Catalog No.:AA008TDW

1089283-49-7 | GSK1904529A

Name: Name:GSK1904529A
Brand: AABLOCKS
SKU: AA008TDW
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1mg

≥95%

in stock

$46.00 $32.00

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5mg

≥95%

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$166.00 $116.00

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10mg

≥95%

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$306.00 $214.00

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25mg

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$652.00 $456.00

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500mg

99% (HPLC)

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$11,355.00 $7,949.00

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1000mg

99% (HPLC)

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$18,133.00 $12,693.00

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Technical Information
Properties
Upstream Synthesis Route
Literature
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Technical Information
Properties
Upstream Synthesis Route
Literature

Technical Information

Catalog Number:

AA008TDW

Chemical Name:

GSK1904529A

CAS Number:

1089283-49-7

Molecular Formula:

C44H47F2N9O5S

Molecular Weight:

851.9631

MDL Number:

MFCD17010271

SMILES:

COc1cc(N2CCC(CC2)N2CCN(CC2)S(=O)(=O)C)c(cc1Nc1nccc(n1)c1c(nc2n1cccc2)c1ccc(c(c1)C(=O)Nc1c(F)cccc1F)OC)CC

Properties

Computed Properties

Complexity:

1530

Covalently-Bonded Unit Count:

Heavy Atom Count:

Hydrogen Bond Acceptor Count:

Hydrogen Bond Donor Count:

Rotatable Bond Count:

XLogP3:

6.8

Upstream Synthesis Route

1089282-91-6

1089278-50-1

1089283-49-7

[1]BioorganicandMedicinalChemistryLetters,2009,vol.19,#3,p.1004-1008

Literature

Title: Identification of potent Yes1 kinase inhibitors using a library screening approach.

Journal: Bioorganic & medicinal chemistry letters 20130801

Title: Antitumor activity of GSK1904529A, a small-molecule inhibitor of the insulin-like growth factor-I receptor tyrosine kinase.

Journal: Clinical cancer research : an official journal of the American Association for Cancer Research 20090501

Title: Discovery and optimization of imidazo[1,2-a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R).

Journal: Bioorganic & medicinal chemistry letters 20090201

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SDS