[1]Locationinpatent:experimentalpartHansen,CamillaP.;Jensen,AndersA.;Christensen,JeppeK.;Balle,Thomas;Liljefors,Tommy;Frølund,Bente[JournalofMedicinalChemistry,2008,vol.51,#23,p.7380-7395]
1152113-37-5 
 
(S)-N-(4-chloro-2-(2-(5-chloro-6-methylpyrazolo1,5-a-pyrimidin-2-yl)piperidine-1-carbonyl)phenyl)methanesulfonamide 
 
C24H29ClN6O3S 
[1]CurrentPatentAssignee:GILEADSCIENCESINC-US2013/273037,2013,A1Locationinpatent:Paragraph1000-1009
1152113-37-5 
 
(1S,5S,6S)-3-((tert-butoxycarbonyl)((2-(trimethylsilyl)ethoxy)methyl)amino)-5-(5-((Z)-2-(5-chloropyridin-2-yl)-2-fluorovinyl)-2-fluorophenyl)-5-methyl-2-thia-4-azabicyclo4.1.0hept-3-ene-1-carboxylicacid 
 
(1S,5S,6S)-3-amino-5-(5-((Z)-2-(5-chloropyridin-2-yl)-2-fluorovinyl)-2-fluorophenyl)-N-(3-hydroxybutyl)-5-methyl-2-thia-4-azabicyclo4.1.0hept-3-ene-1-carboxamide 
[1]CurrentPatentAssignee:AMGENINC-WO2017/24180,2017,A1Locationinpatent:Page/Pagecolumn136
1152113-37-5 
 
(1S,5S,6S)-3-amino-5-(5-((Z)-2-(5-chloropyridin-2-yl)-2-fluorovinyl)-2-fluorophenyl)-5-methyl-2-thia-4-azabicyclo4.1.0hept-3-ene-1-carboxylicacid 
 
((1S,5S,6S)-3-amino-5-(5-((Z)-2-(5-chloropyridin-2-yl)-2-fluorovinyl)-2-fluorophenyl)-5-methyl-2-thia-4-azabicyclo4.1.0hept-3-en-1-yl)(2-methylazetidin-1-yl)methanone 
[1]CurrentPatentAssignee:AMGENINC-WO2017/24180,2017,A1Locationinpatent:Page/Pagecolumn138
1152113-37-5 
 
2-N-3-(3-chloropropoxy)-4-methoxyphenyl-4-N-methylpyrimidine-2,4-diamine 
 
N<SUP>2</SUP>-(4-methoxy-3-(3-(2-methylazetidin-1-yl)propoxy)phenyl)-N<SUP>4</SUP>-methylpyrimidine-2,4-diamine 
[1]CurrentPatentAssignee:EPIZYME,INC.-WO2017/181177,2017,A1Locationinpatent:Paragraph01151-01153