Title: Effects of corticotropin-releasing factor 1 receptor antagonism on the hypothalamic-pituitary-adrenal axis of rodents.
Journal: The Journal of pharmacology and experimental therapeutics 20120601
Title: Effects of corticotropin-releasing hormone receptor antagonists on the ethanol-induced increase of dynorphin A1-8 release in the rat central amygdala.
Journal: Alcohol (Fayetteville, N.Y.) 20111101
Title: Previous ethanol experience enhances synaptic plasticity of NMDA receptors in the ventral tegmental area.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20110406
Title: Exploring the binding site crevice of a family B G protein-coupled receptor, the type 1 corticotropin releasing factor receptor.
Journal: Molecular pharmacology 20101001
Title: Corticotropin-releasing factor receptors induce calcium mobilization through cross-talk with Gq-coupled receptors.
Journal: European journal of pharmacology 20100910
Title: Subtype-specific differences in corticotropin-releasing factor receptor complexes detected by fluorescence spectroscopy.
Journal: Molecular pharmacology 20091201
Title: Cardiovascular responses to microinjections of urocortins into the NTS: role of inotropic glutamate receptors.
Journal: American journal of physiology. Heart and circulatory physiology 20090601
Title: Alanine scanning mutagenesis of the second extracellular loop of type 1 corticotropin-releasing factor receptor revealed residues critical for peptide binding.
Journal: Molecular pharmacology 20090401
Title: Amygdaloid pERK1/2 in corticotropin-releasing hormone overexpressing mice under basal and acute stress conditions.
Journal: Neuroscience 20090317
Title: Residue 17 of sauvagine cross-links to the first transmembrane domain of corticotropin-releasing factor receptor 1 (CRFR1).
Journal: The Journal of biological chemistry 20081219
Title: Corticotropin-releasing factor modulates maternal separation-induced ultrasonic vocalization in rat pups via activation of CRF1 receptor.
Journal: Brain research 20081009
Title: Allosteric ligands for the corticotropin releasing factor type 1 receptor modulate conformational states involved in receptor activation.
Journal: Molecular pharmacology 20080501
Title: Achieving signalling selectivity of ligands for the corticotropin-releasing factor type 1 receptor by modifying the agonist's signalling domain.
Journal: British journal of pharmacology 20070701
Title: 3-(4-Chloro-2-morpholin-4-yl-thiazol-5-yl)-8-(1-ethylpropyl)-2,6-dimethyl-imidazo[1,2-b]pyridazine: a novel brain-penetrant, orally available corticotropin-releasing factor receptor 1 antagonist with efficacy in animal models of alcoholism.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20070307
Title: Corticotropin-releasing hormone skin signaling is receptor-mediated and is predominant in the sebaceous glands.
Journal: Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme 20070201
Title: Evidence that corticotropin-releasing factor receptor type 1 couples to Gs- and Gi-proteins through different conformations of its J-domain.
Journal: British journal of pharmacology 20061201
Title: A centrally acting, anxiolytic angiotensin II AT1 receptor antagonist prevents the isolation stress-induced decrease in cortical CRF1 receptor and benzodiazepine binding.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060601
Title: Peripheral injection of sauvagine prevents repeated colorectal distension-induced visceral pain in female rats.
Journal: Peptides 20050701
Title: Sauvagine analogs selective for corticotropin releasing factor 2 receptor: effect of substitutions at positions 35 and 39 on CRF2R selectivity.
Journal: Peptides 20050501
Title: Stress and central Urocortin increase anxiety-like behavior in the social interaction test via the CRF1 receptor.
Journal: European journal of pharmacology 20050221
Title: Discovery of corticotropin releasing factor 2 receptor selective sauvagine analogues for treatment of skeletal muscle atrophy.
Journal: Journal of medicinal chemistry 20050113
Title: Ethanol versus lipopolysaccharide-induced hypothermia: involvement of urocortin.
Journal: Neuroscience 20050101
Title: Internalization of the human CRF receptor 1 is independent of classical phosphorylation sites and of beta-arrestin 1 recruitment.
Journal: European journal of biochemistry 20041101
Title: Regulation of the coupling to different G proteins of rat corticotropin-releasing factor receptor type 1 in human embryonic kidney 293 cells.
Journal: The Journal of biological chemistry 20040910
Title: Binding differences of human and amphibian corticotropin-releasing factor type 1 (CRF(1)) receptors: identification of amino acids mediating high-affinity astressin binding and functional antagonism.
Journal: Regulatory peptides 20040515
Title: Ligand affinity for amino-terminal and juxtamembrane domains of the corticotropin releasing factor type I receptor: regulation by G-protein and nonpeptide antagonists.
Journal: Biochemistry 20040406
Title: Conformational states of the corticotropin releasing factor 1 (CRF1) receptor: detection, and pharmacological evaluation by peptide ligands.
Journal: Peptides 20031201
Title: Corticotropin-releasing factor (CRF) and related peptides confer neuroprotection via type 1 CRF receptors.
Journal: Neuropharmacology 20031001
Title: A novel water-soluble selective CRF1 receptor antagonist, NBI 35965, blunts stress-induced visceral hyperalgesia and colonic motor function in rats.
Journal: Brain research 20030919
Title: A soluble form of the first extracellular domain of mouse type 2beta corticotropin-releasing factor receptor reveals differential ligand specificity.
Journal: The Journal of biological chemistry 20030502
Title: Mechanism of corticotropin-releasing factor type I receptor regulation by nonpeptide antagonists.
Journal: Molecular pharmacology 20030301
Title: Development of a selective photoactivatable antagonist for corticotropin-releasing factor receptor, type 2 (CRF2).
Journal: European journal of biochemistry 20021101
Title: An artificial peptide with corticotropin-releasing factor receptor-2 (CRF-R2) selective properties: the role of primary structure in the induction of signal transduction pathways.
Journal: The journal of peptide research : official journal of the American Peptide Society 20021001
Title: Sauvagine regulates Ca2+ oscillations and electrical membrane activity of melanotrope cells of Xenopus laevis.
Journal: Journal of neuroendocrinology 20021001
Title: Sauvagine cross-links to the second extracellular loop of the corticotropin-releasing factor type 1 receptor.
Journal: The Journal of biological chemistry 20020906
Title: The highly selective CRF(2) receptor antagonist K41498 binds to presynaptic CRF(2) receptors in rat brain.
Journal: British journal of pharmacology 20020701
Title: N-glycosylation of CRF receptor type 1 is important for its ligand-specific interaction.
Journal: American journal of physiology. Endocrinology and metabolism 20011101
Title: Persistent corticotropin-releasing factor(1) receptor desensitization and downregulation in the human neuroblastoma cell line IMR-32.
Journal: Brain research. Molecular brain research 20010815
Title: An oxidation resistant radioligand for corticotropin-releasing factor receptors.
Journal: Peptides 20010701
Title: Homogeneous cell-based fluorescence polarization assay for the direct detection of cAMP.
Journal: Journal of biomolecular screening 20010401
Title: Amino acid composition and sequence analysis of sauvagine, a new active peptide from the skin of Phyllomedusa sauvagei.
Journal: International journal of peptide and protein research 19810801
Title: A Rühmann, et al. Design, synthesis and pharmacological characterization of new highly selective CRF(2) antagonists: development of 123I-K31440 as a potential SPECT ligand. Peptides. 2002 Mar;23(3):453-60.
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