Title: Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.
Journal: The Journal of organic chemistry 20120504
Title: Characterization of steroid sulfatase in the MC3T3-E1 mouse pre-osteoblastic cell line.
Journal: Steroids 20120501
Title: Synthesis and evaluation of analogues of estrone-3-O-sulfamate as potent steroid sulfatase inhibitors.
Journal: Bioorganic & medicinal chemistry 20120415
Title: Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI.
Journal: European journal of medicinal chemistry 20120301
Title: Inhibition of steroid sulfatase with 4-substituted estrone and estradiol derivatives.
Journal: Bioorganic & medicinal chemistry 20111015
Title: Direct effect of dehydroepiandrosterone sulfate (DHEAS) on PC-12 cell differentiation processes.
Journal: Molecular and cellular endocrinology 20110410
Title: [Steroid sulfatase inhibitor].
Journal: Nihon rinsho. Japanese journal of clinical medicine 20100601
Title: Structures of human carbonic anhydrase II/inhibitor complexes reveal a second binding site for steroidal and nonsteroidal inhibitors.
Journal: Biochemistry 20100427
Title: Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template.
Journal: Journal of medicinal chemistry 20100311
Title: Thiosemicarbazones of formyl benzoic acids as novel potent inhibitors of estrone sulfatase.
Journal: Journal of medicinal chemistry 20070726
Title: Tibolone and its delta-4, 7alpha-methyl norethisterone metabolite are reversible inhibitors of human aromatase.
Journal: The Journal of steroid biochemistry and molecular biology 20070501
Title: 2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.
Journal: Journal of medicinal chemistry 20061228
Title: Inhibition of estrone sulfatase by aromatase inhibitor-based estrogen 3-sulfamates.
Journal: Steroids 20060501
Title: Carbonic anhydrase inhibitors: inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides.
Journal: Bioorganic & medicinal chemistry letters 20051201
Title: Carbonic anhydrase inhibitors: stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II.
Journal: Journal of medicinal chemistry 20050908
Title: A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents.
Journal: Journal of medicinal chemistry 20050811
Title: First crystal structures of human carbonic anhydrase II in complex with dual aromatase-steroid sulfatase inhibitors.
Journal: Biochemistry 20050510
Title: Pregnenolone sulphate attenuates AMPA cytotoxicity on rat cortical neurons.
Journal: The European journal of neuroscience 20050501
Title: Steroid sulfatase: molecular biology, regulation, and inhibition.
Journal: Endocrine reviews 20050401
Title: N-Acyl arylsulfonamides as novel, reversible inhibitors of human steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20050215
Title: The nature of inhibition of steroid sulphatase activity by tibolone and its metabolites.
Journal: The Journal of steroid biochemistry and molecular biology 20050201
Title: Anti-cancer activities of novel D-ring modified 2-substituted estrogen-3-O-sulfamates.
Journal: The Journal of steroid biochemistry and molecular biology 20050201
Title: Stilbene-based inhibitors of estrone sulfatase with a dual mode of action in human breast cancer cells.
Journal: Archiv der Pharmazie 20041201
Title: Pharmacokinetics of the nonsteroidal steroid sulphatase inhibitor 667 COUMATE and its sequestration into red blood cells in rats.
Journal: British journal of cancer 20041004
Title: Estrone formate: a novel type of irreversible inhibitor of human steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20041004
Title: The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates.
Journal: Biochemical and biophysical research communications 20040910
Title: 2-(1-adamantyl)-4-(thio)chromenone-6-carboxylic acids: potent reversible inhibitors of human steroid sulfatase.
Journal: Journal of medicinal chemistry 20040812
Title: 2-Alkylsulfanyl estrogen derivatives: synthesis of a novel class of multi-targeted anti-tumour agents.
Journal: Bioorganic & medicinal chemistry letters 20040621
Title: Inhibition of in vitro angiogenesis by 2-methoxy- and 2-ethyl-estrogen sulfamates.
Journal: International journal of cancer 20040420
Title: Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acid.
Journal: Bioorganic & medicinal chemistry letters 20040209
Title: Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride.
Journal: Bioorganic & medicinal chemistry letters 20040119
Title: Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20040105
Title: 6-(2-adamantan-2-ylidene-hydroxybenzoxazole)-O-sulfamate: a potent non-steroidal irreversible inhibitor of human steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20031215
Title: Nortropinyl-arylsulfonylureas as novel, reversible inhibitors of human steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20031103
Title: Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
Journal: The Journal of steroid biochemistry and molecular biology 20031101
Title: Inhibition of estrone sulfate-induced uterine growth by potent nonestrogenic steroidal inhibitors of steroid sulfatase.
Journal: Cancer research 20031001
Title: The design, synthesis, and in vitro biochemical evaluation of a series of esters of 4-[(aminosulfonyl)oxy]benzoate as novel and highly potent inhibitors of estrone sulfatase.
Journal: Biochemical and biophysical research communications 20030808
Title: Microtiter plate cellular assay for human steroid sulfatase with fluorescence readout.
Journal: Analytical biochemistry 20030715
Title: Inhibition of carbonic anhydrase II by steroidal and non-steroidal sulphamates.
Journal: Biochemical and biophysical research communications 20030613
Title: Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Journal: Journal of medicinal chemistry 20030522
Title: D-ring modified estrone derivatives as novel potent inhibitors of steroid sulfatase.
Journal: Bioorganic & medicinal chemistry 20030417
Title: Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II.
Journal: Bioorganic & medicinal chemistry letters 20030310
Title: Novel D-ring modified steroid derivatives as potent, non-estrogenic, steroid sulfatase inhibitors with in vivo activity.
Journal: The Journal of steroid biochemistry and molecular biology 20030201
Title: Inhibition of MCF-7 breast cancer cell proliferation and in vivo steroid sulphatase activity by 2-methoxyoestradiol-bis-sulphamate.
Journal: The Journal of steroid biochemistry and molecular biology 20030201
Title: Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).
Journal: The Journal of steroid biochemistry and molecular biology 20021101
Title: 2-Substituted 4-(thio)chromenone 6-O-sulfamates: potent inhibitors of human steroid sulfatase.
Journal: Journal of medicinal chemistry 20020912
Title: Inhibition of estrone sulfatase (ES) by derivatives of 4-[(aminosulfonyl)oxy] benzoic acid.
Journal: Bioorganic & medicinal chemistry letters 20020902
Title: Inhibition of steryl sulfatase activity in LNCaP human prostate cancer cells.
Journal: Steroids 20020901
Title: 4,4'-Benzophenone-O,O'-disulfamate: a potent inhibitor of steroid sulfatase.
Journal: Bioorganic & medicinal chemistry letters 20020819
Title: The design, synthesis, and biochemical evaluation of derivatives of biphenyl sulfamate-based compounds as novel inhibitors of estrone sulfatase.
Journal: Biochemical and biophysical research communications 20020531
Title: A novel type of nonsteroidal estrone sulfatase inhibitors.
Journal: Bioorganic & medicinal chemistry letters 20020520
Title: Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20020520
Title: The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds.
Journal: Bioorganic & medicinal chemistry letters 20020506
Title: Synthesis and biochemical evaluation of novel and potent inhibitors of the enzyme oestrone sulphatase (ES).
Journal: The Journal of steroid biochemistry and molecular biology 20020401
Title: Nonsteroidal compounds designed to mimic potent steroid sulfatase inhibitors.
Journal: The Journal of steroid biochemistry and molecular biology 20020301
Title: Determination and use of a transition state for the enzyme estrone sulfatase (ES) from a proposed reaction mechanism.
Journal: Bioorganic & medicinal chemistry letters 20011203
Title: Steroid sulfatase in the human hair follicle concentrates in the dermal papilla.
Journal: The Journal of investigative dermatology 20011201
Title: Tibolone: a compound with tissue specific inhibitory effects on sulfatase.
Journal: Molecular and cellular endocrinology 20011025
Title: Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20010917
Title: Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20010409
Title: Novel inhibitors of the enzyme estrone sulfatase (ES).
Journal: Bioorganic & medicinal chemistry letters 20010326
Title: Non-steroidal and steroidal sulfamates: new drugs for cancer therapy.
Journal: Molecular and cellular endocrinology 20010122
Title: Synthesis and steroid sulphatase inhibitory activity of C19- and C21-steroidal derivatives bearing a benzyl-inhibiting group.
Journal: European journal of medicinal chemistry 20010101
