate receptors by morphine, selective agonists and antagonists and differentiating agents in SH-SY5Y human neuroblastoma cells.
Journal: The Journal of pharmacology and experimental therapeutics19940901
Title: Evidence for a central long-lasting antinociceptive effect of vapreotide, an analog of somatostatin, involving an opioidergic mechanism.
Journal: The Journal of pharmacology and experimental therapeutics19940401
Title: Behavioral and neurochemical studies of opioid effects in the pedunculopontine nucleus and mediodorsal thalamus.
Journal: The Journal of pharmacology and experimental therapeutics19940401
Title: Blockade of neurotensin-induced motor activity by inhibition of protein kinase.
Journal: Psychopharmacology19940201
Title: Pharmacological characterization of the cloned kappa-, delta-, and mu-opioid receptors.
Journal: Molecular pharmacology19940201
Title: Cloning and pharmacological characterization of a rat kappa opioid receptor.
Journal: Proceedings of the National Academy of Sciences of the United States of America19931101
Title: Facilitatory modulation of mesolimbic dopamine neuronal activity by a mu-opioid agonist and nicotine as examined with in vivo microdialysis.
Journal: Brain research19931008
Title: Differential regulation of adenylyl cyclase activity by mu and delta opioids in rat caudate putamen and nucleus accumbens.
Journal: The Journal of pharmacology and experimental therapeutics19931001
Title: Discovery of a novel class of neuromedin B receptor antagonists, substituted somatostatin analogues.
Journal: Molecular pharmacology19931001
Title: Behavioral effects of the mu-opioid peptide agonists DAMGO, DALDA, and PL017 on locomotor activities.
Journal: Pharmacology, biochemistry, and behavior19931001
Title: Differential involvement of ventral tegmental mu, delta and kappa opioid receptors in modulation of basal mesolimbic dopamine release: in vivo microdialysis studies.
Journal: The Journal of pharmacology and experimental therapeutics19930901
Title: Kinetic parameters of antagonism by the delta opioid receptor selective peptide antagonist Boc-Tyr-Pro-Gly-Phe-Leu-Thr against selective and non-selective agonists in the mouse vas deferens.
Journal: Neuropeptides19930801
Title: Investigation of the structural parameters involved in the delta-opioid selectivity of several families of opioid peptides.
Journal: International journal of peptide and protein research19930601
Title: Go mediates the coupling of the mu opioid receptor to adenylyl cyclase in cloned neural cells and brain.
Journal: Proceedings of the National Academy of Sciences of the United States of America19930501
Title: In vivo modulation of gastrointestinal motor activity by Met-enkephalin, morphine and enkephalin analogs in chickens.
Journal: Regulatory peptides19930305
Title: Dexamethasone prevents epileptiform activity induced by morphine in in vivo and in vitro experiments.
Journal: The Journal of pharmacology and experimental therapeutics19921101
Title: Conformationally restricted deltorphin analogues.
Journal: Journal of medicinal chemistry19921016
Title: Opioid receptor antagonists discriminate between presynaptic mu and delta receptors and the adenylate cyclase-coupled opioid receptor complex in the brain.
Journal: The Journal of pharmacology and experimental therapeutics19921001
Title: Evidence for the implication of phosphoinositol signal transduction in mu-opioid inhibition of DNA synthesis.
Journal: Journal of neurochemistry19920901
Title: Modulation of peristalsis in the guinea-pig isolated small intestine by exogenous and endogenous opioids.
Journal: British journal of pharmacology19920801
Title: Spinal interactions between opioid and noradrenergic agonists in mice: multiplicativity involves delta and alpha-2 receptors.
Journal: The Journal of pharmacology and experimental therapeutics19920701
Title: Limbic thalamus in rabbit: architecture, projections to cingulate cortex and distribution of muscarinic acetylcholine, GABAA, and opioid receptors.
Journal: The Journal of comparative neurology19920508
Title: The calcium antagonist diltiazem has antiarrhythmic effects which are mediated in the brain through endogenous opioids.
Journal: Neuropharmacology19920501
Title: Feedback inhibition of met-enkephalin release from the rat spinal cord in vivo.
Journal: Synapse (New York, N.Y.)19920501
Title: Differential development of beta-endorphin and mu opioid binding sites in mouse brain.
Journal: Brain research. Developmental brain research19920320
Title: Opioid control of the in vitro release of cholecystokinin-like material from the rat substantia nigra.
Journal: Journal of neurochemistry19920301
Title: Inhibition of cholinergic neurotransmission in human airways by opioids.
Journal: Journal of applied physiology (Bethesda, Md. : 1985)19920301
Title: Transient expression of opioid receptors in defined regions of developing brain: are embryonic receptors selective?
Journal: Journal of neurochemistry19911201
Title: Neurons in the rat arcuate nucleus are hyperpolarized by GABAB and mu-opioid receptor agonists: evidence for convergence at a ligand-gated potassium conductance.
Journal: Neuroendocrinology19911201
Title: Cyclic somatostatin analogues as potent antagonists at mu-, but not delta- and kappa-opioid receptors mediating presynaptic inhibition of neurotransmitter release in the brain.
Journal: European journal of pharmacology19911119
Title: Binding to opioid receptors of enkephalin derivatives taking alpha-helical conformation and its dimer.
Journal: International journal of peptide and protein research19911001
Title: Characterization and distribution of [3H]ohmefentanyl binding sites in the human brain.
Journal: Synapse (New York, N.Y.)19910701
Title: Kappa- and delta-opioids block sympathetically dependent hyperalgesia.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19910401
Title: A monoclonal anti-idiotypic antibody to mu and delta opioid receptors.
Journal: Brain research. Molecular brain research19910301
Title: Dopaminergic involvement in locomotion elicited from the ventral pallidum/substantia innominata.
Journal: Brain research19910222
Title: Pharmacological profile of various kappa-agonists at kappa-, mu- and delta-opioid receptors mediating presynaptic inhibition of neurotransmitter release in the rat brain.
Journal: British journal of pharmacology19910201
Title: Different profile of electrocortical power spectrum changes after micro-infusion into the locus coeruleus of selective agonists at various opioid receptor subtypes in rats.
Journal: British journal of pharmacology19901101
Title: The effects of opioid peptides on dopamine release in the nucleus accumbens: an in vivo microdialysis study.
Journal: Journal of neurochemistry19901101
Title: Effect of acute and daily neurotensin and enkephalin treatments on extracellular dopamine in the nucleus accumbens.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19900901
Title: Opioids hyperpolarize beta-endorphin neurons via mu-receptor activation of a potassium conductance.
Journal: Neuroendocrinology19900901
Title: Modulation of histamine release in the rat brain by kappa-opioid receptors.
Journal: Journal of neurochemistry19900701
Title: Characterisation and visualisation of [3H]dermorphin binding to mu opioid receptors in the rat brain. Combined high selectivity and affinity in a natural peptide agonist for the morphine (mu) receptor.
Journal: European journal of biochemistry19900520
Title: Modulation of A10 dopamine neurons by gamma-aminobutyric acid agonists.
Journal: The Journal of pharmacology and experimental therapeutics19900501
Title: Modulation of mu, delta and kappa opioid receptors in rat brain by metal ions and histidine.
Journal: Neuropharmacology19900501
Title: Opioids act at mu-receptors to hyperpolarize arcuate neurons via an inwardly rectifying potassium conductance.
Journal: Brain research19900409
Title: Cross-linking of human [125I]beta-endorphin to opioid receptors in rat striatal membranes: biochemical evidence for the existence of a mu/delta opioid receptor complex.
Journal: The Journal of pharmacology and experimental therapeutics19900401
Title: Enkephalinergic and GABAergic modulation of motor activity in the ventral pallidum.
Journal: The Journal of pharmacology and experimental therapeutics19900301
Title: Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
Journal: Neuroscience19900101
Title: Synthesis, biochemical and pharmacological properties of BUBUC, a highly selective and systemically active agonist for in vivo studies of delta-opioid receptors.
Journal: Peptides19900101
Title: Centrally administered opioid peptides stimulate saccharin intake in nondeprived rats.
Journal: Pharmacology, biochemistry, and behavior19890801
Title: Guanine nucleotide regulation of [125I]beta-endorphin binding to NG108-15 and SK-N-SH cell membranes: specific cation requirements.
Journal: Brain research19890724
Title: Dermenkephalin (Tyr-D-Met-Phe-His-Leu-Met-Asp-NH2): a potent and fully specific agonist for the delta opioid receptor.
Journal: Molecular pharmacology19890601
Title: Activation of mu opioid receptors in the nucleus raphe dorsalis blocks apomorphine-induced aggression in rats: serotonin appears not to be involved.
Journal: Brain research19890529
Title: Effects of pentazocine and other opioids on the potassium-evoked release of [3H]noradrenaline from guinea pig cortical slices.
Journal: European journal of pharmacology19890502
Title: Opioid inhibition of spontaneously active neurons of the rat arcuate nucleus in vitro.
Journal: Brain research bulletin19890501
Title: Single potassium channels opened by opioids in rat locus ceruleus neurons.
Journal: Proceedings of the National Academy of Sciences of the United States of America19890501
Title: Paradoxical analgesia produced by low doses of the opiate-antagonist naloxone is mediated by interaction at a site with characteristics of the delta opioid receptor.
Journal: The Journal of pharmacology and experimental therapeutics19890401
Title: Two cell types in rat substantia nigra zona compacta distinguished by membrane properties and the actions of dopamine and opioids.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience19890401
Title: Peripheral opioid receptors mediating antinociception in inflammation. Evidence for involvement of mu, delta and kappa receptors.
Journal: The Journal of pharmacology and experimental therapeutics19890301
Title: Selective opioid antagonist effects on opioid-induced inhibition of release of norepinephrine in guinea pig cortex.
Journal: Neuropharmacology19890201
Title: Mu and delta opioid receptors inhibit serotonin release in rat hippocampus.
Journal: The Journal of pharmacology and experimental therapeutics19890101
Title: Involvement of the mu-opiate receptor in peripheral analgesia.
Journal: Neuroscience19890101
Title: Selectivity of various opioid peptides towards delta-, kappa; and mu-opioid receptors mediating presynaptic inhibition of neurotransmitter release in the brain.
Journal: Neuropeptides19890101
Title: Action of naloxone on myenteric neurons removed from morphine-treated guinea pigs.
Journal: The Journal of pharmacology and experimental therapeutics19881201
Title: Selective tolerance at mu and kappa opioid receptors modulating norepinephrine release in guinea pig cortex.
Journal: The Journal of pharmacology and experimental therapeutics19881201
Title: Identification of endogenous opioid receptor components in rat brain using a monoclonal antibody.
Journal: Molecular pharmacology19881101
Title: Agonists at mu-opioid, M2-muscarinic and GABAB-receptors increase the same potassium conductance in rat lateral parabrachial neurones.
Journal: British journal of pharmacology19881101
Title: Development of conformationally constrained linear peptides exhibiting a high affinity and pronounced selectivity for delta opioid receptors.
Journal: Journal of medicinal chemistry19881001
Title: Inhibition of exocrine pancreatic secretion by opiates is mediated by suppression of cholinergic transmission: characterization of receptor subtypes.
Journal: The Journal of pharmacology and experimental therapeutics19880701
Title: Effects of chronic morphine exposure on opioid inhibition of adenylyl cyclase in 7315c cell membranes: a useful model for the study of tolerance at mu opioid receptors.
Journal: Molecular pharmacology19880501
Title: Comparative binding of mu and delta selective ligands in whole brain and pons/medulla homogenates from rat: affinity profiles of fentanyl derivatives.
Journal: Neuropharmacology19880401
Title: [3H][D-Ser2(O-tert-butyl),Leu5]enkephalyl-Thr6 and [D-Ser2(O-tert-butyl),Leu5]enkephalyl-Thr6(O-tert-butyl). Two new enkephalin analogs with both a good selectivity and a high affinity toward delta-opioid binding sites.
Journal: The Journal of biological chemistry19880325
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