Title: Protective effects of histamine H3-receptor ligands in schizophrenic behaviors in experimental models.
Journal: Pharmacological reports : PR 20120101
Title: Molecular determinants of ligand binding modes in the histamine H(4) receptor: linking ligand-based three-dimensional quantitative structure-activity relationship (3D-QSAR) models to in silico guided receptor mutagenesis studies.
Journal: Journal of medicinal chemistry 20111208
Title: The H4 histamine receptor agonist, clobenpropit, suppresses human cholangiocarcinoma progression by disruption of epithelial mesenchymal transition and tumor metastasis.
Journal: Hepatology (Baltimore, Md.) 20111101
Title: Role of H4 receptor in histamine-mediated responses in human melanoma.
Journal: Melanoma research 20111001
Title: Histamine H(3) receptor-mediated modulation of perivascular nerve transmission in rat mesenteric arteries.
Journal: European journal of pharmacology 20110325
Title: Beneficial interaction between clobenpropit and pyridoxine in prevention of electroshock-induced seizures in mice: lack of histaminergic mechanisms.
Journal: Human & experimental toxicology 20110101
Title: Modulation of hematopoiesis through histamine receptor signaling.
Journal: Frontiers in bioscience (Scholar edition) 20110101
Title: Attenuated expression of HRH4 in colorectal carcinomas: a potential influence on tumor growth and progression.
Journal: BMC cancer 20110101
Title: Withdrawal from repeated administration of morphine alters histamine-induced anxiogenic effects produced by intra-ventral hippocampal microinjection.
Journal: Journal of psychopharmacology (Oxford, England) 20100601
Title: Implementation of a fluorescence-based screening assay identifies histamine H3 receptor antagonists clobenpropit and iodophenpropit as subunit-selective N-methyl-D-aspartate receptor antagonists.
Journal: The Journal of pharmacology and experimental therapeutics 20100601
Title: The H3 receptor antagonist clobenpropit protects against Abeta42-induced neurotoxicity in differentiated rat PC12 cells.
Journal: Die Pharmazie 20100401
Title: Modeling G protein-coupled receptors for structure-based drug discovery using low-frequency normal modes for refinement of homology models: application to H3 antagonists.
Journal: Proteins 20100201
Title: [Effects of clobenpropit and histidine on reinstatement of morphine-induced conditioned place preference].
Journal: Zhejiang da xue xue bao. Yi xue ban = Journal of Zhejiang University. Medical sciences 20091101
Title: The histamine H receptor as a new target for treatment of canine inflammatory skin diseases.
Journal: Veterinary dermatology 20091001
Title: Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studies.
Journal: Bioorganic & medicinal chemistry 20090601
Title: The histamine H4 receptor is functionally expressed on T(H)2 cells.
Journal: The Journal of allergy and clinical immunology 20090301
Title: The role of histamine 3 receptors in the control of food intake in a seasonal model of obesity: the Siberian hamster.
Journal: Behavioural pharmacology 20090301
Title: Histamine H4 receptor antagonism reduces hapten-induced scratching behaviour but not inflammation.
Journal: Experimental dermatology 20090101
Title: Histamine H4 receptors modulate dendritic cell migration through skin--immunomodulatory role of histamine.
Journal: Allergy 20081001
Title: Electrophysiology-based analysis of human histamine H(4) receptor pharmacology using GIRK channel coupling in Xenopus oocytes.
Journal: European journal of pharmacology 20080904
Title: Apomorphine-induced turning behavior in 6-hydroxydopamine lesioned rats is increased by histidine and decreased by histidine decarboxylase, histamine H1 and H2 receptor antagonists, and an H3 receptor agonist.
Journal: Pharmacology, biochemistry, and behavior 20080901
Title: Substance P is involved in the effect of histamine H3 receptor agonist, Sch 50971 on nasal allergic symptoms in mice.
Journal: International immunopharmacology 20080801
Title: Comparison of the effect of an H(3)-inverse agonist on energy intake and hypothalamic histamine release in normal mice and leptin resistant mice with high fat diet-induced obesity.
Journal: Behavioural brain research 20080409
Title: Efficient approaches to S-alkyl-N-alkylisothioureas: syntheses of histamine H3 antagonist clobenpropit and its analogues.
Journal: The Journal of organic chemistry 20080321
Title: Carnosine protects against Abeta42-induced neurotoxicity in differentiated rat PC12 cells.
Journal: Cellular and molecular neurobiology 20080201
Title: The role of histamine in human mammary carcinogenesis: H3 and H4 receptors as potential therapeutic targets for breast cancer treatment.
Journal: Cancer biology & therapy 20080101
Title: Histamine downregulates monocyte CCL2 production through the histamine H4 receptor.
Journal: The Journal of allergy and clinical immunology 20070801
Title: The human histamine H3 receptor couples to GIRK channels in Xenopus oocytes.
Journal: European journal of pharmacology 20070719
Title: The histamine H3 receptor antagonist clobenpropit enhances GABA release to protect against NMDA-induced excitotoxicity through the cAMP/protein kinase A pathway in cultured cortical neurons.
Journal: European journal of pharmacology 20070601
Title: Histamine H3-receptor agonists and imidazole-based H3-receptor antagonists can be thermodynamically discriminated.
Journal: British journal of pharmacology 20070601
Title: Correlation of apparent affinity values from H3-receptor binding assays with apparent affinity (pKapp) and intrinsic activity (alpha) from functional bioassays.
Journal: British journal of pharmacology 20070501
Title: Role of histamine in ghrelin-induced gastroprotection against acute gastric lesions.
Journal: Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20070401
Title: [Reversing effect of histamine on neurotoxicity induced by beta-amyloid1-42].
Journal: Zhejiang da xue xue bao. Yi xue ban = Journal of Zhejiang University. Medical sciences 20070301
Title: Pre-synaptic histamine H3 receptors regulate glutamate, but not GABA release in rat thalamus.
Journal: Neuropharmacology 20070201
Title: Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway.
Journal: Neuropharmacology 20060901
Title: Detection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligand.
Journal: British journal of pharmacology 20060701
Title: Histamine excites neonatal rat sympathetic preganglionic neurons in vitro via activation of H1 receptors.
Journal: Journal of neurophysiology 20060401
Title: Probing the importance of N-glycosylation for [(3)H] clobenpropit binding to human H (3) receptors expressed in HEK 293 cells . 3. Molecular and chemical aspects of the histamine receptors.
Journal: Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20060401
Title: Histamine increases sickle erythrocyte adherence to endothelium.
Journal: British journal of haematology 20060201
Title: Histaminergic neurons protect the developing hippocampus from kainic acid-induced neuronal damage in an organotypic coculture system.
Journal: The Journal of neuroscience : the official journal of the Society for Neuroscience 20060125
Title: Effects of intracerebroventricular administration of ultra low doses of histaminergic drugs on morphine state-dependent memory of passive avoidance in mice.
Journal: Behavioural brain research 20060106
Title: Histamine (H3) receptors modulate the excitatory amino acid receptor response of the vestibular afferents.
Journal: Brain research 20051207
Title: Histamine-3 receptor antagonists reduce superoxide anion generation and lipid peroxidation in rat brain homogenates.
Journal: The Journal of pharmacy and pharmacology 20050601
Title: Histamine H4 receptor stimulation suppresses IL-12p70 production and mediates chemotaxis in human monocyte-derived dendritic cells.
Journal: Journal of immunology (Baltimore, Md. : 1950) 20050501
Title: Inhibition of tryptase release from human colon mast cells by histamine receptor antagonists.
Journal: Asian Pacific journal of allergy and immunology 20050301
Title: Histamine H3 receptors modulate reactive hyperemia in rat gut.
Journal: Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20040901
Title: Presynaptic cannabinoid CB(1) receptors are involved in the inhibition of the neurogenic vasopressor response during septic shock in pithed rats.
Journal: British journal of pharmacology 20040601
Title: Ligand identification for G-protein-coupled receptors: a lead generation perspective.
Journal: Current opinion in chemical biology 20040601
Title: Effect of the histamine H3-antagonist clobenpropit on spatial memory deficits induced by MK-801 as evaluated by radial maze in Sprague-Dawley rats.
Journal: Behavioural brain research 20040505
Title: [Mechanisms of the effect of brain histamine on chronic epilepsy induced by pentylenetetrazole].
Journal: Zhejiang da xue xue bao. Yi xue ban = Journal of Zhejiang University. Medical sciences 20040501
Title: Intracerebroventricular administration of histamine H3 receptor antagonists decreases seizures in rat models of epilepsia.
Journal: Methods and findings in experimental and clinical pharmacology 20040501
Title: Histamine h3 receptor antagonists potentiate methamphetamine self-administration and methamphetamine-induced accumbal dopamine release.
Journal: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20040401
Title: Involvement of central and peripheral histamine H(3) receptors in the control of the vascular tone and oxygen uptake in the mesenteric circulation of the rat.
Journal: Journal of physiology and pharmacology : an official journal of the Polish Physiological Society 20040301
Title: Effects of clobenpropit on pentylenetetrazole-kindled seizures in rats.
Journal: European journal of pharmacology 20031215
Title: Histamine induces cytoskeletal changes in human eosinophils via the H(4) receptor.
Journal: British journal of pharmacology 20031101
Title: Histamine H3 receptors regulate vascular permeability changes in the skin of mast cell-deficient mice.
Journal: International immunopharmacology 20031101
Title: Effects of endogenous histamine on seizure development of pentylenetetrazole-induced kindling in rats.
Journal: Pharmacology 20030901
Title: Molecular and pharmacological characterization of the mouse histamine H3 receptor.
Journal: European journal of pharmacology 20030425
Title: Activation of the extraneuronal monoamine transporter (EMT) from rat expressed in 293 cells.
Journal: British journal of pharmacology 20021101
Title: Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.
Journal: Molecular pharmacology 20020101
Title: Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?
Journal: European journal of pharmacology 20011116
Title: Histamine H3 receptor-mediated inhibition of sympathetically evoked mydriasis in rats.
Journal: European journal of pharmacology 20010504
Title: Histamine H(3) receptor-mediated inhibition of depolarization-induced, dopamine D(1) receptor-dependent release of [(3)H]-gamma-aminobutryic acid from rat striatal slices.
Journal: British journal of pharmacology 20010501
Title: Effect of clobenpropit on regional cerebral blood flow in rat hippocampus.
Journal: Acta pharmacologica Sinica 20010401
Title: Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
Journal: Journal of neurochemistry 20000801
Title: Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.
Journal: Behavioural brain research 19991001
Title: Histamine inhibits the production of interleukin-12 through interaction with H2 receptors.
Journal: The Journal of clinical investigation 19981115
Title: Effect of interleukin-1beta on the ascending and descending reflex in rat small intestine.
Journal: European journal of pharmacology 19981023
Title: Inhibitory H3 receptors on sympathetic nerves of the pithed rat: activation by endogenous histamine and operation in spontaneously hypertensive rats.
Journal: Naunyn-Schmiedeberg's archives of pharmacology 19970201
Title: Short photoperiod-induced decrease of histamine H3 receptors facilitates activation of hypothalamic neurons in the Siberian hamster.
Journal: Endocrinology
