[1]Engler,ThomasA.;Henry,JamesR.;Malhotra,Sushant;Cunningham,Brian;Furness,Kelly;Brozinick,Joseph;Burkholder,TimothyP.;Clay,MichaelP.;Clayton,Joshua;Diefenbacher,Clive;Hawkins,Eric;Iversen,PhilipW.;Li,Yihong;Lindstrom,TerryD.;Marquart,AngelaL.;McLean,Johnathan;Mendel,David;Misener,Elizabeth;Briere,Daniel;O'Toole,JohnC.;Porter,WarrenJ.;Queener,Steven;Reel,JonK.;Owens,RebeccaA.;Brier,RichardA.;Eessalu,ThomasE.;Wagner,JillR.;Campbell,RobertM.;Vaughn,Renee[JournalofMedicinalChemistry,2004,vol.47,#16,p.3934-3937]
[1]Engler,ThomasA.;Henry,JamesR.;Malhotra,Sushant;Cunningham,Brian;Furness,Kelly;Brozinick,Joseph;Burkholder,TimothyP.;Clay,MichaelP.;Clayton,Joshua;Diefenbacher,Clive;Hawkins,Eric;Iversen,PhilipW.;Li,Yihong;Lindstrom,TerryD.;Marquart,AngelaL.;McLean,Johnathan;Mendel,David;Misener,Elizabeth;Briere,Daniel;O'Toole,JohnC.;Porter,WarrenJ.;Queener,Steven;Reel,JonK.;Owens,RebeccaA.;Brier,RichardA.;Eessalu,ThomasE.;Wagner,JillR.;Campbell,RobertM.;Vaughn,Renee[JournalofMedicinalChemistry,2004,vol.47,#16,p.3934-3937]
[1]Engler,ThomasA.;Henry,JamesR.;Malhotra,Sushant;Cunningham,Brian;Furness,Kelly;Brozinick,Joseph;Burkholder,TimothyP.;Clay,MichaelP.;Clayton,Joshua;Diefenbacher,Clive;Hawkins,Eric;Iversen,PhilipW.;Li,Yihong;Lindstrom,TerryD.;Marquart,AngelaL.;McLean,Johnathan;Mendel,David;Misener,Elizabeth;Briere,Daniel;O'Toole,JohnC.;Porter,WarrenJ.;Queener,Steven;Reel,JonK.;Owens,RebeccaA.;Brier,RichardA.;Eessalu,ThomasE.;Wagner,JillR.;Campbell,RobertM.;Vaughn,Renee[JournalofMedicinalChemistry,2004,vol.47,#16,p.3934-3937]
[1]Engler,ThomasA.;Henry,JamesR.;Malhotra,Sushant;Cunningham,Brian;Furness,Kelly;Brozinick,Joseph;Burkholder,TimothyP.;Clay,MichaelP.;Clayton,Joshua;Diefenbacher,Clive;Hawkins,Eric;Iversen,PhilipW.;Li,Yihong;Lindstrom,TerryD.;Marquart,AngelaL.;McLean,Johnathan;Mendel,David;Misener,Elizabeth;Briere,Daniel;O'Toole,JohnC.;Porter,WarrenJ.;Queener,Steven;Reel,JonK.;Owens,RebeccaA.;Brier,RichardA.;Eessalu,ThomasE.;Wagner,JillR.;Campbell,RobertM.;Vaughn,Renee[JournalofMedicinalChemistry,2004,vol.47,#16,p.3934-3937]
[1]Engler,ThomasA.;Henry,JamesR.;Malhotra,Sushant;Cunningham,Brian;Furness,Kelly;Brozinick,Joseph;Burkholder,TimothyP.;Clay,MichaelP.;Clayton,Joshua;Diefenbacher,Clive;Hawkins,Eric;Iversen,PhilipW.;Li,Yihong;Lindstrom,TerryD.;Marquart,AngelaL.;McLean,Johnathan;Mendel,David;Misener,Elizabeth;Briere,Daniel;O'Toole,JohnC.;Porter,WarrenJ.;Queener,Steven;Reel,JonK.;Owens,RebeccaA.;Brier,RichardA.;Eessalu,ThomasE.;Wagner,JillR.;Campbell,RobertM.;Vaughn,Renee[JournalofMedicinalChemistry,2004,vol.47,#16,p.3934-3937]
Title: Fragment and knowledge-based design of selective GSK-3beta inhibitors using virtual screening models.
Journal: European journal of medicinal chemistry 20090601
Title: Glycogen synthase kinase-3 (GSK3): inflammation, diseases, and therapeutics.
Journal: Neurochemical research 20070101
Title: Substituted 3-imidazo[1,2-a]pyridin-3-yl- 4-(1,2,3,4-tetrahydro-[1,4]diazepino-[6,7,1-hi]indol-7-yl)pyrrole-2,5-diones as highly selective and potent inhibitors of glycogen synthase kinase-3.
Journal: Journal of medicinal chemistry 20040729
Title: GSK-3: tricks of the trade for a multi-tasking kinase.
Journal: Journal of cell science 20030401
Title: Zamek-Gliszczynski MJ, et al. Pharmacokinetics, metabolism, and excretion of the glycogen synthase kinase-3 inhibitor LY2090314 in rats, dogs, and humans: a case study in rapid clearance by extensive metabolism with low circulating metabolite exposure. Dr
Title: Atkinson JM, et al. Activating the Wnt/β-Catenin Pathway for the Treatment of Melanoma--Application of LY2090314, a Novel Selective Inhibitor of Glycogen Synthase Kinase-3. PLoS One. 2015 Apr 27;10(4):e0125028.