Title: Toxicologic/transport properties of NCS-382, a γ-hydroxybutyrate (GHB) receptor ligand, in neuronal and epithelial cells: Therapeutic implications for SSADH deficiency, a GABA metabolic disorder.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20180201
Title: In vitro toxicological evaluation of NCS-382, a high-affinity antagonist of γ-hydroxybutyrate (GHB) binding.
Journal: Toxicology in vitro : an international journal published in association with BIBRA 20170401
Title: Novel radioiodinated {gamma}-hydroxybutyric acid analogues for radiolabeling and Photolinking of high-affinity {gamma}-hydroxybutyric acid binding sites.
Journal: The Journal of pharmacology and experimental therapeutics 20101101
Title: Calcium and cAMP signaling induced by gamma-hydroxybutyrate receptor(s) stimulation in NCB-20 neurons.
Journal: Neuroscience 20100428
Title: Neurotoxic effects induced by gammahydroxybutyric acid (GHB) in male rats.
Journal: The international journal of neuropsychopharmacology 20091001
Title: Validation of high-affinity binding sites for succinic acid through distinguishable binding of gamma-hydroxybutyric acid receptor-specific NCS 382 antipodes.
Journal: Bioorganic & medicinal chemistry letters 20081201
Title: Characterization and pharmacology of the GHB receptor.
Journal: Annals of the New York Academy of Sciences 20081001
Title: Differentiating the discriminative stimulus effects of gamma-hydroxybutyrate and ethanol in a three-choice drug discrimination procedure in rats.
Journal: Pharmacology, biochemistry, and behavior 20080601
Title: Gamma-aminobutyric acidB (GABAB)-receptor mediation of different in vivo effects of gamma-butyrolactone.
Journal: Journal of pharmacological sciences 20080201
Title: [Effect of gamma-hydroxybutyric acid receptor on focal cerebral ischemia-reperfusion injury in rats].
Journal: Yao xue xue bao = Acta pharmaceutica Sinica 20070801
Title: Metabolic GHB precursor succinate binds to gamma-hydroxybutyrate receptors: characterization of human basal ganglia areas nucleus accumbens and globus pallidus.
Journal: Journal of neuroscience research 20060701
Title: Succinate semialdehyde dehydrogenase deficiency does not down-regulate gamma-hydroxybutyric acid binding sites in the mouse brain.
Journal: Molecular genetics and metabolism 20060501
Title: Discriminative stimulus effects of flumazenil: perceptual masking by baclofen, and lack of substitution with gamma-hydroxybutyrate and its precursors 1,4-butanediol and gamma-butyrolactone.
Journal: Behavioural pharmacology 20060501
Title: Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Journal: Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
Title: Novel cyclic gamma-hydroxybutyrate (GHB) analogs with high affinity and stereoselectivity of binding to GHB sites in rat brain.
Journal: The Journal of pharmacology and experimental therapeutics 20051001
Title: Drosophila GABA(B) receptors are involved in behavioral effects of gamma-hydroxybutyric acid (GHB).
Journal: European journal of pharmacology 20050920
Title: Involvement of gamma-hydroxybutyrate (GHB) and GABA-B receptors in the acute behavioral effects of GHB in baboons.
Journal: Psychopharmacology 20050701
Title: Discriminative stimulus effects of gamma-hydroxybutyrate (GHB) in rats discriminating GHB from baclofen and diazepam.
Journal: The Journal of pharmacology and experimental therapeutics 20050701
Title: Resuscitative effect of a gamma-aminobutyric acid B receptor antagonist on gamma-hydroxybutyric acid mortality in mice.
Journal: Annals of emergency medicine 20050601
Title: Mechanisms underlying the sympathomimetic cardiovascular responses elicited by gamma-hydroxybutyrate.
Journal: Journal of cardiovascular pharmacology 20041201
Title: Ethanol does not alter the binding of the gamma-hydroxybutyric acid (GHB) receptor ligand [3H]NCS-382 in the rat brain.
Journal: Drug and alcohol dependence 20040906
Title: 4-Hydroxy-trans-2-nonenoic acid is a gamma-hydroxybutyrate receptor ligand in the cerebral cortex and hippocampus.
Journal: Journal of neurochemistry 20040601
Title: Gamma-hydroxybutyrate and ethanol depress spontaneous excitatory postsynaptic currents in dopaminergic neurons of the substantia nigra.
Journal: Brain research 20040130
Title: Effects of gamma-hydroxybutyrate (GHB) on schedule-controlled responding in rats: role of GHB and GABAB receptors.
Journal: The Journal of pharmacology and experimental therapeutics 20040101
Title: A review of pharmacology of NCS-382, a putative antagonist of gamma-hydroxybutyric acid (GHB) receptor.
Journal: CNS drug reviews 20040101
Title: Pathway-specific action of gamma-hydroxybutyric acid in sensory thalamus and its relevance to absence seizures.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20031210
Title: Selective gamma-hydroxybutyric acid receptor ligands increase extracellular glutamate in the hippocampus, but fail to activate G protein and to produce the sedative/hypnotic effect of gamma-hydroxybutyric acid.
Journal: Journal of neurochemistry 20031101
Title: Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA(B)(1)-deficient mice.
Journal: The European journal of neuroscience 20031101
Title: Quantitative autoradiographic analysis of the new radioligand [(3)H](2E)-(5-hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) ethanoic acid ([(3)H]NCS-382) at gamma-hydroxybutyric acid (GHB) binding sites in rat brain.
Journal: Brain research 20030725
Title: Interactions of gamma-hydroxy butyrate with ethanol and NCS 382.
Journal: European journal of pharmacology 20030606
Title: A tertiary alcohol analog of gamma-hydroxybutyric acid as a specific gamma-hydroxybutyric acid receptor ligand.
Journal: The Journal of pharmacology and experimental therapeutics 20030501
Title: Therapeutic intervention in mice deficient for succinate semialdehyde dehydrogenase (gamma-hydroxybutyric aciduria).
Journal: The Journal of pharmacology and experimental therapeutics 20020701
Title: Stereoselectivity of NCS-382 binding to gamma-hydroxybutyrate receptor in the rat brain.
Journal: European journal of pharmacology 20020620
Title: GABA(B)-receptor mediation of the inhibitory effect of gamma-hydroxybutyric acid on intestinal motility in mice.
Journal: Life sciences 20020510
Title: Effects of the putative antagonist NCS382 on the behavioral pharmacological actions of gammahydroxybutyrate in mice.
Journal: Psychopharmacology 20020201
Title: Binding characteristics of the gamma-hydroxybutyric acid receptor antagonist [(3)H](2E)-(5-hydroxy-5,7,8,9-tetrahydro-6H-benzo[a][7]annulen-6-ylidene) ethanoic acid in the rat brain.
Journal: The Journal of pharmacology and experimental therapeutics 20011201
Title: gamma-Hydroxybutyric acid and baclofen decrease extracellular acetylcholine levels in the hippocampus via GABA(B) receptors.
Journal: European journal of pharmacology 20011102
Title: Role of GABA(B) receptors in the sedative/hypnotic effect of gamma-hydroxybutyric acid.
Journal: European journal of pharmacology 20011012
Title: gamma-Hydroxybutyrate modulation of glutamate levels in the hippocampus: an in vivo and in vitro study.
Journal: Journal of neurochemistry 20010901
