Title: Optimization of cellular activity of G9a inhibitors 7-aminoalkoxy-quinazolines.
Journal: Journal of medicinal chemistry 20110908
Title: A chemical probe selectively inhibits G9a and GLP methyltransferase activity in cells.
Journal: Nature chemical biology 20110710
Title: Protein lysine methyltransferase G9a inhibitors: design, synthesis, and structure activity relationships of 2,4-diamino-7-aminoalkoxy-quinazolines.
Journal: Journal of medicinal chemistry 20100812
Title: G9a and Glp methylate lysine 373 in the tumor suppressor p53.
Journal: The Journal of biological chemistry 20100326
Title: Downregulation of histone H3 lysine 9 methyltransferase G9a induces centrosome disruption and chromosome instability in cancer cells.
Journal: PloS one 20080101
Title: Silenced tumor suppressor genes reactivated by DNA demethylation do not return to a fully euchromatic chromatin state.
Journal: Cancer research 20060401
Title: G9a histone methyltransferase plays a dominant role in euchromatic histone H3 lysine 9 methylation and is essential for early embryogenesis.
Journal: Genes & development 20020715
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