[1]CurrentPatentAssignee:KOREARESEARCHINSTITUTEOFCHEMICALTECHNOLOGY-KR2018/57914,2018,ALocationinpatent:Paragraph0064-0065;0069-0071
[2]CurrentPatentAssignee:KOREARESEARCHINSTITUTEOFCHEMICALTECHNOLOGY-KR2020/143148,2020,ALocationinpatent:Paragraph0267;0273-0275
[1]CurrentPatentAssignee:KOREARESEARCHINSTITUTEOFCHEMICALTECHNOLOGY-KR2020/143148,2020,A
Title: Topiramate modulation of β(1)- and β(3)-homomeric GABA(A) receptors.
Journal: Pharmacological research 20110701
Title: The role of GABAbeta2 subunit-containing receptors in mediating the anticonvulsant and sedative effects of loreclezole.
Journal: The European journal of neuroscience 20060701
Title: Fast IPSCs in rat thalamic reticular nucleus require the GABAA receptor beta1 subunit.
Journal: The Journal of physiology 20060415
Title: High-affinity, slowly desensitizing GABAA receptors mediate tonic inhibition in hippocampal dentate granule cells.
Journal: Molecular pharmacology 20060201
Title: Pharmacodynamic and/or pharmacokinetic characteristics of interactions between loreclezole and four conventional antiepileptic drugs in pentylenetetrazole-induced seizures in mice: an isobolographic analysis.
Journal: Epilepsy & behavior : E&B 20051201
Title: Consequence of the presence of two different beta subunit isoforms in a GABA(A) receptor.
Journal: Journal of neurochemistry 20051201
Title: Pharmacodynamic and pharmacokinetic interaction studies of loreclezole with felbamate, lamotrigine, topiramate, and oxcarbazepine in the mouse maximal electroshock seizure model.
Journal: Epilepsia 20050301
Title: Critically timed ethanol exposure reduces GABAAR function on septal neurons developing in vivo but not in vitro.
Journal: Brain research 20040515
Title: Interaction of loreclezole with conventional antiepileptic drugs in amygdala-kindled rats.
Journal: European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20040501
Title: Major differences in inhibitory synaptic transmission onto two neocortical interneuron subclasses.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20031022
Title: Sedation and anesthesia mediated by distinct GABA(A) receptor isoforms.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20030917
Title: Effect of some convulsants on the protective activity of loreclezole and its combinations with valproate or clonazepam in amygdala-kindled rats.
Journal: Polish journal of pharmacology 20030101
Title: Functional characterization of GABA(A) receptors in neonatal hypothalamic brain slice.
Journal: Journal of neurophysiology 20021001
Title: N-Substituted 4-amino-3,3-dipropyl-2(3H)-furanones: new positive allosteric modulators of the GABA(A) receptor sharing electrophysiological properties with the anticonvulsant loreclezole.
Journal: Journal of medicinal chemistry 20020620
Title: Do antiepileptics phenytoin, carbamazepine, and loreclezole show GABA(A) receptor subtype selectivity in rat brain sections?
Journal: Neurochemical research 20010101
Title: Heterogeneity of GABA(A) receptor-mediated responses in the human IMR-32 neuroblastoma cell line.
Journal: Journal of neuroscience research 20000515
Title: Preclinical evaluation of newly approved and potential antiepileptic drugs against cocaine-induced seizures.
Journal: The Journal of pharmacology and experimental therapeutics 19990901
Title: The interactions of hexachlorocyclohexane isomers with human gamma-aminobutyric acid(A) receptors expressed in Xenopus oocytes.
Journal: The Journal of pharmacology and experimental therapeutics 19970901
Title: A novel allosteric modulatory site on the GABAA receptor beta subunit.
Journal: Neuron 19940401
Title: The novel anticonvulsant loreclezole (R 72063) does not produce diazepam-like anterograde amnesia in a passive avoidance test in rats.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 19901101
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