Title: Pharmacokinetics, tolerability, and preliminary efficacy of paquinimod (ABR-215757), a new quinoline-3-carboxamide derivative: studies in lupus-prone mice and a multicenter, randomized, double-blind, placebo-controlled, repeat-dose, dose-ranging study in patients with systemic lupus erythematosus.
Journal: Arthritis and rheumatism 20120501
Title: Specific effect of immunomodulatory quinoline-3-carboxamide ABR-215757 in GM-CSF stimulated bone marrow cell cultures: block of initiation of proliferation of Gr-1+ cells.
Journal: International immunopharmacology 20110801
Title: The impact of a new immunomodulator oxo-quinoline-3-carboxamide on the progression of experimental lupus.
Journal: International immunopharmacology 20041101
Title: Synthesis and biological evaluation of new 1,2-dihydro-4-hydroxy-2-oxo-3-quinolinecarboxamides for treatment of autoimmune disorders: structure-activity relationship.
Journal: Journal of medicinal chemistry 20040408
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