+1 858-523-8231
Login | Register
AA Blocks, Building Blocks, Catalysts, Inhibitors
Login | Register
Home Boronic Acids 1701434-52-7
1701434-52-7,MFCD18733399
Catalog No.:AA00ASPM

1701434-52-7 | 5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyrimidine

Pack Size
Purity
Availability
Price(USD)
Quantity
  
100mg
95%
in stock  
$142.00   $99.00
- +
250mg
95%
in stock  
$193.00   $135.00
- +
1g
95%
in stock  
$468.00   $328.00
- +
5g
95%
in stock  
$1,614.00   $1,130.00
- +
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
  • Request for Quotation
  • Download SDS
  • Technical Information
  • Properties
  • Downstream Synthesis Route
  • Literature
Technical Information
Catalog Number:
AA00ASPM
Chemical Name:
5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyrimidine
CAS Number:
1701434-52-7
Molecular Formula:
C11H14BF3N2O2
Molecular Weight:
274.0473
MDL Number:
MFCD18733399
SMILES:
FC(c1ncc(cn1)B1OC(C(O1)(C)C)(C)C)(F)F
Properties

Downstream Synthesis Route

[1]CurrentPatentAssignee:ROCHEHOLDINGAG-WO2015/52264,2015,A1Locationinpatent:Paragraph01873;01874

[2]CurrentPatentAssignee:BANTAMPHARMACEUTICALLLC-WO2016/196644,2016,A1Locationinpatent:Paragraph772;773

[3]CurrentPatentAssignee:BANTAMPHARMACEUTICALLLC-WO2018/102452,2018,A2Locationinpatent:Paragraph756;757

[4]CurrentPatentAssignee:EISAICOLTD-US2016/332999,2016,A1Locationinpatent:Paragraph0515;0516

[5]CurrentPatentAssignee:EISAICOLTD-EP3330266,2018,A1Locationinpatent:Paragraph0131

[6]Chen,Huifen;Volgraf,Matthew;Do,Steven;Kolesnikov,Aleksandr;Shore,DanielG.;Verma,VishalA.;Villemure,Elisia;Wang,Lan;Chen,Yong;Hu,Baihua;Lu,Ai-Jun;Wu,Guosheng;Xu,Xiaofeng;Yuen,Po-Wai;Zhang,Yamin;Erickson,ShawnD.;Dahl,Martin;Brotherton-Pleiss,Christine;Tay,Suzanne;Ly,JustinQ.;Murray,LesleyJ.;Chen,Jun;Amm,Desiree;Lange,Wienke;Hackos,DavidH.;Reese,RebeccaM.;Shields,ShannonD.;Lyssikatos,JosephP.;Safina,BrianS.;Estrada,AnthonyA.[JournalofMedicinalChemistry,2018,vol.61,#8,p.3641-3659]

[7]CurrentPatentAssignee:ROCHEHOLDINGAG-WO2016/128529,2016,A1Locationinpatent:Paragraph0727;0730;0731

[8]Han,Hua-Bo;Wu,Zheng-Guang;Zheng,You-Xuan[NewJournalofChemistry,2018,vol.42,#16,p.13351-13357]

98027-84-0   
5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyrimidine 
 
5-(2,6-dichloropyridin-4-yl)-2-(trifluoromethyl)pyrimidine 

[1]Patent:WO2015/52264,2015,A1.Locationinpatent:Paragraph02042;02043

[1]CurrentPatentAssignee:ROCHEHOLDINGAG-WO2015/52264,2015,A1Locationinpatent:Paragraph0894;0895

5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyrimidine 
  796851-03-1   
5-(2,5-dichloropyridin-4-yl)-2-(trifluoromethyl)pyrimidine 

[1]Patent:WO2018/15410,2018,A1.Locationinpatent:Paragraph0403-0406

[2]JournalofMedicinalChemistry,2018,vol.61,p.3641-3659

[3]Patent:WO2015/52264,2015,A1.Locationinpatent:Paragraph02066;02067

623585-74-0   
5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyrimidine 
 
methyl5-chloro-2-2-(trifluoromethyl)pyrimidin-5-ylpyridine-4-carboxylate 

[1]Patent:WO2015/52264,2015,A1.Locationinpatent:Paragraph01875;01876

Literature
Quotation Request
Company Name:
*
Contact Person:
*
Email:
*
Quantity Required:
*
Country:
Additional Info:
SDS
Related Products of 1701434-52-7
1025708-31-9

1025708-31-9

 1052686-67-5

1052686-67-5

 321724-19-0

321724-19-0

 1820679-54-6

1820679-54-6

 1235450-87-9

1235450-87-9
Building Blocks
More >
Tags:1701434-52-7 Molecular Formula|1701434-52-7 MDL|1701434-52-7 SMILES|1701434-52-7 5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyrimidine |Heterocyclic_Building_Blocks