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[1]CurrentPatentAssignee:GLAXOSMITHKLINEPLC-EP1051425,2002,B1
Title: Inability to replicate cerebrospinal fluid histamine deficits in the primary hypersomnias: a back to the drawing board moment.
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Title: Development and validation of a sample stabilization strategy and a UPLC-MS/MS method for the simultaneous quantitation of acetylcholine (ACh), histamine (HA), and its metabolites in rat cerebrospinal fluid (CSF).
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Title: Metabolomic profiling for identification of novel potential biomarkers in cardiovascular diseases.
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Title: Histamine potentiates N-methyl-D-aspartate receptors by interacting with an allosteric site distinct from the polyamine binding site.
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Title: CSF levels of the histamine metabolite tele-methylhistamine are only slightly decreased in Alzheimer's disease.
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Title: Inhibition of basophil activation by histamine: a sensitive and reproducible model for the study of the biological activity of high dilutions.
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Title: Bioelimination of histamine in epithelia of the porcine proximal colon of pigs.
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Title: Confirmation of biological effects of high dilutions. Effects of submolecular concentrations of histamine and 1-, 3- and 4-methylhistamines on human basophil activation.
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Title: Antagonist affinity measurements at the Gi-coupled human histamine H3 receptor expressed in CHO cells.
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Title: Early detection of allergic diseases in otorhinolaryngology.
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Title: Hypothalamic neuronal histamine mediates the thyrotropin-releasing hormone-induced suppression of food intake.
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Title: Blockade of brain histamine metabolism alters methamphetamine-induced expression pattern of stereotypy in mice via histamine H1 receptors.
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Title: Hair analysis of histamine and several metabolites in C3H/HeNCrj mice by ultra performance liquid chromatography with electrospray ionization time-of-flight mass spectrometry (UPLC-ESI-TOF-MS): influence of hair cycle and age.
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Title: High-performance liquid chromatographic method for the determination of histamine and 1-methylhistamine in biological buffers.
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Title: Substrate selectivity of monoamine oxidase A, monoamine oxidase B, diamine oxidase, and semicarbazide-sensitive amine oxidase in COS-1 expression systems.
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Title: Rapid determination of histamine and its metabolites in mice hair by ultra-performance liquid chromatography with time-of-flight mass spectrometry.
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Title: N-methyl-D-aspartate receptor antagonists enhance histamine neuron activity in rodent brain.
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Title: Recent advances in molecular pharmacology of the histamine systems: organic cation transporters as a histamine transporter and histamine metabolism.
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Title: Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.
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Title: Glucagon-like peptide-1, corticotropin-releasing hormone, and hypothalamic neuronal histamine interact in the leptin-signaling pathway to regulate feeding behavior.
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Title: Hypothalamic neuronal histamine modulates febrile response but not anorexia induced by lipopolysaccharide.
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Title: Simultaneous fluorometric measurement of histamine and tele-methylhistamine levels in rodent brain by high-performance liquid chromatography.
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Title: Decreased histamine-stimulated phosphoinositide hydrolysis in the cerebral cortex of a rat line selectively bred for high alcohol preference.
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Title: Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain.
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Title: Increased concentrations of histamine and its metabolite, tele-methylhistamine and down-regulation of histamine H3 receptor sites in autopsied brain tissue from cirrhotic patients who died in hepatic coma.
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Title: Evidence of mast cell activation and leukotriene release after mannitol inhalation.
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Title: Brain histamine and histamine H3 receptors following repeated L-histidine administration in rats.
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Title: Ameliorative effects of histamine on 7-chlorokynurenic acid-induced spatial memory deficits in rats.
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Title: Brain histamine turnover and seizure behaviour in two mouse strains: preliminary findings.
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Title: Suppressed weight gain following chronic I-histidine loading--involvement of neuronal histaminergic system?
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Title: Alcoholics show altered histaminergic neurotransmission in several cortical areas--preliminary report.
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Title: Standardised evaluation of urinary excretion of N-tele-methylhistamine in different periods of age in a healthy population.
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Title: Membrane-bound histamine N-methyltransferase in mouse brain: possible role in the synaptic inactivation of neuronal histamine.
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Title: Antimalarial activities of ring-substituted bioimidazoles.
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Title: Increased brain histamine levels in Parkinson's disease but not in multiple system atrophy.
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Title: Human kidney diamine oxidase: heterologous expression, purification, and characterization.
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Title: Real-time monitoring of histamine released from rat basophilic leukemia (RBL-2H3) cells with a histamine microsensor using recombinant histamine oxidase.
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Title: Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
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Title: Effect of alcohol abuse on human brain histamine and tele-methylhistamine.
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Title: Can urinary N-tele methylimidazoleacetic acid (t-MeImAA) serve as a marker of histaminergic activity in hepatic encephalopathy (HE)?
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Title: Acute and chronic effects of methamphetamine on tele-methylhistamine levels in mouse brain: selective involvement of the D(2) and not D(3) receptor.
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Title: Effect of interleukin 1beta on the HPA axis in H1-receptor knockout mice.
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Title: Cerebral and gastric histamine system is altered after portocaval shunt.
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Title: Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?
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Title: Possible involvement of mast-cell activation in aspirin provocation of aspirin-induced asthma.
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Title: Comparison of human, mouse, rat, and guinea pig histamine H4 receptors reveals substantial pharmacological species variation.
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Title: Urinary histamine metabolite elevations during experimental influenza infection.
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Title: Effects of histamine H3-receptor ligands on brain monoamine oxidase in various mammalian species.
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Title: Genomic organization and characterization of splice variants of the human histamine H3 receptor.
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Title: Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow.
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Title: Analysis of histidine and urocanic acid isomers by reversed-phase high-performance liquid chromatography.
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Title: Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles.
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Title: Diazepam-induced decrease in histamine turnover in mouse brain.
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