[1]Evans,KarenA.;Budzik,BrianW.;Ross,SeanA.;Wisnoski,DavidD.;Jin,Jian;Rivero,RalphA.;Vimal,Mythily;Szewczyk,GeorgeR.;Jayawickreme,Channa;Moncol,DavidL.;Rimele,ThomasJ.;Armour,SusanL.;Weaver,SusanP.;Griffin,RobertJ.;Tadepalli,SarvaM.;Jeune,MichaelR.;Shearer,ToddW.;Chen,ZibinB.;Chen,Lihong;Anderson,DonaldL.;Becherer,J.David;DeLosFrailes,Maite;Colilla,FranciscoJavier[JournalofMedicinalChemistry,2009,vol.52,#24,p.7962-7965]
Title: Dipeptidyl peptidase IV inhibition potentiates amino acid- and bile acid-induced bicarbonate secretion in rat duodenum.
Journal: American journal of physiology. Gastrointestinal and liver physiology 20121001
Title: Discovery of 3-aryl-4-isoxazolecarboxamides as TGR5 receptor agonists.
Journal: Journal of medicinal chemistry 20091224
Title: Evans KA, et al. Discovery of 3-aryl-4-isoxazolecarboxamides as TGR5 receptor agonists. J Med Chem. 2009 Dec 24;52(24):7962-5.
Title: Caldwell A, Grundy L, Harrington AM, Garcia-Caraballo S, Castro J, Bunnett NW, Brierley SM. TGR5 agonists induce peripheral and central hypersensitivity to bladder distension. Sci Rep. 2022 Jun 15;12(1):9920.
Title: Castellanos-Jankiewicz A, et al. Hypothalamic bile acid-TGR5 signaling protects from obesity. Cell Metab. 2021 Jul 6;33(7):1483-1492.e10.