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Journal: Oncogene 20170105
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Journal: Endocrine-related cancer 20160401
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Journal: Nature 20150924
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Journal: Cell research 20140701
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Title: Optimization of 3,5-dimethylisoxazole derivatives as potent bromodomain ligands.
Journal: Journal of medicinal chemistry 20130425
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Journal: Nature 20120809
Title: From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151.
Journal: Bioorganic & medicinal chemistry letters 20120415
Title: Fragment-based discovery of bromodomain inhibitors part 2: optimization of phenylisoxazole sulfonamides.
Journal: Journal of medicinal chemistry 20120126
Title: BET bromodomain inhibition as a therapeutic strategy to target c-Myc.
Journal: Cell 20110916
Title: Liver X receptors as regulators of macrophage inflammatory and metabolic pathways.
Journal: Biochimica et biophysica acta 20110801
Title: Discovery and characterization of small molecule inhibitors of the BET family bromodomains.
Journal: Journal of medicinal chemistry 20110609
Title: Suppression of inflammation by a synthetic histone mimic.
Journal: Nature 20101223
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