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Title: Glucose-dependent growth arrest of leukemia cells by MCT1 inhibition: Feeding Warburg's sweet tooth and blocking acid export as an anticancer strategy.
Journal: Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie 20180201
Title: Regulation of Acetate Utilization by Monocarboxylate Transporter 1 (MCT1) in Hepatocellular Carcinoma (HCC).
Journal: Oncology research 20180119
Title: Roles of acid-extruding ion transporters in regulation of breast cancer cell growth in a 3-dimensional microenvironment.
Journal: Molecular cancer 20160101
Title: Effective impairment of myeloma cells and their progenitors by blockade of monocarboxylate transportation.
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Title: A Novel Monocarboxylate Transporter Inhibitor as a Potential Treatment Strategy for γ-Hydroxybutyric Acid Overdose.
Journal: Pharmaceutical research 20150601
Title: Identification of key binding site residues of MCT1 for AR-C155858 reveals the molecular basis of its isoform selectivity.
Journal: The Biochemical journal 20150215
Title: Identification of potent Yes1 kinase inhibitors using a library screening approach.
Journal: Bioorganic & medicinal chemistry letters 20130801
Title: The inhibition of monocarboxylate transporter 2 (MCT2) by AR-C155858 is modulated by the associated ancillary protein.
Journal: The Biochemical journal 20101015
Title: AR-C155858 is a potent inhibitor of monocarboxylate transporters MCT1 and MCT2 that binds to an intracellular site involving transmembrane helices 7-10.
Journal: The Biochemical journal 20100201
Title: Optimization of monocarboxylate transporter 1 blockers through analysis and modulation of atropisomer interconversion properties.
Journal: Journal of medicinal chemistry 20070125
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