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Title: Tight binding of transition-state analogues to a peptidyl-aminoacyl-L/D-isomerase from frog skin.
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Title: Discovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors.
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Title: Synthesis and receptor binding of opioid peptide analogues containing beta3-homo-amino acids.
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Title: Partial ablation of mu-opioid receptor rich striosomes produces deficits on a motor-skill learning task.
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Title: Purification and functional reconstitution of monomeric mu-opioid receptors: allosteric modulation of agonist binding by Gi2.
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Title: Protective effect of dermorphin analogue sedatin on indomethacin-induced injury to the gastric mucosa.
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Title: Neuropathic pain is maintained by brainstem neurons co-expressing opioid and cholecystokinin receptors.
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Title: Conformation-activity relationships of cyclo-constrained micro/delta opioid agonists derived from the N-terminal tetrapeptide segment of dermorphin/deltorphin.
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Title: Amygdala intercalated neurons are required for expression of fear extinction.
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Title: Blood-brain barrier penetration by two dermorphin tetrapeptide analogues: role of lipophilicity vs structural flexibility.
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Title: The use of tritium-labeled dermorphin for studying the interactions of C-terminal dermorphin fragment Tyr-Pro-Ser-NH2 and its stereoisomer Tyr-D-Pro-Ser-NH2 with opioid receptors.
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Title: Methylnaltrexone in the treatment of opioid-induced constipation.
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Title: Effect of synthetic dermorphin analogues on tissue homeostasis in the myocardium of newborn albino rats.
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Title: Effect of sedatin (synthetic dermorphin analog) on the development of Acipenser schrenckii young fish.
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Title: Mechanisms for the effect of arginine-containing dermorphin analogue on proliferative processes in the gastric mucosa of albino rats.
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Title: Ureido group containing cyclic dermorphin(1-7) analogues: synthesis, biology and conformation.
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Title: Receptor binding properties and antinociceptive effects of chimeric peptides consisting of a micro-opioid receptor agonist and an ORL1 receptor antagonist.
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Title: Supranodose vagotomy eliminates respiratory depression evoked by dermorphin in anaesthetized rats.
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Title: Involvement of endogenous opioid peptides in the antinociception induced by the novel dermorphin tetrapeptide analog amidino-TAPA.
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Title: Novel glycosylated [Lys(7)]-dermorphin analogues: synthesis, biological activity and conformational investigations.
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Title: Dependence of the analgesic activities of dermorphin, metenkephalin, and dynorphin A on the ambient temperature.
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Title: Effects of the intravenous administration of [Lys7]dermorphin on local cerebral glucose utilization in the rat.
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Title: Descending facilitation from the rostral ventromedial medulla maintains nerve injury-induced central sensitization.
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Title: Involvement of spinal mu1-opioid receptors on the Tyr-d-Arg-Phe-sarcosine-induced antinociception.
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Title: Targeted drug delivery crossing cytoplasmic membranes of intended cells via ligand-grafted sterically stabilized liposomes.
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Title: Synthesis and biological evaluation of constrained analogues of the opioid peptide H-Tyr-D-Ala-Phe-Gly-NH2 using the 4-amino-2-benzazepin-3-one scaffold.
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Title: Inhibitory control of the acute mu-withdrawal response by indirectly activated adenosine A1 and kappa-opioid systems in the Guinea-pig ileum; reversal by cholecystokinin.
Journal: Neurotoxicology 20051001
Title: Distinguishing and quantifying peptides and proteins containing D-amino acids by tandem mass spectrometry.
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Title: Cyclic enkephalin and dermorphin analogues containing a carbonyl bridge.
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Title: Abbreviated nomenclature for cyclic and branched homo- and hetero-detic peptides.
Journal: The journal of peptide research : official journal of the American Peptide Society 20050601
Title: 6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid mimics active conformation of tyrosine in opioid peptides.
Journal: Bioorganic & medicinal chemistry letters 20050516
Title: New tris-alkoxycarbonyl arginine derivatives for peptide synthesis.
Journal: Journal of peptide science : an official publication of the European Peptide Society 20050101
Title: Synthesis of dermorphin-(1-4) derivatives catalyzed by proteases in organic solvents.
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Title: [Study of thermoregulatory activity of a fragment of natural dermorphin precursor Arg-dermorphin and its analogs].
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Title: [Comparative study of the antiarrhythmic activity of mu- and delta-opioid receptor agonists during acute cardiac ischemia and reperfusion models in rats].
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Title: Tolerance develops in spinal cord, but not in brain with chronic [Dmt1]DALDA treatment.
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Title: Blood-brain barrier permeability of novel [D-arg2]dermorphin (1-4) analogs: transport property is related to the slow onset of antinociceptive activity in the central nervous system.
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Title: Synthesis, conformation and biological activity of dermorphin and deltorphin I analogues containing N-alkylglycine in place of residues in position 1, 3, 5 and 6.
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Title: Potent side-chain to side-chain cyclized dermorphin analogues containing a carbonyl bridge.
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Title: Enhanced evoked excitatory transmitter release in experimental neuropathy requires descending facilitation.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20030910
Title: Opioid peptides: synthesis and biological properties of [(N gamma-glucosyl,N gamma-methoxy)-alpha, gamma-diamino-(S)-butanoyl]4-deltorphin-1-neoglycopeptide and related analogues.
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Title: Expression of EGFP-amino-tagged human mu opioid receptor in Drosophila Schneider 2 cells: a potential expression system for large-scale production of G-protein coupled receptors.
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Title: Endogenous opioid peptides contribute to antinociceptive potency of intrathecal [Dmt1]DALDA.
Journal: The Journal of pharmacology and experimental therapeutics 20030501
Title: Dermorphin tetrapeptide analogues with 2',6'-dimethylphenylalanine (Dmp) substituted for aromatic amino acids have high mu opioid receptor binding and biological activities.
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Title: In vitro and in vivo opioid activity of [DPro(6)]dermorphin, a new dermorphin analogue.
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Title: Dermorphin-based potential affinity labels for mu-opioid receptors.
Journal: The journal of peptide research : official journal of the American Peptide Society 20030101
Title: Vas deferens response to selective opioid receptor agonists in adult mice is impaired following postnatal repeated mild stress.
Journal: European journal of pharmacology 20030101
Title: Dmt and opioid peptides: a potent alliance.
Journal: Biopolymers 20030101
Title: Enhanced spontaneous activity of the mu opioid receptor by cysteine mutations: characterization of a tool for inverse agonist screening.
Journal: BMC pharmacology 20030101
Title: Potent delta-opioid receptor agonists containing the Dmt-Tic pharmacophore.
Journal: Journal of medicinal chemistry 20021205
Title: The mu-selective heptapeptide opioid dermorphin has two conformations around Phe3 psi with no head-to-tail interaction. A quantitative 2-D NMR and molecular modeling analysis.
Journal: Journal of biomolecular structure & dynamics 20021201
Title: Efferent projections from the striatal patch compartment: anterograde degeneration after selective ablation of neurons expressing mu-opioid receptor in rats.
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Title: Urinary peptides in Rett syndrome.
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Title: Lack of involvement of mu(1) opioid receptors in dermorphin-induced inhibition of hypoxic and hypercapnic ventilation in rat pups.
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Title: mu-Opioid receptors: Ligand-dependent activation of potassium conductance, desensitization, and internalization.
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Title: Time-dependent descending facilitation from the rostral ventromedial medulla maintains, but does not initiate, neuropathic pain.
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Title: mu-1 opioid receptor stimulation decreases body temperature in conscious, unrestrained neonatal rats.
Journal: Experimental biology and medicine (Maywood, N.J.) 20020601
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Title: Dermorphin and deltorphin heptapeptide analogues: replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity.
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Title: Evaluation of the Dmt-Tic pharmacophore: conversion of a potent delta-opioid receptor antagonist into a potent delta agonist and ligands with mixed properties.
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Title: [Effect of dermorphin analogs on thermoregulation of rats under various thermal conditions].
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Title: Fetal alveolar epithelial cells contain [D-Ala(2)]-deltorphin I-like immunoreactivity: delta- and mu-opiate receptors mediate opposite effects in developing lung.
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Title: [2',6'-Dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: potent and selective kappa opioid antagonists.
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Title: Inhibition of neuropathic pain by selective ablation of brainstem medullary cells expressing the mu-opioid receptor.
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Title: Receptor binding and biological activity of the dermorphin analog Tyr-D-Arg(2)-Phe-Sar (TAPS).
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Title: The delta-selective opioid peptide dermenkephalin and the mu-selective hybrid peptide dermenkephalin-[1-4]-dermophin-[5-7] display strikingly different conformations despite identical tetrapeptide N-termini. A quantitative 2-D NMR and molecular modeling analysis.
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