Title: Discovery of N6-phenyl-1H-pyrazolo[3,4-d]pyrimidine-3,6-diamine derivatives as novel CK1 inhibitors using common-feature pharmacophore model based virtual screening and hit-to-lead optimization.
Journal: European journal of medicinal chemistry 20121001
Title: IC261 induces cell cycle arrest and apoptosis of human cancer cells via CK1δ/ɛ and Wnt/β-catenin independent inhibition of mitotic spindle formation.
Journal: Oncogene 20110602
Title: Selective inhibition of casein kinase 1 epsilon minimally alters circadian clock period.
Journal: The Journal of pharmacology and experimental therapeutics 20090801
Title: Walton KM, et al. Selective inhibition of casein kinase 1 epsilon minimally alters circadian clock period. J Pharmacol Exp Ther. 2009 Aug;330(2):430-9.
