[1]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1
[2]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1
[3]Watterson,ScottH.;Liu,Qingjie;BeaudoinBertrand,Myra;Batt,DouglasG.;Li,Ling;Pattoli,MarkA.;Skala,Stacey;Cheng,Lihong;Obermeier,MaryT.;Moore,Robin;Yang,Zheng;Vickery,Rodney;Elzinga,PaulA.;Discenza,Lorell;D'Arienzo,Celia;Gillooly,KathleenM.;Taylor,TracyL.;Pulicicchio,Claudine;Zhang,Yifan;Heimrich,Elizabeth;McIntyre,KimW.;Ruan,Qian;Westhouse,RichardA.;Catlett,IanM.;Zheng,Naiyu;Chaudhry,Charu;Dai,Jun;Galella,MichaelA.;Tebben,AndrewJ.;Pokross,Matt;Li,Jianqing;Zhao,Rulin;Smith,Daniel;Rampulla,Richard;Allentoff,Alban;Wallace,MichaelA.;Mathur,Arvind;Salter-Cid,Luisa;Macor,JohnE.;Carter,PercyH.;Fura,Aberra;Burke,JamesR.;Tino,JosephA.[JournalofMedicinalChemistry,2019]Watterson,ScottH.;Liu,Qingjie;BeaudoinBertrand,Myra;Batt,DouglasG.;Li,Ling;Pattoli,MarkA.;Skala,Stacey;Cheng,Lihong;Obermeier,MaryT.;Moore,Robin;Yang,Zheng;Vickery,Rodney;Elzinga,PaulA.;Discenza,Lorell;D'Arienzo,Celia;Gillooly,KathleenM.;Taylor,TracyL.;Pulicicchio,Claudine;Zhang,Yifan;Heimrich,Elizabeth;McIntyre,KimW.;Ruan,Qian;Westhouse,RichardA.;Catlett,IanM.;Zheng,Naiyu;Chaudhry,Charu;Dai,Jun;Galella,MichaelA.;Tebben,AndrewJ.;Pokross,Matt;Li,Jianqing;Zhao,Rulin;Smith,Daniel;Rampulla,Richard;Allentoff,Alban;Wallace,MichaelA.;Mathur,Arvind;Salter-Cid,Luisa;Macor,JohnE.;Carter,PercyH.;Fura,Aberra;Burke,JamesR.;Tino,JosephA.[JournalofMedicinalChemistry,2019,vol.62,#7,p.3228-3250]
[1]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1
[2]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1
[3]Watterson,ScottH.;Liu,Qingjie;BeaudoinBertrand,Myra;Batt,DouglasG.;Li,Ling;Pattoli,MarkA.;Skala,Stacey;Cheng,Lihong;Obermeier,MaryT.;Moore,Robin;Yang,Zheng;Vickery,Rodney;Elzinga,PaulA.;Discenza,Lorell;D'Arienzo,Celia;Gillooly,KathleenM.;Taylor,TracyL.;Pulicicchio,Claudine;Zhang,Yifan;Heimrich,Elizabeth;McIntyre,KimW.;Ruan,Qian;Westhouse,RichardA.;Catlett,IanM.;Zheng,Naiyu;Chaudhry,Charu;Dai,Jun;Galella,MichaelA.;Tebben,AndrewJ.;Pokross,Matt;Li,Jianqing;Zhao,Rulin;Smith,Daniel;Rampulla,Richard;Allentoff,Alban;Wallace,MichaelA.;Mathur,Arvind;Salter-Cid,Luisa;Macor,JohnE.;Carter,PercyH.;Fura,Aberra;Burke,JamesR.;Tino,JosephA.[JournalofMedicinalChemistry,2019]Watterson,ScottH.;Liu,Qingjie;BeaudoinBertrand,Myra;Batt,DouglasG.;Li,Ling;Pattoli,MarkA.;Skala,Stacey;Cheng,Lihong;Obermeier,MaryT.;Moore,Robin;Yang,Zheng;Vickery,Rodney;Elzinga,PaulA.;Discenza,Lorell;D'Arienzo,Celia;Gillooly,KathleenM.;Taylor,TracyL.;Pulicicchio,Claudine;Zhang,Yifan;Heimrich,Elizabeth;McIntyre,KimW.;Ruan,Qian;Westhouse,RichardA.;Catlett,IanM.;Zheng,Naiyu;Chaudhry,Charu;Dai,Jun;Galella,MichaelA.;Tebben,AndrewJ.;Pokross,Matt;Li,Jianqing;Zhao,Rulin;Smith,Daniel;Rampulla,Richard;Allentoff,Alban;Wallace,MichaelA.;Mathur,Arvind;Salter-Cid,Luisa;Macor,JohnE.;Carter,PercyH.;Fura,Aberra;Burke,JamesR.;Tino,JosephA.[JournalofMedicinalChemistry,2019,vol.62,#7,p.3228-3250]
[1]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1
[1]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1Locationinpatent:Paragraph0787
[2]Watterson,ScottH.;Liu,Qingjie;BeaudoinBertrand,Myra;Batt,DouglasG.;Li,Ling;Pattoli,MarkA.;Skala,Stacey;Cheng,Lihong;Obermeier,MaryT.;Moore,Robin;Yang,Zheng;Vickery,Rodney;Elzinga,PaulA.;Discenza,Lorell;D'Arienzo,Celia;Gillooly,KathleenM.;Taylor,TracyL.;Pulicicchio,Claudine;Zhang,Yifan;Heimrich,Elizabeth;McIntyre,KimW.;Ruan,Qian;Westhouse,RichardA.;Catlett,IanM.;Zheng,Naiyu;Chaudhry,Charu;Dai,Jun;Galella,MichaelA.;Tebben,AndrewJ.;Pokross,Matt;Li,Jianqing;Zhao,Rulin;Smith,Daniel;Rampulla,Richard;Allentoff,Alban;Wallace,MichaelA.;Mathur,Arvind;Salter-Cid,Luisa;Macor,JohnE.;Carter,PercyH.;Fura,Aberra;Burke,JamesR.;Tino,JosephA.[JournalofMedicinalChemistry,2019]Watterson,ScottH.;Liu,Qingjie;BeaudoinBertrand,Myra;Batt,DouglasG.;Li,Ling;Pattoli,MarkA.;Skala,Stacey;Cheng,Lihong;Obermeier,MaryT.;Moore,Robin;Yang,Zheng;Vickery,Rodney;Elzinga,PaulA.;Discenza,Lorell;D'Arienzo,Celia;Gillooly,KathleenM.;Taylor,TracyL.;Pulicicchio,Claudine;Zhang,Yifan;Heimrich,Elizabeth;McIntyre,KimW.;Ruan,Qian;Westhouse,RichardA.;Catlett,IanM.;Zheng,Naiyu;Chaudhry,Charu;Dai,Jun;Galella,MichaelA.;Tebben,AndrewJ.;Pokross,Matt;Li,Jianqing;Zhao,Rulin;Smith,Daniel;Rampulla,Richard;Allentoff,Alban;Wallace,MichaelA.;Mathur,Arvind;Salter-Cid,Luisa;Macor,JohnE.;Carter,PercyH.;Fura,Aberra;Burke,JamesR.;Tino,JosephA.[JournalofMedicinalChemistry,2019,vol.62,#7,p.3228-3250]
[3]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-WO2018/45157,2018,A1Locationinpatent:Page/Pagecolumn29-31
[4]Stevens,JasonM.;Simmons,EricM.;Tan,Yichen;Borovika,Alina;Fan,Junying;Forest,RobertV.;Geng,Peng;Guerrero,CarlosA.;Lou,Sha;Skliar,Dimitri;Steinhardt,SarahE.;Strotman,NeilA.[OrganicProcessResearchandDevelopment,2022,vol.26,#4,p.1174-1183]
[1]CurrentPatentAssignee:BRISTOL-MYERSSQUIBBCO-US2016/115126,2016,A1
Title: JR Burke, et al. BMS-986195 Is a Highly Selective and Rapidly Acting Covalent Inhibitor of Bruton’s Tyrosine Kinase with Robust Efficacy at Low Doses in Preclinical Models of RA and Lupus Nephritis. 2017 ACR/ARHP Annual Meeting, September 18, 2017.
Title: Watterson SH, et al. Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid in Vivo Inactivation of Bruton's Tyrosine Kinase (BTK). J Med Chem. 2019 Apr 11;62(7):3228-3250.