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Home Boronic Acids 1352796-65-6
1352796-65-6,MFCD13182191
Catalog No.:AA009FN7

1352796-65-6 | 2-Fluoropyrimidin-5-ylboronic acid pinacol ester

Pack Size
Purity
Availability
Price(USD)
Quantity
  
250mg
95%
in stock  
$45.00   $32.00
- +
500mg
95%
in stock  
$51.00   $36.00
- +
1g
95%
in stock  
$57.00   $40.00
- +
25g
98%
in stock  
$1,407.00   $985.00
- +
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
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  • Download SDS
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
Technical Information
Catalog Number:
AA009FN7
Chemical Name:
2-Fluoropyrimidin-5-ylboronic acid pinacol ester
CAS Number:
1352796-65-6
Molecular Formula:
C10H14BFN2O2
Molecular Weight:
224.0398
MDL Number:
MFCD13182191
SMILES:
CC1(C)OB(OC1(C)C)c1cnc(nc1)F
Properties
Computed Properties
 
Complexity:
252  
Covalently-Bonded Unit Count:
1  
Heavy Atom Count:
16  
Hydrogen Bond Acceptor Count:
5  
Rotatable Bond Count:
1  

Downstream Synthesis Route

[1]CurrentPatentAssignee:PFIZERINC;ELILILLY&CO-WO2018/71447,2018,A1Locationinpatent:Paragraph001278;001279;001280

[1]Pike,KurtG.;Barlaam,Bernard;Cadogan,Elaine;Campbell,Andrew;Chen,Yingxue;Colclough,Nicola;Davies,NicholaL.;De-Almeida,Camila;Degorce,SebastienL.;Didelot,Myriam;Dishington,Allan;Ducray,Richard;Durant,StephenT.;Hassall,LorraineA.;Holmes,Jane;Hughes,GarethD.;Macfaul,PhilipA.;Mulholland,KeithR.;McGuire,ThomasM.;Ouvry,Gilles;Pass,Martin;Robb,Graeme;Stratton,Natalie;Wang,Zhenhua;Wilson,Joanne;Zhai,Baochang;Zhao,Kang;Al-Huniti,Nidal[JournalofMedicinalChemistry,2018,vol.61,#9,p.3823-3841]

163271-08-7   
2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine 
 
tert-butyl(1-(5-(3-cyano-6-(2-morpholinoethoxy)pyrazolo1,5-apyridin-4-yl)pyrimidin-2-yl)-4-methylpiperidin-4-yl)carbamate 

[1]Patent:WO2018/71454,2018,A1.Locationinpatent:Paragraph001248;001250

163271-08-7   
2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine 
 
tert-butyl(4-methyl-1-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidin-2-yl)piperidin-4-yl)carbamate 

[1]Patent:WO2018/71454,2018,A1.Locationinpatent:Paragraph001475;001476;001477

1166997-21-2    1352796-65-6   
CASUnavailable 

[1]CurrentPatentAssignee:PFIZERINC-WO2019/113542,2019,A1Locationinpatent:Paragraph0337

Literature
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SDS
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